| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 08/28/2008 | US20080207598 Indole derivatives |
| 08/28/2008 | US20080207590 Inhibitors of Histone Deacetylase |
| 08/21/2008 | WO2008099022A1 10-sulfonyl-dibenzodiazepinones useful as hepatitis c virus inhibitors |
| 08/21/2008 | WO2008099019A1 6-hydroxy-dibenzodiazepinones useful as hepatitis c virus inhibitors |
| 08/21/2008 | US20080200456 Adenosine A2B receptor antagonists; asthma, allergies, allergic diseases or an autoimmune disease, diarrheal diseases, insulin resistance, diabetes, cancer, ischemia, reperfusion injuries, retinopathy; e.g. 1,3-Dipropyl-8-(6-chloro-3-pyridyl)xanthine |
| 08/21/2008 | US20080200455 1-Aryl- or 1-Alkylsulfonyl-Heterocyclylbenzazoles As 5-Hydroxytryptamine-6 Ligands |
| 08/21/2008 | US20080199940 Cosmids; vectors; prokaryotics; Micromonospora biosynthesis |
| 08/20/2008 | EP1337251B1 Monocyclic or bicyclic carbocycles and heterocycles as factor xa inhibitors |
| 08/19/2008 | US7414049 gamma -secretase inhibitors; treating Alzheimer's disease by blocking the activity of gamma -secretase and reducing or preventing the formation of the various amyloidogenic Abeta peptides; good thermodynamic solubility and bioavailability |
| 08/14/2008 | US20080194546 wherein: one or two of X5, X6 and X8 is N, and the others are CH; R7 is selected from halo, ORO1, SRS1, NRN1RN2, NRN7aC( .dbd. O)RC1, NRN7bSO2RS2a, an optionally substituted C5-20 heteroaryl group, or an optionally substituted C5-20 aryl group, where RO1 and RS1 are selected from H, |
| 08/14/2008 | US20080194520 Sulfonyl Amino Cyclic Derivatives and Use Thereof |
| 08/13/2008 | CN101239953A Antidepressant arylpiperazine derivatives of heterocycle-fused benzodioxans |
| 08/12/2008 | US7410963 Benzo-1,4-diazepin-2-one derivatives as phosphodiesterase PDE2 inhibitors, preparation and therapeutic use thereof |
| 08/12/2008 | CA2304568C Olanzapine pamoate formulations |
| 08/07/2008 | WO2007126935A3 Diazepan orexin receptor antagonists |
| 08/07/2008 | US20080188465 Stable pure anhydrous polymorphic Form I, free of other polymorphs and solvating agents such as water and organic solvents; anti-psychotic agent |
| 08/07/2008 | US20080188462 reversed chloroquines; to treat chloroquine resistant/sensitive malaria parasites; N'-(7-Chloro-quinolin-4-yl)-N-[3-(10,11-dihydro-dibenzo[b,f]azepin-5-yl)-propyl]-N-methyl-propane-1,3-diamine |
| 08/06/2008 | EP1951249A2 Tyrosine kinase inhibitors |
| 08/06/2008 | EP1951205A2 Stable composition for a pharmaceutical formulation containing olanzapine |
| 07/31/2008 | US20080182993 chemical intermediate is 4-(3,5-bi (1,1- dimethylethyl-4-hydroxyphenyl)-N-methyl-2-thiazolemethylamine |
| 07/30/2008 | EP1592684B1 Malonamide derivatives as gamma-secretase inhibitors |
| 07/30/2008 | CN101233117A Multidentate aza ligands able to complex metal ions and the use thereof in diagnostics and therapy |
| 07/30/2008 | CN100406007C Asthma and allergic inflammation modulators |
| 07/29/2008 | CA2409842C 1,4-diazepan-2,5-dione derivatives and their use as nk-1 receptor antagonists |
| 07/29/2008 | CA2175767C Adhesion receptor antagonists |
| 07/24/2008 | WO2008055068A8 Inhibitors of histone deacetylase |
| 07/24/2008 | US20080176849 e.g. N-hydroxy-3-[4-[[(2-hydroxyethyl)[2-(1H-indol-3-yl)ethyl]-amino]methyl]phenyl]-2E-2-propenamide; histone deacetylase inhibitor; anticarcinogenic, antitumor, antiproliferative agents; improved stability |
| 07/24/2008 | US20080176830 Compounds, Compositions, and Methods |
| 07/23/2008 | CN100404535C Organic compounds as agents for the treatment of aldosterone mediated conditions |
| 07/17/2008 | US20080171737 Cyclic sulfonamide derivatives and methods of their use |
| 07/17/2008 | US20080171735 SUCCINOYLAMINO BENZODIAZEPINES AS INHIBITORS OF Abeta PROTEIN PRODUCTION |
| 07/16/2008 | EP1942905A2 Niacin receptor agonists, compositions containing such compounds and methods of treatment |
| 07/16/2008 | EP1326849B1 Benzodiazepine derivatives as inhibitors of gamma secretase |
| 07/15/2008 | CA2421120C Quinolinone derivatives as tyrosine kinase inhibitors |
| 07/10/2008 | WO2008082887A2 Inhibitors of poly(adp-ribose)polymerase |
| 07/10/2008 | WO2008008884A3 Inhibition of beta-amyloid peptide aggregation |
| 07/10/2008 | US20080167289 Pyrimidinohydrodiazepinones, e.g., 2-(1,6-dihydro-4-methyl-6-oxopyridin-3-ylamino)-9-cyclopentyl-8,9-dihydro-5,7,7-trimethyl-5H-pyrimido[4,5-b][1,4]diazepin-6(7H)-one; especially c-Met kinase inhibitors; anticancer agents |
| 07/10/2008 | CA2672860A1 Inhibitors of poly(adp-ribose)polymerase |
| 07/09/2008 | EP1940805A1 Benzodiazepine and benzopiperazine analog inhibitors of histone deacetylase |
| 07/09/2008 | CN100400523C Substituted piperazines,(1,4) diaszepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists |
| 07/03/2008 | US20080161294 Urea derivative, medicinal composition containing the same, and medicinal use of these |
| 07/03/2008 | US20080161292 Inhibitors of poly(adp-ribose)polymerase |
| 07/03/2008 | US20080161291 Antineoplastic agents |
| 07/03/2008 | US20080161290 Serine hydrolase inhibitors |
| 07/03/2008 | US20080161281 Amino-Substituted Tricyclic Derivatives and Methods of Use |
| 07/02/2008 | EP1937252A2 Methods and compositions for stimulating neurogenesis and inhibiting neuronal degeneration |
| 07/02/2008 | EP1730117A4 Thiourea compositions and uses thereof |
| 07/01/2008 | US7393852 analgesics; antiinflammatory agents; antiarthritic agents;Alzheimer's disease; cirrhosis; antiallergens; antihistamines ; anticancer agents; vision defects |
| 06/26/2008 | WO2008002820A3 Substituted benzyl amine compounds |
| 06/26/2008 | US20080153899 Fatty amine drug conjugates |
| 06/26/2008 | US20080153826 substituted aryl cycloalkanoyl derivatives, compositions containing these derivatives, and methods of their use for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorder |
| 06/26/2008 | US20080153814 8-Chloro-2,3-Benzodiazepine Derivatives |
| 06/26/2008 | US20080153812 Novel compounds |
| 06/25/2008 | EP1935885A2 Melanin concentrating hormone receptor ligands : substituted 1-benzyl-4-aryl piperazine analogues. |
| 06/24/2008 | US7390896 Preventing the deposits of amyloid protein, treating neurodegenerative disease, Alzheimer's disease and Down's Syndrome; {[carbamoyl]cycloalkyl}-N-(2-oxo-5-phenyl((S)-3H-benzo[f]1,4-diazepin-3-yl))- or (2-oxo-5-phenyl((S)-3H-benzo[f]1,4-diazepin-3-yl))-carboxamide |
| 06/24/2008 | US7390802 Substituted lactams as inhibitors of Aβ protein production |
| 06/24/2008 | US7390801 Cycloalkyl, lactam, lactone and related compounds, pharmaceutical compositions comprising same, and methods for inhibiting β-amyloid peptide release and/or its synthesis by use of such compounds |
| 06/24/2008 | US7390800 from a soil; 1,3-diazepine-4-one; antibacterial and anticarcinogenic agent; use for ATP synthesis; low toxicity; micromolecule compound |
| 06/24/2008 | US7390797 Fused indazole compounds |
| 06/19/2008 | US20080146547 e.g. 4-Chloro-1-hydroxy-phthalazine-6-carboxylic acid [4-chloro-3'-(2-dimethylamino-ethoxy)-biphenyl-3-yl]-amide; multifunctioning protein kinase inhibitors; anticarcinogenic, antiinflammatory, antidiabetic agent, neurodegenerative diseases |
| 06/18/2008 | EP1931647A2 Selected cgrp antagonists, methods for the production thereof and their use as medicaments |
| 06/18/2008 | EP1931646A2 Selected cgrp antagonists, a method for the production thereof and use in the form of drugs |
| 06/18/2008 | EP1931347A2 Piperazine derivatives |
| 06/18/2008 | EP1443937B1 Substituted 1,4-benzodiazepines and uses thereof for the treatment of cancer |
| 06/18/2008 | CN101203500A Substituted arylamine compounds and uses as 5-HT6 moderator thereof |
| 06/17/2008 | CA2367704C Pyrazolobenzodiazepines as cdk2 inhibitors |
| 06/12/2008 | US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection |
| 06/12/2008 | US20080139538 Tertiary Carbinamines Having Substituted Heterocycles Which Are Active As Beta-Secretase Inhibitors For The Treatment Of Alzheimer's Disease |
| 06/12/2008 | US20080139536 Benzodiazepines for Treating or Preventing Rsv Infection |
| 06/12/2008 | US20080139535 1-(2-naphthylsulfonyl)-4-(5-hydroxyaminocarbonylthiazol-2-yl)piperazine; antiproliferative agent; cell cycle arrest, cellular differentiation, apoptosis and reversal of the transformed phenotype; |
| 06/11/2008 | EP1928845A2 Aminodiazepines as toll-like receptor modulators |
| 06/11/2008 | EP1928465A1 Benzodiazepine derivatives for treating hepatitis c infection |
| 06/10/2008 | US7384935 Phosphate prodrugs of a farnesyl dibenzodiazepinone, processes for their production and their use as pharmaceuticals |
| 06/05/2008 | US20080132490 1-heteroaryl-4-benzoyl-5-(alkyl or cycloalkyl)-1,4-diazepanes; sleep disorders, analgesics, obesity, Parkinson's disease, psychosis and schizophrenia; 6-fluoro-2-{(5R)-5-methyl-4-[2-(2H-1,2,3-triazol-2-yl)benzoyl]-1,4-diazepan-1-yl}quinazoline for example |
| 06/05/2008 | US20080132489 1-aryl-alkyl-substituted-1,4-diazepine derivatives; 1-(4-Chloro-3-methoxy-phenyl)-3,3,5,5-tetramethyl-[1,4]diazepane for example; antidepressants, analgesics, various psychological disorders, dementia, eating disorders, drug abuse; side effect reduction |
| 06/05/2008 | US20080132482 3-(2(R)-Cyclopentylmethyl-3 (S)-hydroxyl-1-oxo-5-phenylpentyl)amino-1-methyl-5-(4-fluoro-phenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one; neurological disorders related to beta -amyloid production, Alzheimer's disease, Down's Syndrome |
| 06/05/2008 | US20080131943 Polynucleotides for production of farnesyl dibenzodiazepinones |
| 06/05/2008 | DE60129697T2 Kondensierte azepinderivate und ihre verwendung als antidiuretisches mittel Condensed azepine derivatives and their use as antidiuretic agent |
| 05/29/2008 | US20080125413 Antagonist for calcitonin gene related peptide (Cgrp); azepinone ligands; migranes; headaches; 1-[(2-methoxyethyl)-2-oxo-6-phenylazepan-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide |
| 05/29/2008 | US20080125412 Containing a diazacycloalkane ring, especially a 1,4-diazepane ring, e.g., N-p-((4-(alpha-phenylmethoxycarbonylmethyl)-1,4-diazepan-1-yl)phenyl)-o-biphenylcarboxamide, for the treatment of hyperlipidemia, obesity and type II diabetes. |
| 05/28/2008 | EP1925614A1 Anxiolytic agents with reduced sedative and ataxic effects |
| 05/27/2008 | US7378411 Substituted thienopyrimidinones as a mitotic kinesin inhibitor |
| 05/22/2008 | WO2008061108A2 Phthalazine derivatives |
| 05/21/2008 | CN101184758A Novel compounds |
| 05/20/2008 | US7375101 N-(7-chloro-2,3-dihydro-1-methyl-2-oxo-5-phenyl-1H-1,4-benzodiazepin-3-yl)-N'-(5isoquinolinyl)-thiourea; bradykinin receptor B2 antagonists;analgesic; septic shock, pancreatitis, edema, rhinitis, asthma, colitis, arthritis, hepatorenal syndrome, cancer, bacterial and viral infections, ulcerative colitis |
| 05/20/2008 | US7375099 Malonamide derivatives |
| 05/15/2008 | US20080114000 Suppressor of excess accumulation of intracellular sodium ions |
| 05/15/2008 | US20080113968 Substituted piperazines and diazepanes |
| 05/14/2008 | EP1485365B1 Sulfonyl-derivatives as novel inhibitors of histone deacetylase |
| 05/13/2008 | US7371753 Dihydropteridinones, processes for preparing them and their use as pharmaceutical compositions |
| 05/08/2008 | WO2008053913A1 Sulfonylurea derivative capable of selectively inhibiting mmp-13 |
| 05/08/2008 | WO2008052638A1 DIAZEPANE-ACETAMIDE DERIVATIVES AS SELECTIVE 11β-HSD1 INHIBITORS |
| 05/08/2008 | WO2008034735A3 4-oxo-2,3,4,5-tetrahydro-benzo[b][1,4]diazepine derivatives |
| 05/08/2008 | US20080108605 Anxiolytic agents with reduced sedative and ataxic effects |
| 05/08/2008 | US20080108601 anticancer agents; catalytic hydrogenation |
| 05/08/2008 | CA2668504A1 Diazepane-acetamide derivatives as selective 11.beta.-hsd1 inhibitors |
| 05/08/2008 | CA2667826A1 Inhibitors of histone deacetylase |
| 05/07/2008 | EP1918285A1 Diazepane-acetamide derivatives as selective 11beta-HSD1 inhibitors |
| 05/07/2008 | EP1918272A1 Pharmaceutically active compounds and methods of use |
| 05/07/2008 | EP1917012A1 Cell migration modulating compounds |