Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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10/27/1994 | WO1994024149A1 1,5-benzodiazepine derivatives having cck antagonistic or agonistic activity |
10/19/1994 | EP0620218A1 Heterocyclic compounds active in gastro-intestinal pathologies |
10/19/1994 | EP0620216A1 Benzamide derivatives and their use as vasopressin antagonists |
10/18/1994 | US5356895 1,4 piperizino inhibitors of non-enzymatic cross-linking of proteins |
10/14/1994 | CA2121112A1 New benzamide derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same |
10/13/1994 | WO1994022840A1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease |
10/13/1994 | WO1994022825A1 Fibrinogen receptor antagonists |
10/13/1994 | CA2159482A1 Fibrinogen receptor antagonists |
10/13/1994 | CA2159442A1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease |
10/12/1994 | EP0619309A1 Process for the preparation of alkylimidazolidone (meth)acrylates |
10/11/1994 | CA1332411C Benzodiazepine analogs |
10/11/1994 | CA1332410C Benzodiazepine analogs |
10/05/1994 | EP0617621A1 Central cholecystokinin antagonists having pharmaceutical activity |
10/05/1994 | EP0617618A1 Aryl-triflates and related compounds |
10/05/1994 | CN1093085A Amine derivatives |
09/29/1994 | WO1994011490A3 Products of the inhibition of advanced glycosylation |
09/28/1994 | EP0616532A1 Use of peripheral-type benzodiazepine sites for treatment of cns trauma or disease |
09/20/1994 | US5349086 Alkylation and salt formation |
09/15/1994 | WO1994020473A1 Compound with vasopressin antagonism |
09/15/1994 | DE4308095A1 Prodrug derivatives of pharmaceutical agents with hydroxyl groups, process for their preparation and their use |
09/01/1994 | WO1994019329A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors |
09/01/1994 | WO1994014776A3 Bicyclic fibrinogen antagonists |
09/01/1994 | CA2156594A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors |
08/30/1994 | US5342839 Useful for therapy of oxygen deficiency diseases of the brain |
08/23/1994 | CA1331564C Redox systems for brain-targeted drug delivery |
08/17/1994 | EP0610334A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII b?III a? RECEPTOR. |
08/10/1994 | EP0609306A1 Benzodiazepine derivatives and their use as antagonists of cholecystokinin and/or gastrin receptors |
07/27/1994 | EP0607697A2 DILAZEP for reduction of elevated intraocular pressure |
07/27/1994 | EP0607355A1 3-ureido-benzodiazepinones useful as antagonists of cck or of gastrine. |
07/27/1994 | EP0607334A1 Cyclic ureas and analogues useful as retroviral protease inhibitiors. |
07/27/1994 | EP0607129A1 Methylpiperazinoazepine derivatives, their preparation and use. |
07/21/1994 | WO1994015924A1 Cholecystokinin antagonists |
07/20/1994 | EP0606658A1 Substituted N-aminoalkylmethansulphoamides as antispasmodic agents |
07/19/1994 | US5331006 Amino acid analogs as CCK antagonists |
07/14/1994 | CA2113032A1 Substituted n-aminoalkylmethane sulfanilide as antispasmodica |
07/13/1994 | EP0605639A1 Air treatment plant for foodstuff comprising a trough with an adjustable width. |
07/07/1994 | WO1994014776A2 Bicyclic fibrinogen antagonists |
07/07/1994 | CA2152631A1 Bicyclic fibrinogen antagonists |
07/05/1994 | US5326758 Low dose temazepam |
07/05/1994 | CA1330613C Amino acid derivatives |
06/28/1994 | US5324838 Forms complex with metals |
06/28/1994 | US5324726 Benzodiazepine analogs |
06/23/1994 | WO1994013648A1 1,4-benzodiazepine derivatives and their use as cck-modulators |
06/23/1994 | CA2150461A1 1,4-benzodiazepine derivatives and their use as cck-modulators |
06/01/1994 | EP0599444A1 Dual action inhibitors |
05/31/1994 | US5317101 Tricyclic heterocycles |
05/31/1994 | US5317021 Analgesics, anticonvulsants |
05/26/1994 | WO1994011490A2 Products of the inhibition of advanced glycosylation |
05/25/1994 | CN1024665C Ring-substituted 2-amino-1,2,3-tetrahydronaphthalenes and its producing process |
05/18/1994 | EP0597540A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents |
05/17/1994 | US5312625 Fused 7-membered cyclic compound and antipsychotic preparation containing the same |
05/11/1994 | CA2104060A1 Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents |
05/04/1994 | EP0594577A1 Novel potent inducers of terminal differentiation and method of use thereof |
04/28/1994 | WO1994008977A1 Substituted caprolactams and derivatives thereof useful for treatment of aids |
04/27/1994 | EP0593603A1 Bicyclic fibrinogen antagonists |
04/27/1994 | EP0593438A1 Fungicidal compositions, fungicidal compounds, their production and use |
04/14/1994 | WO1994008051A1 Complex combinatorial chemical libraries encoded with tags |
04/13/1994 | EP0591529A1 Novel benzodiazepine derivative |
04/12/1994 | US5302715 For binding to antigens, proteins, polypeptides or other labels for preparation of antibodies useful in immunoassays |
04/12/1994 | US5302620 Bisguanidines and fungicides containing them |
04/12/1994 | US5302370 Form complexes with rhenium and technetium |
04/06/1994 | CN1084849A Dual action inhibitors |
04/05/1994 | US5300522 Condensed heterocyclic compounds and pharmaceutical use thereof |
03/31/1994 | WO1994006291A1 Solid phase and combinatorial synthesis of compounds on a solid support |
03/17/1994 | WO1994005671A1 Fullerene derivatives, method of synthesizing them and their use |
03/17/1994 | CA2144051A1 New fullerene derivatives, method of synthesizing them and their use |
03/08/1994 | US5292743 Fungicidal compositions, fungicidal compounds, their production and use |
02/23/1994 | EP0583433A1 Diphosphine ligands |
02/22/1994 | US5288863 Process for the preparation of high-purity 1-(3-chloro-phenyl)-4-methyl-7,8-dimethoxy-5H-2,3-benzodiazepine |
02/22/1994 | US5288514 Linking a protected 2-aminobenzophenone to a substrate; deprotecting and reacting with an amino acid; cyclization; removal from substrate; screening |
02/17/1994 | WO1994003437A1 Benzodiazepine derivatives |
02/17/1994 | CA2140009A1 Benzodiazepine derivatives |
02/16/1994 | EP0508995B1 Muscarinic receptor antagonists |
02/02/1994 | CN1081442A Benzodiazepines |
01/26/1994 | EP0580402A2 Aminediol protease inhibitors |
01/26/1994 | EP0579797A1 Diphosphine ligands |
01/25/1994 | US5281626 Benzenesulfonamide derivatives |
01/21/1994 | CA2100894A1 Aminediol protease inhibitors |
01/06/1994 | WO1994000438A1 Novel benzodiazepine derivative |
01/06/1994 | CA2138129A1 Novel benzodiazepine derivative |
12/23/1993 | CA2112360A1 Bicyclic fibrinogen antagonists |
12/22/1993 | EP0574781A2 2-Amino-5-heterocyclic-substituted-1,4-benzodiazepines and their use in the treatment of aids |
12/21/1993 | US5272165 2-alkylidene-aminoguanidines and methods of use therefor |
12/17/1993 | CA2098063A1 Benzodiazepines |
12/14/1993 | US5270464 Anti-HIV-1 tetrahydroimidazo[1,4]benzodiazepin-2-(thi) ones |
12/07/1993 | US5268476 Substituted 10bH-oxazolo[3,2-c] [1,3] benzoxazine-2(3H), 5-diones |
12/01/1993 | EP0571851A1 Process for the preparation of terminal nitrogen-heterocyclic substituted acrylic- and methacrylicacid alkylesters |
11/24/1993 | EP0570764A2 Asymmetric hydrogenation |
11/23/1993 | US5264432 5-(1-aminoacyl)-5,10-dihydro-11H-dibenzo[b,e](1,4)diazepin-11-ones |
11/16/1993 | US5262152 Amidrazones and derivatives thereof |
11/09/1993 | US5260339 4-phenyl-1,3-benzodiazepines and 2-amino-α-phenylphenethylamines for treating convulsions and protecting neurons |
11/03/1993 | CN1077952A Carbamate derivatives |
11/02/1993 | US5258381 Inhibitors of glycosylation of proteins, antiaging agents, discoloration inhibition of teeth and storage stability of foods |
10/14/1993 | WO1993020067A1 Benzodiazepine derivatives and protein and polypeptide conjugates thereof |
10/14/1993 | CA2132341A1 Benzodiazepine derivatives and protein and polypeptide conjugates thereof |
10/05/1993 | US5250679 Nonpeptidyl platelet aggregation inhibitors having specificity for the GPIIb III.sub. receptor |
09/30/1993 | WO1993019052A1 3-ureido substituted benzodiazepin-2-ones having cholecystokinin and/or gastrin antagonistic activity and their use in therapy |
09/30/1993 | CA2130196A1 Benzodiazepine derivatives |
09/15/1993 | EP0559793A1 Hiv protease inhibitors |
09/07/1993 | US5243071 2-alkylidene-aminoguanidines and methods of use therefor |