Patents
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
11/2000
11/15/2000CN1058487C 1,5-benzodiazepine derivatives having CCK antagoistic or agonistic activity
11/09/2000WO2000066106A2 Use of benzodiazepines for treating autoimmune diseases induced by apoptosis
11/07/2000CA2179306C Dopamine receptor ligands
11/02/2000WO2000064900A1 Pyrazolobenzodiazepines as cdk2 inhibitors
11/01/2000CN1272111A Tricyclic vasopressin agonists
10/2000
10/26/2000WO2000063195A1 Novel heterocyclic amino carbonyl derivatives useful as nitric oxide synthase inhibitors
10/26/2000WO2000063186A1 Process and intermediates for preparing benzodiazepines
10/25/2000CN1271358A Oxazolidinone derivatives and pharmaceutical compositions
10/25/2000CN1271251A 2-methyl-thieno-benzodiazepine formulation
10/24/2000CA2157247C Physical form of dihydro-2,3-benzodiazepine derivative
10/19/2000WO2000061587A1 Pyrido-thieno-diazepines, method for the production thereof and pharmaceutical compositions containing said pyrido-thieno-diazepines
10/19/2000WO2000061569A1 Adamantane derivatives
10/19/2000CA2368829A1 Adamantane derivatives
10/18/2000EP1044023A1 A covalent conjugate of clozapine with a fatty acid and its use for treating schizophrenia
10/17/2000US6133309 Treatment of T-helper cell type 2-mediated immune disease by retinoid antagonists
10/12/2000CA2369238A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/11/2000EP1041989A1 Novel cycloalkenyl substituted compounds
10/11/2000EP0832075B1 n-(2,4-dioxo-2,3,4,5-tetrahydro-1h-1,5-benzodiazepin-3y l)-3-amides
10/05/2000WO2000058294A1 Antibacterial agents
10/03/2000US6127415 Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents
10/03/2000US6127359 Bicyclic fibrinogen antagonists
09/2000
09/28/2000WO2000056721A1 Solid phase synthesis of benzodiazepine diones
09/28/2000WO2000056707A1 Diaryl thioethers, compositions and uses thereof
09/27/2000EP1038868A2 Sulfonamides as antiviral agents
09/27/2000EP0733052B1 Bicyclene derivatives, their production and use
09/27/2000CN1268055A Pharmaceutical suspension comprising nevirapine hemihydrate
09/21/2000WO2000055153A1 Amide derivatives
09/21/2000DE19912638A1 Naphthylcarbonsäureamid-substituierte Sulfonamide Naphthylcarbonsäureamid-substituted sulfonamides
09/20/2000EP1036565A1 Preventives/remedies for diabetes
09/19/2000US6121258 For treatment of arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
09/19/2000US6121256 4-(2,3-(2,5-dimethyl-2,5-hexano)dibenzo(b,f)(1,4)thiazepine-11 -yl)benzoic acid or salt
09/14/2000WO2000053613A1 Chemical vapor deposition precursors and thermochromic materials thereof
09/12/2000US6117940 Solid phase synthesis of compounds such as the imidazoles, benzodiazepines, pyrazines, and steroid mimics.
09/12/2000US6117870 Cyclic amide derivatives
09/12/2000US6117866 For inhibiting platelet aggregation or clot formation and reocclusion of an artery or vein in a mammal following fibrinolytic therapy or angioplasty; for treating stroke, transient ischemia attacks, or myocardial infarction
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/05/2000US6114325 1,2-di-substituted benzene-carboxamide derivative, hair growth promoter and external composition for skin using the same
08/2000
08/30/2000EP1030852A1 Oxazolidinone derivatives and pharmaceutical compositions
08/30/2000EP1030662A2 Treatment of t-helper cell type 2 mediated immune diseases with retinoid antagonists
08/30/2000CN1265109A Thiazolobenzoheterocycles, prepn. and medicines containing same
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/23/2000EP1029859A1 N,N'-Disubstituted unsymmetrical cyclic urea and its use in therapy
08/16/2000EP1027336A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
08/16/2000EP1027042A1 Inhibitors of farnesyl protein transferase
08/15/2000US6103715 Compounds that bind to the dopamine d4 receptor and their use as anxiolytic agents, treatment for schizophrenia, and drug screening; side effect reductioon
08/15/2000US6103459 Lack delivered element-to-carbon bonds to reduce carbon contamination in films produced by vapor deposition; electroconductive polymers; metal complexes of the compounds; di-aza-, phospha-and/or arsa-butadiene type compounds
08/09/2000EP1025092A2 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate
08/09/2000EP1024811A1 Novel benzodiazepine derivatives as antiarrhythmic agents
08/08/2000US6100395 Reductive alkylation of secondary amines with hydrosilane
08/08/2000US6100277 Retroviral protease inhibitor combinations
08/08/2000US6100254 1-benzyl,3-(p-hydroxybenzyl)-5-(p-hydroxyphenyl),7-chloro-1,4 -benzodiazepin-2-one; administering to treat cancer, and diseases caused abnormal nmda channel regulation
08/03/2000WO2000044730A1 2,3,4,5-tetrahydro-1h-[1,4]benzodiazepine-3-hydroxamic acid as matrix metalloproteinase inhibitors
08/03/2000WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
08/03/2000WO2000028947A3 Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress
08/03/2000DE19903126A1 New sulphur substituted sulphonylaminocarboxylic acid N-arylamide derivatives used for treating e.g. cardiovascular diseases and atherosclerosis
08/03/2000CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors
08/03/2000CA2356267A1 2,3,4,5-tetrahydro-1h-¬1,4|benzodiazepine-3-hydroxamic acid as matrix metalloproteinase inhibitors
08/02/2000EP1023072A1 Analgesic compositions
08/01/2000US6096885 Exhibit agonist activity for cck-a receptors thereby enabling them to modulate the hormones gastrin and cholecystokinin in mammals.
08/01/2000US6096741 Oxime derivatives, hydrazone derivatives and use thereof
08/01/2000US6096735 Benzoheterocyclic derivatives
07/2000
07/27/2000WO2000042849A1 COMPLEX OF RAS-FARNESYLTRANSFERASE INHIBITOR AND SULFOBUTYLETHER-7-β-CYCLODEXTRIN OR 2-HYDROXYPROPYL-β-CYCLODEXTRIN AND METHOD
07/26/2000EP1021418A1 Substituted 2,3-benzodiazepin-4-ones and the use thereof
07/26/2000EP1021190A1 Novel amide derivatives
07/25/2000CA2169115C 1-¬2-(substituted vinyl)|-5h-2,3-benzodiazepine derivatives
07/20/2000WO2000042040A1 Tricyclic inhibitors of poly(adp-ribose) polymerases
07/20/2000WO2000041992A1 Reductive alkylation of secondary amines with hydrosilane
07/20/2000CA2359569A1 Reductive alkylation of secondary amines with hydrosilane
07/19/2000EP1019383A2 Process for the aminocarbonylation of benzazepines and benzodiazepines
07/19/2000EP1019058A1 Pharmaceutical suspension comprising nevirapine hemihydrate
07/19/2000EP1018880A1 2-methyl-thieno-benzodiazepine formulation
07/12/2000CN1054380C Condensed cyclic compounds and their use
07/06/2000WO2000039110A1 Homopiperazine derivatives as selective emopamil inhibitors
07/06/2000WO2000039105A1 1,4-diazacycloheptane derivatives useful in the treatment of neurological disorders
07/06/2000WO2000039081A2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
07/06/2000WO2000038618A2 SUCCINOYLAMINO BENZODIAZEPINES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
07/06/2000CA2347671A1 Succinoylamino benzodiazepines as inhibitors of a.beta. protein production
07/05/2000EP0686151B1 Substituted cyclic carbonyls and derivatives thereof useful as retroviral protease inhibitors
06/2000
06/22/2000WO2000006620A3 Polymerization of olefins
06/21/2000EP1010696A1 Method of preparing Oxoquazepam
06/21/2000EP1009739A2 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity
06/21/2000CN1257071A Process for preparation of ketoquazepan
06/14/2000EP1008592A2 Cyclic amide derivatives which inhibit cathepsin K
06/14/2000CN1053438C Benzodiazepin-2-one derivatives, process for their prepn. and pharmaceutical composition containing them
06/14/2000CA2284961A1 Method of preparing oxoquazepam
06/13/2000US6075018 Tranquilizers
06/06/2000US6071903 2,3,4,5-tetrahydro-1H-[1,4]-benzodiazepine-3-hydroxyamic acids
06/06/2000US6071895 Polar-substituted hydrocarbons
06/02/2000WO2000031073A1 Benzoxazole derivatives and drugs containing the same as the active ingredient
06/02/2000CA2351446A1 Benzoxazole derivatives and medicaments comprising said derivatives as active ingredient
05/2000
05/31/2000EP0635016B1 Benzodiazepine derivatives and protein and polypeptide conjugates thereof
05/25/2000WO2000028947A2 Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress
05/25/2000CA2349919A1 Use of a substance binding with the peripheral benzodiazepin receptor for treating skin stress
05/24/2000CN1253954A Heterocyclic alkoxyl amine as regulator in controlled free radical polymerization method
05/18/2000WO2000004892A3 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
05/17/2000EP1000936A1 Novel hexahydro-1,4-diazepine derivatives or salts thereof
05/17/2000EP1000067A1 Thiazolobenzoheterocycles, preparation and medicines containing same
05/17/2000EP1000062A1 Tricyclic vasopressin agonists
05/17/2000CN1253555A Novel 2-(iminomethyl) amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same
05/17/2000CN1253554A Heterocyclic compounds and their use for inhibiting 'beta'-amyloid peptide
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