| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 04/09/2009 | US20090093457 Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions |
| 04/09/2009 | US20090093455 Quinolone analogs and methods related thereto |
| 04/09/2009 | CA2700691A1 New biaryl derivatives |
| 04/09/2009 | CA2694288A1 1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine-6-carboxamide and 2,3,4,5-tetrahydropyrrolo[1,2-a][1,4]-diazepine-7-carboxamide derivatives, preparation and therapeutic use thereof |
| 04/08/2009 | EP2045251A1 Compound that can inhibit ubc13-uev interactions, pharmaceutical compositions and therapeutic uses |
| 04/07/2009 | US7514426 Substituted imidazol[1,5-A][1,2,4]triazolo[1,5-D][1,4]benzodiazepine derivatives |
| 04/02/2009 | WO2007115164A3 Amino acid surrogates for peptidic constructs |
| 04/01/2009 | EP2041088A1 Glycine transporter-1 inhibitors |
| 04/01/2009 | EP1521744B1 Arylsulphonamide derivatives and use thereof as b1 bradykinin receptor antagonists |
| 03/31/2009 | US7511033 Dihydro-benzo[B][1,4]diazepin-2-one sulfonamide derivatives |
| 03/26/2009 | WO2009037642A1 Heterocyclic scaffolds useful for preparation of combinatorial libraries, libraries and methods of preparation thereof |
| 03/26/2009 | WO2009037302A1 5-substituted-1, 4-benz0diazepines as phosphodiesterase inhibitors |
| 03/26/2009 | US20090082339 Novel azacyclyl-substituted arylthienopyrimidinones, process for their preparation and their use as medicaments |
| 03/25/2009 | EP2037741A1 Compositions and methods relating to novel compounds and targets thereof |
| 03/24/2009 | US7507815 Succinoylamino lactams as inhibitors of a-β protein production |
| 03/24/2009 | US7507729 Substituted imidazo-[1,5-a][1,2,4]triazolo[1,5-d][1,4] benzodiazepine derivatives |
| 03/24/2009 | US7507728 for the treatment of cognitive disorders, anxiety, schizophrenia, and Alzheimer's disease; 10-chloro-9H-imidazo[1,5-a][1,2,4]triazolo[1,5-d][1,4]benzodiazepine; ligands; GABA A alpha 5 receptor inhibitors; halogenation |
| 03/19/2009 | US20090075982 Piperazine compounds |
| 03/19/2009 | US20090075980 Pyrazolopyridines and Analogs Thereof |
| 03/19/2009 | US20090075971 Derivatives of 2-alkoxy-3,4,5-trihydroxy-alkyl amides, preparation and use thereof, and compositions containing the same |
| 03/18/2009 | EP2035380A2 Parp inhibitors |
| 03/18/2009 | CN101389600A Optical isomers of dihydro-2,3-benzodiazepine derivatives, process for their stereoselective synthesis |
| 03/18/2009 | CN100469779C Inhibitors of interleukin-1beta converting enzyme |
| 03/17/2009 | US7504436 Bioisosteres of actinonin |
| 03/12/2009 | US20090069304 Mmp-13 selective inhibitor |
| 03/12/2009 | US20090069303 Phthalazinone derivatives |
| 03/12/2009 | US20090069302 Chemical compounds |
| 03/12/2009 | US20090069301 Acridine and Quinoline Derivatives as Sirtuin Modulators |
| 03/12/2009 | US20090069294 Organic Compounds |
| 03/12/2009 | US20090069293 Succinoylamino benzodiazepines as inhibitors of ab protein production |
| 03/12/2009 | US20090069282 Alkyne compounds with mch antagonistic activity and medicaments comprising these compounds |
| 03/11/2009 | CN100467458C Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them |
| 03/10/2009 | US7501510 N,N'-disubstituted thiourea ligand, when complexed with palladium forms a catalyst useful for Heck reaction of arylhalides and olefins and Suzuki cross-coupling reaction of aryl halides with aryl boric acids |
| 03/10/2009 | US7501407 Amide substituted pyrimidine compound; antiarthritic agents; antiischemic agents; antidiabetic agents; inflammatory bowel disease; antiproliferative agents; antiallergens |
| 03/05/2009 | WO2008055068A3 Inhibitors of histone deacetylase |
| 03/05/2009 | US20090062256 LACTAMS SUBSTITUTED BY CYCLIC SUCCINATES AS INHIBITORS OF Abeta PROTEIN PRODUCTION |
| 03/05/2009 | US20090060912 Small molecule pi 3-kinase inhibitors and methods of their use |
| 03/04/2009 | EP2029556A2 Salts and crystal modifications thereof |
| 03/04/2009 | EP2029555A2 Derivatives of 2-alkoxy-3,4,5-trihydroxy-alkyl amides, preparation and use thereof, and compositions containing the same |
| 03/04/2009 | EP1660443B1 Cyclic amine bace-1 inhibitors having a benzamide substituent |
| 03/04/2009 | EP1064300B1 Peptide turn mimetics |
| 03/03/2009 | US7498433 Process and intermediates for the preparation of olanzapine |
| 03/03/2009 | US7498324 Substituted lactams as inhibitors of Aβ protein production |
| 02/26/2009 | WO2009024550A1 N-benzyl, n' -arylcarbonylpiperazine derivatives as lxr modulators |
| 02/26/2009 | US20090054460 Piperazine derivatives and methods of use |
| 02/26/2009 | US20090054416 1,4-Diazabicyclo[3.2.2]nonanecarboxamide Derivatives, Preparation and Therapeutic Use Thereof |
| 02/26/2009 | US20090054409 [4-(4-imidazo[1,2-a]pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-morpholin-4-yl-methanone, used for treating rheumatoid arthritis in mammals |
| 02/26/2009 | US20090054396 Substituted thiophenes and uses thereof |
| 02/26/2009 | US20090054392 Naphthylpyrimidine, naphthylpyrazine and naphthylpyridazine analogs and their use as agonists of the wnt-beta-catenin cellular messaging system |
| 02/26/2009 | CA2694604A1 N-benzyl, n' -arylcarbonylpiperazine derivatives as lxr modulators |
| 02/25/2009 | CN101372477A Method for synthesizing diaza-onium salt |
| 02/24/2009 | US7494984 Substituted imidazo[1,2-a]pyrimidines as HIV viral DNA integrase inhibitors |
| 02/24/2009 | CA2297406C Tricyclic vasopressin agonists |
| 02/19/2009 | WO2009023664A2 Substituted azepine- and diazepine-sulfonamides useful to inhibit 11beta-hydroxysteroid dehydrogenase type-1 |
| 02/19/2009 | WO2009021944A1 New compounds |
| 02/19/2009 | WO2008106128A3 CYCLIC UREA AND CARBAMATE INHIBITORS OF 11β -HYDROXYSTEROID DEHYDROGENASE 1 |
| 02/19/2009 | US20090048238 Novel biaryl derivatives |
| 02/19/2009 | US20090047249 Modulators of toll-like receptor 7 |
| 02/19/2009 | CA2696336A1 Substituted azepine- and diazepine-sulfonamides useful to inhibit 11.beta.-hydroxysteroid dehydrogenase type-1 |
| 02/19/2009 | CA2696261A1 New compounds |
| 02/18/2009 | EP2025673A1 Arylsulfonamides with analgetic activity |
| 02/18/2009 | EP2025672A1 Seven-membered ring compound, production method thereof and pharmaceutical use thereof |
| 02/17/2009 | US7491723 Alkanol and cycloalkanol-amine derivatives and methods of their use |
| 02/12/2009 | WO2008142591A3 3- to 7-membered 1,3-diaza-4-oxo-heterocyclic derivatives capable of releasing active aldehydes or ketones |
| 02/12/2009 | US20090043091 Induce immunology response; anticancer agents; 6-(6-Morpholin-4-yl-4-oxo-4H-pyran-2-yl)-thianthrene-2-carboxylate sodium salt; 6-(4,4,5,5-Tetramethyl-[1,3,2]dioxaborolan-2-yl)-thianthrene-2-carboxylic acid methyl ester |
| 02/12/2009 | US20090042866 Tetrahydrocarbazoles as Active Agents for Inhibiting VEGF Production by Translational Control |
| 02/12/2009 | US20090042865 Dna-pk inhibitors |
| 02/05/2009 | WO2009016286A2 6-cycloamino-3-(pyridin-4-yl)imidazo[1,2-b]pyridazine derivatives, preparation thereof and therapeutic use thereof |
| 02/05/2009 | US20090036430 Pyrido(3,2-d)pyrimidines and pharmaceutical compositions useful for medical treatment |
| 02/05/2009 | CA2691866A1 6-cycloamino-3-(pyridin-4-yl)imidazo[1,2-b]pyridazine derivatives, preparation thereof and therapeutic use thereof |
| 02/04/2009 | CN100457726C Substituted sulfonamide compounds, process for their use as medicament for the treatment of CNS disorders, obestity and type II diabetes |
| 02/03/2009 | CA2259936C Apoptosis inducing adamantyl derivatives and their usage as anti-cancer agents |
| 01/29/2009 | US20090029972 Dibenzodiazepinone Analogues, Processes for Their Production and Their Use as Pharmaceuticals |
| 01/29/2009 | US20090029965 Vasopressin V1a Antagonists |
| 01/27/2009 | US7482439 Caprazene as novel compound and derivatives thereof, and caprazol as novel compound and derivatives thereof |
| 01/27/2009 | US7482346 Carboxylation of the alkylpiperazine; amidation of the carbamate-ester; cannabinoid and vanilloid receptor antagonists |
| 01/27/2009 | US7482338 Non-amide nonanes |
| 01/27/2009 | US7482336 Aminocyclohexanes as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes |
| 01/22/2009 | US20090023711 Piperazines and Piperidines as Mglur5 Potentiators |
| 01/21/2009 | EP0951466B1 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting beta-amyloid peptide release and/or its synthesis by use of such compounds |
| 01/20/2009 | CA2337770C Amide derivatives which are useful as cytokine inhibitors |
| 01/14/2009 | CN100450994C Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors |
| 01/08/2009 | US20090012065 Therapeutic applications of pro-apoptotic benzodiazepines |
| 01/07/2009 | EP2010506A1 Diazepan derivatives modulators of chemokine receptors |
| 01/07/2009 | CN100448449C [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl)amino]alkyl]-acid derivatives for the treatment of pain |
| 01/06/2009 | US7473778 Amidating 2-nitrophenylacetic acid with 4-amino-N-phenylmethylpiperidine; hydrogenating the nitro group; carbamylating the amine formed with a dicarbonate or chloroformate; dissolving product in an aprotic organic solvent; reduction and cyclization; cleaving the benzyl protecting group |
| 01/01/2009 | US20090005365 Therapeutic pyrazolonaphthyridine derivatives |
| 12/31/2008 | WO2009001127A1 Cyanocyclopropylcarboxamides as cathepsin inhibitors |
| 12/31/2008 | EP1051397B1 Method for preparing an n- (aliphatic or aromatic)carbonyl -2-aminoacetamide compound and a cyclyzed compound |
| 12/30/2008 | CA2441771C Dihydro-benzo[b][1,4]diazepin-2-one derivatives as mglur2 antagonists i |
| 12/25/2008 | US20080319189 reacting 4-amino-2-methyl-10H-thieno-[2,3-b][1,5]benzodiazepine and N-methylpiperazine in methanol or ethanol solvent to produce an antipsychotic agent |
| 12/24/2008 | CN100445276C Sulfonylamino-derivatives as novel inhibitors of histone deacetylase |
| 12/23/2008 | CA2442557C Dihydro-benzo¬b|¬1,4|diazepin-2-one derivatives as mglur2 antagonists ii |
| 12/18/2008 | WO2008033764A3 Quinazolinone and isoquinolinone acetamide derivatives |
| 12/18/2008 | WO2007078808A3 Method for isolating (r)-tofisopam |
| 12/18/2008 | US20080312216 Piperazine and [1,4]diazepan derivatives as nk antagonists |
| 12/18/2008 | US20080312215 Substituted [1,4]-diazepanes as CXCR3 antagonists and their use in the treatment of inflammatory disorders |
| 12/17/2008 | EP2001853A1 Novel guanidine derivatives and their medical use |
| 12/17/2008 | EP2001485A2 Diazepan orexin receptor antagonists |
| 12/17/2008 | EP1651623B1 Hexahydrodiazepinones as dipeptidyl peptidase-iv inhibitors for the treatment or prevention of diabetes |