| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 06/06/2002 | WO2002044180A1 Lactam compounds and medicinal use thereof |
| 06/05/2002 | EP1210941A2 Pharmaceutical compositions containing ritonavir (ABT-538) in combination with indinavir (MK-639) and their use for treating AIDS |
| 06/05/2002 | EP1210338A2 1,4-diazepine derivatives for the treatment of diseases related to the central nervous system |
| 06/05/2002 | EP1210332A1 Bleach boosting components, compositions and laundry methods |
| 06/04/2002 | US6399599 Substituted 2-oxo-1,4-diazacycloalkanes |
| 06/04/2002 | US6399598 Diheterocyclic metalloprotease inhibitors |
| 05/30/2002 | WO2001098280A3 5h-2,3-benzodiazepine antagonists of excitatory amino acid receptors |
| 05/29/2002 | EP1208069A1 Process for catalyzing the oxidation of organic compounds |
| 05/23/2002 | US20020062022 Processes for preparation of cyclopenta [b] [1,4] diazepino [6,7,1-hi] indoles and derivatives |
| 05/23/2002 | US20020061887 For therapy and prophylaxis of cardiovascular diseases such as hypertension, angina pectoris, cardiac insufficiency, thromboses or atherosclerosis |
| 05/23/2002 | US20020061878 Diazacycloalkanedione derivatives |
| 05/23/2002 | US20020061874 Substituted lactam; gamma-secretase inhibitor; decreases production of beta-amyloid; treatment for Altzheimer's and Down's syndrome |
| 05/22/2002 | CN1350530A 酰胺衍生物 Amide derivatives |
| 05/22/2002 | CN1350520A Cell adhesive-inhibiting anti inflammatory and immune-suppressive compounds |
| 05/16/2002 | US20020058784 Generation of preferential compound; obtain sample of diamino acid such as 2,3 diaminopropionic acid, incubate with compound with free amino group, recover urein |
| 05/16/2002 | US20020058689 Process for the preparation of 1, 2, 3, 4, 8, 9, 10, 10a-octahydro-7bH-cyclopenta[b] [1, 4]diazepino[6, 7, 1-hi]indole derivatives |
| 05/15/2002 | EP1204644A1 Synthesis of substituted amidines |
| 05/15/2002 | CN1348956A Substituted diazacycloheptane compound, medicine composite contg. same and the use thereof |
| 05/14/2002 | US6387895 Bone disorders; cardiovascular disorders |
| 05/14/2002 | US6387389 Sustained-release derivatives of hydroxylated analogs of substituted 1-[2[bis(aryl)methoxy]ethyl]-piperazines and -homopiperazines and their use |
| 05/10/2002 | WO2002036073A2 Receptor antagonist-lipid conjugates and delivery vehicles containing same |
| 05/09/2002 | US20020055630 Process for preparation of cyclopenta [b] [1,4] diazepino [6,7,1-hi] indole derivatives |
| 05/09/2002 | US20020055504 Acylating a cyclopentaindolemethylamine and cyclizing and reducing the product |
| 05/09/2002 | US20020055501 Treatment of neurological disorders related to beta -amyloid production such as Alzheimer's disease and Down's Syndrome. |
| 05/08/2002 | EP1202988A2 Novel integrin receptor antagonists |
| 05/08/2002 | EP1202977A2 Process for manufacturing diazepine derivatives |
| 05/08/2002 | CN1348455A Pyrazolobenzodiazepines as CDK2 inhibitors |
| 05/08/2002 | CN1347881A 法呢基蛋白转移酶抑制剂 Farnesyl protein transferase inhibitor |
| 05/02/2002 | WO2001082913A3 Use of benzamide derivatives for the treatment of high ocular tension and glaucoma |
| 05/02/2002 | US20020052364 Condensed 2,3-benzodiazepine derivatives and their use as AMPA-receptor inhibitors |
| 05/02/2002 | US20020052360 Hydroxyalkanoylaminolactams and related structures as inhibitors of a beta protein production |
| 05/02/2002 | US20020052358 Methods and compositions related to modulators of annexin and cartilage homeostasis |
| 05/02/2002 | EP1201649A1 Glucocorticoid receptor modulators |
| 05/02/2002 | EP1200442A1 2,3-benzodiazepine derivatives |
| 04/30/2002 | CA2059787C Hydrazine derivative and pesticidal composition comprising said derivative as an effective ingredient |
| 04/25/2002 | US20020049201 Sulfonamide inhibitors of aspartyl protease |
| 04/25/2002 | US20020049194 A benzoazepin or benzodiazepin derivatives, shows excellent anti-vasopressin activity, vasopressin agonistic activity and oxytocin antagonistic activity, and are useful as antagonist |
| 04/25/2002 | US20020049148 Bleach catalyst and composition and method for bleaching a substrate |
| 04/24/2002 | EP1199308A2 Process for the preparation of imidazodiazepine intermediates |
| 04/18/2002 | WO2002030912A1 Benzodiazepine derivatives as inhibitors of gamma secretase |
| 04/18/2002 | WO2001066062A3 Process for preparing pure crystalline lorazepam |
| 04/18/2002 | WO2001015656A9 Tricyclic compounds and their uses as antiarrhythmic antifibrillatory and defibrillatory agents |
| 04/18/2002 | WO2000066106A9 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis |
| 04/18/2002 | US20020045753 E.g., (S)-N-(4-(4-((3,4-dihydro-6-hydroxy-2,5,7,8-tetramethyl-2H-1-benzopyran-2 -yl)-carbonyl)-1-piperazinyl)phenyl)-2-thiophenecarboximidamide , or a salt thereof. |
| 04/18/2002 | CA2424812A1 Benzodiazepine derivatives as inhibitors of gamma secretase |
| 04/17/2002 | EP1196418A1 METHOD FOR PREPARING SUBSTITUTED 1,4]DIAZEPINO 6,7,1- i hi /i ]INDOL-4-ONES |
| 04/17/2002 | EP1196404A1 Piperazine derivatives as modulators of chemokine receptor activity |
| 04/17/2002 | EP1196395A1 Cyclized amino acid derivatives |
| 04/17/2002 | EP0888313B1 2,3-benzodiazepine derivatives and their use as ampa-receptor inhibitors |
| 04/17/2002 | CN1345308A Acetylenic alpha-amino acid based sulfonamide hydroxamic acid TACE inhibitors |
| 04/16/2002 | US6372733 Hexahydro-5-imino-1,4-1,4-thiazepine derivatives as inhibitors of nitric oxide synthases |
| 04/11/2002 | WO2002028842A2 Diazacycloalkanedione derivatives which are useful as lfa-1 antagonist |
| 04/11/2002 | WO2001019797A3 HYDROXYALKANOYL AMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
| 04/11/2002 | US20020042511 New derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them |
| 04/11/2002 | US20020042414 Antiallergens |
| 04/11/2002 | CA2424282A1 Diazacycloalkanedione derivatives which are useful as lfa-1 antagonist |
| 04/09/2002 | US6369221 Anticonvulsants, antiischemic agents; brain and nervous system disorder treatment |
| 04/09/2002 | CA2120229C Methylpiperazinoazepine derivatives, their preparation and their use |
| 04/04/2002 | US20020039998 Administering to human therapeutically effective amount of a combination of drug which is metabolized by cytochrome p450 monooxygenase or pharmaceutically acceptable salt thereof and ritonavir |
| 04/03/2002 | EP1192148A1 Thiochroman derivatives resisting neurological disorders |
| 04/03/2002 | EP1192141A1 1,4-diazacycloheptane derivatives as neuroprotective agents |
| 03/28/2002 | US20020037892 Bis-arylsulfones |
| 03/27/2002 | EP1189890A1 Dihydrobenzodiazepins and their use for treating dyslipidemia |
| 03/27/2002 | CN1342161A Tricyclic inhibitors of poly(ADP-ribose) polymerases |
| 03/26/2002 | US6362193 Antiinflammatory agents |
| 03/21/2002 | WO2002022598A1 Quinolinone derivatives as tyrosine kinase inhibitors |
| 03/21/2002 | WO2002022577A2 Hydroxamate derivatives useful as deacetylase inhibitors |
| 03/20/2002 | EP1187810A2 Heterocyclic analgesic compounds and their use |
| 03/20/2002 | EP1143796A4 Complex of ras-farnesyltransferase inhibitor and sulfobutylether-7-beta-cyclodextrin or 2-hydroxypropyl-beta-cyclodextrin and method |
| 03/20/2002 | EP0944590B1 Aminoguanidines and alkoxyguanidines as protease inhibitors |
| 03/20/2002 | EP0888356B1 Condensed 2,3-benzodiazepine derivatives and their use as ampa-receptor inhibitors |
| 03/14/2002 | WO2002020501A2 Polyarylcarboxamides useful as lipid lowering agents |
| 03/14/2002 | WO2002020477A1 Apoptosis inhibitors |
| 03/14/2002 | US20020032187 Method for stimulating bone formation |
| 03/13/2002 | EP1185529A1 Pyrazolobenzodiazepines as cdk2 inhibitors |
| 03/13/2002 | EP1185512A2 INHIBITORS OF FACTOR Xa |
| 03/13/2002 | EP1185511A2 Inhibitors of factor xa |
| 03/07/2002 | WO2002018327A2 Guanidinobenzamides as mc4-r agonists |
| 03/07/2002 | WO2000069835A3 Process for manufacturing diazepine derivatives |
| 03/06/2002 | EP1183243A1 Short-acting benzodiazepines |
| 03/06/2002 | EP1183242A2 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors |
| 03/06/2002 | EP0906907B1 Compounds potentiating retinoid |
| 03/06/2002 | EP0728748B1 Benzodiazepine derivatives |
| 03/06/2002 | CN1338456A Benzodiazapine compounds containing imidazole propanamido and its preparing process and application |
| 03/05/2002 | US6352982 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists |
| 03/05/2002 | US6352981 Treat disorders which respond to dopamine d.sub.3 ligands such as schistosomiasis, schizophrenia, depression, neuroses or psychoses |
| 02/28/2002 | US20020025958 Psychological disorders |
| 02/28/2002 | US20020025955 Substituted lactams as inhibitors of A beta protein production |
| 02/27/2002 | EP1181279A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof |
| 02/27/2002 | CN1337952A 2,3,4,5-tetrahydro-1H-[1,4] benzodiazepine-3-hydroxamic acid as matrix metalloproteinase inhibitors |
| 02/26/2002 | US6350870 Suspension a lorazepam solvate in solvent; desolventizing |
| 02/21/2002 | WO2001072960A3 Il-8 receptor antagonists |
| 02/21/2002 | WO2001047510A3 Methods and compositions related to modulators of annexin and cartilage homeostasis |
| 02/21/2002 | US20020022636 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
| 02/14/2002 | US20020019013 Combined resin method for high-speed synthesis of combinatorial libraries |
| 02/13/2002 | EP0861250B1 Amidine and isothiourea derivatives as inhibitors of nitric oxide synthase |
| 02/13/2002 | EP0691961B1 Substituted caprolactams and derivatives thereof useful for treatment of hiv disease |
| 02/12/2002 | CA2057504C Process for preparing new n-acyl-2,3-benzodiazepine derivatives, their acid addition salts and pharmaceutical compositions containing the same |
| 02/07/2002 | WO2002009683A2 Aldosterone blocker therapy to prevent or treat inflammation-related disorders |
| 02/07/2002 | US20020016337 Heterocyclic analgesic compounds and methods of use thereof |