Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
08/2001
08/23/2001US20010016657 Substituted isoquinoline derivatives and their use as anticonvulsants
08/23/2001CA2397651A1 Amine derivatives for the treatment of apoptosis
08/22/2001EP1125929A1 Method for making (-)-(2R,4S)-4-[(3,5-bis-trifluoromethyl-benzyl)-methoxycarbonylamino]-2-ethyl-6-trifluoromethyl-3,4-dihydro-2H-quinoline-1-carboxylic acid ethyl ester
08/22/2001EP1125925A1 Amine derivatives for the treatment of apoptosis
08/22/2001EP1124554A1 Pharmaceutical compositions containing tetrahydroisoquinoline compounds
08/21/2001US6277992 Useful as an intermediate for preparing camptothecin derivatives having antitumor activities
08/21/2001US6277861 For treatment and prophylaxis of nervous system disorders, psychological disorders, muscular disorders, drug addiction withdrawal, pain
08/21/2001US6277849 N-sulphonyl and N-sulphinyl amino acid amides as microbiocides
08/16/2001WO2001010842A3 Melanocortin-4 receptor binding compounds and methods of use thereof
08/16/2001EP1123918A1 Aromatic amine derivatives, process for the preparation thereof and agents containing the same
08/16/2001EP1123280A1 Serine protease inhibitor
08/16/2001EP1123272A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
08/16/2001EP1123099A1 Novel indenoisoquinolines as antineoplastic agents
08/15/2001CN1308608A Substituted beta-amino acid inhibitors of methionine aminopeptidase-2
08/15/2001CN1069643C Naphthyridine derivatives and their analogues inhibiting cytomegalovirus
08/14/2001US6274618 Administering (-)-cis-6-phenyl-5-(4-(2-pyrrolidin-1-yl-ethoxy)-phenyl)-5,6,7,8 -tetrahydronphthalen-2-ol to treat vaginal dryness, itching, or painful intercourse
08/14/2001US6274594 Isoquinoline derivatives and their therapeutical use
08/14/2001US6274593 Treating psychological disorders, schizophrenia, and parkinson*s disease
08/14/2001US6274584 Peptide derivatives; bioavailability; enzyme resistance; milk and wool production
08/14/2001CA2159640C Second messenger cell signaling inhibitors
08/14/2001CA2036222C Plating compositions and processes
08/09/2001WO2001056607A1 Integrin expression inhibitors
08/09/2001WO2001019788A3 BENZAMIDES AND RELATED INHIBITORS OF FACTOR Xa
08/09/2001WO2001010834A9 Antibacterial agents
08/09/2001WO2000071511A3 INHIBITORS OF FACTOR Xa
08/09/2001WO2000047554A3 INHIBITORS OF FACTOR Xa
08/09/2001US20010012895 Therapy for hair loss in mammals; drug resistance; nervous system disorders
08/08/2001EP1121342A1 Diaminopropionic acid derivatives
08/08/2001EP1009749B1 Preparation of (s)-n-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxyamide
08/08/2001CN1069309C N-(aminopropyl)-N-phenyl-5,6,7,8-tetrahydronaphtalene-2-carboxamide derivative, preparation and application thereof
08/07/2001US6271235 HIV protease inhibitors
08/02/2001WO2001055146A1 FACTOR Xa INHIBITORS WITH ARYL-AMIDINES AND DERIVATIVES, AND PRODRUGS THEREOF
08/02/2001WO2001055117A1 Novel isoquinoline derivatives, preparation method and pharmaceutical compositions containing them
08/02/2001WO2001016114A3 Heterocyclic compounds and methods for modulating cxcr3 function
08/02/2001WO2000076971A3 Serine protease inhibitors
08/02/2001US20010011134 Cyclic and heterocyclic N-substituted alpha-iminohydroxamic and -carboxylic acids
08/01/2001EP1120114A2 Compositions and methods for treating conditions responsive to estrogen
08/01/2001EP1119550A1 2-substituted heterocyclic sulfonamides
08/01/2001CN1306526A Novel heterocyclically substituted amides with cysteine protease-inhibiting effect
07/2001
07/26/2001WO2001053299A1 Compounds of the saframycin-ecteinascidin series, uses, and synthesis thereof
07/26/2001WO2001053274A1 Amide compounds for inhibiting protein kinases
07/26/2001WO2001053258A1 Nitrogenous cyclic compounds and pharmaceutical compositions containing the same
07/26/2001CA2398409A1 Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound
07/26/2001CA2397597A1 Compounds of the saframycin-ecteinascidin series, uses, and synthesis thereof
07/26/2001CA2394703A1 Amide compounds for inhibiting protein kinases
07/25/2001EP1118323A2 Method of reducing morbidity and the risk of mortality
07/25/2001EP1117640A1 Heterocyclic 2-substituted ketoamides useful for treating hair loss in mammals
07/25/2001EP1117627A1 Transfer hydrogenation process
07/25/2001EP0752857B1 AN IMPROVED METHOD OF SYNTHESIS FOR 6,9-BIS (2-AMINOETHYL)AMINO]BENZO g]ISOQUINOLINE-5,10-DIONE AND ITS DIMALEATE SALT
07/24/2001CA2042112C N'-alkyl-spiro-isoquinoline-pyrrolidine tetrones and analogs thereof useful as aldose reductase inhibitors
07/19/2001WO2001051469A1 Piperidine and piperazine derivatives which function as 5-ht2a receptor antagonists
07/19/2001WO2001004090A3 Neurotrophic tetrahydroisoquinolines and tetrahydrothienopyridines, and related compositions and methods
07/19/2001WO2000076970A3 Serine protease inhibitors
07/19/2001CA2396007A1 Piperidine and piperazine derivatives
07/18/2001EP1116711A2 2-aminoalkyl-1,4-diaminobenzene derivatives and dye composition containing these compounds
07/18/2001EP1115697A1 Unsaturated hydroximic acid derivatives as parp inhibitors
07/18/2001EP1115695A1 (r)-chiral halogenated 1-substitutedamino-(n+1)-alkanols useful for inhibiting cholesteryl ester transfer protein activity
07/18/2001EP1115693A1 SUBSTITUTED POLYCYCLIC ARYL AND HETEROARYL $i(TERTIARY)-HETEROALKYLAMINES USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY
07/18/2001CN1304402A Sulfonamide derivatives
07/17/2001US6262112 Aryl sulfonamides and analogues thereof and their use in the treatment of neurodegenerative diseases
07/17/2001US6262069 1-amino-7-isoquinoline derivatives as serine protease inhibitors
07/17/2001US6262068 Lactam derivatives as antiarrhythmic agents
07/12/2001WO2001049679A1 4-phenyl-1-piperazinyl, -piperidinyl and -tetrahydropyridyl derivatives
07/12/2001WO2001049288A1 Novel compounds and compositions as protease inhibitors
07/12/2001DE10000739A1 New piperidine and piperazine derivatives which are antagonists of certain serotonin receptors, are useful in treatment of, e.g. eating disorders, stroke, anxiety or Parkinson's disease
07/12/2001CA2475413A1 Compositions and methods for treating conditions responsive to estrogen
07/12/2001CA2475393A1 Compositions and methods for treating conditions responsive to estrogen
07/12/2001CA2396257A1 Novel compounds and compositions as protease inhibitors
07/12/2001CA2331059A1 Method of reducing morbidity and the risk of mortality
07/11/2001CN1303372A New heterocyclically substituted amides, their production and their use
07/11/2001CN1303365A Benzamide and sulfonamide substituted aminoguanidines and alkoxyguanidines as protease inhibitors
07/11/2001CN1302800A Method for preparing 4-carboxyamino-2-substituted-1,2,3,4-tetrahydroquinoline
07/11/2001CN1068308C Substituted benzoylguanide, its preparing process and medicine and application of same
07/10/2001US6258822 Urokinase inhibitors
07/05/2001WO2001047891A1 Heterocyclic compounds having sulfonamide groups
07/05/2001WO2001047868A1 Novel phenylalanine derivatives
07/05/2001WO2001009065A3 Nitration in a static micromixer
07/05/2001WO2000055137A8 Compounds and methods for modulation of estrogen receptors
07/05/2001WO2000050376A3 Efficient synthesis of alkyl carbonates
07/04/2001EP1113007A1 Tetrahydroisoquinoline compounds as estrogen agonists/antagonists
07/04/2001EP1112456A1 Tube for lining pipes and channels, and a method and device for the production thereof
07/04/2001CN1302292A Aminoisoquinoline derivatives
07/04/2001CN1067991C Aminoalkyl substituted benzo-heterocyclic compounds
07/03/2001US6255349 Alph-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
07/03/2001US6255318 Antiviral compounds
06/2001
06/28/2001WO2001046200A1 Novel piperidine and piperazine derivatives
06/28/2001WO2001010834A3 Antibacterial agents
06/28/2001CA2394095A1 Novel piperidine and piperazine derivatives
06/27/2001EP1110945A2 Azocompounds for the antemortem diagnosis of Alzheimer's disease and in vivo imaging and prevention of amyloid deposition
06/27/2001EP0718281B1 Cyclohexanediurea derivative and process for producing the same
06/27/2001CN1301265A Novel substituted arylhydroxamic acids as metalloproteinase inhibitors
06/27/2001CN1301161A Serotonergic 5HT receptor compounds for treating ocular and CNS disorders
06/27/2001CN1301154A Amide derivatives and nociceptin antagonists
06/26/2001US6252090 Compounds having activity as inhibitors of cytochrome P450RAI
06/26/2001US6252085 Oxazoline derivative
06/26/2001US6252077 1-(N′-(arylalkylaminoalkyl) aminoisoquinolines; a new class of dopamine receptor subtype specific ligands
06/26/2001US6252076 Process for preparation of pyrimidine derivatives
06/24/2001CA2329516A1 Tetrahydroisoquinoline compounds as estrogen agonists/antagonists
06/21/2001WO2001044179A1 Novel succinate compounds, compositions and methods of use and preparation
06/21/2001WO2001044178A1 Novel urea compounds, compositions and methods of use and preparation
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