| Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924) |
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| 12/25/2007 | US7312208 Quaternary ammonium compounds |
| 12/19/2007 | EP1347967B1 Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists |
| 12/19/2007 | CN101090894A Macrocyclic compounds and compositions useful as BACE inhibitors |
| 12/12/2007 | EP1863776A1 N-hydroxyamides omega-substituted with tricyclic groups as histone deacetylase inhibitors, their preparation and use in pharmaceutical formulations |
| 12/12/2007 | CN100354281C Process for preparation of 9-amino substituted 9,10-dihydropyrrolo [2,1-b] [1,3] benzotiazepines |
| 12/06/2007 | WO2006056772A3 Salts of quetiapine |
| 12/05/2007 | EP1861385A1 Novel anti-arrythmic and heart failure drugs that target the leak in the ryanodine receptor (ryr2) |
| 12/04/2007 | US7304047 Method of treating substance abuse with quetiapine |
| 11/22/2007 | WO2007062336A3 Salt forms |
| 11/22/2007 | US20070270402 (+) or (-)-9-(piperazin-1-yl)-9,10-dihydropyrrolo[2,1-b][1,3]benzothiazepine; schizophrenia, paranoid states, manic-depressive states, social regression, personality regression, hallucination, appetite disorders |
| 11/21/2007 | EP1856073A1 A PROCESS FOR THE PREPARATION OF AN 11-(4-SUBSTITUTED-I-PIPERAZINYL)DIBENZO[b,f][1,4]THIAZEPINE DERIVATIVE |
| 11/15/2007 | WO2007062338A3 Solid formulations |
| 11/14/2007 | EP1853569A1 Ligands for g-protein coupled receptors |
| 11/13/2007 | US7294622 Lactams and uses thereof |
| 10/25/2007 | US20070249582 Method of Treating Substance Abuse with Quetiapine |
| 10/24/2007 | EP1846382A2 Controlled release compositions comprising an antipsychotic agent |
| 10/18/2007 | WO2007117180A1 Azaheterocycles, combinatory library, focused library, pharmaceutical composition and methods for the production thereof |
| 10/17/2007 | EP1845089A1 Novel lactams and uses thereof |
| 10/11/2007 | WO2007008226A3 Palladium-catalyzed carbon-carbon bond forming reactions |
| 10/10/2007 | EP1841751A1 INDUSTRIAL PREPARATION OF 11-(4-(2-(2-HYDROXYETHOXY ETHYL)-1-PIPERAZINYL)DIBENZO (b,f)-1(1, 4)THIAZEPINE |
| 10/09/2007 | US7279582 For example (2S, 3S, 5S)-2-(2,6-dimethylphenoxyacetyl)amino-3-hydroxy-5-(2S-(1-tetrahydro-pyrimid-2-onyl)-3-methyl butanoyl)amino-1,6-diphenylhexane; HIV therapy |
| 10/09/2007 | US7279573 Benzodiazepine derivatives that may be fused to a pyrroline or piperidine ring; e.g., N-[1 (R)-(3-Aminopropylcarbamoyl)-2-(naphthalen-2-yl)ethyl]-3-(5,11-dioxo-2,3-dihydro-1H-(11aS)-pyrrolo[2,1-c][1,4]benzodiazepin-10-yl)propionamide; increasing levels of endogenous growth hormones in humans and animals |
| 10/04/2007 | WO2007111026A1 Optical film |
| 10/03/2007 | EP1838680A2 Macrocyclic compounds and compositions useful as bace inhibitors |
| 09/27/2007 | US20070225494 Process for the Preparation of 11-(4-[2-(2-Hydroxyethoxy)Ethyl]-I-Piperazinyl)Dibenzo[b,f][I,4]Thiazepine |
| 09/26/2007 | EP1554250B1 Novel lactams and uses thereof |
| 09/20/2007 | WO2007104933A1 Chemical compounds |
| 09/20/2007 | US20070219180 Muscle Relaxtion Accelerator and Therapeutic Agent for Muscular Tissue Diseases Such as Muscle Relaxation Failure |
| 09/13/2007 | WO2007101347A1 Bir domain binding compounds |
| 09/13/2007 | US20070213364 Alkoxyphenylpropanoic Acid Derivatives |
| 09/13/2007 | CA2642659A1 Process for preparing dibenzothiazepine compounds |
| 08/30/2007 | US20070203336 Process for preparing dibenzothiazepine compounds |
| 08/30/2007 | US20070203115 Novel quaternary ammonium compounds |
| 08/29/2007 | EP1660469B1 Process for the preparation of 11-(1-piperazinyl)dibenzo 'b, f! '1 ,4!-thiazepine, an intermediate in the synthesis of the antipsychotic drug quetiapine |
| 08/22/2007 | EP1819679A2 2-alcoxy-3,4,5-trihydroxy-alkylamides, preparation thereof, compositions containing them and use thereof |
| 08/16/2007 | US20070190041 Novel benzothiazepine and bensothiepine compounds |
| 08/01/2007 | EP1294698B1 Fused azepine derivatives and their use as antidiuretic agents |
| 07/18/2007 | EP1660468B1 Procedure for preparing 11-(4-[2-(2-hydroxyethoxy)ethyl]-1-piperazinyl)-dibenzo[b,f][1,4]thiazepine |
| 07/12/2007 | US20070160537 In vivo screening method of therapeutic agent for memory/learning dysfunctions by schizophrenia |
| 07/03/2007 | US7238686 stable, reproducible two crystalline forms; prepared by dissolving quetiapine free base and fumaric acid in suitable solvent and crystallizing fumarate salt; suitable solvents are ketones like acetone, methyl iso butyl ketone; esters like ethyl acetate, ethyl formate, methyl acetate; and mixture |
| 06/13/2007 | EP1795199A2 Quetiapine for the treatment of substance dependence or substance abuse |
| 06/13/2007 | EP1794137A2 Specific kinase inhibitors |
| 06/12/2007 | US7229984 Dibenzoxazepinone derivatives and uses thereof |
| 06/12/2007 | US7229983 antibacterial; beta -lactam antibiotics |
| 06/05/2007 | USRE39679 Substituted heterocycle fused gamma-carbolines |
| 05/24/2007 | US20070117787 N-[(3R,5S)-1-(3-Acetoxy-2,2-dimethylpropyl)-7-chloro-5-(2,3-dimethoxyphenyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetyl]piperidine-4-acetic acid; in combination with a statin, lowering cholesterol-level and lowering triglyceride-level |
| 05/17/2007 | US20070111987 cyclization using phosphorus oxychloride; antipsychotic or neuroleptic agent for psychological disorders |
| 05/17/2007 | US20070111986 comprises the ring closure and deprotection of an intermediate; 11-(4-[2-(2-hydroxyethoxy)ethyl]-1-piperazinyl]dibenzo[b,f]-1,4-thiazepine; used as an antipsychotic or neuroleptic |
| 05/09/2007 | EP1781646A1 Process for the preparation of 11-(4-[2-(2-hydroxyethoxy)ethyl]-i-piperazinyl)dibenzo[b,f][1,4]thiazepine |
| 05/08/2007 | US7214793 Reacting dithiodisalicylic acid with 1-chloro-2-nitrobenzene in a basic aqueous solution; reducing the nitro group of the 2-(2-nitrophenylthio)benzoic acid formed with hydrogen gas, a solvent and a heterogeneous metal catalyst; and cyclizing the product in an organic solvent |
| 05/08/2007 | CA2342950C New process for preparing 11-amino-3-chloro-6,11-dihydro-5,5-dioxo-6-methyl-dibenzo[c,f][1,2]-thia zepine and application in the synthesis of tianeptine |
| 05/03/2007 | WO2007049532A1 Aminodihydrothiazine derivative |
| 05/03/2007 | WO2007048870A1 Quetiapine hemifumarate purification by crystallization |
| 05/03/2007 | US20070099848 Rapamycin carbohydrate derivatives |
| 05/03/2007 | CA2628074A1 Aminodihydrothiazine derivative |
| 04/26/2007 | WO2007047737A1 Cb-1 modulating compounds and their use |
| 04/26/2007 | CA2625423A1 Cb-1 modulating compounds and their use |
| 04/25/2007 | EP1776160A1 Novel serotonin receptor ligands and their uses thereof |
| 04/25/2007 | EP1359919B1 Use of quetiapine for the treatment of cocaine dependence |
| 04/19/2007 | WO2007009656A3 Novel 1,4-benzothiazepine-1,1-dioxide derivative having improved properties, method for the production thereof, medicaments containing said compound, and use thereof |
| 04/19/2007 | US20070088020 Agonists to a cannabinoid type 2 receptor; antiinflammatory agents; immunosuppressants; nephritis |
| 04/18/2007 | EP1345918B1 1,5 benzothiazepines and their use as antihyperlipidemics |
| 04/17/2007 | US7205334 vacuolar-type (H+)-ATPase-inhibiting macrocyclic lactams belonging to the chondropsin class useful in cancer chemotherapy |
| 04/17/2007 | CA2295792C A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent |
| 04/10/2007 | US7202256 Proline CCI-779, production of and uses therefor, and two-step enzymatic synthesis of proline CCI-779 and CCI-779 |
| 04/05/2007 | WO2007036599A1 New crystallization process of quetiapine hemifumarate |
| 04/04/2007 | CN1308313C Fused azepine drivatives and their use as antidiuretic agents |
| 03/29/2007 | US20070072792 Macrocyclic lactams and pharmaceutical use thereof |
| 03/22/2007 | US20070066589 Method of preparing 10th-dibenzo[b,f][11,4]thiazepin-11-one |
| 03/20/2007 | US7192950 Psychological disorders; eating disorders; dietetics |
| 03/20/2007 | US7192948 Bicyclic heterocycles as HIV integrase inhibitors |
| 03/20/2007 | US7192947 Peptides derivatives comprising thiazepine group for the treatment of hyperlipidemic conditions |
| 03/20/2007 | US7192946 Hyperlipemia agents; bile acid transport inhibitors |
| 03/20/2007 | US7192945 Benzothiazepine derivatives |
| 03/13/2007 | CA2264063C Cryptophycin compounds |
| 03/07/2007 | CN1923794A Process for production of high-purity enamines |
| 03/01/2007 | WO2006117700A3 Process for preparing quetiapine and quetiapine fumarate |
| 03/01/2007 | WO2005030711A3 Bridged macrocyclic module compositions |
| 02/22/2007 | WO2007020011A1 Processes for the preparation of thiazepines |
| 02/22/2007 | WO2006081347B1 Controlled release compositions comprising an antipsychotic agent |
| 02/14/2007 | EP1751168A1 Proline cci-779 (proline-rapamycin 42-ester with 2,2-bis (hydroxymethyl) propionic acid) and two-step enzymatic synthesis of proline cci-779 and cci-779 using microbial lipase |
| 02/14/2007 | CN1914214A Tricycle indole hydroxyethlamine derivatives and their use in the treatment of alzheimer's disease |
| 02/13/2007 | US7176195 Treatment of nocturnal enuresis, nocturia, polyuria resulting from central diabetes insipidus, urinary incontinence or bleeding disorders such a hemophilia |
| 02/07/2007 | CN1907977A Process for preparing diltiazem intermediate |
| 02/01/2007 | WO2006049734A3 Quetiapine analogs and methods of use thereof |
| 01/25/2007 | WO2007009655A1 1,4-benzothiazepine 1,1-dioxide derivative, process for its preparation, medicaments comprising this compound, and use thereof as a hypolipidaemic |
| 01/25/2007 | DE102005033100B3 Neues 1,4-Benzothiazepin-1,1-Dioxidderivat mit verbesserten Eigenschaften, diese Verbindung enthaltene Arzneimittel und Verfahren zu deren Herstellung New 1,4-benzothiazepine-1,1-Dioxidderivat with improved properties, these drug compound contained and processes for their preparation |
| 01/25/2007 | CA2614697A1 Novel 1,4-benzothiazepine-1,1-dioxide derivative having improved properties, method for the production thereof, medicaments containing said compound, and use thereof |
| 01/25/2007 | CA2614524A1 1,4-benzothiazepine 1,1-dioxide derivative, process for its preparation, medicaments comprising this compound, and use thereof as a hypolipidaemic |
| 01/24/2007 | CN1902182A Macrocyclic lactams and pharmaceutical use thereof |
| 01/17/2007 | EP1743895A1 Muscle relaxation accelerator and therapeutic agent for muscular tissue diseases such as muscle relaxation failure |
| 01/17/2007 | EP1742707A2 Treatment of cns disorders using cns target modulators |
| 01/11/2007 | WO2007004234A1 A PROCESS FOR THE PREPARATION OF 2-[2-(4-DIBENZO[b,f] [L,4] THIAZEPIN-11-yl-1- PIPERAZINYL)ETHOXY] ETHANOL FUMARATE |
| 01/09/2007 | CA2394720C Cyanomethylene compounds and fungicidal compositions |
| 12/28/2006 | WO2006081347A3 Controlled release compositions comprising an antipsychotic agent |
| 12/27/2006 | EP1427423B1 Benzothiazepine and benzothiadiazepine derivatives with ileal bile acid transport (ibat) inhibitory activity for the treatment hyperlipidaemia |
| 12/21/2006 | WO2006135544A1 SYNTHESIS OF 11-(4[-(2-HYDROXYETHOXY)ETHYL]-PIPERAZINYL)-DIBENZO[b,f][1,4]THIAZEPINE AND ITS FUMARATE SALT |
| 12/13/2006 | EP1731505A1 Alkoxyphenylpropanoic acid derivatives |
| 12/06/2006 | EP1345610B1 Quetiapine for treating of dyskinesia in non-psychotic patients |
| 12/06/2006 | CN1872846A Method of preparing 2-benzothiazepines derivative |