Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
12/2002
12/19/2002US20020189033 Substituted 2-aminoalkyl-1,4diaminobenzene compounds and oxidation dye precursor compositions containing same
12/19/2002DE10128331A1 New 2-(heteroarylsulfonyl-amino)-benzamide derivatives, which are potassium ion channel blocking antiarrhythmic agents, useful for e.g. treating atrial fibrillation or flutter
12/19/2002DE10115227A1 Optischer Datenträger enthaltend in der Informationsschicht eine lichtabsorbierende Verbindung mit mehreren chromophoren Zentren Optical data storage medium in the information layer containing a light absorbing compound having a plurality of chromophoric centers
12/19/2002CA2450628A1 Benzothiophene compounds having antiinfective activity
12/19/2002CA2450625A1 Isoquinoline compounds having antiinfective activity
12/19/2002CA2450271A1 Novel phenylalkyl diamine and amide analogs
12/19/2002CA2450269A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002CA2450265A1 Hiv protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis
12/19/2002CA2449256A1 Modulators of peroxisome proliferator activated receptors
12/19/2002CA2445653A1 Substituted sulfonamide compounds, process for their use as medicament for the treatment of cns disorders, obesity and type ii diabetes
12/18/2002EP1265867A1 Novel malonic acid derivates, processes for their preparation, their use as inhibitor of factor xa activity and pharmaceutical compositions containing them
12/18/2002EP1265853A1 Carboxylic acid derivatives as ip antagonists
12/18/2002EP0946502B1 Sulfonamide interleukin-beta converting enzyme inhibitors
12/17/2002US6495562 Such as 6-(2-(4,4-diethyl-1-isopropyl-3,4-dihydro-6-isoquinolinyl)cyclopropyl)-2 -naphthalenecarboximidamide
12/17/2002US6495552 Treatment or prevention of the diseases and conditions which respond to treatment by retinoids and or which in healthy mammals, including humans, are controlled by natural retinoic acid.
12/12/2002WO2002098426A1 Substituted tetrahydroisoquinolines for use in the treatment of inflammatory diseases
12/12/2002WO2002098406A1 Novel compounds and compositions as cathepsin inhibitors
12/12/2002US20020188004 Heterocycle carboxamides as antiviral agents
12/12/2002CA2449021A1 Novel compounds and compositions as cathepsin inhibitors
12/11/2002EP1264820A1 Novel amide compounds
12/11/2002EP1263730A1 Amine derivatives for the treatment of apoptosis
12/11/2002EP0966436B1 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
12/11/2002EP0782567B2 Isothiourea derivatives as no synthase inhibitors
12/11/2002EP0752813B1 Inhibitors of metazoan parasite proteases
12/11/2002EP0628030B1 2,3,4,5-TETRAHYDRO-1H --3-BENZAZEPINES HAVING ANTI-PSYCHOTIC ACTIVITY, AND SYNTHESIS OF $g(a)-SUBSTITUTED-ARYLACETAMIDES
12/10/2002US6492520 Substituted pyrido-or pyrimido-containing 6,6- or 6,7-bicyclic derivatives
12/10/2002US6492388 Such as n-(5-chloro-1,2,3,4-tetrahydroisoquinolin-7-yl)-4-ethoxybenzamide
12/10/2002US6492378 Substituted isoquinoline derivatives and their use as anticonvulsivants
12/09/2002WO2002004403A1 Biphenylcarboxylic acid amides, production thereof and use thereof as medicaments
12/09/2002CA2412116A1 Biphenylcarboxylic acid amides, the preparation thereof and the use thereof as medicaments
12/05/2002WO2002096880A1 Novel heterocyclic compound and medicinal use thereof
12/05/2002WO2002096858A1 Cinnamide derivatives as kcnq potassium channel modulators
12/05/2002WO2002096424A1 Hetereocyclic beta-aminoacids and their use as anti-epileptogenic agents
12/05/2002WO2002011707A3 Drugs for incontinence
12/05/2002US20020183342 For use as insecticides against a variety of insects, including larvae, such as tobacco budworm
12/05/2002CA2448894A1 Cinnamide derivatives as kcnq potassium channel modulators
12/05/2002CA2448634A1 Novel heterocyclic compound and medicinal use thereof
12/05/2002CA2448160A1 Heterocyclic beta-amino acids and their use as anti-epileptogenic agents
12/03/2002US6489479 Process for the preparation of mixed anhydrides
12/03/2002US6489352 Antiepileptic agents; nervous system disorders
11/2002
11/28/2002WO2002094815A1 Process for the production of quinazolines
11/28/2002WO2002094790A1 Fused heterocyclic compound and medicinal use thereof
11/28/2002WO2002078745A3 Use of mglur5 antagonists in the manufacture of a medicament in the treatment of autism, mental retardation, schizophrenia
11/28/2002US20020177605 3-substituted isoquinolin-1-yl derivatives
11/28/2002CA2447233A1 Process for the production of quinazolines
11/27/2002EP1259485A2 BENZAMIDES AND RELATED INHIBITORS OF FACTOR Xa
11/26/2002US6486340 Method for producing an α-aminonitrile from a tertiary anime and a cyanide through oxidation with oxygen by using a transition metal catalyst
11/26/2002US6486175 Diester prodrugs of a decahydroisoquinoline-3-carboxylic acid
11/26/2002US6486174 Treatment of tumor growth, metastasis, restenosis, osteoporosis, inflammation, macular degeneration, diabetic retinopathy, rheumatoid arthritis, sickle cell anemia, nerve system disorders
11/26/2002US6486173 Serotonin-7 (5-ht7); treatment of central nervous system disorders such as sleep disorders, depression and schizophrenia; for example 1,3-dihydro-2-((4-(4-fluorophenyl)-4-oxobutyl))isoindole
11/26/2002CA2231364C Novel n-aminoalkylfluorenecarboxamides; a new class of dopamine receptor subtype specific ligands
11/21/2002US20020173521 Inhibitors of copper-containing amine oxidases
11/21/2002US20020172793 Optical data store comprising an axially substituted cobalt phthalocyanine in the light-writeable information layer
11/20/2002EP1258252A1 Integrin expression inhibitors
11/20/2002CN1380289A Amide capable of inhibiting ApoB-secretion/MTP
11/20/2002CN1380288A Tetrahydroisoquinoline hydroximic acid sulfamide compound, its synthesis method and its application
11/19/2002US6482849 Inhibitors of α4β1 mediated cell adhesion
11/19/2002US6482832 Heterocyclically substituted amides, their production and their use
11/14/2002WO2002090347A1 Amide compounds
11/14/2002WO2002090334A1 Isoquinolinone derivatives as parp inhibitors
11/14/2002WO2002090314A1 Pyruvate derivatives
11/14/2002WO2002089749A2 Arylsulfonamide ethers, and methods of use thereof
11/14/2002US20020169326 Fatty acid derivatives
11/14/2002US20020169185 Quinolinyl and benzothiazolyl modulators
11/14/2002CA2445923A1 Arylsulfonamide ethers, and methods of use thereof
11/14/2002CA2444531A1 Isoquinolinone derivatives as parp inhibitors
11/13/2002EP0760658B1 Compounds for inhibiting osteoclast-mediated bone resorption
11/12/2002US6479436 Hetaroyl cyclohexanedione derivatives with herbicidal effect
11/07/2002WO2002089128A1 An optical data storage medium containing a diaza hemicyanine dye as the light-absorbing compound in the information layer
11/07/2002WO2002088101A2 Inhibitors of bace
11/07/2002WO2002088088A1 Process for preparing 1-methyl-1,2,3,4-tetrahydroisoquinoline or a salt thereof
11/07/2002WO2002088071A1 20-hydroxyeicosatetraenoic acid production inhibitors
11/07/2002US20020165394 Inhibition of RAF kinase using quinolyl, isoquinolyl or pyridyl ureas
11/07/2002US20020165236 Such as 3-(3-(4-(4-sulfamoyl-benzylsulfamoyl-phenyl)-ureido)-benzamidine for treatment of malaria
11/07/2002US20020165230 Gamma-ketoacid dipeptides as inhibitors of caspase-3
11/07/2002US20020165202 Antiinflammatory agents; antiproliferative agents
11/07/2002US20020165201 Cyanoguanidine prodrugs
11/07/2002US20020165167 Bacterial polypeptide deformylase (PDF) inhibitors, N-formyl hydroxylamine derivatives
11/06/2002EP1254895A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
11/06/2002EP1254140A1 Compounds of the saframycin-ecteinascidin series, uses, and synthesis thereof
11/06/2002EP1254136A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF
11/06/2002EP0901488B1 2,4-diaminopyrimidine derivatives
11/06/2002CN1378446A Method of inhibiting amyloid protein aggregation and imaging amyloid deposits
11/05/2002US6476232 4-(2-amino-1-hydroxyethyl)oxazoline derivative and method for producing same
11/05/2002US6476047 Good bioavailability and powerful analgesic activity based on calcium channel blockade.
11/05/2002CA2038379C Trifluoromethyl mercaptan and mercaptoacyl derivatives and method of using same
10/2002
10/31/2002WO2002086879A1 Optical data support comprising a hemicyanin dye in the information layer as light-absorbing compound
10/31/2002WO2002086878A2 Optical data carrier whose information layer contains a light-absorbing compound having a number of chromophoric centers
10/31/2002WO2002086078A2 Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
10/31/2002WO2002085859A1 HETEROARYL UREAS CONTAINING NITROGEN HETERO-ATOMS AS p38 KINASE INHIBITORS
10/31/2002WO2002085820A2 Chiral organic compounds and metal coordination complexes thereof
10/31/2002US20020161236 2-methyl-3-(protected hydroxy) benzyl chloride; use making nelfinavir mesylate
10/31/2002US20020161234 Forming a diastereoselective epoxide from a chiral alpha-amino aldehyde
10/31/2002US20020161231 Intermediate for preparing camptothecin derivatives
10/31/2002US20020161189 Used in the antagonism and agonism of delta and mu opioid receptors
10/30/2002EP1252146A1 Amide compounds for inhibiting protein kinases
10/30/2002EP0854863B1 Esters and amides as pla2 inhibitors
10/30/2002CN1377336A Carboxylic acid derivatives and drugs containing the same
10/29/2002US6472534 Treating tetrahydrofuran derivativ with an oxophilic electrophilic reagent in a manner that is effective to provide the oxazoline compound
10/29/2002US6472405 Glycoprotein IIB/IIIA antagonists
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