Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
09/2000
09/28/2000CA2367963A1 Hydroxamic and carboxylic acid derivatives
09/27/2000EP1038868A2 Sulfonamides as antiviral agents
09/27/2000EP1037878A2 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
09/27/2000EP1037633A1 Antiviral compounds
09/27/2000EP0901465B1 Compounds with anti-inflammatory and immunosuppressive activities
09/27/2000CN1267670A Two aporphine-benzyl isoquinoline compounds with antineoplastic activity
09/27/2000CN1056832C Fused dihydropyridine derivate, its producing process, and its pharmaceutical composition
09/26/2000US6124461 Compounds, compositions, and methods for treating erectile dysfunction
09/21/2000WO2000055137A1 Compounds and methods for modulation of estrogen receptors
09/21/2000DE19912638A1 Naphthylcarbonsäureamid-substituierte Sulfonamide Naphthylcarbonsäureamid-substituted sulfonamides
09/21/2000CA2367895A1 Compounds and methods for modulation of estrogen receptors
09/20/2000EP1035843A2 I h?-MODULATORS
09/20/2000CN1056602C Esters and amides as PLAZ inhibitors
09/19/2000US6121283 N-substituted-6-(2-(4-trifluoromethylphenyl)phenylcarbonyl-amino) -1,2,3,4-tetrahydroisoquinolines; treating disorders including obesity, hyperlipidemia, and diabetes; microsomal triglyceride transfer protein (mtp); apolipoprotein b (apo-b)
09/19/2000US6121278 Di-n-heterocyclic compounds, methods, and compositions for inhibiting parp activity
09/19/2000US6119687 Partial liquid breathing of fluorocarbons
09/14/2000WO2000024717A3 Isoquinoline derivatives
09/13/2000EP1034164A1 Substituted beta-alanine derivatives as cell adhesion inhibitors
09/12/2000US6118010 Catalytic reduction of the 1-alkoxycarbonyl-3-oxo-3-phenylpropyl derivative
09/12/2000US6117999 Chemical intermediate for nelfinavir
09/12/2000US6117910 Bicyclic fibrinogen antagonists
09/08/2000WO2000051971A1 Oxamic acids and derivatives as thyroid receptor ligands
09/08/2000WO2000051970A1 Amide compounds for the potentiation of cholinergic activity
09/08/2000WO2000034260A3 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
09/06/2000EP1032570A1 Isoquinoline derivatives and their therapeutical use
09/06/2000EP1032559A1 Aminoalkylphenol derivatives and related compounds
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/06/2000CN1265669A Compounds which inhibit leukocyte adhesion mediated by VLA-4
09/06/2000CN1265645A Urokinase inhibitors
09/05/2000US6114530 Isoquiolinamines and phthalazinamines useful in treating stress related disorderes such as post traumatic stress disorder as well as depression, headache and anxiety
09/05/2000US6114529 Useful for preparing camptothecin derivatives having antitumor activities
09/05/2000US6114175 Amyloid-binding compounds which are non-azo derivatives of chrysamine g to determine degree of brain deposits quantitatively characterized by amyloidosis; down's syndrome; prevent cell degeneration; radioactive imaging
08/2000
08/31/2000WO2000050872A2 A system for cell-based screening
08/31/2000WO2000050406A1 Isoquinoline derivatives and isoquinoline combinatorial libraries
08/31/2000WO2000050389A1 Efficient carbamate synthesis
08/31/2000WO2000050377A1 Efficient synthesis of secondary amines by selective alkylation of primary amines
08/31/2000WO2000050376A2 Efficient synthesis of alkyl carbonates
08/30/2000EP1031563A1 Sulfonyl derivatives
08/29/2000US6110934 Substituted benzamide derivatives and their use as anticonvulsants
08/29/2000US6110933 Amino acid derivatives and their use as phospholipase A2 inhibitor
08/29/2000US6110922 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
08/24/2000WO2000015992A3 Tube for lining pipes and channels, and a method and device for the production thereof
08/22/2000US6107331 Use of estrogen antagonists and estrogen agonists in inhibiting pathological conditions
08/17/2000WO2000047554A2 INHIBITORS OF FACTOR Xa
08/17/2000WO2000047553A2 ALKENYL AND ALKYNYL COMPOUNDS AS INHIBITORS OF FACTOR Xa
08/17/2000CA2362375A1 Alkenyl and alkynyl compounds as inhibitors of factor xa
08/17/2000CA2361428A1 Inhibitors of factor xa
08/16/2000EP1027336A1 Heteroaryl diazacycloalkanes as cholinergic ligands at nicotinic acetylcholine receptors
08/16/2000EP1027052A1 Novel combination
08/16/2000CN1055468C Alkylaminoindane compounds process for preparing them and pharmaceutical compositions containing them,and use
08/10/2000WO2000046204A1 Tetrahydro isoquino linealkanol derivatives and pharmaceutical compositions containing same
08/10/2000CA2361805A1 Tetrahydro isoquino linealkanol derivatives and pharmaceutical compositions containing same
08/09/2000EP1025090A1 Vitronectin receptor antagonists
08/09/2000EP1025087A1 Substituted isoquinoline derivatives and their use as anticonvulsants
08/09/2000EP0820434B1 Phenoxyethylamine derivatives having high affinity for the 5-ht 1a receptor, preparation thereof, use thereof as drugs, and pharmaceutical compositions containing said derivatives
08/09/2000CN1262677A Preparation of fused polycyclic alkaloids by ring closure of azomethine ylides, noval compounds thereof and their use as chemotherapeutic agents
08/09/2000CN1262620A Beta-Alkoxyacrylates against malaria
08/09/2000CN1262272A HIV proteinase inhibitor
08/08/2000US6100404 Erythromycin compounds
08/08/2000US6100277 Retroviral protease inhibitor combinations
08/03/2000WO2000044713A1 Alkynyl containing hydroxamic acid compounds as tace inhibitors
08/03/2000WO2000044709A2 ACETYLENIC α-AMINO ACID-BASED SULFONAMIDE HYDROXAMIC ACID TACE INHIBITORS
08/03/2000CA2356346A1 Alkynyl containing hydroxamic acid compounds as tace inhibitors
08/03/2000CA2356299A1 Acetylenic .alpha.-amino acid-based sulfonamide hydroxamic acid tace inhibitors
08/02/2000EP1023269A1 Beta3-adrenoreceptor agonists, agonist compositions and methods of using
08/02/2000EP1023268A1 Isoquinolines as urokinase inhibitors
08/02/2000CN1261906A Alkyl, alkenyl and alkynyl chrysamine G derivatives for the antemortem diagnosis of alzheimer's disease and in vivo imaging and prevention of amyloid deposition
08/02/2000CN1261883A Novel compounds
08/01/2000US6096752 Method for the preparation of tertiary amines, a compound useful therefor and alpha-2-receptor active tetrahydroisoquinoline derivatives
08/01/2000US6096712 Tripeptide derivative; antiallergens, male contraceptives, antiinflammatory agents, antispasmodics, hypertensive agents
08/01/2000CA2209925C 5,6-diaryl-5,6,7,8-tetrahydronaphthalenes and their analogs as estrogen agonists/antagonists
08/01/2000CA2019335C Phenylalkan (en)oic acids
07/2000
07/27/2000WO1999057098A3 Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
07/26/2000EP0736011B1 Anellated dihydropyridines and their use in the production of pharmaceutical preparations
07/26/2000CN1261350A Tetrahydroisoquinoline derivatives as modulators of dopamine D3 receptors
07/26/2000CN1261278A Methods for treating inflammatory diseases using padprt inhibitors
07/25/2000US6093731 Isoquinolines
07/25/2000US6093730 Substituted isoquinoline-3-carboxamides, their preparation and their use as pharmaceuticals
07/25/2000US6093729 Substituted bicyclic heteroaroylguanidines, a process for their preparation, their use as a medicament or a diagnostic agent, and a medicament containing them
07/20/2000WO2000042071A2 Compounds and methods to inhibit or augment an inflammatory response
07/20/2000CA2697598A1 Compounds and methods to inhibit or augment an inflammatory response
07/19/2000EP1020445A1 Fused pyridine derivatives
07/19/2000EP1019367A1 Derivatives of 2,5- and 3,5-disubstituted anilines, their preparation and use
07/19/2000EP0902781A4 Preparation of (s)-decahydroisoquinoline-3-carboxylic acid t-butylamide
07/13/2000WO2000040560A1 Aminoalcohol derivatives and their use as beta 3 adrenergic agonists
07/12/2000EP1017664A1 C3a receptor ligands
07/12/2000EP1017382A1 Biarylalkanoic acids as cell adhesion inhibitors
07/06/2000WO2000039081A2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
07/06/2000WO2000039070A1 Ortho-diphenol compounds, methods and pharmaceutical compositions for inhibiting parp
07/06/2000CA2358315A1 Ortho-diphenol compounds, methods and pharmaceutical compositions for inhibiting parp
07/05/2000EP1015444A1 Novel pyrimidine derivatives and processes for the preparation thereof
07/05/2000EP1015432A1 Separation of enantiomers of octahydroisoquinoline
07/05/2000CN1259126A Pharmacological agents
07/05/2000CN1259119A Substituted 3,3-diamino-2-propenenitriles their preparation and use
07/04/2000US6084120 β-Alkoxyacrylates against malaria
06/2000
06/29/2000WO2000037429A2 INHIBITORS OF α4β1 MEDIATED CELL ADHESION
06/28/2000EP1012166A1 1-amino-7-isoquinoline derivatives as serine protease inhibitors
06/28/2000EP1012145A1 Alkoxy-substituted compounds, methods, and compositions for inhibiting parp activity
06/28/2000EP1011651A1 Method of treating diabetes and related disease states
06/28/2000CN1053899C Acylguanidine, its preparation process and use, and pharmaceutical composition contg. same
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