Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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10/10/2002 | WO2002079172A1 Method for preparing monocyclic $i(n)-acyl-aminolactam compounds and combinatorial libraries thereof |
10/10/2002 | WO2002078680A1 Gaba-receptor modulators for the treatment of neurodegenerative diseases of the eye |
10/10/2002 | WO2002078628A2 Cyanamide, alkoxyamino, and urea derivatives of 1,3-benzodiazapines as hiv reverse transcriptase inhibitors |
10/10/2002 | CA2439842A1 Gaba-receptor modulators for the treatment of neurodegenerative diseases of the eye |
10/09/2002 | EP1246819A1 A method for the preparation of substituted benzene derivatives |
10/08/2002 | US6462064 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents, especially for cervical cancers and dysplasias |
10/08/2002 | US6462037 Such as 7-chloro-3-methyl-5-(2-cyclopropylethynyl)-1,5-dihydro-5-(trifluoromethyl) -1,4-benzodiazepin-2-one; protease inhibitors |
10/08/2002 | CA2066083C Benzodiazepine analogs as cholecystokinin antagonists |
10/03/2002 | WO2002076925A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses |
10/03/2002 | WO2002076404A2 Fatty alcohol drug conjugates |
10/03/2002 | WO2002076402A2 Fatty amine drug conjugates |
10/03/2002 | CA2441080A1 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses |
10/02/2002 | EP1244624A1 Anthracene derivatives as anti-cancer agents |
10/02/2002 | EP1244457A2 Methods and compositions related to modulators of annexin and cartilage homeostasis |
10/02/2002 | EP0871465B1 Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids |
10/02/2002 | EP0679641B1 Sulfonamide and sulfonic ester derivatives each having tricyclic hetero ring |
10/01/2002 | US6458784 Vitronectin receptor antagonists |
10/01/2002 | US6458783 Non-imidazole benzodiazepine inhibitors of farnesyl protein transferase |
10/01/2002 | US6458782 Treatments of diabetes and complications of diabetes. |
09/26/2002 | US20020137939 Novel guanidinobenzamides |
09/26/2002 | US20020137737 1-(3-methyl-1-(1,3-dihydro-1-methyl-2-oxo-5-phenyl-2H-1,4 -benzodiazepin-3-ylcarbamoyl)-butyl)-cyclopent-3-enecarboxylic amide, for example; gamma-secretase inhibitors; Alzhemier's disease, Down's Syndrome |
09/25/2002 | EP1181279A4 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof |
09/24/2002 | US6455529 Adhesion receptor antagonists |
09/24/2002 | US6455523 Inhibitors of farnesyl protein transferase |
09/19/2002 | WO2002072570A2 Non-imidazole compounds as histamine h3 antagonists |
09/18/2002 | EP0757681B1 CONDENSED HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE AS GnRH ANTAGONISTS |
09/18/2002 | CN1370174A 2,3-benzodiazepine derivatives |
09/17/2002 | US6452001 1,4-diazepine-2-one derivatives as neurokinin antagonist |
09/17/2002 | US6452000 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate |
09/12/2002 | WO2002070493A1 Bisaryl derivatives having fsh receptor modulatory activity |
09/12/2002 | WO2002069895A2 Heterocyclic analgesic compounds and methods of use thereof |
09/12/2002 | WO2001012600A9 INHIBITORS OF FACTOR Xa |
09/12/2002 | US20020128262 Styrylbenzodiazepines |
09/12/2002 | US20020128261 Cyclohepta [b] [1,4] diazepino [6,7, 1-hi] indoles and derivatives |
09/12/2002 | CA2434184A1 Bisaryl derivatives having fsh receptor modulatory activity |
09/06/2002 | WO2002022577A3 Hydroxamate derivatives useful as deacetylase inhibitors |
09/04/2002 | EP1105392B1 Process for the preparation of imidazodiazepine intermediates |
09/04/2002 | CN1367769A Process for catalyzing oxidation of organic compounds |
08/29/2002 | US20020119966 Central nervous system disorders |
08/28/2002 | EP1234818A1 Calcium salts of 1,5-benzodiazepine derivatives, process for producing the salts and drugs containing the same |
08/27/2002 | US6441172 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof |
08/27/2002 | US6440959 Inhibitors of cyclin-dependent kinases |
08/27/2002 | US6440588 1,4-diazepine compound with electron attractive group selected from the group consisting of cyano group, an acyl group, and an alkoxy group |
08/27/2002 | CA2224738C Use of ritonavir (abt-538) for improving the pharmacokinetics of drugs metabolized by cytochrome p450 in a method of treating aids |
08/22/2002 | WO2002064545A1 Acylated indanyl amines and their use as pharmaceuticals |
08/22/2002 | US20020115724 Methods and agents for inhibiting protein aging |
08/22/2002 | US20020115660 Labled isotopes of phenyl 4-(1,4-diazepin-1-yl)-2-amino phenyl sulfone derivatives used in nuclear magnetic resonance imaging and positron emission tomography |
08/08/2002 | WO2002060870A2 Delta agonist analgesics |
08/08/2002 | WO2002018327A3 Guanidinobenzamides as mc4-r agonists |
08/08/2002 | US20020107392 Quinolinone derivatives |
08/08/2002 | US20020107242 Cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
08/08/2002 | US20020107239 Cyclized amide derivatives |
08/08/2002 | US20020107235 Carbamate and hydroxy groups containing phenanthrene derivatives; useful to treat obesity, diabetes and inflammation |
08/07/2002 | CN1362960A Method for preparing substituted [1,4] diazepino (6,7,1-hi) indol-4-ones |
08/07/2002 | CN1362949A 1,5-benzodiazepine derivatives as cck-A receptor agonists |
08/01/2002 | WO2002059102A2 Urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and use |
08/01/2002 | WO2001098279A3 Bis-arylsulfones |
08/01/2002 | US20020103184 Cyclic malonamides as inhibitors of a beta protein production |
08/01/2002 | CA2435647A1 Urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and use |
07/31/2002 | EP1226139A2 Cyclized amide derivatives for treating or preventing neuronal damage |
07/31/2002 | EP1226122A1 Bicyclic vasopressin agonists |
07/30/2002 | US6426413 Inhibitors of caspases |
07/25/2002 | WO2002057230A1 Il-8 receptor antagonists |
07/24/2002 | EP1224175A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists |
07/24/2002 | EP1224174A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists |
07/24/2002 | EP1102743B1 Amide derivatives which are useful as cytokine inhibitors |
07/23/2002 | US6423840 Forming n-acylamino compound |
07/17/2002 | EP1222176A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION |
07/17/2002 | CN1359377A Dihydrobenzodiazepins and their use for treating dyslipidemia |
07/16/2002 | CA2059704C [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl)amino]alkyl]-acid derivatives |
07/11/2002 | US20020091256 2,3-dicyano-5-amino-5-hydroxy-6-phenylmethylidene-7-methyl-4H-1,4 -diazepine for example; electroluminescence; charge transfer agents; electroluminescence device |
07/10/2002 | EP1221440A1 Benzoheterocyclic derivatives useful as vasopressin or oxytocin modulators |
07/10/2002 | EP1220852A1 Substituted diazepans |
07/10/2002 | EP1140786A4 Reductive alkylation of secondary amines with hydrosilane |
07/09/2002 | US6417183 1,4-diazacycloheptane derivatives |
07/04/2002 | WO2002051838A1 Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists |
07/04/2002 | WO2002051831A1 Oxybenzamides derivatives as factor xa inhibitors |
07/04/2002 | WO2002051232A2 Novel benzazepines and related heterocyclic derivatives |
07/04/2002 | US20020086860 For treatment or prevention of disorders such as obsessive-compulsive disorder, depression, anxiety, schizophrenia |
07/03/2002 | EP1218377A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION |
07/02/2002 | USRE37781 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors |
07/02/2002 | US6414144 Such as (2s)-(rel-7br,10ar)-2-methyl-1,2,3,4,8,9,10,10a-octahydro-7bh -cyclopenta(b)(1,4)diazepino(6,7,1-hi)indole; for treatment of obesity |
06/27/2002 | WO2002050044A1 Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient |
06/27/2002 | WO2002020501A3 Polyarylcarboxamides useful as lipid lowering agents |
06/26/2002 | EP1217000A1 Inhibitors of factor Xa and factor VIIa |
06/26/2002 | CN1086705C Stereoselective process and intermediates for producing dihydro-2,3-benzodiazepine derivatives |
06/18/2002 | US6407094 Glutamate receptor antagonists |
06/13/2002 | WO2002028842A3 Diazacycloalkanedione derivatives which are useful as lfa-1 antagonist |
06/13/2002 | DE10041671C1 Verfahren zur Herstellung von Imidazo[1,2-c][2,3]benzodiazepinen sowie Phenylessigsäureester und Oxazol-Derivate als Zwischenprodukte bei deren Herstellung Benzodiazepines process for the preparation of imidazo [1,2-c] [2,3] oxazole and phenylacetic acid esters and derivatives, as intermediates in the preparation thereof |
06/12/2002 | EP1212306A2 Hydroxyalkanoylaminolactams and related structures as inhibitors of abeta protein production |
06/12/2002 | EP1212305A2 1,5-benzodiazepine derivatives as cck-a receptor agonists |
06/12/2002 | EP1212269A1 Methods for preparing n- (aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds |
06/12/2002 | EP0885204B1 Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds |
06/12/2002 | CN1353702A Adamantane derivatives |
06/12/2002 | CN1353691A Cell adhesion-inhibiting anti inflammatory and immune-suppresive compounds |
06/11/2002 | US6403738 Polymerization of olefins |
06/11/2002 | US6403607 Sulfonamide derivatives and drugs containing the same as the active ingredient |
06/11/2002 | US6403595 Anticoagulants |
06/11/2002 | US6403578 Anticoagulants, cardiovascular disorders |
06/11/2002 | US6403112 Ectoin and ectoin derivatives as moisturizers in cosmetics |