| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 10/10/2001 | EP1140786A1 Reductive alkylation of secondary amines with hydrosilane |
| 10/10/2001 | CN1072664C Novel aryl glycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compound |
| 10/04/2001 | WO2001072960A2 Il-8 receptor antagonists |
| 10/04/2001 | EP0830350B1 n-(1-alkyl-5-phenyl-2,3,4,5-tetrahydro-1h-benzo[b][1,5]diazepin-3-yl)-acetamides |
| 10/04/2001 | CA2403787A1 Il-8 receptor antagonists |
| 10/03/2001 | CN1315953A Process for preparation of imidazodiazepine intermediates |
| 09/20/2001 | US20010023305 By direct reaction of an amine with an alpha, gamma-dihaloalkane or an alpha, gamma-dihaloalkene; tertiary aminoalkylorganometallics can be made by then reacting the tert haloalkylamines with an alkali metals |
| 09/19/2001 | EP1134220A1 Benzoxazole derivatives and drugs containing the same as the active ingredient |
| 09/19/2001 | EP0538297B1 Antiviral tetrahydroimidazo 1,4]benzodiazepin-2-(thio)ones |
| 09/19/2001 | CN1313280A Benzheterocyclic derivatives |
| 09/18/2001 | US6291452 Cholecystokinin antagonists. |
| 09/13/2001 | WO2001066534A2 Cyclic and bicyclic diamino histamine-3 receptor antagonists |
| 09/13/2001 | WO2001066062A2 Process for preparing pure crystalline lorazepam |
| 09/13/2001 | US20010021388 Cyclization of a triether with a diamine compound |
| 09/13/2001 | CA2401928A1 Process for preparing pure crystalline lorazepam |
| 09/12/2001 | EP1131039A2 Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress |
| 09/07/2001 | WO2001055111A8 Biaryl compounds, their preparation and their use in therapy |
| 09/06/2001 | US20010020093 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermeidate |
| 09/06/2001 | US20010020019 Novel halo-alkoxycarbonyl prodrugs |
| 09/05/2001 | EP0832061B1 Benzamide derivatives and their use as vasopressin antagonists |
| 09/05/2001 | CN1311779A Succinoylamino lactams as inhibitors and as A beta protein production |
| 09/04/2001 | US6284767 Retroviral protease inhibiting compounds |
| 08/30/2001 | WO2001015656A3 Tricyclic compounds and their uses as antiarrhythmic antifibrillatory and defibrillatory agents |
| 08/29/2001 | CN1310629A Coadministration of ACAT and MMP inhibitors for the treatment of atherosclerotic lesions |
| 08/28/2001 | US6281353 Method of making diazepine derivatives |
| 08/23/2001 | WO2001060826A2 SUCCINOYLAMINO CARBOCYCLES AND HETEROCYCLES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
| 08/23/2001 | US20010016583 Therapeutic application of pro-apoptotic benzodiazepines |
| 08/23/2001 | CA2395862A1 Succinoylamino carbocycles and heterocycles as inhibitors of a.beta. protein production |
| 08/22/2001 | EP1124556A1 Use of optically pure (r)-tofisopam for treating and preventing anxiety disorders and composition thereof |
| 08/22/2001 | CN1309122A Process for synthesizing 2-alkoxycarbonylmethyl-1,4-benzodiazepine |
| 08/16/2001 | WO2000066106A3 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis |
| 08/16/2001 | US20010014738 Process for the preparation of imidazodiazepine intermediates |
| 08/16/2001 | EP1143946A3 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis |
| 08/16/2001 | EP1123928A1 1,5-benzodiazepine compounds, process for producing the same, and medicine |
| 08/15/2001 | CN1308606A Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use pharmaceutical preparations comprising them |
| 08/14/2001 | CA2162838C Process for preparing an alkylimidazolidone (meth)acrylate |
| 08/09/2001 | WO2001056563A1 Adamantyl derivatives as anti-cancer agents |
| 08/08/2001 | CN1307567A 1,5 benzodiazepine derivatives |
| 08/02/2001 | WO2001055121A1 Azepine derivatives |
| 08/02/2001 | WO2001055111A1 Biaryl compounds, their preparation and their use in therapy |
| 08/02/2001 | US20010011087 Vitronectin receptor antagonists, their preparation and their use |
| 07/31/2001 | US6267973 Ectoin and ectoin derivatives as moisturizers in cosmetics |
| 07/26/2001 | WO2001053258A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same |
| 07/26/2001 | WO2001053255A1 Gamma-secretase inhibitors |
| 07/26/2001 | CA2398409A1 Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound |
| 07/26/2001 | CA2397543A1 Gamma-secretase inhibitors |
| 07/18/2001 | EP1115758A2 Polymerization of olefins |
| 07/12/2001 | WO2001049681A1 A method for the preparation of substituted benzene derivatives |
| 07/12/2001 | WO2001002358A3 Cyclized amide derivatives for treating or preventing neuronal damage |
| 07/10/2001 | US6258948 An n-acylamino compound; antiinflammatory agents, autoimmune diseases |
| 07/10/2001 | CA2226691C Combinatorial 1,4-benzodiazepin-2,5-dione library |
| 07/05/2001 | WO2001047899A1 Substituted piperazine derivatives as mtp inhibitors |
| 07/05/2001 | WO2001047510A2 Methods and compositions related to modulators of annexin and cartilage homeostasis |
| 07/05/2001 | DE19963235A1 Substituierte Piperazinderivate, ihre Herstellung und ihre Verwendung als Arzneimittel Substituted piperazine derivatives, their preparation and their use as medicaments |
| 07/05/2001 | CA2394644A1 Substituted piperazine derivatives,the preparation thereof and their useas medicaments |
| 07/04/2001 | EP1112250A1 Therapeutic compounds and methods |
| 07/03/2001 | US6255481 Treating aqueous suspension of anhydrous nevirapine with hydrochloric acid then treating with sodium hydroxide yields the free base as a precipitate/hemihydrate which is then filtered from solution and water washed |
| 06/27/2001 | CN1301257A Substituted 1,3-diaza-2-(thi)oxo-cycloalkanes |
| 06/27/2001 | CN1301156A Treatment of T-Helper cell tyre 2 mediated immune diseases with retinoid antagonists |
| 06/26/2001 | US6252067 Reacting 2,2,2-trifluoromethane sulfonate with corresponding amide compound in presence of potassium carbonate; refluxing |
| 06/26/2001 | US6251949 Oxime derivatives, hydrazone derivatives and use thereof |
| 06/21/2001 | WO2001044190A1 Anthracene derivatives as anti-cancer agents |
| 06/21/2001 | CA2395170A1 Anti-cancer agents (iii) |
| 06/14/2001 | WO2001042243A2 Protein kinase inhibitors |
| 06/14/2001 | WO2001002373A8 Dihydrobenzodiazepins and their use for treating dyslipidemia |
| 06/13/2001 | EP1105392A1 Process for the preparation of imidazodiazepine intermediates |
| 06/13/2001 | EP1105359A1 Solid phase synthesis of compounds by carbon-carbon bond forming mitsunobu reactions |
| 06/12/2001 | US6245767 Cardiovascualr disorders |
| 06/07/2001 | WO2001040197A1 Calcium salts of 1,5-benzodiazepine derivatives, process for producing the salts and drugs containing the same |
| 06/06/2001 | EP1104754A1 Novel sulfonyl derivatives |
| 05/30/2001 | EP1102752A1 Succinoylamino lactams as inhibitors of a beta protein production |
| 05/30/2001 | EP1102743A1 Amide derivatives which are useful as cytokine inhibitors |
| 05/29/2001 | US6239131 1,5 Benzodiazepine derivatives |
| 05/25/2001 | WO2000039081A3 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
| 05/23/2001 | EP1100504A2 Pharmaceutical compositions and their uses for treatment of demyelinating disorders |
| 05/22/2001 | US6235778 Anticoagulants |
| 05/16/2001 | EP1098897A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation |
| 05/16/2001 | EP1098662A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions |
| 05/15/2001 | CA2238978C Retroviral protease inhibiting compounds |
| 05/10/2001 | WO2001004122A3 New 2,3-benzodiazepine derivatives |
| 05/09/2001 | EP0855397B1 (r)-5-bromo-n-(1-ethyl-4-methylhexahydro-1h-1,4-diazepin-6-yl)-2-methoxy-6-methylamino-3-pyridine-carboxamide, process for producing the same and medicinal composition containing the same |
| 05/03/2001 | WO2001030769A2 Process for alkylation of benzodiazepindione compounds |
| 05/02/2001 | EP1095016A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
| 05/02/2001 | CN1293666A Benzenesulfonamide-derivatives and their use as medicaments |
| 05/02/2001 | CN1293663A 2,3,4,5-tetrahydro-1H-[1,4] benzodiazepine-3-hydroxamix acids as matrix metal-protease |
| 05/01/2001 | US6225465 Process for the aminocarbonylation of benzazepines and benzodiazepines |
| 05/01/2001 | CA2037299C Gamma emitting, cck-a antagonists for pancreatic imaging |
| 04/26/2001 | WO2001029012A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists |
| 04/26/2001 | WO2001029011A2 Benzodiazepine derivatives as metabotropic glutamate receptor antagonists |
| 04/26/2001 | WO2001029005A1 Bicyclic vasopressin agonists |
| 04/26/2001 | CA2387886A1 Bicyclic vasopressin agonists |
| 04/25/2001 | EP1093372A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING $g(b)-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS |
| 04/25/2001 | CN1064960C Method for preparation of nitrazepam |
| 04/24/2001 | US6222032 Conducting the c-alkylation or n-alkylation reaction in the presence of a slightly nucleophilic strong base comprising a phosphorus compound |
| 04/19/2001 | WO2001027108A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
| 04/19/2001 | WO2001027102A1 Substituted diazepanes |
| 04/19/2001 | WO2001027091A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
| 04/19/2001 | CA2387493A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production |
| 04/19/2001 | CA2384544A1 Amino lactam sulfonamides as inhibitors of a.beta. protein production |
| 04/18/2001 | EP1091944A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors |