Patents
Patents for C07D 243 - Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms (5,961)
10/2012
10/24/2012CN102753528A Diphenyl azepine derivatives as monoamine reuptake inhibitors
10/24/2012CN101628897B Method for preparing 2,3-dihydro-1H-1,4-benzodiazepine compounds
10/18/2012US20120264746 Cell migration modulating compounds
10/17/2012EP2509600A1 Therapeutically active compounds for use in the treatment of cancer characterized as having an idh mutation
10/11/2012WO2012035549A3 An improved process for the synthesis of beta amino acid derivatives
10/11/2012US20120259111 Seven-membered ring compound and pharmaceutical use therefor
10/11/2012US20120258960 Novel multifunctional peptidase inhibitors, especially for medical use
10/11/2012US20120255898 Semipermeable polymers and method for producing same
10/10/2012EP2508515A1 Ligands for g-protein coupled receptors
10/10/2012EP2507215A1 Diphenyl azepine derivatives as monoamine reuptake inhibitors
10/10/2012CN101821245B New compounds
10/10/2012CN101616919B Inhibitors of poly(adp-ribose)polymerase
10/04/2012US20120252792 Methods and compositions for modulating rho-mediated gene transcription
10/03/2012CN101679290B 3- to 7-membered 1,3-diaza-4-oxo-heterocyclic derivatives capable of releasing active aldehydes or ketones
10/02/2012US8278334 Cyclic amine BACE-1 inhibitors having a benzamide substituent
09/2012
09/27/2012WO2012129353A1 Bis(fluoroalkyl)-1,4-benzodiazepinone compounds
09/27/2012US20120245151 Bisfluoroalkyl-1,4-benzodiazepinone compounds
09/27/2012US20120245141 Activators of human pyruvate kinase
09/27/2012CA2830902A1 Bis(fluoroalkyl)-1,4-benzodiazepinone compounds
09/26/2012CN102690239A Synthesis method of 1, 5-benzodiazepine derivative
09/26/2012CN101448796B Salts and crystal modifications thereof
09/20/2012WO2012124696A1 Guanidine compound
09/20/2012US20120238518 Diazeniumdiolated compounds, pharmaceutical compositions, and method of treating cancer
09/20/2012CA2830157A1 Guanidine compound
09/19/2012EP2498599A1 Analgesic that binds filamin a
09/18/2012US8268894 Compositions and methods for the treatment of infectious diseases
09/18/2012US8268803 5, 6-ring annulated indole derivatives and use thereof
09/13/2012WO2011100838A8 Derivatives of 1-phenyl-1,5-dihydro-benzo[b] [1.4]diazepine-2.4-dione as inhibitors of hiv replication
09/13/2012US20120232067 Benzodiazepinone compounds and methods of treatment using same
09/12/2012CN102666500A Seven-membered ring compound and pharmaceutical use therefor
09/11/2012US8263781 Substituted aminothiazolone indazoles as estrogen related receptor-alpha modulators
09/11/2012CA2576862C A process for producing pure form of 2-methyl-4-(4-methyl-1-piperazinyl)-10h-thieno[2,3-b][1,5]benzodiazepine
09/11/2012CA2572811C Method for producing 3-(4-piperidinyl)-2,3,4,5-tetrahydro-1,3-benzodiazepin-2(1h)-one
09/06/2012US20120225866 Nitrogen-containing compounds and pharmaceutical compositions thereof for the treatment of atrial fibrillation
09/05/2012CN101304743B Methods and compositions for stimulating neurogenesis and inhibiting neuronal degeneration
08/2012
08/30/2012WO2012115608A2 Polyamine inhibitors for the treatment and prevention of parkinson's disease
08/29/2012EP2491022A1 Diazepam derivatives as modulators of chemokine receptors
08/28/2012US8252786 Compound that can inhibit UBC13-UEV interactions, pharmaceutical compositions and therapeutic uses
08/23/2012US20120214801 Compositions and methods relating to novel compounds and targets thereof
08/23/2012US20120214792 Thieno- adn furo-pyrimidine modulators of the histamine h4 receptor
08/22/2012EP2489657A2 Inhibitors of histone deacetylase
08/22/2012EP1820798B1 7-membered ring compound, process for producing the same, and medicinal use thereof
08/15/2012EP2485728A1 Wnt pathway antagonists
08/15/2012CN102639512A Process for producing benzo[b][1,4]diazepine-2,4-dione compound
08/15/2012CN101495463B Seven-membered ring compound, production method thereof and pharmaceutical use thereof
08/14/2012US8242264 Process for preparing 4-acetyl-2,3,4,5-tetrahydro-benzo[1,4]diazepine and the intermediates thereof
08/14/2012US8242118 Arylsulfonamide derivatives for use as CCR3 antagonists in the treatment of inflammatory and immunological disorders
08/14/2012US8242108 Cell migration modulating compounds
08/14/2012US8242107 Diazepane-acetamide derivatives as selective 11β-HSD1 inhibitors
08/09/2012US20120202800 Dual small molecule inhibitors of cancer and angiogenesis
08/09/2012US20120202793 Rho kinase inhibitors
08/07/2012US8236949 Tetrazine-based bio-orthogonal coupling reagents and methods
08/07/2012US8236793 Diazabicyclic aryl derivatives as cholinergic receptor modulators
08/07/2012US8236792 Substituted pyrrolidine amides as modulators of the histamine H3 receptor
08/07/2012CA2412782C Cyclic urea compounds and preparation thereof
08/01/2012EP2480538A1 [1,4]-benzodiazepines as vasopressin v2 receptor antagonists
07/2012
07/26/2012WO2012097682A1 Bicyclic inhibitors of alk
07/26/2012US20120189614 Inhibitors of filovirus entry into host cells
07/26/2012CA2824871A1 Bicyclic inhibitors of alk
07/19/2012US20120184537 [1,4]-benzodiazepines as vasopressin v2 receptor antagonists
07/18/2012EP2476756A1 Amine-containing lipids and uses thereof
07/17/2012US8222243 Therapeutic isoxazole compounds
07/10/2012US8217029 Oxazolidinone antibiotics
07/10/2012CA2537440C Malonamide derivatives blocking the activity of gama-secretase
07/10/2012CA2360003C Tricyclic inhibitors of poly(adp-ribose) polymerases
07/04/2012EP2470020A1 Benzodiazepinone compounds and methods of treatment using same
07/04/2012CN101516859B 4-oxo-2,3,4,5-tetrahydro-benzo[b][1,4]diazepine derivatives
06/2012
06/27/2012EP2468733A1 Process for producing benzo[b][1,4]diazepine-2,4-dione compound
06/27/2012EP2467364A2 Nitrogen-containing compounds and pharmaceutical compositions thereof for the treatment of atrial fibrillation
06/27/2012CN102512424A Compositions and methods relating to novel compounds and targets thereof
06/21/2012WO2012031090A9 Small molecule inhibitors of ebola and lassa fever viruses and methods of use
06/20/2012EP2300473B1 Fumarate salt of 4-bromophenyl 1,4-diazabicyclo[3.2.2]nonane-4-carboxylate, crystalline forms thereof, preparation thereof and therapeutic use thereof
06/20/2012EP1663996B1 (thio)carbamoyl-cyclohexane derivatives as d3/d2 receptor antagonists
06/20/2012CN102510859A [1,4]-benzodiazepines as vasopressin v2 receptor antagonists
06/19/2012USRE43481 Diazepan derivatives or salts thereof
06/19/2012US8203001 Chemical compounds
06/19/2012US8202989 One step process for the preparation of substituted 5, 10-dihydrodibenzo [b,e][1, 4]diazepine-11-ones
06/14/2012US20120149899 Process for producing benzo[b][1,4]diazepine-2,4-dione compound
06/07/2012WO2012072620A1 7-nitro-5-phenyl-1-(pyrrolidin-1-ylmethyl)-1h-benzo[e][1,4]diazepin-2(3h)-one and other benzodiazepine derivatives
06/07/2012US20120142674 N-phenyl-(homo)piperazinyl-benzenesulfonyl or benzenesulfonamide compounds suitable for treating disorders that respond to the modulation of the serotonin 5-ht6 receptor
06/06/2012CN101472904B Diazepan derivatives modulators of chemokine receptors
06/05/2012US8193178 Thieno- and furo-pyrimidine modulators of the histamine H4 receptor
05/2012
05/30/2012CN102482234A Nitrogen-containing compound and pharmaceutical composition
05/29/2012US8188072 Benzodiazepinone compounds useful in the treatment of skin conditions
05/29/2012CA2496585C Novel 1,4-diazabicycloalkane derivatives, their preparation and use
05/24/2012US20120129939 Polyamine inhibitors for the treatment and prevention of parkinson's disease
05/23/2012CN102464623A 1,4-二氮杂环辛烷-6-甲酸酯衍生物的制备方法 Preparation of 1,4-diazabicyclo octane-6-carboxylic acid ester derivative
05/18/2012WO2012064483A1 Transamination of nitrogen-containing compounds to make cyclic and cyclic/acyclic polyamine mixtures
05/16/2012EP1904460B1 Multidentate aza ligands able to complex metal ions and the use thereof in diagnostics and therapy
05/16/2012CN102459200A 适用于治疗响应于调节血清素5-ht6受体的疾病的苯磺酰基苯胺化合物 Applicable to the treatment response to serotonin 5-ht6 regulating receptor diseases Phenylsulfonylaniline compound
05/16/2012CN102459199A 适于治疗响应于5-羟色胺5-HT<sub>6</sub>受体调节的病症的苯磺酰苯胺化合物 Adapted to therapeutic response to serotonin 5-HT <sub> 6 </ sub> receptor modulated disorder benzenesulfonyl aniline compound
05/16/2012CN102459178A 2,5-disubstituted arylsulfonamide ccr3 antagonists
05/16/2012CN102452991A Synthetic technology of hapten 3-(3-chlorine-propyl)diazepam
05/16/2012CN102452990A Homopiperazine acethydrazide derivative with low neurotoxicity and preparation method and application thereof
05/15/2012US8178545 Dual small molecule inhibitors of cancer and angiogenesis
05/10/2012WO2012059432A1 N-phenyl-(homo)piperazinyl-benzenesulfonyl or benzenesulfonamide compounds suitable for treating disorders that respond to the modulation of the 5-ht6 receptor
05/10/2012US20120116073 P2x4 receptor antagonist
05/10/2012US20120115851 Compound inhibiting in vivo phosphorus transport and medicine containing the same
05/09/2012EP2448582A1 Therapeutic compounds and compositions
05/09/2012EP1423107B1 Fatty alcohol drug conjugates
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