Patents
Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924)
01/1995
01/03/1995US5378698 Benzothiazepine derivatives
12/1994
12/28/1994CN1096782A Process for preparation benzothiazepine derivatives
12/22/1994WO1994029286A1 Analgesic dibenzoxazepines and dibenzothiazepines
12/22/1994WO1994028901A1 Amino acid derivative
12/22/1994CA2165159A1 Analgesic dibenzoxazepines and dibenzothiazepines
12/22/1994CA2140553A1 Amino acid derivative
12/07/1994EP0626952A1 Hypolipidaemic benzothiazepine compounds
11/1994
11/30/1994EP0626377A1 Method for producing benzylidene derivatives
11/24/1994WO1994026719A1 Mercapto-amide derivatives useful as neutral endopeptidase and ace inhibitors
11/23/1994EP0549666B1 Novel aminobenzosultam derivatives as lipoxygenase inhibitors
11/16/1994CN1026585C Preparation of aryltrioxalone
11/08/1994CA1332943C Process for preparing perhydrothiazepine derivatives
10/1994
10/13/1994WO1994022840A1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease
10/13/1994CA2159442A1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease
10/11/1994US5354747 2-, 3-, 4-, 5-, 6-, 7-, 8-, 9- and/or 10-substituted dibenzoxazepine and dibenzthiazepine compounds, pharmaceutical compositions and methods of use
09/1994
09/21/1994EP0615971A1 5-(Piperazinylalkyl)-1,5-benzothiazepinones useful as calcium antagonists
09/20/1994US5348965 N-substituted azaheterocyclic carboxylic acids
09/07/1994EP0613472A1 10-acyl-dibenz(b,f) (1,4)-oxazepines and their thiazepines analo gues useful as prostaglandin antagonists
09/06/1994US5344828 Piperazinealkanoic acid and a pharmaceutical composition comprising the same
09/01/1994WO1994019329A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
08/1994
08/31/1994EP0612737A1 Process for preparing 1,5-benzothiazepine derivatives
08/18/1994WO1994018184A1 Hypolipidaemic compounds
08/18/1994WO1994018183A1 Hypolipidaemic condensed 1,4-thiazepines
08/18/1994CA2156184A1 Hypolipidaemic condensed 1, 4-thiazepines
08/18/1994CA2156183A1 Hypolipidaemic compounds
08/03/1994EP0609031A1 Process for preparing benzothiazepine derivatives
07/1994
07/28/1994CA2114036A1 Process for preparing benzothiazepine derivatives
07/13/1994EP0357750B1 Urethane-protected amino acid-n-carboxyanhydrides
06/1994
06/28/1994US5324722 2-, 3-, 5-, 8-, 10- and/or 11-substituted dibenzoxazepine compounds, pharmaceutical compositions and methods for treating pain
06/23/1994WO1994013828A1 Chiral arylpropionates and their use
06/23/1994WO1994013651A1 Benzazepinone derivatives
06/23/1994CA2151384A1 Benzazepinone derivatives
06/01/1994EP0599444A1 Dual action inhibitors
06/01/1994CN1087338A Therapeutic agents
05/1994
05/31/1994US5317017 N-biphenyl-3-amido substituted benzolactams stimulate growth hormone release
05/26/1994WO1994011360A1 1,4-benzothiazepines useful as neurological agents
05/26/1994CA2148584A1 Therapeutic agents
05/24/1994US5315005 Process for the single crystallization of enatiomeric ratio's (2S,3S):(2R,3R) of substituted 1,5-benzothiazepinone
05/17/1994US5312625 Fused 7-membered cyclic compound and antipsychotic preparation containing the same
05/10/1994US5310904 Process for preparing optically active benzothiazepine compounds by asymmetric reduction
05/10/1994US5310737 Benzo-fused lactams that promote the release of growth hormone
05/03/1994CA1329214C 2-hydroxy-3-(4-methoxyphenyl)-3-(2- aminophenylthio)propionic acid, 8'-phenylmenthyl ester, especially for diltiazem
04/1994
04/28/1994WO1994008977A1 Substituted caprolactams and derivatives thereof useful for treatment of aids
04/27/1994EP0594101A1 A process for the preparation of diltiazem
04/27/1994EP0593603A1 Bicyclic fibrinogen antagonists
04/24/1994CA2108950A1 A process for the preparation of diltiazem
04/14/1994WO1994007483A1 Benzo-fused lactams promote release of growth hormone
04/14/1994CA2142974A1 Benzo-fused lactams promote release of growth hormone
04/06/1994CN1084849A Dual action inhibitors
04/05/1994US5300522 Condensed heterocyclic compounds and pharmaceutical use thereof
03/1994
03/17/1994WO1994005634A1 Benzo-fused lactams promote release of growth hormone
03/15/1994US5294706 Process for preparing 1,5-benzothiazepine derivatives
03/09/1994CN1083485A Benzothiazepine and benzoxazepine derivatives
02/1994
02/23/1994EP0583408A1 Substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
02/23/1994EP0583317A1 Dibenzothiazepinthione as antiviral agents
02/23/1994EP0583288A1 Antivizal dibenzothiazepinone derivatives
02/15/1994CA1327006C Process for preparing a retard product containing diltiazem for a single daily administration
02/01/1994US5283241 Animal growth regulators
02/01/1994US5283240 Administering prostaglandin antagonists
01/1994
01/25/1994US5281590 2-H and 3-alkoxy or hydroxy-8-substituted-dibenz[b,f]-[1,4]oxazepine-10(11)-carboxylic acid, substituted hydrazides for the treatment of osteoporosis
01/20/1994WO1994001421A1 Benzothiazepine and benzoxazepine derivatives as cholecystokinin receptor antagonists
01/20/1994CA2139417A1 Benzothiazepine and benzoxazepine derivatives
01/05/1994CN1023399C Preparation of 8-substituted-2-aminotetralines
12/1993
12/28/1993US5274300 Enzymatic hydrolysis of glycidate esters in the presence of bisulfite anion
12/23/1993CA2112360A1 Bicyclic fibrinogen antagonists
12/08/1993EP0368994B1 Benzothiazepines for the preparation of medicaments for the amelioration of epileptic seizures
10/1993
10/19/1993US5254682 Cyclic renin inhibitors containing 3(S)-amino-4-cyclohexyl-2(R)-hydroxy-butanoic acid or 4-cyclo-hexyl-(2R, 3S)-dihydroxybutanoic acid or related analogs
10/13/1993CN1022412C Method for preparing urethane-protected amino acid-N-carboxyanhydrides
10/05/1993US5250680 Heterogeneous synthesis of azepinones from esters
09/1993
09/29/1993EP0561861A1 A process for the preparation of diltiazem.
09/14/1993US5244803 Stereoselective hydrolysis by microorganism in culture
09/07/1993US5242912 Cyclic anthranilic acid derivatives and process of preparing the same
08/1993
08/19/1993WO1993016055A1 Hypolipidaemic benzothiazepine compounds
08/19/1993CA2117485A1 Hypolipidaemic benzothiazepine compounds
08/18/1993EP0294375B1 Herbicidal aryl triazolinones
08/18/1993CN1021821C Aryl triazolineone herbicide
08/11/1993EP0555042A1 Pharmaceutical composition for inhibiting platelet aggregation
08/10/1993CA1321280C Urethane-protected amino acid-n-carboxyanhydrides
07/1993
07/14/1993EP0551076A1 Process for preparing optically active benzothiazepine compounds by asymmetric reduction
07/11/1993CA2086862A1 Process for preparing optically active benzothiazepine compounds by asymmetric reduction
07/08/1993WO1993013082A1 Substituted dibenzoxazepines or dibenzothiazepines and their use as prostaglandin e2 antagonists
07/06/1993US5225557 Process for making optically active naphtho[1,2-b]thiazepin-4(5H)-ones
06/1993
06/29/1993US5223612 Process for the preparation of benzothiazepines by cyclization with phosphonic acids
06/22/1993CA1319364C Fused heterocyclic compounds
06/16/1993CN1073168A Benzothiazepine derivatives
06/02/1993CN1021047C 1,5-benzothiazepine derivative and preparation thereof
05/1993
05/19/1993CN1020726C Process for preparing cyclic compounds containing sulfur
05/13/1993WO1993009104A1 10-acyl-dibenz(b,f) (1,4)-oxazepines and their thiazepines analo gues useful as prostaglandin antagonists
05/13/1993CA2118688A1 Substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
05/12/1993EP0541263A1 5-piperazinylalkyl-1,5-benzothiazepinones useful as calcium antagonists
05/12/1993CN1020605C Process for preparing azacycloparaffin derivatives
05/11/1993CA1317593C Method of ameliorating epileptic seizures
04/1993
04/28/1993CN1071333A Calcium receptor active molecules
04/27/1993US5206235 Animal growth regulators; stimulants
04/27/1993US5206233 Substituted thiazepines as central nervous system agents
04/22/1993CA2080671A1 Benzothiazepine derivatives
04/15/1993WO1993007132A1 10-acyl-dibenz(b,f)(1,4)-oxazepines and their thiazepines and diazepines analogues useful as prostaglandin antagonists
03/1993
03/30/1993US5198557 Reaction with mercapto compound for cardiovascular disorders
03/16/1993US5194605 Cyclic renin inhibitors containing 2-substituted (3S,4S)-4-amino-5-cyclohexyl-3-hydroxy pentanoic acid, 2-substituted (3S,4S)-5-cyclohexyl-3,4-di-hydroxy pentanoic acid or 2-substituted (4S,5S)-5-amino-6-cyclohexyl-4-hydroxyhexanoic acid or its analogs
03/04/1993WO1993004373A1 Calcium receptor active molecules
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