| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 04/15/1999 | CA2306077A1 Novel cycloalkenyl substituted compounds |
| 04/15/1999 | CA2304513A1 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate |
| 04/14/1999 | EP0907644A1 Pharmaceutical preparation |
| 04/14/1999 | EP0907643A1 Compounds with growth hormone releasing properties |
| 04/14/1999 | CN1214047A Novel aromatic piperazines derived from substituted cycloazanes, method for prepairing same, pharmaceutical compsns, and use thereof as drugs |
| 04/14/1999 | CN1214045A Process for aminocarbonylation of benzazepines and benzodiazepines |
| 04/08/1999 | WO1999016313A1 2-methyl-thieno-benzodiazepine formulation |
| 04/07/1999 | EP0906907A1 Compounds potentiating retinoid |
| 04/06/1999 | US5891871 Substituted 2,3-benzodiazepin-4-ones and the use thereof |
| 03/31/1999 | EP0904540A1 Methods for spatially-dispersed positionally-encoded combinatorial library synthesis |
| 03/31/1999 | CN1212692A Substituted A2a-and diazacycloheptane and cyclooctane compounds and their use |
| 03/31/1999 | CN1212689A Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds |
| 03/30/1999 | US5888992 Polar substituted hydrocarbons |
| 03/24/1999 | EP0903349A2 CCR-3 receptor antagonists |
| 03/24/1999 | EP0903343A1 Alpha-Substituted phenylpropionic acid derivative and medicine containing the same |
| 03/24/1999 | CN1211572A Cyclic amine derivatives-CCR-3 receptor antagonists |
| 03/19/1999 | CA2247772A1 .alpha.-substituted phenylpropionic acid derivative and medicine containing the same |
| 03/16/1999 | US5883261 Esterification reaction in the presence of sodium methoxide |
| 03/11/1999 | WO1999012034A1 Amine compounds and combinatorial libraries comprising same |
| 03/11/1999 | WO1999011649A2 Parp inhibitors, pharmaceutical compositions comprising same, and methods of using same |
| 03/11/1999 | WO1999011624A1 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
| 03/11/1999 | CA2294118A1 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
| 03/11/1999 | CA2294074A1 Parp inhibitors, pharmaceutical compositions comprising same, and methods of using same |
| 03/10/1999 | CN1210538A Condensed 2,3-benzodiazepine derivatives and their use as ampa-receptor inhibitors |
| 03/09/1999 | US5880295 Process for the preparation of diamine intermediates useful in the synthesis of HIV protease inhibitors |
| 03/04/1999 | WO1999009991A1 Novel amide derivatives |
| 03/04/1999 | WO1999009990A1 Pharmaceutical suspension comprising nevirapine hemihydrate |
| 03/04/1999 | CA2301566A1 N-acylated lipophilic amino acid derivatives |
| 03/03/1999 | EP0899264A1 7-Phenyl-1,4-diazepane derivatives as neurokinine receptor antagonists |
| 03/03/1999 | EP0500952B1 Process for producing nitrogenous heterocycle |
| 03/03/1999 | CN1209744A Vitronectin receptor antagonists |
| 03/02/1999 | US5877312 Method for preparing alkylating agents for their use for alkylating cyclic ureas |
| 03/02/1999 | US5877278 Solid phase synthesis using two submonomers-an acylating agent, e.g. a haloacetic acid, and a primary amine; cyclization to produce mimetics of drugs; elimination of the necessity of protection groups |
| 03/02/1999 | US5877170 Substitute caprolactams and derivatives thereof useful for treatment of HIV disease |
| 02/25/1999 | DE19837386A1 New CCR-3 antagonist piperazine derivatives and analogues |
| 02/24/1999 | CN1209126A Novel compounds with analgesic effect |
| 02/23/1999 | CA1340402C Quinoline derivatives and processes for preparation thereof |
| 02/18/1999 | CA2245043A1 Ccr-3 receptor antagonists |
| 02/17/1999 | CN1208405A Retroviral protease inhibiting compounds |
| 02/16/1999 | US5872115 Compounds for treatment of hypercholesterolemia, ischemic heart disease, cerebrovascular disease or atherosclerosis |
| 02/11/1999 | WO1999006409A1 Tricyclic vasopressin agonists |
| 02/09/1999 | US5869483 Tricyclic benzazepine vasopressin antagonists |
| 02/04/1999 | WO1999005147A1 Thiazolobenzoheterocycles, preparation and medicines containing same |
| 02/04/1999 | WO1999005124A1 Novel hexahydro-1,4-diazepine derivatives or salts thereof |
| 02/04/1999 | CA2289572A1 Novel hexahydro-1,4-diazepine derivatives or salts thereof |
| 02/03/1999 | CN1041921C Bicyclic fibrinogen antagonists |
| 01/28/1999 | WO1998046576A3 Halo-alkoxycarbonyl prodrugs |
| 01/27/1999 | EP0892797A1 Inhibitors of farnesyl protein transferase |
| 01/27/1999 | CN1206006A Novel hexahydro-1,4-diazepine derivative and its salt |
| 01/26/1999 | US5863914 Administering to human n,n-dimethylbenzene or n,n-dimethylnaphthalene-cyclic urea derivative to treat a disease-state caused by inhibition of factor xa |
| 01/20/1999 | EP0891337A1 Inhibitors of farnesyl-protein transferase |
| 01/12/1999 | US5859007 Treatment of diabetes, obesity |
| 01/12/1999 | US5859005 Inhibitors of thrombin and factor xa |
| 01/07/1999 | EP0888356A1 Condensed 2,3-benzodiazepine derivatives and their use as ampa-receptor inhibitors |
| 01/07/1999 | EP0888313A1 2,3-benzodiazepine derivatives and their use as ampa-receptor inhibitors |
| 12/30/1998 | EP0594577B1 Novel potent inducers of terminal differentiation and method of use thereof |
| 12/30/1998 | CN1041420C Process for preparing N-acyl-2,3-benzodiazepine derivatives |
| 12/29/1998 | US5854274 Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives |
| 12/29/1998 | US5854236 Tricyclic benzazepine vasopressin antagonists |
| 12/23/1998 | EP0885204A1 Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds |
| 12/22/1998 | US5852010 Inhibitors of farnesyl-protein transferase |
| 12/16/1998 | CN1202160A Compounds potentiating retinoid |
| 12/15/1998 | US5849735 Tricyclic benzazepine vasopressin antagonists |
| 12/15/1998 | US5849732 Phenol compound having antioxidative activity and the process for preparing the same |
| 12/09/1998 | EP0882024A1 Retroviral protease inhibiting compounds |
| 12/08/1998 | US5846969 Tricyclic heterocyclic sulfonamide and sulfonic ester derivatives |
| 12/03/1998 | WO1998054229A1 Use of ylides of phosphorus as slightly nuceophilic strong bases |
| 12/03/1998 | CA2291345A1 Use of ylides of phosphorus as slightly nuceophilic strong bases |
| 12/02/1998 | EP0881235A1 Phosphorus ylides, their preparation and use thereof as low-nucleophilic strong-basic compounds |
| 12/02/1998 | EP0880512A1 Novel aromatic piperazines derived from substituted cycloazanes, method for preparing same, pharmaceutical compositions, and use thereof as drugs |
| 12/02/1998 | CN1200374A Vitronectin receptor antagonists, their prepn. and their use |
| 12/02/1998 | CN1200373A Vitronectin receptor antagonists, their prepn. and use |
| 12/01/1998 | US5843952 Tricyclic benzazepine vasopressin antagonists |
| 12/01/1998 | US5843941 Ras farnesyl transferase inhibitors |
| 11/24/1998 | US5840960 Potent inducers of terminal differentiation and method of use thereof |
| 11/18/1998 | EP0877744A1 Substituted aza- and diazacycloheptane and cyclooctane compounds and their use |
| 11/10/1998 | US5834463 Condensed heterocyclic compounds, their production and use |
| 11/10/1998 | US5834462 Antitumor agents; anticarcinogenic agents particularly for nasopharyngel, pulmonary, intestinal, mammary, uterus, gastric, ovarian or liver cancer and also leukemia |
| 11/03/1998 | US5831089 Process to produce midazolam |
| 10/29/1998 | WO1998047882A1 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists |
| 10/29/1998 | CA2285664A1 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists |
| 10/28/1998 | EP0873322A1 Novel compounds with analgesic effect |
| 10/22/1998 | WO1998046591A1 SELECTIVE FACTOR Xa INHIBITORS |
| 10/22/1998 | WO1998046576A2 Halo-alkoxycarbonyl prodrugs |
| 10/22/1998 | CA2285335A1 Selective factor xa inhibitors |
| 10/21/1998 | EP0871465A1 Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids |
| 10/21/1998 | EP0710229B1 1,5-benzodiazepine derivatives useful as cck or gastrin antagonists |
| 10/20/1998 | US5824676 Piperazinyl-dibenz(b,f)(1,4)oxazepine derivatives |
| 10/14/1998 | EP0869967A2 INHIBITORS OF INTERLEUKIN-1$g(b) CONVERTING ENZYME |
| 10/14/1998 | EP0869787A1 Vitronectin receptor antagonists |
| 10/08/1998 | WO1998028268A3 CYCLOALKYL, LACTAM, LACTONE AND RELATED COMPOUNDS AS β-AMYLOID PEPTIDE RELEASE INHIBITORS |
| 10/07/1998 | EP0850238A4 Combinatorial 1,4-benzodiazepin-2,5-dione library |
| 10/06/1998 | US5817655 Treatment of nervous system disorders |
| 10/06/1998 | US5817602 Herbicidal thiadiazabicyclodecanes |
| 10/01/1998 | WO1998042696A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same |
| 09/22/1998 | US5811422 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors |
| 09/16/1998 | EP0710230B1 1,5-benzodiazepine derivatives useful as cck or gastrin antagonists |
| 09/15/1998 | US5807851 2,3-Benzodiazepine Derivatives as non-competitive AMPA |
| 09/09/1998 | CN1192729A Benzamide derivatives and their use as vasopressin antagonists |
| 09/03/1998 | WO1998038177A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR INHIBITING β-AMYLOID PEPTIDE |