Patents
Patents for C07D 261 - Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings (11,459)
06/1999
06/02/1999EP0918761A1 Certain amido- and amino-substituted benzylamine derivatives; a new class of neuropeptite y1 specific ligands
06/02/1999CN1218460A Substituted 4-hydroxy-phenylalcanoic acid derivatives with activity to ppar-'gamma'
06/01/1999US5908931 Preorganized hexadentate ligands useful in radiographic imaging agents
06/01/1999US5908863 Geminal carboxylic acids and esters thereof pharmaceutical formulations containing them useful in the treatment of bone dysmetabolism
05/1999
05/27/1999WO1999025701A1 NOVEL HETEROCYCLICALLY SUBSTITUTED α-HYDROXYCARBOXLIC ACID DERIVATIVES, METHOD FOR PRODUCING THE SAME AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS
05/27/1999WO1999025686A1 Cyclic amine derivatives and their use as drugs
05/27/1999CA2308746A1 Novel heterocyclically substituted .alpha.-hydroxycarboxylic acid derivatives, method for producing the same and their use as endothelin receptor_antagonists
05/26/1999EP0917528A1 New amidino derivatives and their use as thrombin inhibitors
05/26/1999CN1217711A Aryl substituted cyclic amines as selective dopamine D3 ligands
05/20/1999WO1999024409A1 Isoxazole derivatives and their use as herbicides
05/20/1999WO1999024394A2 Compounds for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition
05/20/1999WO1999016753A3 Tricyclic 3-oxo-propanenitrile compounds
05/20/1999DE19750529A1 New heterocyclic alpha-hydroxycarboxylic acid derivatives useful for treating hypertension, chronic coronary insufficiency, asthma, prostate cancer etc.
05/20/1999CA2309626A1 Compounds for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition
05/19/1999EP0916661A1 Process for the preparation of 3,5-dimethylisoxazol-4-sulfochloride
05/19/1999EP0916658A1 Assays utilizing improved chemiluminescent esters, thioesters and amides
05/19/1999EP0915847A1 Substituted sulfonamides as selective beta3 agonists for the treatment of diabetes and obesity
05/19/1999CN1216986A Isoxazole derivatives
05/18/1999US5905080 Central nervous system, psychological, eating disorders; cognition activators, parkinson*s disease
05/14/1999WO1999023063A1 Substituted anilides
05/14/1999WO1999022720A2 Selective cyclooxygenase-2 inhibitors against premature labor
05/14/1999CA2308639A1 Method of using cyclooxygenase-2 inhibitors in maintaining the fetal ductus ateriosus during treatment and prevention of preterm labor
05/12/1999EP0914319A1 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists
05/12/1999CN1216543A Novel benzene derivatives substituted by heterocycles and herbicides
05/12/1999CN1216534A Novel heterocycle-substituted benzene derivatives and herbicides
05/06/1999WO1999021842A1 Herbicidal 4-benzoylisoxazoles derivatives
05/06/1999EP0912499A1 Pesticides
05/05/1999CN1216043A Substd. benzenesulfonamide derivs as prodrugs of COX-2 inhibitors
04/1999
04/28/1999EP0910564A1 D-amino acid derived inhibitors of cysteine and serine proteases
04/22/1999WO1999019300A1 Prostaglandin agonists and their use to treat bone disorders
04/22/1999WO1999019299A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999WO1999018941A2 Ih-MODULATORS
04/22/1999CA2305353A1 Heterocycles useful in the treatment of benign prostatic hyperplasia and intermediates thereof
04/22/1999CA2305180A1 Ih-modulators
04/21/1999CN1214678A Butadiene derivatives and process for preparing thereof
04/15/1999WO1999018090A1 An efficient method for the conversion of nitriles to amidines
04/15/1999WO1999018076A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/15/1999CA2305746A1 An efficient method for the conversion of nitriles to amidines
04/15/1999CA2303449A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/14/1999EP0908457A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents
04/14/1999EP0907634A1 Pesticides
04/14/1999EP0907625A1 Fluorous reaction and separation systems
04/14/1999CN1214046A 4,5-dihydronaphth [1,2-C] isoxazoles and derivatives thereof having CNS activity
04/14/1999CN1214041A Sulfonated amino acid derivatives and metalloproteinase inhibitors contg. same
04/14/1999CN1214039A Carbamoyloxy derivatives of mutiline and their use as antibacterials
04/08/1999WO1999016753A2 Tricyclic 3-oxo-propanenitrile compounds
04/08/1999WO1999016751A1 Benzamidine derivatives as factor xa inhibitors
04/08/1999WO1999003823A3 Novel polyamine analogues as therapeutic and diagnostic agents
04/08/1999WO1998054161A9 Oxazolidinone antibacterial agents having a thiocarbonyl functionality
04/08/1999DE19743435A1 Benzamidinderivate Benzamidine derivatives
04/08/1999CA2305568A1 Benzamidinderivates
04/08/1999CA2302025A1 Tricyclic 3-oxo-propanenitrile compounds
04/07/1999CN1213302A Preparation containing combination of N-5-methylisoxazole-4-carboxylic acid-(4-trifluoromethyl)-anilide and N-(4 trifluoromethylphenyl)-2-cyano-3-hyroxycrotonic acid amide
04/06/1999US5892117 Oxidation of secondary amine using hydrogen peroxide and sodium tungstate
04/06/1999US5892052 Process for making retroviral protease inhibiting compounds
03/1999
03/31/1999EP0904079A1 Antidiabetic agents
03/31/1999EP0904077A2 Methods for the preparation of biphenyl isoxazole sulfonamides
03/31/1999EP0877733A4 Process for production of piperidine derivatives
03/31/1999EP0733035B1 Tricyclic derivatives, pharmaceutical compositions containing them
03/31/1999EP0638074B1 Isoxazole carboxylic acid amides, process for producing them and their use
03/30/1999US5889059 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
03/30/1999US5889035 1-(Arylthioalkyl, arylaminoalkyl or arylmethylenealkyl)-3-(heteroaryl) pyrrolidines and related compounds useful as antipsychotics and analgesics
03/30/1999US5889004 4-heteroaryl-1-piperazinealkylthiols and derivatives thereof and their therapeutic utility
03/25/1999WO1999014216A1 Substituted 3(-1,2-benzisothiazol or isoxazol-5 yl)-substituted pyrimidine as herbicides
03/25/1999WO1999014210A1 Process for the preparation of substituted 5,6-dihydro-2h-pyran-2-ones
03/24/1999EP0903345A1 Crystal form of N-(4-trifluoromethylphenyl)-5-methylisoxazole-4-carboxamid
03/24/1999CN1211976A Isoxazole derivatives and their use as herbicides
03/24/1999CN1042631C Substituted salicylic acids, its medicinal composition and use
03/23/1999US5886175 Tetracycline antibiotics
03/23/1999US5886036 Treating hiv infections
03/23/1999US5886033 Use of isoxazole and crotonamide derivatives for the treatment of carcinomatous disorders
03/23/1999US5886015 Applying fungicide or insecticide to the locus of the seed, plant or soil
03/17/1999EP0901479A1 Isoxazole derivatives and their use as herbicides
03/17/1999CN1211241A New intermediates to pesticides
03/17/1999CN1211183A Methods for preparation of biphenyl isoxazole sulfonamides
03/17/1999CA2246221A1 3-(1,2-benzisothiazol- and isoxazol-5-yl)-2,4(1h,3h)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-yl)-4(3h)-pyrimidinone or thione herbicidal agents
03/16/1999US5883125 Benzyloxy substituted aromatics and their use as fungicides and insecticides
03/11/1999WO1998056771A3 Piperazine derivatives and their use as anti-inflammatory agents
03/10/1999EP0900795A1 Benzene derivatives substituted by heterocycles and herbicides
03/09/1999US5880121 Serotonin 5ht3 antagonist, useful for treating anxiety, phychiatric disorders, nausea, vomiting and drug dependency
03/04/1999WO1999010313A1 N-aroylphenylalanine derivatives
03/04/1999WO1999010312A1 N-alkanoylphenylalanine derivatives
03/04/1999DE19838138A1 New isoxazole-5-one derivatives
03/04/1999CA2300121A1 N-alkanoylphenylalanine derivatives
03/03/1999EP0898566A1 Substituted benzylamines and their use for the treatment of depression
03/03/1999CN1042334C Herbicide composition containing 4-benzoyl-isoxazole derivative and use thereof
02/1999
02/25/1999WO1999009009A1 Method for producing organic compounds
02/25/1999WO1999009008A1 Method for producing substituted-2-nitroguanidine derivatives
02/25/1999CA2301172A1 Method for the producing substituted-2-nitroguanidine derivatives
02/25/1999CA2300808A1 Method for the producing substituted-2-nitroguanidine derivatives
02/24/1999CN1042225C Substituted isoxazole derivatives prepn. method
02/23/1999US5874467 Phenylacetic acid derivatives and use as fungicides
02/23/1999US5874451 Hypolipidemic agents
02/23/1999US5874435 Psychological disorders; analgesics
02/23/1999CA2176255C Isoxazoline compounds as antiinflammatory agents
02/18/1999WO1999007697A1 Substituted 4-benzoyl-pyrazoles
02/18/1999WO1999007688A1 2-benzoyl-cyclohexane-1,3-diones
02/18/1999WO1999007670A1 Anthranilic acid analogs
02/18/1999CA2298589A1 Substituted 4-benzoyl-pyrazoles
02/18/1999CA2298574A1 2-benzoyl-cyclohexane-1,3-diones
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