Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
04/2000
04/04/2000US6045773 Method of detecting cyclooxygenase-2
03/2000
03/29/2000EP0988293A1 Bisimino-substituted phenyl compounds and their use as pesticides
03/29/2000EP0988292A2 Piperazine derivatives and their use as anti-inflammatory agents
03/29/2000EP0988278A1 Preparation and uses of n-methylnitrone
03/28/2000US6043374 Benzisothiazolidine Compounds
03/28/2000US6043265 Isoxazolyl endothelin antagonists
03/28/2000US6043240 Useful as antipsychotic and analgesic agents
03/22/2000EP0987256A1 Crystal form of N-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamid
03/22/2000EP0986384A1 Inhibitors of protein isoprenyl transferases
03/22/2000CN1248255A 3-heterocyclyl-substituted benzoyl derivatives
03/22/2000CN1050603C Prepn. of intermediate product used in process for diastereoselective synthesis of nucleosides
03/21/2000US6040463 Sordarin derivatives
03/15/2000EP0984947A1 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
03/15/2000EP0984923A1 O-benzyl oxime ethers and their use as pesticides
03/15/2000EP0984914A1 Substituted 2-(3-alkenyl-benzoyl)-cyclohexane-1,3-diones
03/15/2000CN1247530A Acrylonitrile compounds, process for their prodn. and pesticides containing them
03/09/2000WO2000012084A1 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
03/09/2000CA2342222A1 Geometrically restricted 2-indolinone derivatives as modulators of protein kinase activity
03/02/2000WO2000010566A1 Novel isoxazolinone antibacterial agents
03/02/2000CA2341271A1 Novel isoxazolinone antibacterial agents
03/01/2000CN1246116A Sulphonamide derivatives, process for their preparation and their use as medicaments
02/2000
02/29/2000US6031110 Ortho-substituted 2-methoxyiminophenyl-N-methylacetamides
02/29/2000US6030991 Adjusting the binding of an endothelin peptide to endothelin a or, particularly, endothelin b receptors, i.e. inhibiting or stimulating; antiinflammatory agent; asthma; kidneys; gastrointestinal, cardioascular disorders; hypotensive agents
02/29/2000US6030964 Binds to retinoic acid receptors and useful for treating psoriasis, autoimmune diseases, tumors, rheumatoid arthritis and for inducing immunosuppression in organ transplantation
02/23/2000EP0980369A1 Sulfonamides for treatment of endothelin-mediated disorders
02/23/2000CN1049651C Metalloproteinase inhibitors
02/17/2000WO2000008001A1 Substituted isoxazole as estrogen receptor modulators
02/17/2000WO2000007996A2 Pyrazoles as estrogen receptor modulators
02/17/2000WO2000007991A1 Amide derivatives useful as inhibitors of the production of cytokines
02/17/2000WO2000007980A1 Amide derivatives which are useful as cytokine inhibitors
02/17/2000CA2338121A1 Amide derivatives useful as inhibitors of the production of cytokines
02/16/2000EP0979226A1 Isoxazole derivatives
02/16/2000EP0979077A1 Method of using cyclooxygenase-2 inhibitors in the prevention of cardiovascular disorders
02/16/2000CN1244862A Endothelin antagonists: N-[[2'-[[4,5-dimethyl-3-isoxazolyl) amino] sulfonyl]-4-(2-oxazolyl) [1,1'-biphenyl]-2-yl] methyl]
02/16/2000CN1049336C Isoxazole derivatives for the treatment of irritable bowels system in preparing composition
02/10/2000WO2000006537A1 N-substituted sulfonamide derivatives
02/10/2000WO2000006529A1 Diketoacid-derivatives as inhibitors of polymerases
02/10/2000WO2000006525A2 Synthesis of combinatorial libraries of compounds reminiscent of natural products
02/10/2000CA2338490A1 Diketoacid-derivatives as inhibitors of polymerases
02/09/2000EP0977815A1 ALKYL, ALKENYL AND ALKYNYL CHRYSAMINE G DERIVATIVES FOR THE ANTEMORTEM DIAGNOSIS OF ALZHEIMER'S DISEASE AND $i(IN VIVO) IMAGING AND PREVENTION OF AMYLOID DEPOSITION
02/09/2000CN1244196A 3-amino-1,2-benzoisoxazole derivatives, process for preparation,a nd use thereof
02/09/2000CN1244122A Method of using cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia
02/08/2000US6022977 Dynamic resolution of isoxazoline thioesters to isoxazoline carboxylic acids
02/08/2000US6022870 4-(heterocycle-substituted-phenyl)-1,2,4-triazol-3-ones
02/03/2000WO2000005201A1 N-benzocycloalkyl-amide derivatives and their use as medicaments
02/03/2000DE19834557A1 New (hetero)aryl 1,2,4-triazole or isoxazole derivatives useful as fungicides, insecticides, acaricides and nematocides
02/03/2000CA2338198A1 N-benzocycloalkyl-amide derivatives and their use as medicaments
02/02/2000EP0975588A1 Antipicornaviral compouds, compositions containing them, and methods for their use
02/02/2000EP0975587A1 Oxime ether compounds, their use and intermediates for preparations of the same
02/01/2000US6020497 3-substitutes isoxazolidines as chiral auxiliary agents
02/01/2000US6020372 Use of isoxazole and crotonamide derivatives for the treatment of carcinomatous disorders
02/01/2000US6020371 Antipicornaviral compounds compositions containing them and methods for their use
02/01/2000US6020368 Microbiocides
01/2000
01/27/2000WO2000003988A1 Novel benzoic acid derivatives and processes for the preparation thereof
01/26/2000EP0973748A1 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses
01/26/2000EP0973728A1 Acrylic acid phenylester derivatives
01/26/2000CN1048719C Novel 7-(substituted)-8-(substituted)-9-(substituted amino)-6-demethyl-6-deoxytetracyclines, prepn. method, their compositions and use thereof
01/25/2000US6018069 (2s,3s,5s)-2,5-diamine-1,6-diphenyl-3-hydroxyhexane compounds are purified by obtaining the acid addition salt from a mixture with its (2s,3s,5r) stereoisomer; useful as intermediates to hiv protease inhibitor synthesis
01/25/2000US6017956 N,N-disubstituted amic acid derivatives
01/25/2000US6017928 Retroviral protease inhibiting compounds
01/20/2000WO2000002851A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them
01/20/2000WO1999048851A3 Processes for preparing intermediates
01/19/2000EP0971906A1 Lipase catalyzed dynamic resolution of isoxazoline thioesters to isoxazoline carboxylic acids
01/19/2000EP0672038B1 Herbicides
01/18/2000US6015909 Arylidene compound and silver halide photographic material
01/18/2000US6015908 IL-8 receptor antagonists
01/18/2000US6015227 Thermoplastic foam extrusion screw with circulation channels
01/13/2000WO2000001666A1 C-TERMINAL MODIFIED OXAMYL DIPEPTIDES AS INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
01/13/2000WO2000001389A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
01/13/2000WO1999018941A3 Ih-MODULATORS
01/13/2000DE19830430A1 New sulfur-substituted sulfonylamino-carboxylic acid N-arylamide derivatives useful as guanylate cyclase activators in treatment of e.g. cardiovascular disorders, asthma and diabetes
01/13/2000CA2336714A1 Biphenyl sulfonamides as dual angiotensin endothelin receptor antagonists
01/12/2000EP0970950A2 Novel isoxazoline and isoxazole fibrinogen receptor antagonists
01/12/2000EP0970061A1 Fungicidal alkoximinomethyldioxazine derivatives
01/12/2000EP0810999B1 Isoxazolyl-benzoyl derivatives
01/11/2000US6013837 Aromatic amides, method for preparing and compositions containing same, and use thereof as pesticides
01/11/2000US6013805 Pentafluorothio-substituted isoxazoles
01/06/2000WO2000000481A1 Cyclic carbamates and isoxazolidines as iib/iiia antagonists
01/06/2000WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2333647A1 Cyclic carbamates and isoxazolidines as iib/iiia antagonists
01/05/2000EP0968179A1 N-sulphonyl and n-sulphinyl amino acid amides as microbiocides
12/1999
12/29/1999WO1999067229A1 New 2-aminocarbonyl-5(2h)-isoxazolones as ligands of a dfp-binding site for treatment of cns-diseases
12/29/1999EP0966452A1 Process for preparing sulphurous 2-chloro-3-(4,5-dihydroisoxazol-3-yl)-benzoic acids
12/29/1999EP0612314B1 2-pyrazinylethylamine derivatives and their use as pharmaceuticals
12/29/1999CA2335190A1 New 2-aminocarbonyl-5(2h)-isoxazolones as ligands of a dfp-binding site for treatment of cns-diseases
12/28/1999US6007739 Liquid crystal compound, liquid crystal composition, and liquid crystal display device using the same
12/23/1999WO1999065871A2 Thiolesters and uses thereof
12/23/1999WO1999065310A1 Il-8 receptor antagonists
12/23/1999DE19827387A1 Use of ligands of the high affinity binding site of diisopropyl-fluorophosphate in treatment of central nervous system disorders
12/23/1999CA2335464A1 Novel thiolesters and uses thereof
12/23/1999CA2335292A1 Il-8 receptor antagonists
12/22/1999EP0904077A4 Methods for the preparation of biphenyl isoxazole sulfonamides
12/21/1999US6005116 Isoxazole compounds useful for the prophylaxis or treatment of nervous diseases
12/21/1999US6004955 Cyclic carbamates and isoxazolidines as IIb/IIIa antagonists
12/21/1999US6004903 2-Anylocyclohexanediones having improved herbicidal properties
12/16/1999WO1999064404A1 Heterocycle-bearing thio phenol compounds, intermediates for the preparation of the same and processes for the preparation of both
12/15/1999EP0963984A1 Heteroarylpiperidines and piperazines and their use as antipsychotics and analgetics
12/15/1999CN1238766A 3-alkoxyisoxazol-4-yl-substituted 2-amino carboxylic acid compounds
12/15/1999CN1238760A N-(aryl/heteroaryl/alkyl acetyl) amino acid esters, pharmaceutical composition comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds
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