Patents for C07D 281 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms (1,924) |
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10/26/2012 | CA2833320A1 Dibenzothiazepine derivatives and their use in the treatment of cns disorders |
10/17/2012 | CN101891707B Method for preparing Quetiapine or pharmaceutically acceptable fumarate thereof |
10/10/2012 | EP2508515A1 Ligands for g-protein coupled receptors |
09/19/2012 | CN102686602A Lanthionine derivative |
08/02/2012 | WO2012063085A3 Drug derivatives |
07/11/2012 | CN102558093A Agents for preventing and treating disorders involving modulation of the ryr receptors |
06/12/2012 | US8198268 Tianeptine sulfate salt forms and methods of making and using the same |
05/30/2012 | CN101337948B 1,5-benzothiazepines compounds, preparation method and application thereof |
05/18/2012 | CA2816000A1 Drug derivatives |
05/16/2012 | CN1854128B Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds |
05/10/2012 | US20120114588 Ibat inhibitors for treatment of metabolic disorders and related conditions |
05/02/2012 | CN102432562A Quetiapine fumarate compound and new preparation method thereof |
04/25/2012 | EP1719768B1 Novel benzothiazepine and benzothiepine compounds |
04/24/2012 | US8163730 Fused tricyclic compounds as inhibitors of tumor necrosis factor-alpha |
04/17/2012 | US8158618 Dibenzothiazepine derivatives and uses thereof—424 |
03/28/2012 | CN102391208A New crystal form I of quetiapine fumarate and preparation method thereof |
03/27/2012 | US8143242 Malonamide derivatives with antithrombotic activity |
03/22/2012 | US20120071429 Novel antibacterial agents |
02/23/2012 | US20120046198 Ligand Libraries for Screening GPCRs |
02/02/2012 | US20120029188 Substituted Aniline Derivatives |
01/31/2012 | US8106023 1,4-benzothiepin-1, 1-dioxide derivatives with improved properties method for producing the same, drugs containing said compounds and the use thereof |
01/26/2012 | US20120022249 Aminodihydrothiazine derivatives |
01/24/2012 | US8101597 Quetiapine salts and their polymorphs |
01/24/2012 | US8101583 1,4-benzothiepin-1,1-dioxide derivatives which are substituted with fluorine, method for producing the same, drugs containing said compounds and use thereof |
01/19/2012 | US20120016116 Aminodihydrothiazine derivatives |
01/19/2012 | US20120015925 Novel benzothiazepine and benzothiepine compounds |
01/11/2012 | EP2403841A1 Process for the preparation of quetiapine fumarate |
12/28/2011 | CN102293773A 含有苯并硫氮杂卓和苯并虑平化合物的药物 Benzothiazepine and benzo drugs containing compounds doxepin |
12/07/2011 | EP2392567A1 Benzothiazine derivatives and their use as lxr modulators |
12/07/2011 | EP2250159B1 Process for preparing benzothiazepines from gamma-aminoalkylbenzenes |
11/29/2011 | US8067585 Photocoupling; cyclization and sulfonimidation of disulfonyl fluoride compound by reaction with ammonia; heating, alkylation, electrolysis, quaternization, salt formation; chemical intermediates |
11/29/2011 | US8067584 Benzothiazepine derivatives |
11/22/2011 | US8063037 Progesterone receptor modulators |
11/03/2011 | US20110269743 Phenylthiophenyldihydrobenzothiazepine inhibitors of store operated calcium release |
11/03/2011 | CA2795543A1 Chemical compounds |
11/02/2011 | EP1535913B1 Novel quaternary ammonium compounds |
11/01/2011 | US8048876 Process for preparing quetiapine and quetiapine fumarate |
10/25/2011 | US8044039 Quetiapine hemifumarate purification by crystallization |
10/25/2011 | US8044038 Crystallization process of quetiapine hemifumarate |
10/13/2011 | WO2011126071A1 Agent for inhibiting viral infection and/or treating infectious disease, and method for inhibiting viral infection and/or treating infectious disease |
10/11/2011 | US8034805 Methods for the preparation of salts of 2-[2-(4-dibenzo[B,F][1,4]thiazepin-11-yl-1-piperazinyl)ethoxyl]ethanol (quetiapine) and for the purification thereof |
10/06/2011 | WO2011121602A1 Process for preparation of dibenzothiazepinone compounds |
10/05/2011 | CN102206195A Crystalline quetiapine fumarate and pharmaceutical compositions thereof |
09/28/2011 | EP2367806A2 Process and intermediates for the preparation of 7-((3-chloro-6-methyl-5,5-dioxo-6,11-dihydrodibenzo(c,f)(1,2) thiazepin-11-yl)amino)heptanoate |
09/21/2011 | CN101360725B Solid formulations |
09/20/2011 | US8022203 Amino derivatives of beta-homoandrostanes and beta-heteroandrostanes |
09/20/2011 | US8022059 Indazole acrylic acid amide compound |
09/20/2011 | US8022058 Agents for preventing and treating disorders involving modulation of the RyR receptors |
09/20/2011 | CA2115828C Calcium receptor active molecules |
09/09/2011 | WO2011107248A1 NOVEL COMPOUNDS FOR MODULATION OF ORPHAN NUCLEAR RECEPTOR RAR-RELATED ORPHAN RECEPTOR-GAMMA (RORγ GAMMA, NR1F3) ACTIVITY AND FOR THE TREATMENT OF CHRONIC INFLAMMATORY AND AUTOIMMUNE DISEASE |
09/06/2011 | US8012943 Antibacterial agents |
08/24/2011 | CN102161644A Ligands for g-protein coupled receptors |
08/18/2011 | WO2010070510A3 A process for preparing quetiapine fumarate |
08/17/2011 | EP2357474A1 Lurasidone for use in the treatment of memory or learning dysfunction by schizophrenia |
08/11/2011 | US20110195945 Compounds, Compositions and Methods for Treating or Preventing Hypoxic or Ischemic Injury |
08/03/2011 | EP2349276A2 Hiv integrase inhibitors |
07/20/2011 | CN1930137B Novel benzothiazepine and benzothiepine compounds |
07/20/2011 | CN102131791A Dibenzothiazepine derivatives and use thereof |
07/14/2011 | US20110172190 Agents for preventing and treating disorders involving modulation of the ryanodine receptors |
07/13/2011 | EP2343286A1 Dibenzo[b,f][1,4]oxazepine derivatives as inhibitors of histone deacetylase |
07/07/2011 | WO2011081184A1 Lanthionine derivative |
07/07/2011 | CA2784310A1 Lanthionine derivatives |
07/05/2011 | US7973030 Benzothiazepine and benzothiepine compounds |
06/28/2011 | US7968707 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection |
06/16/2011 | US20110144087 Short acting benzothiazepine calcium channel blockers and uses thereof |
06/15/2011 | EP2330895A1 Short acting benzothiazepine calcium channel blockers and uses thereof |
05/31/2011 | CA2493390C A process for production of high-purity enamines |
05/12/2011 | US20110112068 Human immunodeficiency virus protease inhibitors |
04/28/2011 | US20110098273 Oligomer-Calcium Channel Blocker Conjugates |
04/20/2011 | EP2311464A1 Agents for preventing and treating disorders involving modulation of the ryr receptors |
04/13/2011 | EP2307389A1 Dibenzothiazepine derivatives and use thereof |
03/30/2011 | EP0933354B1 Calcium receptor-active compounds |
03/24/2011 | WO2011034051A1 Novel cyclic squaramide derivatives |
03/17/2011 | US20110065667 Phenylpyrazole derivatives |
03/08/2011 | US7902355 Process for the preparation of an 11-(4-substituted-1-piperazinyl)dibenzo[b,f][1,4]thiazepine derivative |
02/16/2011 | CN101977902A Process for preparing benzothiazepines from gamma-aminoalkylbenzenes |
02/08/2011 | CA2480940C Non-steroidal progesterone receptor modulators |
02/08/2011 | CA2431461C 1,5 benzothiazepines and their use as antihyperlipidemics |
02/02/2011 | CN101962369A Amino substituted diaryl[a,d]cycloheptene analogs as muscarinic agonists and methods of treatment of neuropsychiatric disorders |
02/01/2011 | US7879840 Ryanodine receptors (RyRs) modulators comprising 1,4-benzothiazepine derivatives, that regulate calcium channel functioning in cells, used for the treatment of cardiovascular disorders and muscular disorders |
02/01/2011 | CA2459449C Benzothiazepine and benzothiadiazepine derivatives with ileal bile acid transport (ibat) inhibitory activity for the treatment hyperlipidaemia |
01/19/2011 | EP1664009B1 Preparation method for quetiapine |
01/04/2011 | US7863441 cyclization using phosphorus oxychloride; antipsychotic or neuroleptic agent for psychological disorders |
01/04/2011 | US7863277 antipsychotic (ziprasidone and quetiapine) encapsulated in cyclodextrin, and a dermatologically acceptable carrier consisting of ethoxy diglycol, lecithin soya, isopropyl palmitate, poloxamer and water; schizophrenia; Bipolar disorders |
12/28/2010 | US7858777 comprises the ring closure and deprotection of an intermediate; 11-(4-[2-(2-hydroxyethoxy)ethyl]-1-piperazinyl]dibenzo[b,f]-1,4-thiazepine; used as an antipsychotic or neuroleptic |
12/28/2010 | US7858776 (2,3-cis)-3-amino-2-phenyl-2,3-dihydro-1,5-benzoxazepin-4(5H)-one; for treatment of neurological disorders related to amyloid beta protein production such as Alzheimer's disease; inhibit gamma secretase and thereby inhibit the production of amyloid beta protein |
12/22/2010 | CN101925587A Process for preparation of quetiapine |
12/09/2010 | US20100311718 Treatment of Psychoses with Dibenzothiazepine Antipsychotic |
12/07/2010 | US7847094 Industrial preparation of 11-[4-{2-(2-hydroxyethoxy) ethyl}-1-piperazinyl] dibenzo [b,f]-[1,4]thiazepine |
12/02/2010 | US20100305094 Fused tricyclic compounds as inhibitors of tumor necrosis factor-alpha |
11/24/2010 | EP2253315A1 Alkoxyphenylpropanoic acid derivatives |
11/24/2010 | CN101891707A Method for preparing Quetiapine or pharmaceutically acceptable fumarate thereof |
11/24/2010 | CN101891706A 3,4-dihydrobenzo[f][1,4]thiazepine compound or salts of same and medical use of same |
11/17/2010 | EP2250159A1 Process for preparing benzothiazepines from gamma-aminoalkylbenzenes |
11/03/2010 | EP2245021A1 A process for the preparation of quetiapine |
10/19/2010 | US7816408 (N-{5-[(4-chlorophenyl)thio]pentyl}-N-[(1R)-1-(1-naphthyl)ethyl]amine); mimics/blocks effect of extracellular calcium in parathyroid cells, juxtaglomerular/proximal tubule kidney cells, parafollicular thyroid cells, bone osteoclasts, keratinocytes or placental trophoblasts; hyperparathyroidism |
10/14/2010 | WO2010070667A3 Process and intermediates for the preparation of 7-( (3-chloro-6-methyl-5,5-dioxo-6,ll-dihydrodibenzo (c, f) (1,2) thiazepin-11-yd amino) heptanoate |
10/07/2010 | US20100256082 Metallo-hydrolase inhibitors using metal binding moietes in combination with targeting moieties |
10/05/2010 | US7807827 reacting 2-(4-dibenzo[b,f][1,4]thiazepine-11-il-piperazine-1-il)ethanol and 2-(2-chloroethoxy)-tetrahydro-2H-pyran and tetrabutylammonium hydrogen sulfate in presence of NaOH base to form quetiapine; high degree of purity; antipsychotic or neuroleptic |
09/28/2010 | US7803792 benzothiazepine compounds having a thioamide bond and a quaternary ammonium substituent, exhibiti a potent ileal bile acid transporter inhibiting activity, used for for treating hyperlipidemia or arteriosclerosis |