Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924) |
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09/05/2000 | US6114523 Process for the recycle of a waste product of diltiazem synthesis |
09/05/2000 | US6114322 Anticholesterol agent |
08/30/2000 | CN1265109A Thiazolobenzoheterocycles, prepn. and medicines containing same |
08/30/2000 | CN1265101A Crystalline dibentothiazepine derivatives and its use as antipsychotic agent |
08/23/2000 | EP1029071A1 Process for preparing (2r,3s)-3-(4-lower alkoxyphenyl)glycidic acid esters |
08/17/2000 | WO2000047568A2 1,2-benzothiazepines for the treatment of hyperlipidemic diseases |
08/17/2000 | CA2362147A1 1,2-benzothiazepines for the treatment of hyperlipidemic diseases |
08/09/2000 | EP1025080A1 Process for the recycle of a waste product of diltiazem synthesis |
08/03/2000 | WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS |
08/03/2000 | CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors |
07/26/2000 | EP1021190A1 Novel amide derivatives |
07/20/2000 | WO2000042031A2 Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
07/20/2000 | CA2359562A1 Substituted 2-arylimino heterocycles and compositions containing them, for use as progesterone receptor binding agents |
07/12/2000 | CN1054380C Condensed cyclic compounds and their use |
07/06/2000 | WO2000038728A1 Combinations of ileal bile acid transport inhibitors and bile acid sequestring agents for cardiovascular indications |
07/06/2000 | CA2356156A1 Combinations of ileal bile acid transport inhibitors and bile acid sequestring agents for cardiovascular indications |
07/05/2000 | EP0686151B1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors |
06/14/2000 | EP1007051A1 Integrin receptor antagonists |
05/17/2000 | EP1000067A1 Thiazolobenzoheterocycles, preparation and medicines containing same |
05/17/2000 | EP1000043A1 A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent |
05/17/2000 | CN1052479C Process for preparing 1,5-benzothiazepine derivatives |
05/10/2000 | CN1252795A 4,1-benzoxazepines, their analogues,and their use as somatostatin agonists |
04/27/2000 | WO2000023416A1 New compounds, their preparation and use |
04/13/2000 | WO2000020006A1 Use of diltiazem for treating retinal pathologies |
04/12/2000 | CN1051226C Preparation of medicine for treating imbalance of memory and recognition with tri-cyclic compound |
03/30/2000 | WO2000017384A1 Process for the enzymatic kinetic resolution of 3-phenylglycidates by transesterification with aminoalcohols |
03/29/2000 | EP0988297A2 Process for preparing optically active phenyloxirane compounds |
03/28/2000 | US6043361 Polymerisable monomers and polymers |
03/28/2000 | US6043358 Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases |
03/01/2000 | CN1245802A Preparation method of 1,5-benzothia azatropy lidene derivative |
02/23/2000 | EP0792268B1 Hypolipidemic benzothiazepines |
02/16/2000 | EP0979227A1 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists |
02/15/2000 | US6025506 Process for preparing an optically active phenylglycidyl acid derivative |
02/15/2000 | US6025355 Substituted indolinyl and derivatives thereof, neurological injury and neurodegenerative disorders. |
02/03/2000 | WO2000005246A1 Thioazepinone derivatives, preparation method and intermediates therefor, use as medicines and pharmaceutical compositions containing same |
02/01/2000 | US6020330 Hypolipidemic 1,4-benzothiazepine-1,1-dioxides |
01/19/2000 | CN1242007A Cycloalkyl, lactam lactone and related compounds as 'beta'-amyloid peptide release inhibitors |
01/19/2000 | CN1048484C A process for preparing a composition containing benzoheterocycles |
01/06/2000 | CA2330110A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors |
12/29/1999 | WO1999067230A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION |
12/29/1999 | WO1999067219A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
12/29/1999 | WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS |
12/29/1999 | CA2342778A1 Inhibitors of .alpha.4.beta.1 mediated cell adhesion |
12/29/1999 | CA2324475A1 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds |
12/29/1999 | CA2324474A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
12/28/1999 | US6008214 Inhibiting platelet aggregation and bone resorption, treating stroke, transient ischemia attacks, or myocardial infarction, treating osteoporosis |
12/22/1999 | EP0964682A1 A method of treating liver disease and like indications with vasodilating agents |
12/21/1999 | US6004948 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclooxygenase II |
12/16/1999 | WO1999063992A1 Novel calcium channel drugs and uses |
12/16/1999 | CA2318901A1 Novel calcium channel drugs and uses |
12/07/1999 | US5998637 Process for preparing optically active trans-3-substituted glycidic acid ester |
12/07/1999 | US5998400 Atherosclerosis |
11/18/1999 | WO1999058531A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors |
11/18/1999 | CA2330108A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors |
11/16/1999 | US5985869 Benzoheterocyclic compounds |
11/03/1999 | CN1233957A Pharmaceutical compositions |
10/27/1999 | EP0951466A2 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds |
10/20/1999 | CN1232457A 1,4-heterocyclic metalloprotease inhibitors |
10/19/1999 | US5968924 Benzo-fused lactams promote release of growth hormone |
10/13/1999 | CN1231661A Aralkyl and aralkylidene heterocyclic lactams and imides |
10/12/1999 | US5965553 Anticholesterol agents, hypotriglyceridemic agents, antiatherosclerosis agents, antifungal agents, alzheimer's agents or anti-acne agents |
10/06/1999 | EP0946180A1 Method for stimulating bone formation |
09/15/1999 | CN1228773A Heterocyclic metalloprotease inhibitors |
09/15/1999 | CN1228772A Heterocyclic metalloprotease inhibitors |
08/31/1999 | US5945533 Process for preparing optically active benzothiazepine compound and intermediate therefor |
08/18/1999 | CN1226164A Method for treating liver disease and like indications with vasodilating agent |
08/17/1999 | US5939412 Bicyclic fibrinogen antagonists |
08/12/1999 | WO1998008505A8 Pharmaceutical compounds |
08/11/1999 | EP0934065A1 Pharmaceutical compounds |
08/04/1999 | EP0933354A1 Calcium receptor-active compounds |
08/04/1999 | CN1225083A Calcium receptor-active compounds |
07/27/1999 | US5929069 Compounds activating pharmacological effects of retinoids |
07/27/1999 | US5929068 Intermediates for preparing diltiazem can be readily obtained without using an expensive optically active resolving agent |
07/21/1999 | EP0929528A1 Aralkyl and aralkylidene heterocyclic lactams and imides |
07/21/1999 | CN1044238C Method for preparing benzylidene derivatives |
07/15/1999 | WO1999035135A1 Hypolipidemic benzothiazepine compounds |
07/15/1999 | CA2317651A1 Hypolipidemic benzothiazepine compounds |
06/30/1999 | EP0925300A1 Pharmaceutically active compounds and methods of use |
06/30/1999 | EP0925287A1 Heterocyclic metalloprotease inhibitors |
06/23/1999 | EP0923563A1 1,4-heterocyclic metallprotease inhibitors |
06/23/1999 | EP0923561A1 Heterocyclic metalloprotease inhibitors |
06/22/1999 | US5914332 Retroviral protease inhibiting compounds |
06/08/1999 | US5910494 Hypolipidemic 1,4-benzothiazepine-1,1-dioxides |
05/06/1999 | WO1999022014A1 Process for preparing (2r,3s)-3-(4-lower alkoxyphenyl)glycidic acid esters |
05/04/1999 | CA2150766C Method for the manufacture of benzothiazepine derivatives |
04/29/1999 | WO1999020603A1 Process for the recycle of a waste product of diltiazem synthesis |
04/29/1999 | CA2304371A1 Process for the recycle of a waste product of diltiazem synthesis |
04/27/1999 | CA2087743C Pharmaceutical composition for inhibiting platelet aggregation |
04/15/1999 | WO1998038182A9 Hypolipidemic bicyclic derivatives |
04/14/1999 | EP0626952B1 Hypolipidaemic benzothiazepine compounds |
04/07/1999 | EP0906907A1 Compounds potentiating retinoid |
03/30/1999 | US5888542 Matrix tablet allowing the prolonged release of the sodium salt of tianeptine after administration by the oral route |
03/25/1999 | WO1998056762A3 Process for preparing optically active phenyloxirane compounds |
03/16/1999 | US5883264 Subjecting racemic trans-3-phenylglycidamide compound to optical resolution using a microorganism having ability of preferentially hydrolyzing one of (2s,3r) isomer or (2r,3s) isomer thereof |
03/09/1999 | US5880295 Process for the preparation of diamine intermediates useful in the synthesis of HIV protease inhibitors |
03/04/1999 | WO1999009991A1 Novel amide derivatives |
03/04/1999 | CA2301566A1 N-acylated lipophilic amino acid derivatives |
03/02/1999 | US5877170 Substitute caprolactams and derivatives thereof useful for treatment of HIV disease |
02/18/1999 | WO1999007875A1 Process for preparing (2r,3s)-3-(substituted or unsubstituted phenyl)glycidamide compounds by asymmetric amidation |
02/17/1999 | CN1208405A Retroviral protease inhibiting compounds |