Patents
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
10/2002
10/10/2002WO2002079172A1 Method for preparing monocyclic $i(n)-acyl-aminolactam compounds and combinatorial libraries thereof
10/10/2002WO2002078680A1 Gaba-receptor modulators for the treatment of neurodegenerative diseases of the eye
10/10/2002WO2002078628A2 Cyanamide, alkoxyamino, and urea derivatives of 1,3-benzodiazapines as hiv reverse transcriptase inhibitors
10/10/2002CA2439842A1 Gaba-receptor modulators for the treatment of neurodegenerative diseases of the eye
10/09/2002EP1246819A1 A method for the preparation of substituted benzene derivatives
10/08/2002US6462064 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents, especially for cervical cancers and dysplasias
10/08/2002US6462037 Such as 7-chloro-3-methyl-5-(2-cyclopropylethynyl)-1,5-dihydro-5-(trifluoromethyl) -1,4-benzodiazepin-2-one; protease inhibitors
10/08/2002CA2066083C Benzodiazepine analogs as cholecystokinin antagonists
10/03/2002WO2002076925A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/03/2002WO2002076404A2 Fatty alcohol drug conjugates
10/03/2002WO2002076402A2 Fatty amine drug conjugates
10/03/2002CA2441080A1 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
10/02/2002EP1244624A1 Anthracene derivatives as anti-cancer agents
10/02/2002EP1244457A2 Methods and compositions related to modulators of annexin and cartilage homeostasis
10/02/2002EP0871465B1 Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids
10/02/2002EP0679641B1 Sulfonamide and sulfonic ester derivatives each having tricyclic hetero ring
10/01/2002US6458784 Vitronectin receptor antagonists
10/01/2002US6458783 Non-imidazole benzodiazepine inhibitors of farnesyl protein transferase
10/01/2002US6458782 Treatments of diabetes and complications of diabetes.
09/2002
09/26/2002US20020137939 Novel guanidinobenzamides
09/26/2002US20020137737 1-(3-methyl-1-(1,3-dihydro-1-methyl-2-oxo-5-phenyl-2H-1,4 -benzodiazepin-3-ylcarbamoyl)-butyl)-cyclopent-3-enecarboxylic amide, for example; gamma-secretase inhibitors; Alzhemier's disease, Down's Syndrome
09/25/2002EP1181279A4 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
09/24/2002US6455529 Adhesion receptor antagonists
09/24/2002US6455523 Inhibitors of farnesyl protein transferase
09/19/2002WO2002072570A2 Non-imidazole compounds as histamine h3 antagonists
09/18/2002EP0757681B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS
09/18/2002CN1370174A 2,3-benzodiazepine derivatives
09/17/2002US6452001 1,4-diazepine-2-one derivatives as neurokinin antagonist
09/17/2002US6452000 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate
09/12/2002WO2002070493A1 Bisaryl derivatives having fsh receptor modulatory activity
09/12/2002WO2002069895A2 Heterocyclic analgesic compounds and methods of use thereof
09/12/2002WO2001012600A9 INHIBITORS OF FACTOR Xa
09/12/2002US20020128262 Styrylbenzodiazepines
09/12/2002US20020128261 Cyclohepta [b] [1,4] diazepino [6,7, 1-hi] indoles and derivatives
09/12/2002CA2434184A1 Bisaryl derivatives having fsh receptor modulatory activity
09/06/2002WO2002022577A3 Hydroxamate derivatives useful as deacetylase inhibitors
09/04/2002EP1105392B1 Process for the preparation of imidazodiazepine intermediates
09/04/2002CN1367769A Process for catalyzing oxidation of organic compounds
08/2002
08/29/2002US20020119966 Central nervous system disorders
08/28/2002EP1234818A1 Calcium salts of 1,5-benzodiazepine derivatives, process for producing the salts and drugs containing the same
08/27/2002US6441172 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
08/27/2002US6440959 Inhibitors of cyclin-dependent kinases
08/27/2002US6440588 1,4-diazepine compound with electron attractive group selected from the group consisting of cyano group, an acyl group, and an alkoxy group
08/27/2002CA2224738C Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids
08/22/2002WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals
08/22/2002US20020115724 Methods and agents for inhibiting protein aging
08/22/2002US20020115660 Labled isotopes of phenyl 4-(1,4-diazepin-1-yl)-2-amino phenyl sulfone derivatives used in nuclear magnetic resonance imaging and positron emission tomography
08/08/2002WO2002060870A2 Delta agonist analgesics
08/08/2002WO2002018327A3 Guanidinobenzamides as mc4-r agonists
08/08/2002US20020107392 Quinolinone derivatives
08/08/2002US20020107242 Cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
08/08/2002US20020107239 Cyclized amide derivatives
08/08/2002US20020107235 Carbamate and hydroxy groups containing phenanthrene derivatives; useful to treat obesity, diabetes and inflammation
08/07/2002CN1362960A Method for preparing substituted [1,4] diazepino (6,7,1-hi) indol-4-ones
08/07/2002CN1362949A 1,5-benzodiazepine derivatives as cck-A receptor agonists
08/01/2002WO2002059102A2 Urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and use
08/01/2002WO2001098279A3 Bis-arylsulfones
08/01/2002US20020103184 Cyclic malonamides as inhibitors of a beta protein production
08/01/2002CA2435647A1 Urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and use
07/2002
07/31/2002EP1226139A2 Cyclized amide derivatives for treating or preventing neuronal damage
07/31/2002EP1226122A1 Bicyclic vasopressin agonists
07/30/2002US6426413 Inhibitors of caspases
07/25/2002WO2002057230A1 Il-8 receptor antagonists
07/24/2002EP1224175A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
07/24/2002EP1224174A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists
07/24/2002EP1102743B1 Amide derivatives which are useful as cytokine inhibitors
07/23/2002US6423840 Forming n-acylamino compound
07/17/2002EP1222176A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION
07/17/2002CN1359377A Dihydrobenzodiazepins and their use for treating dyslipidemia
07/16/2002CA2059704C [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl)amino]alkyl]-acid derivatives
07/11/2002US20020091256 2,3-dicyano-5-amino-5-hydroxy-6-phenylmethylidene-7-methyl-4H-1,4 -diazepine for example; electroluminescence; charge transfer agents; electroluminescence device
07/10/2002EP1221440A1 Benzoheterocyclic derivatives useful as vasopressin or oxytocin modulators
07/10/2002EP1220852A1 Substituted diazepans
07/10/2002EP1140786A4 Reductive alkylation of secondary amines with hydrosilane
07/09/2002US6417183 1,4-diazacycloheptane derivatives
07/04/2002WO2002051838A1 Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
07/04/2002WO2002051831A1 Oxybenzamides derivatives as factor xa inhibitors
07/04/2002WO2002051232A2 Novel benzazepines and related heterocyclic derivatives
07/04/2002US20020086860 For treatment or prevention of disorders such as obsessive-compulsive disorder, depression, anxiety, schizophrenia
07/03/2002EP1218377A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION
07/02/2002USRE37781 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
07/02/2002US6414144 Such as (2s)-(rel-7br,10ar)-2-methyl-1,2,3,4,8,9,10,10a-octahydro-7bh -cyclopenta(b)(1,4)diazepino(6,7,1-hi)indole; for treatment of obesity
06/2002
06/27/2002WO2002050044A1 Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient
06/27/2002WO2002020501A3 Polyarylcarboxamides useful as lipid lowering agents
06/26/2002EP1217000A1 Inhibitors of factor Xa and factor VIIa
06/26/2002CN1086705C Stereoselective process and intermediates for producing dihydro-2,3-benzodiazepine derivatives
06/18/2002US6407094 Glutamate receptor antagonists
06/13/2002WO2002028842A3 Diazacycloalkanedione derivatives which are useful as lfa-1 antagonist
06/13/2002DE10041671C1 Verfahren zur Herstellung von Imidazo[1,2-c][2,3]benzodiazepinen sowie Phenylessigsäureester und Oxazol-Derivate als Zwischenprodukte bei deren Herstellung Benzodiazepines process for the preparation of imidazo [1,2-c] [2,3] oxazole and phenylacetic acid esters and derivatives, as intermediates in the preparation thereof
06/12/2002EP1212306A2 Hydroxyalkanoylaminolactams and related structures as inhibitors of abeta protein production
06/12/2002EP1212305A2 1,5-benzodiazepine derivatives as cck-a receptor agonists
06/12/2002EP1212269A1 Methods for preparing n- (aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
06/12/2002EP0885204B1 Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds
06/12/2002CN1353702A Adamantane derivatives
06/12/2002CN1353691A Cell adhesion-inhibiting anti inflammatory and immune-suppresive compounds
06/11/2002US6403738 Polymerization of olefins
06/11/2002US6403607 Sulfonamide derivatives and drugs containing the same as the active ingredient
06/11/2002US6403595 Anticoagulants
06/11/2002US6403578 Anticoagulants, cardiovascular disorders
06/11/2002US6403112 Ectoin and ectoin derivatives as moisturizers in cosmetics
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