| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 05/10/2000 | CN1252795A 4,1-benzoxazepines, their analogues,and their use as somatostatin agonists |
| 05/09/2000 | US6060586 Ureins derived from alpha, omega-diamono acids and process for their preparation |
| 05/09/2000 | US6060071 Ectoin and ectoin derivatives as moisturizers in cosmetics |
| 05/04/2000 | WO2000024400A1 Use of optically pure (r)-tofisopam for treating and preventing anxiety disorders and composition thereof |
| 05/04/2000 | CA2348281A1 Use of optically pure (r)-tofisopam for treating and preventing anxiety disorders and composition thereof |
| 05/03/2000 | CN1052000C Preparation of alkylimidazolidone (meth) acrylates |
| 05/03/2000 | CN1051999C Preparation of alkylimidazolidine (meth) acrylate (S) |
| 04/27/2000 | WO2000023487A1 Amino-ketone solid support templates |
| 04/27/2000 | WO2000023428A1 1,5-benzodiazepine compounds, process for producing the same, and medicine |
| 04/27/2000 | CA2347938A1 1,5-benzodiazepine compounds, their production and use |
| 04/27/2000 | CA2347243A1 Amino-ketone solid support templates |
| 04/25/2000 | US6054597 Reacting the corresponding dimethyl ester with reducing agent; then hydrazine |
| 04/25/2000 | US6054457 Benzamide derivatives and their use as vasopressin antagonists |
| 04/20/2000 | DE19949352A1 Heterocyclic alkoxyamine polymerization composition useful as regulator in free-radical polymerization to obtain low-polydispersity polymeric resins |
| 04/18/2000 | CA2087604C Diamine compounds and cerebral protective drugs containing the same |
| 04/16/2000 | CA2286375A1 Heterocyclic alkoxyamines as regulators in controlled radical polymerization processes |
| 04/05/2000 | CN1051079C Benzodiazepine derivs. their preparation method and pharmaceutical composition contg. same |
| 03/29/2000 | CN1050835C 1,5-benzodiazepine derivatives and its preparation process and use in medicine |
| 03/28/2000 | US6043358 Hexahydro-5-imino-1,4-heteroazepine derivatives as inhibitors of nitric oxide synthases |
| 03/22/2000 | EP0986585A1 Use of ylides of phosphorus as slightly nuceophilic strong bases |
| 03/22/2000 | EP0830349B1 Method for preparing n, n'-disubstitued cyclic ureas |
| 03/22/2000 | CN1248250A Novel 1,4-diazacycloheptane derivatives and their use in hair oxidation dyes |
| 03/21/2000 | US6040303 7-phenyl-1, 4-diazepane compounds, process for their preparation, and pharmaceutical compositions containing them |
| 03/16/2000 | WO2000014073A1 Benzodiazepinone derivatives, preparation method and intermediates therefor, use as medicines and compositions |
| 03/16/2000 | WO2000014063A1 Therapeutic compounds and methods |
| 03/16/2000 | CA2342858A1 Method of screening compounds useful in the treatment of a desease caused by or exacerbated by mpv |
| 03/15/2000 | CN1050353C Process for prepn. of alkylimidazolidone (meth)-acrylates |
| 03/14/2000 | US6037157 Method for improving pharmacokinetics |
| 03/14/2000 | CA2009542C Cyclic guanidines as calcium antagonists |
| 03/08/2000 | CN1246850A 1,5-benzodiazepine derivatives |
| 03/02/2000 | WO2000010942A1 Solid phase synthesis of compounds by carbon-carbon bond forming mitsunobu reactions |
| 03/02/2000 | CA2338563A1 Solid phase synthesis of compounds by carbon-carbon bond forming mitsunobu reactions |
| 03/01/2000 | CN1246157A Enzymatic resolution of benzodiazepine-acetic acid esters with lipase |
| 02/24/2000 | WO2000009480A1 Novel sulfonyl derivatives |
| 02/24/2000 | CA2340100A1 Novel sulfonyl derivatives |
| 02/22/2000 | CA2157248C Crystalline form of dihydro-2, 3 benzodiazepine derivative |
| 02/17/2000 | WO2000007995A1 SUCCINOYLAMINO LACTAMS AS INHIBITORS OF Aβ PROTEIN PRODUCTION |
| 02/17/2000 | WO2000007980A1 Amide derivatives which are useful as cytokine inhibitors |
| 02/17/2000 | CA2338944A1 Succinoylamino lactams as inhibitors of a.beta. protein production |
| 02/16/2000 | EP0979227A1 4,1-benzoxazepines, their analogues, and their use as somatostatin agonists |
| 02/10/2000 | WO2000006620A2 Polymerization of olefins |
| 02/10/2000 | CA2338686A1 Polymerization of olefins |
| 02/09/2000 | CN1049217C 1,5-benzodiazepine derivatives |
| 02/08/2000 | US6022969 Symmetrical bis(aminoalkyl), bis(amidinoalkyl) and bis(guanidinoalkyl) cycloalkanes |
| 02/03/2000 | WO2000004892A2 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions |
| 02/03/2000 | CA2335062A1 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions |
| 02/02/2000 | EP0975625A1 SELECTIVE FACTOR Xa INHIBITORS |
| 02/02/2000 | EP0975608A2 Halo-alkoxycarbonyl prodrugs |
| 01/27/2000 | WO2000004020A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation |
| 01/27/2000 | CA2337377A1 Compounds, compositions, and methods for stimulating neuronal growth and elongation |
| 01/26/2000 | EP0973763A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and pharmaceutical compositions containing same |
| 01/20/2000 | WO2000002851A1 Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them |
| 01/19/2000 | CN1242007A Cycloalkyl, lactam lactone and related compounds as 'beta'-amyloid peptide release inhibitors |
| 01/19/2000 | CN1048484C A process for preparing a composition containing benzoheterocycles |
| 01/13/2000 | WO2000001376A2 Pharmaceutical compositions and their uses for treatment of demyelinating disorders |
| 01/12/2000 | EP0693067B1 Fibrinogen receptor antagonists |
| 01/06/2000 | WO2000000479A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors |
| 01/06/2000 | WO2000000202A1 Method for inhibiting c-jun expression using jak-3 inhibitors |
| 01/06/2000 | CA2337999A1 Method for inhibiting c-jun expression using jak-3 inhibitors |
| 01/06/2000 | CA2330110A1 1,3-benzodiazepin-2-ones and 1,3-benzoxazepin-2-ones useful as hiv reverse transcriptase inhibitors |
| 01/05/2000 | EP0968198A1 HETEROCYCLIC COMPOUNDS AND THEIR USE FOR INHIBITING $g(b)-AMYLOID PEPTIDE |
| 01/04/2000 | US6011045 Inhibitors of bone resorption; anticancer agents |
| 01/04/2000 | US6011029 Benzodiazepine compounds |
| 12/29/1999 | WO1999067221A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999067220A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999067219A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS |
| 12/29/1999 | EP0966449A1 Novel 1,4-diazacycloheptane derivatives and their use in hair oxidation dyes |
| 12/29/1999 | CA2325389A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | CA2325388A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/29/1999 | CA2324475A1 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds |
| 12/29/1999 | CA2324474A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis |
| 12/28/1999 | US6008216 Process for preparing 2-methyl-thieno-benzodiazepine |
| 12/28/1999 | US6008214 Inhibiting platelet aggregation and bone resorption, treating stroke, transient ischemia attacks, or myocardial infarction, treating osteoporosis |
| 12/23/1999 | WO1999065870A2 Sulfonamide inhibitors of aspartyl protease |
| 12/22/1999 | EP0964928A1 Enzymatic resolution of benzodiazepine-acetic acid esters with a lipase |
| 12/16/1999 | WO1999064403A1 1,5-benzodiazepine derivatives |
| 12/16/1999 | CA2334798A1 1,5-benzodiazepine derivatives |
| 12/15/1999 | CN1238689A Vitronectin receptor antagonists |
| 12/14/1999 | US6001579 Supports and combinatorial chemical libraries thereof encoded by non-sequencable tags |
| 12/08/1999 | CN1237961A Aminoguanidines and alkoxyguanidines as protease inhibitors |
| 12/07/1999 | US5998614 Preparation of asymmetric cyclic ureas using an alkali metal in liquid ammonia process |
| 12/07/1999 | US5998414 Troponyl piperazines as dopamine D4 receptor ligands |
| 12/07/1999 | US5998407 Inhibitors of farnesyl-protein transferase |
| 12/07/1999 | US5998406 Bactericides |
| 12/07/1999 | CA2013037C Aminobenzenesulfonic acid derivative |
| 12/01/1999 | EP0960104A1 N-(amidinophenyl)-n'-(subst.)-3h-2,4-benzodiazepin-3-one derivatives as factor xa inhibitors |
| 11/25/1999 | WO1999059977A1 Substituted 1,3-diaza-2-(thi)oxo-cycloalkanes |
| 11/25/1999 | DE19822678A1 New 1,3-diaza-2-oxo-cycloalkane derivatives, useful as pre- or post-emergence, total or selective herbicides |
| 11/25/1999 | CA2332443A1 Substituted 1,3-diaza-2-(thi)oxo-cycloalkanes |
| 11/24/1999 | EP0957917A1 Vitronectin receptor antagonists |
| 11/23/1999 | US5990145 Antiinflammatory,-carcinogenic,-tumor,-metastasis agents; cardiovascular disorders, e.g., arteriosclerosis, restenosis; retinopaathies and nephropathies; osteoporosis |
| 11/23/1999 | US5990113 Monohydrate of 2-(1-piperazinyl)-5-methylbenzenesulfonic acid, free of anhydrous crystals; free from weight change due to moisture absorption and can be weighed accurately in manufacturing a pharmaceutical composition for heart diseases |
| 11/17/1999 | CN1235602A 1-(3-aminoindazol-5-yl)-3-phenylmethyl-cyclic urea useful as HIV protease inhibitors |
| 11/17/1999 | CN1046501C Thiourea compositions and preparation of nitryl, aromatic and imino heterocyclic compounds |
| 11/16/1999 | US5986114 Benzopyranol derivatives |
| 11/16/1999 | US5985869 Benzoheterocyclic compounds |
| 11/16/1999 | CA2120215C 2,3-dihydro-4(1h)-quinazolinones active in gastro-intestinal pathologies |
| 11/10/1999 | EP0776208B1 2,3-dihydro-1-(2,2,2-trifluoroethyl)-2-oxo-5-phenyl-1h-1,4-benzodiazepines |
| 11/04/1999 | WO1999055684A1 Solid supported synthesis of sulfonated 2-oxopiperazines |