| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 08/06/2009 | US20090197872 Novel 1,4-diaza-bicyclo[3.2.2]nonyl pyrimidinyl derivatives and their medical use |
| 08/06/2009 | US20090197859 Pyridinyl Amides for the Treatment of CNS and Metabolic Disorders |
| 08/05/2009 | EP1742707A4 Treatment of cns disorders using cns target modulators |
| 08/05/2009 | CN101500997A PARP inhibitors |
| 07/30/2009 | WO2009093269A1 Novel heterocyclic compounds |
| 07/30/2009 | US20090192138 compounds |
| 07/30/2009 | CA2712685A1 Novel heterocyclic compounds |
| 07/29/2009 | EP2083014A2 Inhibitors of interleukin-1ß converting enzyme |
| 07/29/2009 | EP1409468B9 Guanidinobenzamides as mc4-r agonists |
| 07/29/2009 | CN101495463A Seven-membered ring compound, production method thereof and pharmaceutical use thereof |
| 07/28/2009 | US7566715 Substituted sulfonamide compounds useful for the prophylaxis and treatment of conditions relating to obesity, type II diabetes and/or disorders of the central nervous system |
| 07/28/2009 | US7566707 For example, 2-[3-(Tert-butyloxycarbonylamino)-piperidin-1-yl]-3-(2-butyn-1-yl)-5-[(dibenzo[b,f][1,4]-oxazepin-11-yl)methyl]-3,5-dihydro-imidazo[4,5-d]pyridazin-4-one; inhibiting effect on activity of the enzyme dipeptidylpeptidase-IV; use in treatment of diabetes mellitus, arthritis, obesity |
| 07/23/2009 | WO2009043747A3 N-heterocyclic biaryl carboxamides as ccr receptor antagonists |
| 07/23/2009 | WO2009023664A3 Substituted azepine- and diazepine-sulfonamides useful to inhibit 11beta-hydroxysteroid dehydrogenase type-1 |
| 07/23/2009 | WO2008061796A3 Compounds for the treatment of diseases associated with amyloid or amyloid-like proteins |
| 07/23/2009 | US20090186881 1(R)-1-(4-methyl-2-oxo-2,3-dihydro-benzoxazol-6-ylmethyl)-2-oxo-2-[4-(tetrahydropyran-4-yl)-piperazin-1-yl]-ethyl 4-(2-oxo-1,2,4,5-tetrahydro-1,3-benzodiazepin-3-yl); calcitonin gene related peptide antagonist; analgesic, antidiabetic agent; migraine or cluster headaches, non-insulin-dependent diabetes |
| 07/23/2009 | US20090186878 Crystalline forms of a farnesyl dibenzodiazepinone |
| 07/16/2009 | WO2009061916A3 Benzodiazepinone compounds useful in the treatment of skin conditions |
| 07/16/2009 | US20090181951 Parp inhibitors |
| 07/15/2009 | EP2078001A1 Diazepane-acetamide derivatives as selective 11 -hsd1 inhibitors |
| 07/14/2009 | US7560547 chemical synthesis of N-[2,4-dibromo-6-methylpyridin-3-yl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]acetamide; used as drugs and chemical intermediates |
| 07/14/2009 | CA2532818C (thio) carbamoyl-cyclohexane derivatives as d3/d2 receptor antagonists |
| 07/09/2009 | US20090176800 In vivo screening method of therapeutic agent for memory/learning dysfunctions by schizophrenia |
| 07/09/2009 | US20090176771 Gyrase inhibitors and uses thereof |
| 07/09/2009 | US20090176770 e.g. 1-(3,4-dibromo-benzyl)-2-[4-(1-methyl-piperidin-4-yl)-piperazin-1-yl]-2-oxo-ethyl 4-(2-oxo-1,2,4.5-tetrahydro-1,3-benzodiazepin-3-yl)-piperidine-1-carboxylate; calcitonin gene related peptide antagonist; analgesic, antidiabetic agent; migraine or cluster headaches, non-insulin-dependent diabetes |
| 07/09/2009 | US20090176767 Biphenyl-2-ylcarbamic Acid 1-(2-{5-[2-(4-Hydroxyphenyl)ethylamino]pentylcarbamoyl}ethyl)piperidin-4-yl Ester, used for the treatment of respiratory system disorders such as chronic obstructive pulmonary disease and asthma |
| 07/09/2009 | US20090176766 Imidazolidinone and imidazolidinethione derivatives |
| 07/09/2009 | US20090176763 Azaindoles useful as inhibitors of JAK and other protein kinases |
| 07/08/2009 | EP2076491A1 New benzamide derivatives as bradykinin antagonists |
| 07/02/2009 | WO2009081349A1 5-phenyl-lh-benz0 [e] [1, 4] diazepine compounds substituted with an hydroxamic acid group as histone deacetylase inhibitors |
| 07/02/2009 | US20090170836 New inhibitors of histone deacetylase |
| 07/02/2009 | US20090170831 Substituted lactams as inhibitors of abeta protein production |
| 07/01/2009 | EP2074083A1 New sulfonamide derivatives as bradykinin antagonists |
| 07/01/2009 | EP1851207B1 Alkyl substituted homopiperazine derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 07/01/2009 | CN101472904A Diazepan derivatives modulators of chemokine receptors |
| 06/30/2009 | US7553976 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them |
| 06/25/2009 | US20090163478 Salts and Crystal Modifications Thereof |
| 06/25/2009 | US20090163476 N-Phenyl Benzamide Derivatives as Sirtuin Modulators |
| 06/23/2009 | US7550456 substituted aryl cycloalkanoyl derivatives, compositions containing these derivatives, and methods of their use for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorder |
| 06/23/2009 | CA2420694C Guanidinobenzamides as mc4-r agonists |
| 06/18/2009 | WO2009075691A1 Cb-1 modulating compounds and their use |
| 06/18/2009 | WO2007027532A3 Niacin receptor agonists, compositions containing such compounds and methods of treatment |
| 06/17/2009 | EP2069317A2 4-oxo-2,3,4,5-tetrahydro-benzo[b][1,4]diazepine derivatives |
| 06/17/2009 | EP2069315A2 Quinazolinone and isoquinolinone acetamide derivatives |
| 06/17/2009 | EP1171428B1 Fab i inhibitors |
| 06/11/2009 | US20090149448 Phenoxyacetic Acid Derivatives Useful for Treating Respiratory Diseases |
| 06/10/2009 | CN101454296A Derivatives of 2-alkoxy-3,4,5-trihydroxy-alkyl amides, preparation and use thereof, and compositions containing the same |
| 06/04/2009 | WO2009068595A1 Novel carboxylic acid 4-phenylazo-phenyl ester derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 06/04/2009 | WO2001060458A3 Inhibitors of prenyl-protein transferase |
| 06/04/2009 | US20090143365 Derivatives of alkylpiperazine- and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors |
| 06/04/2009 | US20090143361 Pyrido[3,2-E]Pyrazines, Process For Preparing The Same, And Their Use As Inhibitors Of Phosphodiesterase 10 |
| 06/04/2009 | US20090143354 P2X7 Receptor Antagonists and Their Use |
| 06/04/2009 | CA2706974A1 Novel carboxylic acid 4-phenylazo-phenyl ester derivatives and their use as monoamine neurotransmitter re-uptake inhibitors |
| 06/03/2009 | CN101448796A Salts and crystal modifications thereof |
| 06/02/2009 | US7541383 Use of carboxylic acid derivatives which modulate the function and/or expression of proteins involved in atopic diseases, inflammatory conditions and cancer; treatment of asthma, allergic diseases and immunologic diseases |
| 06/02/2009 | US7541355 Conversion process for 2,3-benzodiazepine enantiomers |
| 05/28/2009 | US20090137562 Substituted benzyl amine compounds |
| 05/27/2009 | EP2062583A2 Therapeutic applications of pro-apoptotic benzodiazepines |
| 05/26/2009 | US7538114 Glycine transporter-1 inhibitors |
| 05/26/2009 | CA2459432C Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders |
| 05/21/2009 | US20090131415 Cycloalkyloxy-and heterocycloalkyloxypyridine compounds as modulators of the histamine h3 receptor |
| 05/14/2009 | WO2009061916A2 Benzodiazepinone compounds useful in the treatment of skin conditions |
| 05/14/2009 | WO2009060208A1 Pyrrolobenzodiazepines |
| 05/14/2009 | US20090124604 4-oxoquinazolin-3-yl benzamide derivatives for the treatment of cytokine diseases |
| 05/14/2009 | US20090124603 Diazepan Orexin Receptor Antagonists |
| 05/14/2009 | US20090124602 Kinase inhibitors |
| 05/14/2009 | DE102007052900A1 Stereospezifische Hydroxylierung Stereospecific hydroxylation |
| 05/14/2009 | CA2703005A1 Benzodiazepinone compounds useful in the treatment of skin conditions |
| 05/13/2009 | EP2058304A1 P2x4 receptor antagonist |
| 05/13/2009 | EP1587795B1 N- (1-benzyl-2-oxo-2- (1-piperazinyl) ethyl) -1-piperidincarboxamid-derivatives and related compounds use as cgrp-antagonists for treating a headache |
| 05/12/2009 | US7531543 Phenylpiperazine cycloalkanol derivatives and methods of their use |
| 05/07/2009 | WO2009059047A2 Tricyclic compounds and methods for using the same |
| 05/07/2009 | WO2009058238A1 Substituted diazepan orexin receptor antagonists |
| 05/07/2009 | US20090118263 Novel Adenine Compound |
| 05/07/2009 | US20090118244 Benzodiazepinone compounds useful in the treatment of skin conditions |
| 05/07/2009 | CA2703904A1 Substituted diazepan orexin receptor antagonists |
| 05/06/2009 | EP2054398A1 New heterocyclic compounds containing nitrogen atoms or pharmaceutically acceptable salts thereof, process for the preparation thereof and pharmaceutical composition comprising the same for treatment of cancer |
| 05/06/2009 | CN101426771A Process for manufacturing diazepine derivatives |
| 05/05/2009 | US7528249 Amidating a cyclic carboxylic acid (methyl 1-[N-(3-methylbutyl)carbamoyl]cyclopentane-carboxylic acid) with an aminobenzodiazepinone (3-amino-1-methyl-5-phenyl-3H-benzoazepin-2-one) |
| 05/05/2009 | US7528154 Polyarylcarboxamides useful as lipid lowering agents |
| 05/05/2009 | US7528128 Pyrrolo[2,1-C][1,4]benzodiazepine hybrids and a process for the preparation thereof |
| 04/30/2009 | WO2009053763A1 New non-peptide derivatives as bradykinin b1 antagonists |
| 04/30/2009 | WO2007021545A3 Piperazine derivatives |
| 04/30/2009 | US20090111796 7-membered ring compound and method of production and pharmaceutical application thereof |
| 04/30/2009 | US20090111793 Hydroxyalkanoylaminolactams and related structures as inhibitors of a beta protein production |
| 04/30/2009 | CA2703290A1 New non-peptide derivatives as bradykinin b1 antagonists |
| 04/29/2009 | CN101421257A Agents that disrupt cellular replication and their use in inhibiting pathological conditions |
| 04/23/2009 | US20090105228 Heterocyclic benzodiazepine cgrp receptor antagonists |
| 04/23/2009 | US20090105215 Heterocyclic compounds, methods for the preparation thereof, and uses thereof |
| 04/22/2009 | EP2049473A2 Substituted benzyl amine compounds |
| 04/22/2009 | CN100480248C Malonamide derivatives as gamma-secretase inhibitors |
| 04/21/2009 | US7521222 Farnesyl dibenzodiazepinone and processes for its production |
| 04/21/2009 | US7521062 Thiosemicarbazones as anti-virals and immunopotentiators |
| 04/15/2009 | EP1711470B1 Malonamide derivatives blocking the activtiy of gamma-secretase |
| 04/14/2009 | CA2409841C Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| 04/14/2009 | CA2408934C Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists |
| 04/09/2009 | WO2009044007A2 1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazine-6-carboxamide and 2,3,4,5-tetrahydropyrrolo[1,2-a][1,4]-diazépine-7-carboxamide derivatives, preparation and therapeutic use thereof |
| 04/09/2009 | WO2009043747A2 N-heterocyclic biaryl carboxamides as ccr receptor antagonists |
| 04/09/2009 | US20090093464 Naphthalene Derivatives as Modulators of the Glucocorticoid Receptor |
| 04/09/2009 | US20090093463 Novel compounds of substituted and unsubtituted adamantyl amides |