Patents
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
04/2001
04/18/2001EP1091739A1 Method for inhibiting c-jun expression using jak-3 inhibitors
04/17/2001US6218534 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermediate
04/17/2001US6218375 Complex of ras-farnesyltransferase inhibitor and sulfobutylether-7-β-cyclodextrin or 2-hydroxypropyl-β-cyclodextrin and method
04/11/2001EP1089981A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis.
04/11/2001EP1089980A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001EP1089977A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
04/11/2001CN1064354C Trilcyclic benzazepine vasopressin antagnonists
04/10/2001US6214823 Benzodiazepine derivatives as antiarrhythmic agents
04/10/2001US6214822 Substituted aza and diazacycloheptane and cyclooctane compounds and their use
04/05/2001WO2000073284A3 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
04/04/2001CN1290254A Sulfonamide derivatives process for producing the same and utilization thereof
04/03/2001US6211228 Compositions and methods for treating mast-cell mediated conditions
04/03/2001US6211183 Selective factor Xa inhibitors
03/2001
03/28/2001EP1086076A1 Sulfonamide inhibitors of aspartyl protease
03/28/2001CN1289324A Method for preparing an N-[(aliphatic or aromatic) carbonyl]-2-aminoacetamide compound and a cyclyzed compound
03/27/2001US6207663 Vitronectin receptor antagonists, their preparation and use
03/22/2001WO2001019797A2 HYDROXYALKANOYL AMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF Aβ PROTEIN PRODUCTION
03/22/2001WO2000063195A8 Novel heterocyclic amino carbonyl derivatives useful as nitric oxide synthase inhibitors
03/22/2001WO2000001376A3 Pharmaceutical compositions and their uses for treatment of demyelinating disorders
03/22/2001CA2377221A1 Hydroxyalkanoyl aminolactams and related structures as inhibitors of a.beta. protein production
03/21/2001EP1085014A1 1,5-benzodiazepine derivatives
03/20/2001US6204262 1,3-Benzodiazepin-2-ones and 1,3-Benzoxazepin-2-ones useful as HIV reverse transcriptase inhibitors
03/20/2001US6204261 Inhibitors of interleukin-1β Converting enzyme inhibitors
03/15/2001WO1999065870A3 Sulfonamide inhibitors of aspartyl protease
03/13/2001US6201119 Antiretroviral tetrahydroimidazo[1,4]benzodiazepin-2(thi) ones
03/13/2001US6200970 For treating a disease associated with overstimulation of an ampa receptor, or hyperactivity of an excitatory amino acid
03/08/2001WO2001016110A1 Bleach boosting components, compositions and laundry methods
03/08/2001WO2001015656A2 Tricyclic compounds and their uses as antiarrhythmic antifibrillatory and defibrillatory agents
03/08/2001CA2381892A1 Bleach boosting components, compositions and laundry methods
03/07/2001EP1080077A1 Substituted 1,3-diaza-2-(thi)oxo-cycloalkanes
03/06/2001US6197764 Clozapine compositions and uses thereof
03/01/2001WO2000071516B1 INHIBITORS OF FACTOR Xa
03/01/2001WO2000068209A3 1,5-benzodiazepine derivatives as cck-a receptor agonists
02/2001
02/22/2001WO2001012600A1 INHIBITORS OF FACTOR Xa
02/15/2001WO2001010847A2 Novel integrin receptor antagonists
02/15/2001WO2001010846A2 1,4-diazepine derivatives for the treatment of diseases related to the central nervous system
02/15/2001WO2001010799A1 Methods for preparing n-[(aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
02/15/2001WO2001010797A1 Process for catalyzing the oxidation of organic compounds
02/15/2001WO2001010216A1 Antiarrhythmic compounds
02/15/2001DE19936780A1 Neue Antagonisten von Integrinrezeptoren New antagonists of integrin
02/15/2001CA2381260A1 Novel 1,4-benzodiazepine compounds and derivatives thereof
02/15/2001CA2380851A1 Process for catalyzing the oxidation of organic compounds
02/15/2001CA2379977A1 Novel integrin receptor antagonists
02/08/2001WO2001055118A1 Benzene-fused heterocycle derivatives and drugs containing the same as the active ingredient
02/07/2001EP1073644A1 Solid supported synthesis of sulfonated 2-oxopiperazines
01/2001
01/31/2001EP1072587A1 Sulfonamide derivatives and drugs containing the same as the active ingredient
01/31/2001CN1282322A 1,4-diazacycloheptane derivatives
01/25/2001WO2000071515A3 INHIBITORS OF FACTOR Xa
01/24/2001EP0694039B1 1,5-benzodiazepine derivatives having cck antagonistic and or agonistic activity
01/18/2001WO2001004122A2 New 2,3-benzodiazepine derivatives
01/18/2001WO2001004103A1 Benzazepinones and quinazolines
01/18/2001WO2000071516A3 INHIBITORS OF FACTOR Xa
01/18/2001CA2378305A1 New 2,3-benzodiazepine derivatives
01/11/2001WO2001002403A1 METHOD FOR PREPARING SUBSTITUTED [1,4]DIAZEPINO[6,7,1-hi]INDOL-4-ONES
01/11/2001WO2001002381A1 Piperazine derivatives as modulators of chemokine receptor activity
01/11/2001WO2001002373A1 Dihydrobenzodiazepins and their use for treating dyslipidemia
01/11/2001WO2001002372A1 Cyclized amino acid derivatives
01/11/2001WO2001002358A2 Cyclized amide derivatives for treating or preventing neuronal damage
01/11/2001CA2376707A1 Process for the preparation of substituted ¬1,4|diazepino¬6,7,1-hi|indol-4-ones
01/10/2001EP1067103A2 Process for producing halogenated benzene compound
01/09/2001US6172059 Controlling particle size
01/04/2001WO2001000625A1 Process for the preparation of imidazodiazepine intermediates
01/04/2001CA2341524A1 Process for the preparation of imidazodiazepine intermediates
01/03/2001EP1064300A1 Peptide turn mimetics
01/03/2001EP1064274A1 Benzenesulfonamide derivatives and their use as medicaments
01/03/2001CN1278797A Oxo-substituted compouns, process of making, and compositions and methods for inhibiting parp activity
01/02/2001US6169084 2-methyl-thieno-benzodiazepine formulation
12/2000
12/28/2000WO2000078744A1 Thiochroman derivatives against neurological disorders
12/28/2000WO2000078736A1 1,4-diazacycloheptane derivatives as neuroprotective agents
12/28/2000WO2000078725A1 Synthesis of substituted amidines
12/27/2000EP1062210A1 1,2-diazepane derivatives as interleukin-1beta converting enzyme inhibitors
12/26/2000US6166005 Heterocyclic metalloprotease inhibitors
12/26/2000US6165230 For dyeing keratinous fibers; brilliance, color tone, colorfastness, thermal stability, level dyeing
12/21/2000WO2000044709A3 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
12/20/2000EP1060169A1 1,4-diazacycloheptane derivatives
12/20/2000CN1277604A Heteraryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
12/12/2000US6160133 Stereospecific biosynthesis of the alcohol by enzymatic reduction of the corresponding aldehyde or ketone using a candida, zygosaccaromyces, or mortierrela microorganism
12/07/2000WO2000073284A2 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
12/07/2000CA2370141A1 1,4-benzodiazepin-2-ones useful as hiv reverse transcriptase inhibitors
12/06/2000EP1056727A1 Solid support synthesis of 2-oxopiperazines
12/06/2000CN1275912A Novel amide derivatives
12/05/2000CA2195974C 2,3-dihydro-1-(2,2,2-trifluoroethyl)-2-oxo-5-phenyl-1h-1,4-benzodiazepines
11/2000
11/30/2000WO2000071518A2 Heterocyclic analgesic compounds and their use
11/30/2000WO2000071516A2 INHIBITORS OF FACTOR Xa
11/30/2000WO2000071515A2 INHIBITORS OF FACTOR Xa
11/30/2000CA2374788A1 Inhibitors of factor xa
11/30/2000CA2372887A1 Heterocyclic analgesic compounds and their use
11/30/2000CA2371904A1 Inhibitors of factor xa
11/23/2000WO2000069836A1 Short-acting benzodiazepines
11/23/2000WO2000069835A2 Process for manufacturing diazepine derivatives
11/23/2000WO2000069830A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
11/23/2000CA2373590A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
11/22/2000EP1054005A1 Sulfonamide derivatives, process for producing the same and utilization thereof
11/22/2000CN1058710C Benzamide derivatives, process for prepn. thereof and pharmaceutical compsn. comprising same
11/21/2000US6150370 1,3-dinitrocyclic compound treats numerous diseases caused by undesired metalloprotease activity, such as tumor metastasis, osteoarthritis, rheumatoid arthritis, skin inflammation, ulcerations, and periodontitis
11/16/2000WO2000068209A2 1,5-benzodiazepine derivatives as cck-a receptor agonists
11/16/2000CA2370801A1 1,5-benzodiazepine derivatives as cck-a receptor agonists
11/15/2000EP1051407A1 2,3,4,5-tetrahydro-1h-[1,4]-benzodiazepine-3-hydroxamic acids as matrix metalloproteinase inhibitors
11/15/2000EP1051397A1 Method for preparing an n- (aliphatic or aromatic)carbonyl]-2-aminoacetamide compound and a cyclyzed compound
11/15/2000CN1273586A Method for preparation of asymmetric cyclic ureas through monoaylated diamine
1 ... 28 29 30 31 32 33 34 35 36 37 38 39 40 41 42 43 44 45 46 47 48 ... 60