Patents
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
10/2007
10/17/2007CN101056842A Prodrugs of (2R)-2-propyloctanoic acid for treatment of stroke
10/17/2007CN100343285C Heterocyclic alkoxyl amine as regulator in controlled free radical polymerization method
10/16/2007US7282496 Rheumatic diseases; bone disorders; Aids; antiinflammatory agents
10/16/2007US7282494 Heteroaryl diazacycloalkanes, their preparation and use
10/11/2007US20070238723 Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine receptors
10/10/2007EP1381608B1 Cyclohexylphenyl vasopressin agonists
10/09/2007US7279582 For example (2S, 3S, 5S)-2-(2,6-dimethylphenoxyacetyl)amino-3-hydroxy-5-(2S-(1-tetrahydro-pyrimid-2-onyl)-3-methyl butanoyl)amino-1,6-diphenylhexane; HIV therapy
10/09/2007US7279573 Benzodiazepine derivatives that may be fused to a pyrroline or piperidine ring; e.g., N-[1 (R)-(3-Aminopropylcarbamoyl)-2-(naphthalen-2-yl)ethyl]-3-(5,11-dioxo-2,3-dihydro-1H-(11aS)-pyrrolo[2,1-c][1,4]benzodiazepin-10-yl)propionamide; increasing levels of endogenous growth hormones in humans and animals
10/04/2007WO2007110363A1 Novel guanidine derivatives and their medical use
10/04/2007US20070232594 Aromatic amide derivatives, medicinal compositions containing the same, medical uses of both
10/03/2007EP1839662A1 Antitumor agent
10/03/2007CN101048391A Tetracyclic indole derivatives as antiviral agents
10/02/2007US7276496 Cyclic malonamides as inhibitors of Aβ protein protection
10/02/2007US7276495 Substituted lactams as inhibitors of Aβ protein production
10/02/2007US7276348 Using benzodiazepine derivatives to treat and prevent defects in programed cell death, autoimmune, inflammatory and cell proliferative diseases
09/2007
09/27/2007WO2007107352A1 Agents that disrupt cellular replication and their use in inhibiting pathological conditions
09/27/2007CA2646541A1 Agents that disrupt cellular replication and their use in inhibiting pathological conditions
09/26/2007CN101041669A Non nucleoside reverse transcriptase inhibitors
09/20/2007WO2007105225A1 PROCESS FOR PRODUCING PURE AND STABLE FORM OF 2-METHYL-4-(4- METHYL- 1 -PIPERAZINYL)-10H-THIENO[2,3-b] [ 1,5]BENZODIAZEPINE
09/19/2007CN101039927A Serotonin 5-HT3 receptor agonist
09/18/2007US7271164 Therapy , prevention of obsessive-complusive disorders; antidepressants; anxiety; schizophrenia; eating disorders; obesity; antiepileptic agents central nervous system disorders; sleep disorders
09/18/2007US7271163 Cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
09/18/2007US7271162 Cycloocta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives
09/13/2007WO2007102936A2 Polynucleotides for production of farnesyl dibenzodiazepinones
09/13/2007WO2007102392A1 Mmp-13-selective inhibitor
09/13/2007US20070213316 N,N'-substituted-1,3-diamino-2-hydroxypropane derivatives
09/12/2007CN101033232A Method of preparing olanzapine crystal system I
09/11/2007US7268128 Increase the intracellular cAMP level and further inhibit the activation of T cells; allergic diseases, inflammatory or immunological diseases
09/11/2007CA2373506C Process for manufacturing diazepine derivatives
09/11/2007CA2143848C Complex combinatorial chemical libraries encoded with tags
09/07/2007WO2007100852A1 Therapeutic piperazines as pde4 inhibitors
09/07/2007CA2644069A1 Therapeutic piperazines as pde4 inhibitors
09/06/2007US20070208008 Substituted sulfonamides and ureas useful for inhibiting kinase activity
09/05/2007EP1828160A1 Sulfonyl amino cyclic derivatives and use thereof as mmp inhibitors
09/05/2007EP1057815B1 Cyclic amide compounds
09/04/2007US7265106 Chromatography; separation of enantiomorphs
09/04/2007US7265104 Tetraazabenzo[e]azulene derivatives and analogs thereof
08/2007
08/29/2007EP1417184B1 Composition for dyeing keratinous fibres containing a paraphenylenediamine substituted by a diazacycloheptane radical
08/28/2007US7262188 Phenyl sulfone derivatives and their use in the treatment of CNS disorders
08/28/2007US7262187 Substituted oxazolo- and thizaolopyrimidinones as a mitotic kinesin inhibitor
08/28/2007US7262186 Kinesin spindle protein inhibitor; antiproliferative agents; anticancer agents; 4-(2,5-difluorophenyl0-N-3-fluoropyrrolidin-3-yl)-2-hydroxymethyl-2-phenyl-2,5-dihydro-1N-pyrrol-1-carboxamide
08/22/2007EP1820799A1 2,3,4,5-tetrahydro-1h-1,5-benzodiazepine derivative and medicinal composition
08/22/2007EP1820798A1 7-membered ring compound, process for producing the same, and medicinal use thereof
08/21/2007US7259160 Hexahydrodiazepinones as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes
08/21/2007CA2379445C Lactams substituted by cyclic succinates as inhibitors of a.beta. protein production
08/16/2007WO2007074130A3 3-(4-piperidinyl)-2,3,4,5-tetrahydro-1,3-benzodiazepine-2(1h)-one
08/16/2007US20070191312 Novel heterocyclic compounds, preparation process and intermediates, and use as medicaments, in particular as beta-lactamase inhibitors and antibacterials
08/16/2007US20070191309 a 7 or 8-hydroxy; a protected oxygen at position 11; carbamate protecting group at the N10 position (oxycarbonyl); reaction with a diiodoalkane; antitumour anthramycin antibiotic
08/16/2007US20070190523 Method and compositions for identifying anti-hiv therapeutic compounds
08/15/2007EP1818326A1 Nitrogen-containing heterocyclic compounds and pharmaceutical composition containing the compounds
08/15/2007EP1817294A1 1,2,3,4-tetrahydropyrazin-2-yl acetamides and their use as bradykinin antagonists for the treatment of inflammation related disorders
08/15/2007CN101018774A Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof
08/09/2007US20070185094 Novel 3-substitued-1,4-benzodiazepines
08/09/2007CA2640627A1 Crystalline forms of a farnesyl dibenzodiazepinone
08/08/2007CN101012294A Method of preparing benzodiazepines pharmaceutical molecular engram solid phase extractant
08/07/2007US7253157 Containing a diazacycloalkane ring, especially a 1,4-diazepane ring, e.g., N-p-((4-(alpha-phenylmethoxycarbonylmethyl)-1,4-diazepan-1-yl)phenyl)-o-biphenylcarboxamide, for the treatment of hyperlipidemia, obesity and type II diabetes.
08/01/2007EP1813603A1 Aromatic amide derivatives, medicinal compositions containing the same, medical uses of both
08/01/2007EP1461038B1 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders
08/01/2007EP1294698B1 Fused azepine derivatives and their use as antidiuretic agents
08/01/2007CN1329382C Novel arylsusfonamide compounds for treatment of obesity, type II diabetes and CNS-disorders
07/2007
07/31/2007US7250410 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses thereof
07/26/2007US20070173502 Novel urea derivatives, method for preparing same, use thereof as medicines, pharmaceutical compositions and novel use
07/26/2007US20070173491 Substituted lactams as inhibitors of Abeta protein production
07/25/2007EP1809612A1 Dibenzodiazepinone analogues, processes for their production and their use as pharmaceuticals
07/25/2007EP1809296A2 Novel [1,4]benzodiazepines as vasopressin v2 receptor antagonists
07/24/2007USRE39743 Antibiotics, bactericides
07/19/2007WO2007080140A1 Cyclohexyl piperazinyl methanone derivatives and their use as histamine h3 receptor modulators
07/19/2007WO2007035722A3 Methods and compositions for stimulating neurogenesis and inhibiting neuronal degeneration
07/19/2007US20070167436 Cyclohexyl piperazinyl methanone derivatives
07/19/2007CA2635719A1 Cyclohexyl piperazinyl methanone derivatives and their use as histamine h3 receptor modulators
07/18/2007EP1807403A2 Tetracyclic indole derivatives as antiviral agents
07/18/2007EP1509537B1 Cellular accumulation of phosphonate analogs of hiv protease inhibitor compounds and the compounds as such
07/18/2007CN1326857C Novel 1,4-diazabicycloalkane derivatives, their preparation and use
07/17/2007US7244843 Modulators of serotonin receptors
07/17/2007US7244723 Kinesin spindle protein (KSP) inhibitors, e.g., 3-benzyl-2-(1-{(4-bromobenzyl)[2-(dimethylamino)ethyl]amino}propyl)furo[2,3-d]pyrimidin-4(3H)-one; antiproliferative and -carcinogenic agents; side effects reduction; cancers of the brain, genitourinary tract, lymphatic system, stomach, larynx and lung
07/12/2007WO2007079078A1 Diamine derivatives as inhibitors of leukotriene a4 hydrolase
07/12/2007WO2007079003A2 Amide inhibitors of leukotriene a4 hydrolase
07/12/2007WO2007078808A2 Method for isolating (r)-tofisopam
07/12/2007WO2007077469A1 Optical isomers of dihydro-2,3-benzodiazepines and their stereoselective synthesis
07/12/2007US20070161628 Phosphodiesterase inhibitors
07/12/2007US20070160537 In vivo screening method of therapeutic agent for memory/learning dysfunctions by schizophrenia
07/12/2007CA2633804A1 Optical isomers of dihydro-2,3-benzodiazepines and their stereoselective synthesis
07/12/2007CA2633285A1 Method for isolating (r)-tofisopam
07/11/2007EP1806341A2 (+)Phenyl-(4-{4-[(4'-trifluoromethyl-biphenyl-2-carbonyl)-amino]-phenyl}-piperidin-1-yl)-acetic acid methyl ester as lipid lowering agent
07/10/2007US7241787 Substituted N-cycloexylimidazolinones, process for their preparation and their use as medicaments
07/10/2007US7241767 And thiones, 1-substituted with a pyrazolyl(thio)carbonyl group, e.g., 6-Bromo-1-[[3-bromo-1-(3-chloro-2-pyridinyl)-1H-pyrazol-5-yl]carbonyl]-8-methyl-3-(1-methylethyl)-2,4(1H,3R)-quinazolinedione; especially for use in growing and stored agronomic crops
07/10/2007US7241765 Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues
07/10/2007US7241317 For the oxidation dyeing of keratinous fibers, in particular human hair
07/10/2007CA2466340C Farnesyl dibenzodiazepinone, processes for its production and its use as a pharmaceutical
07/05/2007WO2007076555A2 A location based wireless collaborative environment with a visual user interface
07/05/2007WO2007026254A3 Benzodiazepine derivatives , their preparation and the therapeutic use thereof
07/05/2007US20070155730 Benzodiazepine And Benzopiperazine Analog Inhibitors Of Histone Deacetylase
07/05/2007US20070155727 Amide inhibitors of leukotriene A4 hydrolase
07/05/2007US20070155725 N-(1-Aza-bicyclo[2.2.2]oct-3-yl)-5-cyano-2-(3,5-dichloro-phenoxy)-benzenesulfonamide; asthma, allergic rhinitis or lung granuloma, HIV; CC type chemokine receptor antagonist
07/05/2007CA2633932A1 3-(4-piperidinyl)-2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1h)-one
07/04/2007EP1803711A1 Multidentate aza ligands able to complex metal ions and the use thereof in diagnostics and therapy
07/03/2007US7238688 For therapy of allergy, allergy-induced airway responses, congestion, hypotension, cardiovascular disease, hypotension, diseases of the GI tract, hyper and hypo motility and acidic secretion of the gastrointestinal tract, obesity, sleep
07/03/2007US7238685 E.g., substituted 2,3,5,10b-tetraaza-benzo[e]azulen-6-yl)-acetic acids, 2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepin-5-yl)-(4,6-dimethoxy-pyrimidin-2-yloxy)-acetic acids and 2,3,4,5-tetrahydro-benzo[e][1,4]diazepin-1-ylmethyl}-benzoates; treating vasoconstriction, proliferation and inflammation
06/2007
06/28/2007WO2007072974A1 P2x4 receptor antagonist
06/27/2007CN1989114A Process for the preparation of 3-(4-piperidinyl)- 2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1H)-on
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