| Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924) |
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| 09/28/2010 | CA2415475C Pyrrolo[2,1-b][1,3]benzothiazepines and their use for the preparation of medicaments with antipsychotic activity |
| 09/10/2010 | WO2010100623A1 Process for the preparation of quetiapine fumarate |
| 09/07/2010 | CA2485349C A11-piperazinyldibenzo (b, f) (1, 4) oxazepines and thiazepines as atypical antipsychotic agents having low affinity for the d2 receptor |
| 08/26/2010 | US20100216763 Heteroaryl Amide Derivatives |
| 08/18/2010 | EP1781646B1 PROCESS FOR THE PREPARATION OF 11-(4-[2-(2-HYDROXYETHOXY)ETHYL]-1-PIPERAZINYL)DIBENZO[b,f][1,4]THIAZEPINE |
| 08/12/2010 | US20100203135 Skin Equivalent Culture |
| 08/05/2010 | WO2010085976A1 Process for the synthesis of quetiapine |
| 07/21/2010 | CN101781271A Simple industrial technology for preparing diltiazem from chiral intermediates |
| 07/20/2010 | CA2431982C Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists |
| 06/24/2010 | WO2010070667A2 Novel process for the preparation of 7-((3-chloro-6-methyl-5,5-dioxo-6,11-dihydrodibenzo(c,f)(1,2) thiazepin-11-yl)amino)heptanoate |
| 06/24/2010 | US20100160627 (2,3-cis)-3-amino-2-phenyl-2,3-dihydro-1,5-benzoxazepin-4(5H)-one; for treatment of neurological disorders related to amyloid beta protein production such as Alzheimer's disease; inhibit gamma secretase and thereby inhibit the production of amyloid beta protein |
| 06/24/2010 | US20100160290 Pharmaceutical composition for treating alzheimer's disease |
| 06/17/2010 | US20100152440 NOVEL ANTI-ARRHYTHMIC AND HEART FAILURE DRUGS THAT TARGET THE LEAK IN THE RYANODINE RECEPTOR (RyR2) |
| 06/16/2010 | CN1872846B Method of preparing 2-benzothiazepines derivative |
| 06/16/2010 | CN101735211A Applications of 2,3-dihydro[1,5] benzothiazepine compounds or salts thereof in preparation of GSK-3beta inhibitor |
| 06/10/2010 | US20100144715 Substituted Benzodiazepinones, Benzoxazepinones and Benzothiazepinones as Sodium Channel Blockers |
| 06/03/2010 | WO2010062565A1 Muscarinic agonists |
| 06/03/2010 | WO2010042392A3 Hiv integrase inhibitors |
| 06/03/2010 | US20100137282 Tricyclic nitrogen containing compounds as antibacterial agents |
| 05/27/2010 | US20100130474 Alpha7 nicotinic acetylcholine receptor inhibitors |
| 05/12/2010 | EP1856073B1 A PROCESS FOR THE PREPARATION OF AN 11-(4-SUBSTITUTED-I-PIPERAZINYL)DIBENZO[b,f][1,4]THIAZEPINE DERIVATIVE |
| 05/12/2010 | CN101704799A Novel anti-arrhythmic and heart failure drugs that target the leak in the ryanodine receptor (RyR2) and uses thereof |
| 05/11/2010 | US7713966 Heterobicyclic metalloprotease inhibitors |
| 05/06/2010 | WO2010051239A1 Tianeptine sulfate salt forms and methods of making and using the same |
| 05/06/2010 | US20100112051 Tianeptine sulfate salt forms and methods of making and using the same |
| 04/27/2010 | US7704990 4-(Piperidinomethylaminosulfonyl),7-(methoxy-)-1,4-benzothiazepineprepared by the reaction of 7-(methoxy-)-1,4-benzothiazepine andpiperidinomethylaminosulfonyl chloride using a basic catalyst; ranodinereceptors that regulate calcium channel functioning in cells; skeletal muscular, cardiac disorders |
| 04/21/2010 | EP2177224A2 Agents for preventing and treating disorders involving modulation of the RyR receptors |
| 04/15/2010 | WO2010042392A2 Hiv integrase inhibitors |
| 04/15/2010 | WO2010042391A2 Hiv integrase inhibitors |
| 04/15/2010 | CA2738814A1 Hiv integrase inhibitors |
| 04/08/2010 | US20100087419 Hiv integrase inhibitors |
| 03/30/2010 | US7687622 Process for preparing quetiapine fumarate |
| 03/25/2010 | WO2010033270A1 Dibenzothiazepine modulators of dopamine, alpha adrenergic, and serotonin receptors |
| 03/24/2010 | CN101676275A preparation method of quetiapine fumarate |
| 03/18/2010 | US20100069356 Dibenzothiazepine modulators of dopamine, alpha adrenergic, and serotonin receptors |
| 03/16/2010 | US7678902 Reacting 2,2'-dithiosalicylic acid with 1-chloro-2-nitrobenzene in basic aqueous solution, conducting nitro group reduction reaction, simultaneously cyclizing and chlorinating in solvent, and halogenating; environmentally friendly, cost efficiency |
| 03/04/2010 | US20100056494 Purine compounds and compositions as kinase inhibitors for the treatment of plasmodium related diseases |
| 03/02/2010 | US7671195 Process for preparing dibenzothiazepine compounds |
| 02/25/2010 | WO2010021149A1 Spiro compound capable of inhibiting acid secretion |
| 02/18/2010 | US20100041638 Chemical Compounds 293 |
| 02/10/2010 | EP2151435A1 Pharmaceutical composition for treatment of alzheimer's disease |
| 02/09/2010 | CA2557576C Novel benzothiazepine and benzothiepine compounds |
| 02/04/2010 | US20100029612 2-Aminoethyl Substituted Pyrimidin-2-Ones Cyclopropanes, Pyrazolines, Pyrimidines and Benzothiazepines and Their Uses as Urotensin II and Somatostatin 5 Receptor Ligands |
| 01/28/2010 | US20100022513 Organic compounds |
| 01/28/2010 | US20100022509 Inhibitors of MshC and Homologs Thereof, and Methods of Identifying Same |
| 01/28/2010 | US20100022500 Macrocyclic Lactams and Pharmaceutical Use Thereof |
| 01/26/2010 | US7652003 Macrocyclic β-secretase inhibitors |
| 01/21/2010 | US20100016579 Crystalline forms of quetiapine hemifumarate |
| 01/20/2010 | EP2144892A2 Improved process for preparing quetiapine fumarate |
| 01/13/2010 | EP2035400B1 Method for the preparation of salts of 2-[2-(4-dibenzo[b,f][1,4]thiazepin-11-yl-1-piperazinyl)ethoxy]ethanol (quetiapine) |
| 01/06/2010 | EP1427713B1 Benzothiazepine derivatives for the treatment of hyperlipidemia |
| 01/06/2010 | CN101619047A Preparation process of quetiadine hemifumarate |
| 01/06/2010 | CN100577653C Process for producing dibenzo thionitrogen tropilidine derivative |
| 12/30/2009 | EP2137157A1 Polymorphs of 7-[(3-chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid s,s dioxide and methods of making and using the same |
| 12/23/2009 | WO2009154563A1 Dibenzothiazepine derivatives and use thereof |
| 12/23/2009 | EP1664007B1 Preparation of quetiapine |
| 12/23/2009 | CA2728675A1 Dibenzothiazepine derivatives and use thereof |
| 12/17/2009 | WO2009151392A1 Novel derivatives of 11-piperazin-l-yldibenzo [b,f] [1,4] thiazepine for treating at least one syndrome or condition associated with schizophrenia and other psychotic disorders |
| 12/16/2009 | CN100569761C Method for preparing pharmaceutical pure quetiapine fumarate |
| 12/02/2009 | EP2124908A1 Compounds and uses thereof |
| 12/01/2009 | US7625887 e.g. 2-[3,5-trans-5-(3-aminophenyl)-7-chloro-1-neopentyl-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]-N-(2-fluorobenzyl)acetamide; G-protein-coupled receptor (TGR5) agonist; central nervous system diseases; antiinflammatory agent; learning enhancement; angina pectoris, arrhythmia, bronchial asthma |
| 11/25/2009 | EP2120957A1 Compounds and uses thereof |
| 11/25/2009 | EP2120563A1 Compounds and uses thereof |
| 11/12/2009 | US20090281077 Cyclic sulfones useful as mitochondrial sodium-calcium exchangers |
| 11/10/2009 | US7615536 Hyperlipidemia, arteriosclerosis and hypercholesterolemia treatment |
| 11/05/2009 | WO2009004480A3 Quetiapine salts and their polymorphs |
| 11/03/2009 | US7612055 Macrocyclic lactams and pharmaceutical use thereof |
| 10/27/2009 | CA2415050C Process for the preparation of 9-amino substituted 9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepines |
| 10/20/2009 | CA2379294C Process for preparing dibenzothiazepine derivatives |
| 10/13/2009 | US7601695 11-N-[4-(4-Pyridin-3-yl-imidazol-1-yl)-butyl]-6-O-methyl-5-O-(3-dimethylamino-2-hydroxy-propoxy)-3-oxo-erythronolide A, 11,12-carbamate; functionalized macrolides; antiviral, antiprotozoal, anticancer and antigastrointestinal |
| 10/07/2009 | EP1000043B1 A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent |
| 10/06/2009 | US7598237 7-aryl 1,5-dihydro-4,1-benzoxazepin-2(3H)-one derivatives and their use as progesterone receptor modulators |
| 09/30/2009 | EP1243584B1 Cyanomethylene compounds, process for producing the same, and agricultural or horticultural bactericide |
| 09/16/2009 | EP2099459A1 Compounds and uses thereof |
| 09/11/2009 | WO2009111463A1 Process for preparing benzothiazepines from gamma-aminoalkylbenzenes |
| 09/11/2009 | CA2717523A1 Process for preparing benzothiazepines from .gamma.-aminoalkylbenzenes |
| 09/10/2009 | US20090227788 Process for preparing benzothiazepines from gamma-aminoalkylbenzenes |
| 08/20/2009 | US20090209593 Novel antibacterial agents |
| 08/19/2009 | CN101511804A Cyclic sulfones useful as mitochondrial sodium-calcium exchangers |
| 08/18/2009 | US7576198 A hydroxy compound containing substituted orpyridine, pyrazine, pyrimidine, oxazole, thiadiazole, quinoline, isoquinoline etc. as anti HIV agent, for treating AIDS |
| 08/06/2009 | WO2009095529A1 A process for the preparation of quetiapine |
| 08/06/2009 | CA2711395A1 A process for the preparation of quetiapine |
| 08/05/2009 | EP1742707A4 Treatment of cns disorders using cns target modulators |
| 08/05/2009 | EP1430040B1 Benzothiazepine derivatives |
| 08/05/2009 | CN101500576A Agents for preventing and treating disorders involving modulation of the RYR receptors |
| 07/28/2009 | US7566707 For example, 2-[3-(Tert-butyloxycarbonylamino)-piperidin-1-yl]-3-(2-butyn-1-yl)-5-[(dibenzo[b,f][1,4]-oxazepin-11-yl)methyl]-3,5-dihydro-imidazo[4,5-d]pyridazin-4-one; inhibiting effect on activity of the enzyme dipeptidylpeptidase-IV; use in treatment of diabetes mellitus, arthritis, obesity |
| 07/22/2009 | EP1567524B1 Thia-epothilone derivatives for the treatment of cancer |
| 07/22/2009 | CN100516022C Process for production of high-purity enamines |
| 07/21/2009 | US7563785 Quetiapine analogs and methods of use thereof |
| 07/09/2009 | US20090176993 (N-{5-[(4-chlorophenyl)thio]pentyl}-N-[(1R)-1-(1-naphthyl)ethyl]amine); mimics/blocks effect of extracellular calcium in parathyroid cells, juxtaglomerular/proximal tubule kidney cells, parafollicular thyroid cells, bone osteoclasts, keratinocytes or placental trophoblasts; hyperparathyroidism |
| 07/09/2009 | US20090176800 In vivo screening method of therapeutic agent for memory/learning dysfunctions by schizophrenia |
| 07/09/2009 | DE10297841B3 Preparation of diltiazem useful to treat angina involves synthesizing (2R,3S)-(-)-ethyl-2,3-dihydroxy-3-(4-methoxyphenyl)propionate using multifunctional catalyst, ring opening of the cyclic sulfite by 2-aminothiophenol and cyclization |
| 06/18/2009 | WO2009075691A1 Cb-1 modulating compounds and their use |
| 06/17/2009 | EP2069319A1 Cyclic sulfones useful as mitochondrial sodium-calcium exchangers |
| 06/11/2009 | US20090149442 Atypical antipsychotic agents having low affinity for the D2 receptor |
| 06/09/2009 | US7544678 Anti-arrythmic and heart failure drugs that target the leak in the ryanodine receptor (RyR2) |
| 06/03/2009 | CN100494185C Novel quaternary ammonium compounds |
| 05/27/2009 | EP0934287B1 Heterocyclic esters and amides |
| 05/27/2009 | CN100491333C Process for production of high-purity enamines |
| 05/19/2009 | CA2338651C Pyrrolo[2,1-b][1,3]benzothiazepines with atypical antipsychotic activity |