| Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865) |
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| 03/14/2001 | EP1082306A1 Conformationally constrained amino acid compounds having affinity for the alpha2delta subunit of a calcium channel |
| 03/13/2001 | US6201020 Effective poly(adenosine 5'-diphospho-ribose) polymerase (parp) inhibitor for treatment of tissue damage by necrosis or apoptosis; side effect reduction |
| 03/13/2001 | US6201013 Inosine monophosphate dehydrogenase (impdh) inhibitor; side effect reduction, non-drug resistant |
| 03/13/2001 | US6200995 Pyridyloxybenzenesulfonamide derivatives; diabetes, obesity |
| 03/13/2001 | US6200978 For preventing or treating inflammatory diseases such as arthritis, psoriasis, asthma, or inflammatory bowel disease, disorders of respiratory function, gastrointestinal disorders such as functional bowel disease, as analgesics |
| 03/13/2001 | US6200976 Antithrombotic quinoxazolines |
| 03/13/2001 | US6200967 Used as thrombin inhibitors, coagulation inhibitors and agents for the treatment of thromboembolic disorders |
| 03/08/2001 | WO2001016114A2 Heterocyclic compounds and methods for modulating cxcr3 function |
| 03/08/2001 | WO2001002367A3 Diester prodrugs of a decahydroisoquinoline-3-carboxylic acid |
| 03/08/2001 | WO2000050872A3 A system for cell-based screening |
| 03/08/2001 | WO1999039704A8 Antibacterial agents |
| 03/07/2001 | EP1081142A2 Novel N-Aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands |
| 03/07/2001 | EP1080083A1 Novel heterocyclically substituted amides with cysteine protease-inhibiting effect |
| 03/07/2001 | EP1080074A1 New heterocyclically substituted amides, their production and their use |
| 03/07/2001 | EP1079821A1 Protease inhibitors |
| 03/07/2001 | EP1079763A2 Serotonergic 5ht 7? receptor compounds for treating ocular and cns disorders |
| 03/07/2001 | EP0641325B1 Retroviral protease inhibitors |
| 03/06/2001 | US6197785 Cardiovascular disorders |
| 03/06/2001 | US6197771 Nervous system disorders; antiischemic agents; alzheimer'sdisease; parkinson's disease; huntington's disease |
| 03/06/2001 | CA1341196C Process for the preparation of substituted imino diacids |
| 03/01/2001 | WO2001014879A1 4-unsubstituted dihydroisoquinolinone derivatives and combinatorial libraries thereof |
| 03/01/2001 | WO2001014328A2 Substituted ureas as cell adhesion inhibitors |
| 03/01/2001 | WO2001014320A1 Compounds that inhibit tryptase activity |
| 03/01/2001 | DE19939910A1 Neue Verbindungen, die Tryptase-Aktivität hemmen Novel compounds that inhibit tryptase activity |
| 03/01/2001 | CA2381096A1 Compounds that inhibit tryptase activity |
| 02/28/2001 | EP1077978A1 Novel substituted aryl hydroxamic acids as metalloproteinase inhibitors |
| 02/28/2001 | EP1077945A1 Isoquinolines as urokinase inhibitors |
| 02/28/2001 | EP1077944A1 Carboxamide compounds, compositions, and methods for inhibiting parp activity |
| 02/28/2001 | EP1077698A1 Metabolites of ecteinascidin 743 |
| 02/28/2001 | CN1285820A Metabotropic glutamate receptor antagonists for treating central nervous system disease |
| 02/27/2001 | US6194451 Prevent release tumor necrosis factor; antiinflammatory agents |
| 02/27/2001 | US6194409 Heterocyclic derivatives and their use as antithrombotic agents |
| 02/22/2001 | WO2000071500A8 Halogen compounds |
| 02/21/2001 | EP1076649A1 Isoquinoline compound melanocortin receptor ligands and methods of using same |
| 02/21/2001 | CN1284946A Substituted isoquinoline derivatives and their use as anticonvulsants |
| 02/21/2001 | CN1062266C Amidine derivative and platelet agglutination inhibitor containing said amidine derivative |
| 02/15/2001 | WO2001010843A1 4-(substituted phenyl)-5-halopyrimidine derivatives and herbicides containing the same as the active ingredient |
| 02/15/2001 | WO2001010842A2 Melanocortin-4 receptor binding compounds and methods of use thereof |
| 02/15/2001 | WO2001010839A2 Multivalent substituted ketoamides and amides for treating hair loss |
| 02/15/2001 | WO2001010838A1 Multivalent compounds |
| 02/15/2001 | WO2001010835A1 Antibacterial agents |
| 02/15/2001 | WO2001010834A2 Antibacterial agents |
| 02/15/2001 | CA2381008A1 Melanocortin-4 receptor binding compounds and methods of use thereof |
| 02/14/2001 | CN1283995A Antiviral compounds |
| 02/13/2001 | US6187789 Muscle relaxants for emergency intubation and surgery |
| 02/08/2001 | WO2001009101A1 Isoquinoline derivatives, pharmaceutical compositions containing the same, and a process for the preparation of the active substance |
| 02/08/2001 | WO2001009100A1 Reductive methylation of tetrahydroisochinoline in a static micromixer |
| 02/08/2001 | WO2001009065A2 Nitration in a static micromixer |
| 02/07/2001 | EP1074545A1 Isoquinolinesulfonamide derivatives and drugs containing the same as the active ingredient |
| 02/07/2001 | EP1073633A2 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2 |
| 02/07/2001 | EP1073624A1 Aminomethyl-benzoic ester derivatives as tryptase inhibitors |
| 02/07/2001 | EP0922035B1 Tetrahydroisoquinoline derivatives and their pharmaceutical use |
| 02/07/2001 | CN1282738A Improved method for sgnthesizing 6,9-bis[(2-aminoethyl) amino] benz[g] isoquinoline-5, 10-diketone and its dimaleate |
| 02/07/2001 | CN1282732A 'alpha'-hydroxy-'beta' amino acid ester and its preparation method |
| 02/01/2001 | WO2001007412A1 Antiviral tetrahydroisichinolinsulfonamides |
| 02/01/2001 | DE19935694A1 Reduktive Methylierung von Aminen im statischen Mikromischer Reductive methylation of amines in the static micromixer |
| 02/01/2001 | DE19935692A1 Nitrierung in einem statischen Mikromischer Nitration in a static micromixer |
| 01/31/2001 | EP1072587A1 Sulfonamide derivatives and drugs containing the same as the active ingredient |
| 01/31/2001 | EP1072263A1 Amide derivatives and nociceptin antagonists |
| 01/31/2001 | EP1071669A1 Bicyclic compounds having an anti-thrombitic effect |
| 01/30/2001 | US6180675 IL-8 receptor antagonists |
| 01/30/2001 | US6180646 Retroviral protease inhibitors |
| 01/30/2001 | US6180645 Antiepilepic agent |
| 01/30/2001 | US6180619 Prenyl transferase inhibitors |
| 01/25/2001 | WO2001005783A1 Bradykinin b1 receptor antagonists |
| 01/25/2001 | DE19934272A1 New N-phenyl-tetrahydroisoquinoline-sulfonamide derivatives are antiviral agents especially useful for treating cytomegalovirus infections |
| 01/25/2001 | CA2379064A1 Bradykinin b1 receptor antagonists |
| 01/24/2001 | EP1070049A1 Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors |
| 01/24/2001 | EP1069901A1 Calcilytic compounds and method of use |
| 01/24/2001 | CN1281362A Novel combination medicine |
| 01/23/2001 | US6177445 Substituted isoquinolines as ultra short acting neuromuscular blockers |
| 01/18/2001 | WO2001004090A2 Neurotrophic tetrahydroisoquinolines and tetrahydrothienopyridines, and related compositions and methods |
| 01/18/2001 | WO2001004087A1 Sulfonamide substituted benzylamine derivatives and their use as medicaments |
| 01/17/2001 | EP1069110A1 Sulfonamide derivatives |
| 01/17/2001 | EP1067917A2 Method of treating dopaminergic and gaba-nergic disorders |
| 01/17/2001 | EP0983258A4 N-hydroxy 4-sulfonyl butanamide compounds |
| 01/17/2001 | EP0725059B1 2,3-diaminopropionic acid derivative |
| 01/16/2001 | US6174924 Treating nerve cell death comprising administering to a subject exhibiting symptoms of nerve cell death or susceptible to nerve cell death a substituted guanidine compound |
| 01/11/2001 | WO2001002368A1 N-heterocyclic derivatives with neuronal activity |
| 01/11/2001 | WO2001002367A2 Diester prodrugs of a decahydroisoquinoline-3-carboxylic acid |
| 01/11/2001 | WO2001002366A2 Substituted isoquinoline derivatives and their use as inticonvulsants |
| 01/11/2001 | CA2527931A1 Substituted isoquinoline derivatives and their use as anticonvulsants |
| 01/11/2001 | CA2376495A1 Substituted isoquinoline derivatives and their use as anticonvulsants |
| 01/04/2001 | WO2001000573A1 Indanyl-substituted benzole carbonamide, method for the production of the same, use thereof as a medicament and pharmaceutical preparations containing the same |
| 01/04/2001 | WO2001000206A1 Vla-4 inhibitor compounds |
| 01/04/2001 | CA2377087A1 Indanyl-substituted benzole carbonamide, method for the production of the same, use thereof as a medicament and pharmaceutical preparations containing the same |
| 01/04/2001 | CA2369308A1 Vla-4 inhibitor compounds |
| 01/03/2001 | EP1065200A1 Aminoisoquinoline derivatives |
| 01/03/2001 | CN1278797A Oxo-substituted compouns, process of making, and compositions and methods for inhibiting parp activity |
| 01/03/2001 | CN1278793A Sulfonyl derivatives |
| 01/02/2001 | US6169088 1,3 diazines with platelet-derived growth factor receptor inhibitory activity |
| 01/02/2001 | US6169085 A viricide for preventing and treating retroviral infection or the spread of a retrovirus, inhibiting replication of a retrovirus and treating aids |
| 01/02/2001 | US6168776 Alkyl, alkenyl and alkynyl Chrysamine G derivatives for the antemortem diagnosis of Alzheimer's disease and in vivo imaging and prevention of amyloid deposition |
| 12/28/2000 | WO2000078145A1 Macrophage scavenger receptor antagonists |
| 12/28/2000 | DE19929076A1 New indanyl-substituted benzenesulfonamide derivatives, as potassium channel blockers useful as safe antiarrhythmic agents, e.g. for treating atrial fibrillation or flutter |
| 12/28/2000 | CA2377288A1 Macrophage scavenger receptor antagonists |
| 12/27/2000 | EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) |
| 12/27/2000 | EP1062217A1 Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives |
| 12/27/2000 | CN1278250A Vitronectin receptor antagonists |
| 12/27/2000 | CN1059902C Estrogen excitant/antagonist |