| Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961) |
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| 04/18/2006 | US7029918 For reference standards in immunoassays; drug screening |
| 04/13/2006 | US20060079512 10-farnesyl-4,6,8-tri(bisbenzyloxyphosphoryloxy)-5,10-dihydro-dibenzo[b,e][1,4]diazepin-11-one; antitumor, anticarcinogenic agent; solid (pancreatic, prostate, colorectal, lung, ovarian cancer) or hematopoietic (leukemia or lymphoma) neoplasm; bactericide, inhibitor of 5-lipoxygenase, cyclooxygenase-2 |
| 04/13/2006 | US20060079509 Antineoplastic agents; inhibitors of cancer cell growth, mammalian lipoxygenase, acute and chronic inflammation |
| 04/13/2006 | US20060079508 10-farnesyl-4,6,8-trihydroxy-dibenzodiazepin-11-one; ECO-4601; anticarcinogenic, antitumor agent; early stage of cancer; reducing side-effects on normal cells |
| 04/13/2006 | US20060079506 Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors |
| 04/06/2006 | WO2006034567A1 Use of compositions comprising farnesyl dibenzodiazepinones for treating neoplastic cells and conditions |
| 04/06/2006 | WO2006001866A3 Crystalline forms of n-desmethylclozapine |
| 04/06/2006 | CA2581658A1 Dibenzodiazepinone analogues, processes for their production and their use as pharmaceuticals |
| 04/05/2006 | EP1294720B1 Non-nucleoside reverse transcriptase inhibitors |
| 04/04/2006 | CA2256492C Diarylalkyl cyclic diamine derivatives as chemokine receptor antagonists |
| 04/04/2006 | CA2241787C Substituted aza- and diazacycloheptane and cyclooctane compounds and their use |
| 03/30/2006 | US20060069088 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
| 03/30/2006 | US20060069083 Pesticidal dibenzo(hetero)azepine derivatives |
| 03/29/2006 | EP1640368A2 Cyclic ureas and processes for their preparation |
| 03/29/2006 | EP1064300A4 Peptide turn mimetics |
| 03/28/2006 | US7019000 administering nitrogen-sulfur compounds, e.g. 4,4-dithiodimorpholine to inhibit binding of the E6 protein by human papilloma virus; treatment of cervical cancer |
| 03/28/2006 | US7018998 substituted 4,5-dihydro-1H-benzo[b][1,4]-diazepin-2-one; amidation of a substituted monoprotected 1,2-diaminobenzene with an ester, deprotecting, cyclization; chronic neurological disorders, psychosis, schizophrenia, Alzheimer's disease |
| 03/23/2006 | WO2006008133A3 Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof |
| 03/23/2006 | DE19547099B4 Verfahren zur Herstellung von (Meth)acrylsäureestern Acrylic acid esters, process for the preparation of (meth) |
| 03/22/2006 | EP1636197A1 Novel 3-substituted-1,4-benzodiazepines |
| 03/21/2006 | US7015214 Such as 7-chloro-2-cyanoimino-5-(cyclopropylmethyloxy)-1,5-dihydro-5-trifluoromethyl-1,3-benzodiazepine |
| 03/21/2006 | US7015213 Use of diazepines for preparing medicines for treating pathological conditions or diseases involving one of the growth hormone release inhibiting factor receptors |
| 03/21/2006 | CA2186285C Carbonyl containing compounds and their derivatives as multi-functional fuel and lube additives |
| 03/16/2006 | WO2006028161A1 Serotonin 5-ht3 receptor agonist |
| 03/15/2006 | EP1403249B1 Cyclic diamine compounds bearing six-membered cyclic groups |
| 03/15/2006 | CN1747938A Novel substituted 2,3-benzodiazepine derivatives |
| 03/09/2006 | WO2005091697A3 Thiourea compositions and uses thereof |
| 03/09/2006 | US20060052597 Aryloxyalkylamine derivatives as h3 receptor ligands |
| 03/09/2006 | US20060052396 Arylamines for the treatment of conditions associated with gsk-3 |
| 03/08/2006 | CN1745083A Pyrrolo[2,1-c][1,4] benzodiazepines as vasopressin agonists |
| 03/08/2006 | CN1745076A Malonamide derivatives as gamma-secretase inhibitors |
| 03/07/2006 | US7008945 Amide derivatives |
| 03/07/2006 | US7008938 Benzene-fused heteroring derivatives and pharmaceutical agents comprising the same as active ingredient |
| 03/02/2006 | WO2005113542A3 N-cyclic sulfonamido inhibitors of gamma secretase |
| 03/02/2006 | CA2578370A1 Triazolobenzodiazepines and their use as vasopressin antagonists |
| 03/01/2006 | CN1740173A Inhibitors of interleukin-1beta converting enzyme |
| 03/01/2006 | CN1243724C Amide derivatives which are useful as cell factor inhibitors |
| 02/23/2006 | US20060040923 1,1-Diethyl-3-(2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)-urea; respiratory syncytial virus; cost efficient replacement for Synagis (palivizumab) used for RSV; respiratory system disorders; asthna; viral diseases; myxoviruses; mumps; flaviviruses; dengue, West Nile, parainfluenza viruses |
| 02/23/2006 | US20060040921 Process and intermediates for the preparation of olanzapine |
| 02/23/2006 | CA2577060A1 Substituted benzofused heterocycles |
| 02/23/2006 | CA2575979A1 Novel serotonin receptor ligands and their uses thereof |
| 02/23/2006 | CA2573730A1 1,2,3,4-tetrahydropyrazin-2-yl acetamides and their use as bradykinin antagonists for the treatment of inflammation related disorders |
| 02/22/2006 | CN1738820A Novel diazabicyclic aryl derivatives |
| 02/22/2006 | CN1738805A N- (1-benzyl-2-oxo-2- (1-piperazinyl) ethyl) -1-piperidincarboxamid-derivatives and related compounds use as CGRP-antagonists for treating a headache |
| 02/22/2006 | CN1242992C Cyclic diamine compounds bearing six-membered cyclic groups |
| 02/16/2006 | US20060035884 N-cyclic sulfonamido inhibitors of gamma secretase |
| 02/16/2006 | US20060034773 Multidentate AZA ligands able to complex metal ions and the use thereof in diagnostics and therapy |
| 02/15/2006 | CN1735609A Diazepanes derivatives useful as LFA inhibitors |
| 02/09/2006 | WO2003090691A3 Method and compositions for identifying anti-hiv therapeutic compounds |
| 02/09/2006 | US20060030553 Cell adhesion inhibitors |
| 02/08/2006 | EP1622865A2 Novel bioisosteres of actinonin |
| 02/08/2006 | EP1183243B1 Short-acting benzodiazepines |
| 02/07/2006 | US6995269 Guanidinobenzamides |
| 02/07/2006 | US6995155 Imines such as 4-(3-((3-(2,4-dichlorophenyl)propanoyl)amino)-1-(3-(morpholin-4-yl)propyl)-2-oxo-2,3-dihydro-1H-1,4-benzodiazepin-5-yl)benzamide, administered for prophylaxis of Alzheimer's disease |
| 02/07/2006 | CA2360308C Glucocorticoid receptor modulators |
| 02/02/2006 | WO2006010511A1 Method for producing 3-(4-piperidinyl)-2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1h)-on |
| 02/02/2006 | US20060025407 Succinoylaminobenzodiazepines as inhibitors of Abeta protein production |
| 02/02/2006 | US20060025404 Such as 1-(4-{[1-(1-methylethyl)-4-piperidinyl]oxy}phenyl)-4-{[4-(methylsulfonyl)phenyl]carbonyl}piperazine; neurodegenerative disorders including Alzheimer's disease; allergic rhinitis |
| 02/02/2006 | US20060024832 Water-soluble derivatives of lipophilic drugs |
| 02/01/2006 | EP1620445A2 Method and compositions for identifying anti-hiv therapeutic compounds |
| 02/01/2006 | CN1729158A Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors |
| 02/01/2006 | CN1239158C 2-methyl-thieno-benzodiazepine formulation |
| 01/26/2006 | US20060020041 substituted ethylene diamines such as N-Geranyl-N'-(2-adamanthyl)ethane-1,2-diamine, used for the treatment of leprosy or tuberculosis caused by mycobacterial infections |
| 01/26/2006 | CA2574237A1 Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof |
| 01/25/2006 | EP1619189A1 N-(3-acyl-2-hydroxyalkyl) cycloalkyl amide derivatives |
| 01/25/2006 | EP1619187A1 Process for the preparation of 3-(4-piperidinyl)- 2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1H)-on |
| 01/25/2006 | EP1618096A1 11-phenyl-dibenzodiazepine derivatives as rxr-antagonists |
| 01/25/2006 | EP1617807A2 Substituted 1,4-diazepines and uses thereof |
| 01/25/2006 | CN1726201A Substituted piperazines,(1,4) diaszepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine h1 and/or h3 antagonists or histamine h3 reverse antagonists |
| 01/18/2006 | EP1616867A1 Hydroxycarboxylic acid derivatives |
| 01/18/2006 | EP1616859A1 Substituted cyclohexyl carboxylic acid compounds |
| 01/18/2006 | EP1615699A2 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors |
| 01/18/2006 | EP1220852B1 Substituted diazepans |
| 01/12/2006 | WO2005103037A3 Selected cgrp antagonists, methods for the production thereof, and use thereof as medicaments |
| 01/12/2006 | US20060009517 Tricyclic inhibitors of poly(ADP-ribose) polymerases |
| 01/12/2006 | US20060009446 New compounds |
| 01/12/2006 | CA2572874A1 Urea derivative |
| 01/12/2006 | CA2570185A1 Stereospecific anxiolytic and anticonvulsant agents with reduced muscle-relaxant, sedative-hypnotic and ataxic effects |
| 01/11/2006 | EP1614678A2 Sulfur substituted sulfonylaminocarboxylic acid N-heteroarylamides, their preparation, their use and pharmaceutical preparations comprising them |
| 01/10/2006 | US6984637 Cyclic amine derivatives-CCR-3 receptor antagonists |
| 01/10/2006 | US6984626 For therapy and prophylaxis of Alzheimer's disease |
| 01/10/2006 | CA2370411C Diazabicyclo compounds for the treatment of schizophrenia and other disorders |
| 01/10/2006 | CA2129990C Benzodiazepin derivatives useful as cck-receptor antagonists |
| 01/05/2006 | WO2006001866A2 Crystalline forms of n-desmethylclozapine |
| 01/05/2006 | CA2560671A1 Crystalline forms of n-desmethylclozapine |
| 01/04/2006 | EP1611110A1 Adenosine deaminase inhibitor and novel bacillus sp. iada-7 strain which produces it |
| 12/29/2005 | US20050288275 New compounds |
| 12/28/2005 | EP1608650A1 Pyrene-linked pyrrolo(2,1-c)(1,4)benzodiazepine derivatives useful as anticancer agents |
| 12/28/2005 | EP1608374A1 2-phenoxy- and 2-phenylsulfomamide derivatives with ccr3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders |
| 12/28/2005 | EP0945445B9 1,5-benzodiazepine derivatives |
| 12/22/2005 | WO2005103041A9 Treatment of cns disorders using cns target modulators |
| 12/22/2005 | US20050282800 Method of synthesis and isolation of solid N-desmethylclozapine and crystalline forms thereof |
| 12/21/2005 | EP1606268A1 Heterocyclic kinase inhibitors |
| 12/20/2005 | US6977298 Tricyclic inhibitors of poly(ADP-ribose) polymerases |
| 12/15/2005 | WO2005117876A1 Dual small molecule inhibitors of cancer and angiogenesis |
| 12/15/2005 | CA2568622A1 Dual small molecule inhibitors of cancer and angiogenesis |
| 12/08/2005 | WO2005116034A1 Tetraazabenzo[e]azulene derivatives and analogs thereof |
| 12/08/2005 | WO2004096134A3 Substituted 1,4-diazepines and uses thereof |
| 12/08/2005 | CA2568056A1 Tetraazabenzo[e]azulene derivatives and analogs thereof |
| 12/07/2005 | EP0957917B1 Vitronectin receptor antagonists |