| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 11/04/1999 | CA2328934A1 Solid supported synthesis of sulfonated 2-oxopiperazines |
| 10/28/1999 | WO1999054321A1 Substituted diamines and their use as cell adhesion inhibitors |
| 10/27/1999 | EP0951466A2 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds |
| 10/21/1999 | DE19816889A1 New piperazine derivatives useful in treatment of e.g. cardiovascular, renal and central nervous system disorders, obesity and diabetes, in antibody production and as analytical and diagnostics aids |
| 10/20/1999 | EP0949926A1 Benzodiazepine hydrazide derivatives as inhibitors of hiv integrase |
| 10/20/1999 | CN1232457A 1,4-heterocyclic metalloprotease inhibitors |
| 10/19/1999 | US5968736 Methods for recording the reaction history of a solid support |
| 10/19/1999 | US5968478 N- methyl piperazine compounds having dopamine receptor affinity |
| 10/12/1999 | CA2134430C Process for the preparation of alkyl-imidazolidone (meth)acrylate |
| 10/07/1999 | WO1999050237A1 Sulfonamide derivatives and drugs containing the same as the active ingredient |
| 10/07/1999 | CA2325997A1 Sulfonamide derivatives and drugs containing the same as the active ingredient |
| 10/06/1999 | EP0946180A1 Method for stimulating bone formation |
| 10/05/1999 | US5962451 Gastrointestinal disorders; antiulcer agent; anticancer agents; side-effect reduction |
| 10/05/1999 | US5962337 Attaching amino-protected alpha aminoacid which may be n-alkylated to solid support via carboxyl group, cleaving amino protecting group, acylating with 2-azidobenzoyl chloride, cyclizing via aza-wittig ring closure |
| 09/29/1999 | EP0945445A1 1,5-benzodiazepine derivatives |
| 09/29/1999 | EP0944590A2 Aminoguanidines and alkoxyguanidines as protease inhibitors |
| 09/29/1999 | CN1230111A Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents |
| 09/29/1999 | CN1230110A Cell adhesion inhibitors |
| 09/23/1999 | WO1999047508A1 Benzenesulfonamide-derivatives and their use as medicaments |
| 09/23/1999 | CA2323783A1 Benzenesulfonamide-derivatives and their use as medicaments |
| 09/22/1999 | CN1229412A Inhibitors of interleukin-1'beta' converting emzyme |
| 09/16/1999 | WO1999046248A1 1,2-diazepane derivatives as interleukin-1beta converting enzyme inhibitors |
| 09/15/1999 | CN1228773A Heterocyclic metalloprotease inhibitors |
| 09/15/1999 | CN1228772A Heterocyclic metalloprotease inhibitors |
| 09/15/1999 | CN1228771A 1,3-diheterocyclic metalloprotease inhibitors |
| 09/14/1999 | US5952352 Heterocyclic compounds |
| 09/14/1999 | CA1340734C Substituted bridged-diazabicycloalkyl quinolone carboxylic acids |
| 09/08/1999 | EP0940388A1 Oxime derivatives, hydrazone derivatives, and use thereof |
| 09/02/1999 | WO1999043662A1 Solid support synthesis of 2-oxopiperazines |
| 09/02/1999 | CA2321302A1 Solid support synthesis of 2-oxopiperazines |
| 09/01/1999 | CN1227550A Troponyl piperazines as selective dopamine D4 receptor ligands |
| 08/31/1999 | US5945415 (R)-5-bromo-N-(1-ethyl-4-methylhexahydro-1H-1,4-diazepin-6-yl)-2-methoxy-6-methylamino-3-pyridinecarboxamide, process for producing the same and medicinal composition containing the same |
| 08/25/1999 | EP0937067A1 1-(3-aminoindazol-5-yl)-3-phenylmethyl-cyclic ureas useful as hiv protease inhibitors |
| 08/25/1999 | EP0937053A1 Sustained-release derivatives of hydroxylated analogs of substituted 1- 2 bis(aryl)methoxy]ethyl]-piperazines and -homopiperazines and their use as noncompetitive antagonists of dopamine reuptake |
| 08/24/1999 | US5942614 Process to produce midazolam |
| 08/24/1999 | US5942506 1- 2-(substituted vinyl)!-5H-2,3-benzodiazepine derivatives |
| 08/19/1999 | WO1999024024A3 Treatment of t-helper cell type 2 mediated immune diseases with retinoid antagonists |
| 08/17/1999 | US5939414 Benzodiazepine hydrazide derivatives as inhibitors of HIV integrase |
| 08/17/1999 | US5939412 Bicyclic fibrinogen antagonists |
| 08/12/1999 | WO1999040075A1 Sulfonamide derivatives, process for producing the same and utilization thereof |
| 08/12/1999 | CA2317017A1 Sulfonamide derivatives, their production and use |
| 08/11/1999 | EP0934282A1 1,4-benzodiazepinones and their uses as cck antagonists |
| 08/11/1999 | CN1225621A Inhibition of matrix metalloproteases by substituted biaryl oxobutyric acids |
| 08/05/1999 | WO1999038844A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound |
| 08/05/1999 | CA2318601A1 Method for preparing an n-[(aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound |
| 07/29/1999 | WO1999037625A1 2,3,4,5-tetrahydro-1h-[1,4]-benzodiazepine-3-hydroxamic acids as matrix metalloproteinase inhibitors |
| 07/29/1999 | WO1999019306A3 2,3-benzodiazepin-2-one derivatives, their preparation and their use as inhibitors of protein tyrosine kinases |
| 07/29/1999 | CA2317546A1 2,3,4,5-tetrahydro-1h-¬1,4|-benzodiazepine-3-hydroxamic acids as matrix metalloproteinase inhibitors |
| 07/27/1999 | US5929069 Compounds activating pharmacological effects of retinoids |
| 07/27/1999 | CA2032355C Process for the preparation of alkyl imidazolidone (meth)acrylate |
| 07/21/1999 | EP0929537A1 Troponyl piperazines as selective dopamine d4 receptor ligands |
| 07/20/1999 | US5925635 N-(amidinophenyl) cyclourea analogs as factor XA inhibitors |
| 07/13/1999 | US5922892 Process to produce midazolam |
| 07/07/1999 | EP0927168A1 1,3-diheterocyclic metalloprotease inhibitors |
| 07/06/1999 | US5919954 Stereoselective process for producing dihydro-2,3-benzodiazepine derivatives |
| 07/06/1999 | CA2120594C Process for the preparation of (meth)acrylate(s) of alkylimidazolidone |
| 07/01/1999 | WO1999032461A1 1,4-diazacycloheptane derivatives |
| 07/01/1999 | CA2312070A1 1,4-diazacycloheptane derivatives |
| 06/30/1999 | EP0926138A1 Diamide compounds and drugs containing the same |
| 06/30/1999 | EP0925287A1 Heterocyclic metalloprotease inhibitors |
| 06/30/1999 | EP0756602B1 Cck or gastrin modulating 5-heterocyclic-1,5-benzodiazepines |
| 06/24/1999 | WO1999018085A3 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate |
| 06/23/1999 | EP0923563A1 1,4-heterocyclic metallprotease inhibitors |
| 06/23/1999 | EP0923561A1 Heterocyclic metalloprotease inhibitors |
| 06/23/1999 | EP0923530A1 Inhibition of matrix metalloproteases by substituted biaryl oxobutyric acids |
| 06/23/1999 | CN1220262A 7-phenyl-1,4-stable derivative, its preparing method and medicine containing said compound |
| 06/23/1999 | CN1220261A Novel process for preparation of clonidine derivatives |
| 06/22/1999 | US5914332 Retroviral protease inhibiting compounds |
| 06/17/1999 | WO1999029324A1 Preventives/remedies for diabetes |
| 06/17/1999 | CA2312716A1 Medicament for prevention and treatment of diabetes |
| 06/16/1999 | EP0922696A2 Urea derivatives of alpha, omega-diaminoacids and peptides |
| 06/09/1999 | EP0920312A1 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents |
| 06/09/1999 | EP0755514A4 Complex combinatorial chemical libraries encoded with tags |
| 06/03/1999 | WO1999026661A1 A covalent conjugate of clozapine with a fatty acid and its use for treating schizophrenia |
| 06/02/1999 | EP0918773A1 Process for the production of 8-chloro-6-(2-fluorophenyl)-1-methyl-4h-imidazo 1,5-a]benzodiazepine |
| 05/26/1999 | EP0917462A1 Cell adhesion inhibitors |
| 05/20/1999 | WO1999024428A1 Oxazolidinone derivatives and pharmaceutical compositions |
| 05/20/1999 | WO1999024024A2 Treatment of t-helper cell type 2 mediated immune diseases with retinoid antagonists |
| 05/20/1999 | CA2303959A1 Oxazolidinone derivatives and pharmaceutical compositions |
| 05/12/1999 | EP0914605A1 Molecular model for vla-4 inhibitors |
| 05/12/1999 | EP0914319A1 Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists |
| 05/12/1999 | EP0583433B1 Diphosphine ligands |
| 05/12/1999 | CN1216537A Compounds with growth hormone releasing properties |
| 05/06/1999 | WO1999021834A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors |
| 04/29/1999 | WO1999020599A1 Pharmaceutically active compounds and methods of use |
| 04/29/1999 | WO1999020281A1 Novel benzodiazepine derivatives as antiarrhythmic agents |
| 04/29/1999 | CA2307597A1 Pharmaceutically active compounds and methods of use |
| 04/29/1999 | CA2306960A1 Novel benzodiazepine derivatives as antiarrhythmic agents |
| 04/28/1999 | EP0911320A2 1,2-Di-substituted benzenecarboxamide derivative, hair growth promoter and external composition for skin using the same |
| 04/28/1999 | CN1215054A Bychclic fibrinogen antagonists |
| 04/28/1999 | CN1215051A 'Alpha' substituted benzyl propionate derivant and medicine containing same |
| 04/22/1999 | WO1999019306A2 2,3-benzodiazepin-2-one derivatives, their preparation and their use as inhibitors of protein tyrosine kinases |
| 04/22/1999 | WO1999018967A1 Analgesic compositions |
| 04/22/1999 | WO1999018951A1 Inhibitors of farnesyl protein transferase |
| 04/22/1999 | WO1999011624B1 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
| 04/22/1999 | CA2304473A1 Inhibitors of farnesyl protein transferase |
| 04/21/1999 | EP0579797B1 Diphosphine ligands |
| 04/21/1999 | CN1214685A Inhibitors of farnesyl protein transferase |
| 04/15/1999 | WO1999018085A2 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate |
| 04/15/1999 | WO1999017776A1 Novel cycloalkenyl substituted compounds |