Patents
Sitemap › C07 - Organic chemistry › C07D - Heterocyclic compounds › C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
08/2010
08/04/2010EP2010506B1 Diazepan derivatives modulators of chemokine receptors
07/2010
07/29/2010WO2010084979A1 Benzodiazepin-2-on derivatives
07/29/2010US20100190688 Tetrapeptide analogs
07/29/2010US20100189762 Triarylmethane analogs and their use in treating cancers
07/29/2010CA2749700A1 Benzodiazepin-2-on derivatives
07/27/2010US7763605 [1,4]benzodiazepines as vasopressin V2 receptor antagonists
07/22/2010US20100183712 Acylated indanyl amines and their use as pharmaceuticals
07/20/2010US7759354 Bicyclic guanidine derivatives as asparyl protease inhibitors, compositions, and uses thereof
07/20/2010US7759346 [[2-(amino-3,4-dioxo-1-cyclobuten-1-yl)amino]alkyl]-acid derivatives for the treatment of pain
07/20/2010US7759338 Programmed cell death, autoimmunity, inflammation, hyperproliferation; easy formulation, shelf life
07/20/2010US7759337 N-cyclopropyl-4-methyl-3-{1-[(2R)-2-methylpiperazin-1-yl]phthalazin-6-yl}benzamide, useful for the prophylaxis and treatment of protein kinase mediated diseases including rheumatoid arthritis, psoriasis and other inflammation disorders
07/20/2010CA2431982C Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
07/14/2010EP2206704A1 Pharmaceutically active diazepanes
07/14/2010EP2205583A2 N-heterocyclic biaryl carboxamides as ccr receptor antagonists
07/13/2010US7754711 Pyridazine derivatives and their use as therapeutic agents
07/13/2010US7753965 Hair dye composition
07/08/2010US20100173896 Organic Compounds
07/06/2010US7750150 Process for producing acid adduct salt of polyacidic base compound
07/01/2010US20100166887 DIBENZO[b,e][1,4]DIAZEPINE MODULATORS OF DOPAMINE RECEPTORS, SEROTONIN RECEPTORS, ADRENERGIC RECEPTORS, ACETYLCHOLINE RECEPTORS, AND/OR HISTAMINE RECEPTORS
06/2010
06/29/2010US7745431 leukotriene B4 inhibitor; optically pure R-enantionmer of tofisopam
06/24/2010US20100160299 Dendrimer conjugates
06/24/2010US20100160297 Compounds for pim kinase inhibition and for treating malignancy
06/24/2010US20100160291 Tricyclic spiro-oxindole derivatives and their uses as therapeutic agents
06/24/2010US20100160280 Aminopyridine and carboxypyridine compounds as phosphodiesterase 10 inhibitors
06/23/2010EP2199295A1 Compounds with 7-member cycle and the pharmaceutical use thereof for preventing and treating diabetes and metabolism syndrome
06/23/2010EP2197855A1 Heterocyclic scaffolds useful for preparation of combinatorial libraries, libraries and methods of preparation thereof
06/22/2010US7741318 used for treating central nervous system diseases such as depression, cognitive diseases and neurodegenerative diseases such as Parkinson's disease, alzheimer's disease or psychoses, and stroke
06/17/2010US20100152171 CGRP Antagonists
06/17/2010US20100152168 Substituted benzimidazolone derivatives, medicaments comprising them and their use
06/17/2010US20100152138 Cyclic amine bace-1 inhibitors having a benzamide substituent
06/17/2010US20100150831 Modulators of cxcr7
06/16/2010CN101735159A Method for producing monoacetylated homopiperazine
06/16/2010CN101270093B Novel method for synthesizing 2,3,4,5-tetrahydric--1H-1,4-benzodiazepine
06/15/2010US7737272 Diazaphosphacycle transition metal complexes
06/15/2010US7737142 (Thio) carbamoyl-cyclohexane derivatives as D3/D2 receptor antagonists
06/10/2010US20100144715 Substituted Benzodiazepinones, Benzoxazepinones and Benzothiazepinones as Sodium Channel Blockers
06/10/2010US20100144708 Heterocyclic compounds containing nitrogen atoms or pharmaceutically acceptable salts thereof, process for the preparation thereof and pharmaceutical composition comprising the same for treatment of cancer
06/10/2010US20100144707 Pharmacokinetically improved compounds
06/09/2010CN1694874B Benzodiazepine derivatives and pharmaceutical compositions containing them
06/03/2010US20100137287 Aryl-and heteroaryl-substituted tetrahydrobenzo-1,4-diazepines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
06/03/2010US20100135999 Quinoline-carboxamide derivatives as p2y12 antagonists
06/02/2010EP2190827A1 N-benzyl, n' -arylcarbonylpiperazine derivatives as lxr modulators
06/02/2010EP1608650B1 Pyrene-linked pyrrolo(2,1-c)(1,4)benzodiazepine derivatives useful as anticancer agents
06/02/2010CN1938280B Thiourea compositions and uses thereof
06/01/2010US7728069 Ring-opening reaction of a substituted 2-oxo-1,3-dioxolane or a substituted 2-oxo-1,3-diazepane with a biomolecule, a polymer or a surface to prepare a finish, dispersant, emulsifier, adhesion promoter, adhesive or contact adhesive for modifying surfaces or for immobilizing active substances
06/01/2010US7727997 N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives
06/01/2010US7727982 N-(5-bromo-2-pyridinyl)-(2-4-[(2-aminosulfonyl)phenyl]phenylcarbonylamino)phenylcarboxamide; potent and highly selective inhibitors; coagulation disorders; antithrombotic agents; diagnostic reagents; good bioavailability and/or solubility
05/2010
05/27/2010US20100130483 Novel diazabicyclic aryl derivatives
05/27/2010US20100130482 Diazabicyclic aryl derivatives as nicotinic acetylcholine receptor ligands
05/27/2010US20100130481 Anticonvulsant and anxiolytic methods of using receptor subtype selective agents
05/27/2010US20100130474 Alpha7 nicotinic acetylcholine receptor inhibitors
05/27/2010US20100129473 AMINO SUBSTITUTED DIARYL[a,d]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS
05/26/2010EP2188269A1 New compounds
05/26/2010EP1874739B1 Pharmaceutically active diazepanes
05/26/2010CN1910137B Aryl aniline derivatives as beta2 adrenergic receptor agonists
05/25/2010CA2431761C Novel 2,3-benzodiazepine derivatives and pharmaceutical compositions containing the same as the active ingredient
05/20/2010US20100125065 Carboline derivatives useful in the inhibition of angiogenesis
05/19/2010EP2185561A2 1,2,3,4-tetrahydropyrroloý1,2-a¨pyrazine-6-carboxamide and 2,3,4,5-tetrahydropyrroloý1,2-a¨ý1,4¨-diazépine-7-carboxamide derivatives, preparation and therapeutic use thereof
05/19/2010EP1371646B1 Aryl-substituted alicyclic compound and medical composition comprising the same
05/18/2010US7718795 Succinoylamino benzodiazepines as inhibitors of aβ protein production
05/18/2010US7718658 Saturated ring with 2 nitrogens, 1 of which is 2-(o-(difluoromethyl)phenyl)quinazol-4-yl-substituted and the other is oxyalkanoyl-substituted; inhibitors of voltage-gated sodium channels and calcium channels; treating acute, chronic, neuropathic, or inflammatory pain
05/18/2010US7718650 Piperazino or diazepino-substituted arylsulfonamides; obesity, type II diabetes and/or central nervous system disorders; 4-chloro-N-[5-(4-methyl-1,4-diazepan-1-yl)-2-nitrophenyl]benzenesulfonamide for example; Serotonin 5-HT6 receptor antagonist activity
05/13/2010US20100121049 Indenoisoquinolinone analogs and methods of use thereof
05/12/2010EP2078001B1 Diazepane-acetamide derivatives as selective 11 -hsd1 inhibitors
05/12/2010CN101503394B High piperazine acetydrazide derivatives, and preparation and use thereof
05/11/2010US7713963 Acylated indanyl amines and their use as pharmaceuticals
05/11/2010CA2462110C Phenyl-piperazine derivatives as serotonin reuptake inhibitors
05/06/2010WO2010051206A1 Novel cyclic benzimidazole derivatives useful anti-diabetic agents
05/06/2010US20100113771 Novel benzothiazole and benzoxazole linked pyrrolo[2,1-c] [1, 4] benzodiazepine hybrids as novel antitumour agents and process for the preparation thereof
05/06/2010US20100113428 Diazabicyclic aryl derivatives as cholinergic receptor modulators
05/06/2010US20100113424 N-benzyl pyrrolidine derivatives
05/06/2010US20100113414 Thiazolyl-dihydro-indazoles
05/06/2010US20100113391 Bicyclic heterocyclic compound
05/06/2010CA2741672A1 Novel cyclic benzimidazole derivatives useful anti-diabetic agents
05/04/2010US7709487 Sulfonyl-derivatives as novel inhibitors of histone deacetylase
05/04/2010US7709470 retinopathy, nephropathy, neuropathy, and hyperlipidemia, obesity, dyslipidemia, and osteoporosis; Retinoid X receptors (RXRs); 4-(2-Cyano-5,7,7,10,10-pentamethyl-7,8,9,10-tetrahydro-5H-5,13-diaza-benzo[4,5]-cyclohepta[1,2-b]naphthalen-12-yl)-2-fluoro-benzoic Acid
04/2010
04/29/2010WO2010048138A1 Synthesis of intermediates useful for the production of certain cgrp inhibitors and intermediates used in such synthesis
04/29/2010WO2010047982A1 Novel cyclic benzimidazole derivatives useful anti-diabetic agents
04/29/2010WO2010046929A2 Novel polymorphic forms of temazepam and processes for preparing the same
04/29/2010US20100105894 Cyclopropane compounds and pharmaceutical use thereof
04/29/2010CA2741125A1 Novel cyclic benzimidazole derivatives useful anti-diabetic agents
04/27/2010US7705143 Benzoimidazole compounds
04/27/2010US7704998 Sulfonyl-derivatives as novel inhibitors or histone deacetylase
04/27/2010US7704997 Amino-tetrazole analogues and methods of use
04/22/2010US20100099665 Isoquinolinone derivatives
04/21/2010EP1272175B1 N,n'-diaryl guanidines as il-8 receptor antagonists
04/21/2010CN101696144A Method for preparing amine from ammonium salts
04/20/2010US7700628 Aromatic ether derivatives useful as thrombin inhibitors
04/20/2010US7700591 to prevent or treat inflammatory and immunoregulatory disorders and diseases, allergic diseases, atopic conditions including allergic rhinitis, dermatitis, conjunctivitis, and asthma, as well as autoimmune pathologies such as rheumatoid arthritis and atherosclerosis
04/20/2010US7700587 Haloperidol analogs
04/20/2010US7700586 Arylsulfonamide derivatives for use as ccr3 antagonists in the treatment of inflammatory and immunological disorders
04/15/2010US20100093704 Novel psychotropic agents having glutamate nmda activity
04/15/2010US20100093055 Remedy for diabetes
04/14/2010EP1694410B1 Cyclopropane derivatives and pharmaceutical use thereof
04/13/2010CA2336807C Sulfur substituted sulfonylaminocarboxylic acid n-arylamides, their preparation, their use and pharmaceutical preparations comprising them
04/08/2010WO2009053763A8 New non-peptide derivatives as bradykinin b1 antagonists
04/08/2010US20100087410 Aryl aniline derivatives as beta2 adrenergic receptor agonists
04/07/2010CN1872854B Antibiotic in lactam class, and prepartion method
04/06/2010US7691837 e.g. 1-{[1,5-bis(4-cholorophenyl)-2-methylpyrrol-3-yl]methyl}-4-(4-fluoro-phenyl)piperazine; Mycobacterium tuberculosis, drug resistant Mycobacterium tuberculosis, Mycobacterium avium-intracellulare complex, Mycobacterium fortuitum or Mycobacterium kansasi
03/2010
03/25/2010US20100075954 Substituted imidazo[1,5-a][1,2,4]triazolo[1,5-d][1,4]benzodiazepine derivatives
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