Patents
Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924)
02/1999
02/11/1999WO1999006381A1 A crystalline dibenzothiazepine derivative and its use as an antipsychotic agent
02/11/1999WO1999006049A1 Integrin receptor antagonists
02/11/1999CA2298544A1 Integrin receptor antagonists
02/10/1999CN1207681A Sustained-release microgranules contg. diltiazem as active principle
02/09/1999US5869697 Process for preparing diltiazem
02/09/1999US5869483 Tricyclic benzazepine vasopressin antagonists
02/04/1999WO1999005147A1 Thiazolobenzoheterocycles, preparation and medicines containing same
01/1999
01/12/1999US5859241 Process for the preparation of a benzothiazepine
01/12/1999US5859240 Reduction of imine group; oxidation; salt formation
01/12/1999US5859239 Mercaptoalkanoylamino and acylmercaptoalkanoylamino benzoxazepines and benzothiazepines
01/05/1999US5856477 Hypotensive agents; congestive heart failure
01/05/1999US5856476 Processes for preparing azepiones useful as intermediates in the preparation of inhibitors of angiotensin converting enzyme and neutral endopeptidase
12/1998
12/29/1998US5854274 Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives
12/29/1998US5854236 Tricyclic benzazepine vasopressin antagonists
12/29/1998US5854233 Method of treating liver disease and like indications with vasodilating agents
12/17/1998WO1998056762A2 Process for preparing optically active phenyloxirane compounds
12/17/1998CA2293404A1 Process for preparing optically active phenyloxirane compounds
12/16/1998CN1202160A Compounds potentiating retinoid
12/09/1998EP0882024A1 Retroviral protease inhibiting compounds
12/08/1998US5847122 Process for preparing 1,5-benzothiazepine derivative
12/08/1998US5846969 Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives
12/08/1998US5846967 Natriuretic and anti-hypertensive compounds
12/01/1998US5843952 Tricyclic benzazepine vasopressin antagonists
11/1998
11/25/1998CN1199733A Process for preparing optically active trans-3-substituted glycidic acid ester
11/18/1998CN1040751C Process for preparation of benzothiazepine derivs.
11/10/1998US5834462 Antitumor agents; anticarcinogenic agents particularly for nasopharyngel, pulmonary, intestinal, mammary, uterus, gastric, ovarian or liver cancer and also leukemia
10/1998
10/29/1998WO1998047882A1 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists
10/29/1998CA2285664A1 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists
10/28/1998CN1197070A Process for preparing optically active phenylglycidyl acid derivative
10/08/1998WO1998028268A3 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS
10/07/1998EP0868184A1 Sustained-release microgranules containing diltiazem as the active principle
10/07/1998CN1194979A Hypolipidemic 1,4-benzothiazepine-1, 1-dioxides
10/06/1998US5817653 Endothelin receptor antagonists
10/06/1998US5817652 Hypolipidaemic condensed 1,4-thiazepines
09/1998
09/24/1998WO1998041510A1 Novel benzolactam derivatives and medicinal compositions comprising the same
09/22/1998US5811422 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
09/16/1998EP0864582A2 Hypolipidemic 1,4-benzothiazepine-1,-dioxides
09/03/1998WO1998038182A1 Hypolipidemic bicyclic derivatives
09/02/1998EP0861834A1 Process for preparing optically active trans-3-substituted glycidic acid ester
09/02/1998EP0861250A1 Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase
09/02/1998EP0861238A1 Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases
08/1998
08/27/1998CA2230299A1 Process for preparing optically active trans-3-substituted glycidic acid ester
08/26/1998EP0860439A1 Process for preparing an optically active phenylglycidyl acid derivative
08/21/1998CA2228196A1 Process for preparing an optically active phenylglycidyl acid derivative
08/20/1998WO1998035941A1 New benzolactam derivatives and medicinal compositions containing the same
08/20/1998WO1998035939A1 Malonic diamide derivatives and use thereof
08/19/1998EP0858999A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
08/18/1998CA2037298C Processes for preparing 1,5-benzothiazepine derivatives
07/1998
07/28/1998US5786353 Tricyclic benzazepine vasopressin antagonists
07/14/1998CA2025226C Process for preparing optically active 3-phenylglycidic acid esters
07/08/1998CN1039008C Dual action inhibitors in angiotensin invertase and neutral endopeptidase
07/02/1998WO1998028268A2 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS
07/02/1998CA2272305A1 Cycloalkyl, lactam, lactone and related compounds as .beta.-amyloid peptide release inhibitors
06/1998
06/24/1998EP0848703A1 Derivatives of benzosulphonamides as inhibitors of the enzyme cyclo-oxygenase ii
06/23/1998US5770594 Naphthyl-benzoxazepines or -benzothiazepines as squalene synthetase inhibitors
06/16/1998CA2042535C Process for the preparation of intermediates useful for the synthesis of benzothiazepines
06/02/1998US5760221 Subjecting 1,8-dicarboxylic acid ester to dieckmann condensation reaction
06/02/1998US5760031 Kidney diseases
05/1998
05/19/1998US5753642 Agriculture, medicine
05/05/1998US5747487 Tricyclic benzazepine vasopressin antagonists
04/1998
04/16/1998WO1998015278A1 Method for stimulating bone formation
04/15/1998EP0799220A4 Polymerisable monomers and polymers
04/14/1998US5739128 Administering for treatment of diseases characterized by excess renal reabsorption of water
04/09/1998WO1998014433A1 Aralkyl and aralkylidene heterocyclic lactams and imides
04/07/1998US5736538 Treats in mammal the disease characterized by excess renal reabsorption of water, is congestive heart failure, nephrotic syndrome, hyponatremia, coronary and renal vasospasm, cardiac ischemia, liver cirrhosis and brain edema
04/01/1998EP0832879A1 Process for preparing intermediates for thrombin inhibitors
03/1998
03/20/1998CA2185950A1 Process for preparing intermediates for thrombin inhibitors
03/11/1998EP0667866B1 1,4-benzothiazepines useful as neurological agents
03/05/1998WO1998008827A1 Heterocyclic metalloprotease inhibitors
03/05/1998WO1998008825A1 1,4-heterocyclic metalloprotease inhibitors
03/05/1998WO1998008823A1 Heterocyclic metalloprotease inhibitors
03/05/1998WO1998008505A1 Pharmaceutical compounds
03/05/1998CA2264045A1 Heterocyclic metalloprotease inhibitors
03/05/1998CA2263932A1 1,4-heterocyclic metalloprotease inhibitors
03/05/1998CA2263917A1 Heterocyclic metalloprotease inhibitors
03/04/1998EP0826678A1 Process for preparing optically active benzothiazepine compound, and intermediate therefor
03/04/1998CN1174837A Process for preparing optically active benzothiazepine compound, and intermediate therefor
03/03/1998US5723602 Angiotensin converting enzyme and endopeptidase inhibitors, cardiovascular disorders
03/03/1998US5723458 1,4-benzothiazepines
03/03/1998US5723457 Acylmercaptoalkanoylamino and mercaptoalkanoylamino benzazepines
02/1998
02/12/1998WO1998005657A1 2,3-dihydro-1,4-benzothiazepines, their preparation and their use as intermediates
01/1998
01/15/1998WO1998001417A1 Calcium receptor-active compounds
01/15/1998WO1998001164A1 Tricyclic radiolabeled d4 receptor ligands
01/06/1998US5705638 Process for preparing optically active 3-hydroxy-1,5-benzothiazepine derivative and intermediate therefor
12/1997
12/31/1997CN1168878A Process for preparing optically active 2-halogeno-3-hydroxypropionic acid ester
12/31/1997CN1168792A Matrix table allowing prolonged release of sodium salt of tianeptine after administration by oral route
12/30/1997CA2142707C Benzo-fused lactams promote release of growth hormone
12/29/1997EP0814080A1 Squalene synthetase inhibitors
12/24/1997WO1997048396A1 A method of treating liver disease and like indications with vasodilating agents
12/24/1997CA2258696A1 A method of treating liver disease and like indications with vasodilating agents
12/20/1997CA2208174A1 Squalene synthetase inhibitors
12/18/1997WO1997047625A1 Tricyclic benzazepine vasopressin antagonists
12/16/1997US5698691 Condensed cyclic compounds and their use
12/02/1997US5693636 Bicyclic fibrinogen antagonists
12/02/1997US5693635 Tricyclic benzazepine vasopressin antagonists
11/1997
11/26/1997EP0808824A2 Process for preparing optically active 2-halogeno-3-hydroxypropionic acid ester
11/12/1997CN1164856A Novel alkylamino derivatives as sigma 2 selective ligands
11/11/1997US5686445 Pyridobenzoxazepine and pyridobenzothiazepine vasopressin antagonists
11/05/1997CN1164230A Hypolipidemic benzothiazepines
10/1997
10/29/1997EP0803253A1 Matrix-type oral sustained-release tablets containing tianeptine sodium salt
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