Patents
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
10/1994
10/27/1994WO1994024149A1 1,5-benzodiazepine derivatives having cck antagonistic or agonistic activity
10/19/1994EP0620218A1 Heterocyclic compounds active in gastro-intestinal pathologies
10/19/1994EP0620216A1 Benzamide derivatives and their use as vasopressin antagonists
10/18/1994US5356895 1,4 piperizino inhibitors of non-enzymatic cross-linking of proteins
10/14/1994CA2121112A1 New benzamide derivatives, processes for the preparation thereof and pharmaceutical composition comprising the same
10/13/1994WO1994022840A1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease
10/13/1994WO1994022825A1 Fibrinogen receptor antagonists
10/13/1994CA2159482A1 Fibrinogen receptor antagonists
10/13/1994CA2159442A1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease
10/12/1994EP0619309A1 Process for the preparation of alkylimidazolidone (meth)acrylates
10/11/1994CA1332411C Benzodiazepine analogs
10/11/1994CA1332410C Benzodiazepine analogs
10/05/1994EP0617621A1 Central cholecystokinin antagonists having pharmaceutical activity
10/05/1994EP0617618A1 Aryl-triflates and related compounds
10/05/1994CN1093085A Amine derivatives
09/1994
09/29/1994WO1994011490A3 Products of the inhibition of advanced glycosylation
09/28/1994EP0616532A1 Use of peripheral-type benzodiazepine sites for treatment of cns trauma or disease
09/20/1994US5349086 Alkylation and salt formation
09/15/1994WO1994020473A1 Compound with vasopressin antagonism
09/15/1994DE4308095A1 Prodrug derivatives of pharmaceutical agents with hydroxyl groups, process for their preparation and their use
09/01/1994WO1994019329A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
09/01/1994WO1994014776A3 Bicyclic fibrinogen antagonists
09/01/1994CA2156594A1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
08/1994
08/30/1994US5342839 Useful for therapy of oxygen deficiency diseases of the brain
08/23/1994CA1331564C Redox systems for brain-targeted drug delivery
08/17/1994EP0610334A1 NONPEPTIDYL INTEGRIN INHIBITORS HAVING SPECIFICITY FOR THE GPII b?III a? RECEPTOR.
08/10/1994EP0609306A1 Benzodiazepine derivatives and their use as antagonists of cholecystokinin and/or gastrin receptors
07/1994
07/27/1994EP0607697A2 DILAZEP for reduction of elevated intraocular pressure
07/27/1994EP0607355A1 3-ureido-benzodiazepinones useful as antagonists of cck or of gastrine.
07/27/1994EP0607334A1 Cyclic ureas and analogues useful as retroviral protease inhibitiors.
07/27/1994EP0607129A1 Methylpiperazinoazepine derivatives, their preparation and use.
07/21/1994WO1994015924A1 Cholecystokinin antagonists
07/20/1994EP0606658A1 Substituted N-aminoalkylmethansulphoamides as antispasmodic agents
07/19/1994US5331006 Amino acid analogs as CCK antagonists
07/14/1994CA2113032A1 Substituted n-aminoalkylmethane sulfanilide as antispasmodica
07/13/1994EP0605639A1 Air treatment plant for foodstuff comprising a trough with an adjustable width.
07/07/1994WO1994014776A2 Bicyclic fibrinogen antagonists
07/07/1994CA2152631A1 Bicyclic fibrinogen antagonists
07/05/1994US5326758 Low dose temazepam
07/05/1994CA1330613C Amino acid derivatives
06/1994
06/28/1994US5324838 Forms complex with metals
06/28/1994US5324726 Benzodiazepine analogs
06/23/1994WO1994013648A1 1,4-benzodiazepine derivatives and their use as cck-modulators
06/23/1994CA2150461A1 1,4-benzodiazepine derivatives and their use as cck-modulators
06/01/1994EP0599444A1 Dual action inhibitors
05/1994
05/31/1994US5317101 Tricyclic heterocycles
05/31/1994US5317021 Analgesics, anticonvulsants
05/26/1994WO1994011490A2 Products of the inhibition of advanced glycosylation
05/25/1994CN1024665C Ring-substituted 2-amino-1,2,3-tetrahydronaphthalenes and its producing process
05/18/1994EP0597540A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents
05/17/1994US5312625 Fused 7-membered cyclic compound and antipsychotic preparation containing the same
05/11/1994CA2104060A1 Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents
05/04/1994EP0594577A1 Novel potent inducers of terminal differentiation and method of use thereof
04/1994
04/28/1994WO1994008977A1 Substituted caprolactams and derivatives thereof useful for treatment of aids
04/27/1994EP0593603A1 Bicyclic fibrinogen antagonists
04/27/1994EP0593438A1 Fungicidal compositions, fungicidal compounds, their production and use
04/14/1994WO1994008051A1 Complex combinatorial chemical libraries encoded with tags
04/13/1994EP0591529A1 Novel benzodiazepine derivative
04/12/1994US5302715 For binding to antigens, proteins, polypeptides or other labels for preparation of antibodies useful in immunoassays
04/12/1994US5302620 Bisguanidines and fungicides containing them
04/12/1994US5302370 Form complexes with rhenium and technetium
04/06/1994CN1084849A Dual action inhibitors
04/05/1994US5300522 Condensed heterocyclic compounds and pharmaceutical use thereof
03/1994
03/31/1994WO1994006291A1 Solid phase and combinatorial synthesis of compounds on a solid support
03/17/1994WO1994005671A1 Fullerene derivatives, method of synthesizing them and their use
03/17/1994CA2144051A1 New fullerene derivatives, method of synthesizing them and their use
03/08/1994US5292743 Fungicidal compositions, fungicidal compounds, their production and use
02/1994
02/23/1994EP0583433A1 Diphosphine ligands
02/22/1994US5288863 Process for the preparation of high-purity 1-(3-chloro-phenyl)-4-methyl-7,8-dimethoxy-5H-2,3-benzodiazepine
02/22/1994US5288514 Linking a protected 2-aminobenzophenone to a substrate; deprotecting and reacting with an amino acid; cyclization; removal from substrate; screening
02/17/1994WO1994003437A1 Benzodiazepine derivatives
02/17/1994CA2140009A1 Benzodiazepine derivatives
02/16/1994EP0508995B1 Muscarinic receptor antagonists
02/02/1994CN1081442A Benzodiazepines
01/1994
01/26/1994EP0580402A2 Aminediol protease inhibitors
01/26/1994EP0579797A1 Diphosphine ligands
01/25/1994US5281626 Benzenesulfonamide derivatives
01/21/1994CA2100894A1 Aminediol protease inhibitors
01/06/1994WO1994000438A1 Novel benzodiazepine derivative
01/06/1994CA2138129A1 Novel benzodiazepine derivative
12/1993
12/23/1993CA2112360A1 Bicyclic fibrinogen antagonists
12/22/1993EP0574781A2 2-Amino-5-heterocyclic-substituted-1,4-benzodiazepines and their use in the treatment of aids
12/21/1993US5272165 2-alkylidene-aminoguanidines and methods of use therefor
12/17/1993CA2098063A1 Benzodiazepines
12/14/1993US5270464 Anti-HIV-1 tetrahydroimidazo[1,4]benzodiazepin-2-(thi) ones
12/07/1993US5268476 Substituted 10bH-oxazolo[3,2-c] [1,3] benzoxazine-2(3H), 5-diones
12/01/1993EP0571851A1 Process for the preparation of terminal nitrogen-heterocyclic substituted acrylic- and methacrylicacid alkylesters
11/1993
11/24/1993EP0570764A2 Asymmetric hydrogenation
11/23/1993US5264432 5-(1-aminoacyl)-5,10-dihydro-11H-dibenzo[b,e](1,4)diazepin-11-ones
11/16/1993US5262152 Amidrazones and derivatives thereof
11/09/1993US5260339 4-phenyl-1,3-benzodiazepines and 2-amino-α-phenylphenethylamines for treating convulsions and protecting neurons
11/03/1993CN1077952A Carbamate derivatives
11/02/1993US5258381 Inhibitors of glycosylation of proteins, antiaging agents, discoloration inhibition of teeth and storage stability of foods
10/1993
10/14/1993WO1993020067A1 Benzodiazepine derivatives and protein and polypeptide conjugates thereof
10/14/1993CA2132341A1 Benzodiazepine derivatives and protein and polypeptide conjugates thereof
10/05/1993US5250679 Nonpeptidyl platelet aggregation inhibitors having specificity for the GPIIb III.sub. receptor
09/1993
09/30/1993WO1993019052A1 3-ureido substituted benzodiazepin-2-ones having cholecystokinin and/or gastrin antagonistic activity and their use in therapy
09/30/1993CA2130196A1 Benzodiazepine derivatives
09/15/1993EP0559793A1 Hiv protease inhibitors
09/07/1993US5243071 2-alkylidene-aminoguanidines and methods of use therefor
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