Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865) |
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06/28/2000 | CN1053895C Substd. sulfonic acid amide, preparation process and pharmaceutical composition of same |
06/27/2000 | US6080790 Selective and potent inhibitors of phosphodiesterase iv and are useful for the prophylaxis and treatment of inflammatory diseases and the alleviation of conditions associated with central nervous malfunction |
06/27/2000 | US6080773 Benzylamine derivatives which are useful in treating psychiatric disorders |
06/22/2000 | WO2000035883A1 Continuous process for the preparation of optically pure decahydroisoquinolinecarboxamide |
06/22/2000 | WO2000035882A1 1,2,3,4-tetrahydronaphthalenes and their pharmaceutical use |
06/22/2000 | WO2000035860A2 Acyl isothiocyanate resins and their use in solid-supported synthesis of guanidines |
06/22/2000 | WO2000035280A1 Exo-r-mecamylamine formulation and use in treatment |
06/22/2000 | WO2000035279A1 Exo-s-mecamylamine formulation and use in treatment |
06/22/2000 | CA2393442A1 Exo-r-mecamylamine formulation and use in treatment |
06/21/2000 | EP1009758A1 Meta-benzamidine derivatives as serine protease inhibitors |
06/21/2000 | EP1009749A1 Preparation of (s)-n-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxyamide |
06/21/2000 | EP1009739A2 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
06/21/2000 | EP1009405A1 Pyrrolidine and piperidine modulators of chemokine receptor activity |
06/21/2000 | CN1257483A Substituted isoquinolines as ultra short acting neuromuscular blockers |
06/15/2000 | WO2000034268A1 Thiourea inhibitors of herpes viruses |
06/15/2000 | WO2000034260A2 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group |
06/15/2000 | WO2000034238A1 Thiourea inhibitors of herpes viruses |
06/15/2000 | WO2000034237A2 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses |
06/15/2000 | CA2351403A1 Thiourea inhibitors of herpes viruses |
06/15/2000 | CA2350996A1 Thiourea inhibitors of herpes viruses |
06/15/2000 | CA2350899A1 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses |
06/15/2000 | CA2350833A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group |
06/14/2000 | EP0777645B1 Oxime ethers and their use as pesticides |
06/07/2000 | EP1005459A1 Substituted isoquinolines as anticonvulsivants |
06/07/2000 | EP1005446A1 N-aroylphenylalanine derivatives |
06/07/2000 | CN1255917A Anti-convulsant isoquinolyl-benzamide derivatives |
06/06/2000 | US6071969 Substituted aminoguanidines and methods of use thereof |
06/06/2000 | US6071929 Selective blockers of n-methyl-d-aspartic acid for teatment of nervous system and brain disorders or injuries |
06/06/2000 | US6071906 Inhibits or modulates the inducible isoform of nitric oxide synthase over the the constitutive isoforms; antiarthritic, -diabetic, ischemic, thrombosis agents; cardiovascular disorders; toxic shock syndrome; autoimmune diseases |
06/02/2000 | WO2000031036A1 Novel naphthalene derivatives |
05/31/2000 | EP1004306A2 Estrogen agonists/antagonists |
05/31/2000 | CN1255124A Substituted isoquinoline derivatives and their use as anticonulsants |
05/31/2000 | CN1052984C New erythromycin derivative and its preparing process and application in medicine |
05/31/2000 | CN1052976C Substituted benzenesulfonylureas and -thioureas, preparation process and possible uses of pharmaceutical preparation therefor |
05/25/2000 | WO2000029380A1 Tetrahydroisoquinoline derivatives as lhrh antagonists |
05/25/2000 | CA2351187A1 Tetrahydroisoquinoline derivatives as lhrh antagonists |
05/24/2000 | EP1001973A1 Compounds which inhibit leukocyte adhesion mediated by vla-4 |
05/24/2000 | CN1254337A N-hydroxy 4-sulfonyl butyramide compounds |
05/23/2000 | US6066650 Inhibitors of microsomal triglyceride transfer protein and method |
05/18/2000 | WO2000027790A1 Mutilin compounds |
05/18/2000 | WO2000004892A3 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions |
05/17/2000 | EP1000999A1 Compounds for organic el devices and organic el devices |
05/17/2000 | EP1000018A2 Urokinase inhibitors |
05/17/2000 | EP0848701B1 O-benzyl oxime ether derivatives and their use in crop protection compositions |
05/17/2000 | CN1253559A Sulfonyl divalent aryl alpha-hydroxamic acid compounds |
05/17/2000 | CN1253548A HIV protease inhibitors |
05/17/2000 | CN1253547A 1,4-substituted cyclic amine derivatives |
05/17/2000 | CN1253545A Aryl sulfonamides and analogues thereof and their use in treatment of neurodegenerative diseases |
05/17/2000 | CN1253474A Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds |
05/17/2000 | CN1253133A Method for purifying isoquinoline |
05/17/2000 | CN1253019A Method for preparing medicine composition capable of inhibiting post infective virus proteinase |
05/16/2000 | US6063925 Separation of enantiomers of octahydroisoquinoline |
05/16/2000 | US6063789 Antiinflammatory agents |
05/16/2000 | US6063784 Heteroaryloxyethylamines, method of preparation, application as medicine and pharmaceutical compositions containing them |
05/11/2000 | WO2000025777A1 SUBSTITUTED PHENETHYLSULFONES AND METHOD OF REDUCING TNFαLEVELS |
05/10/2000 | EP0999256A1 Compounds for organic el element and organic el element |
05/10/2000 | EP0999210A1 Process for the purification of isoquinoline |
05/10/2000 | EP0999208A1 Nitrogenous heterocyclic compounds and hyperlipemia remedy containing the same |
05/10/2000 | EP0998451A1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use |
05/10/2000 | CN1252792A Process and intermediates for the preparation of 4'-trifluoromethyl-bipheyl-2-carboxylic acid (1,2,3,4-tetrahydro-isoquinolin-6-yl)-amide |
05/10/2000 | CN1052240C Method for preparing inhibitor of retroinfection viral protease |
05/09/2000 | US6060503 Antiestrogenic, anticarcinogenic stereospecific benzopyran derivative; breast cancer |
05/04/2000 | WO2000024718A1 Serine protease inhibitor |
05/04/2000 | WO2000024717A2 Isoquinoline derivatives |
05/04/2000 | CA2346990A1 Serine protease inhibitor |
05/03/2000 | EP0997147A1 Amino acid derivatives |
05/03/2000 | EP0996439A1 $g(b)-ALKOXYACRYLATES AGAINST MALARIA |
05/03/2000 | CN1252058A Preparation of butylthio-isoquinoline and intermediate thereof |
05/03/2000 | CN1051998C Isoquinolines preparation thereof and its medicinal compositions |
05/02/2000 | US6057358 Amine derivatives, processes for producing them and a use of them as antiarrhythmic drugs |
05/02/2000 | US6057313 Treating central nervous system disorders |
04/27/2000 | WO2000023421A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES |
04/27/2000 | WO2000023420A1 Aromatic amine derivatives, process for the preparation thereof and agents containing the same |
04/27/2000 | WO2000023078A1 Pharmaceutical compositions containing tetrahydroisoquinoline compounds |
04/27/2000 | CA2348159A1 Aromatic amine derivatives, their production and use |
04/27/2000 | CA2347792A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases |
04/26/2000 | EP0994862A2 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation |
04/26/2000 | CN1251586A Noval pyrimidine derivatives and process and preparing thereof |
04/20/2000 | WO2000021920A1 Diaminopropionic acid derivatives |
04/20/2000 | WO2000021537A1 Novel indenoisoquinolines as antineoplastic agents |
04/13/2000 | WO2000020413A1 Novel 2-[3-phenyl-2-propenyl]-1,2,3,4-tetrahydroxyisoquinoline derivatives, preparation method and use as fungicides |
04/13/2000 | WO2000002850A3 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators |
04/12/2000 | EP0992502A1 2-(3-Phenyl-2-propenyl)-1,2,3,4-tetrahydro-isochinolin derivatives, process for their preparation and their use as fungicides |
04/12/2000 | EP0992495A1 Process for obtaining quinapryl hydrochloride and solvates useful for isolating and purifying quinapryl hydrochloride |
04/12/2000 | EP0991624A1 Phenylalkyl derivatives with thrombin-inhibiting effect |
04/12/2000 | EP0991619A1 INHIBITORS OF $g(a) 4?$g(b) 1?MEDIATED CELL ADHESION |
04/11/2000 | US6048854 2,3-diaminopropionic acid derivative |
04/11/2000 | CA2016656C Enzyme inhibitors |
04/06/2000 | WO2000018735A1 2-substituted heterocyclic sulfonamides |
04/06/2000 | WO2000018733A1 Heterocyclic 2-substituted ketoamides useful for treating hair loss in mammals |
04/06/2000 | WO2000018724A1 (R)-CHIRAL HALOGENATED 1-SUBSTITUTEDAMINO-(n+1)-ALKANOLS USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY |
04/06/2000 | WO2000018721A1 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity |
04/06/2000 | WO2000018708A1 Transfer hydrogenation process |
04/04/2000 | US6046211 Amidino derivatives useful as nitric oxide synthase inhibitors |
04/04/2000 | US6046210 Antipsychotic agents |
04/04/2000 | US6046191 Combination |
03/29/2000 | EP0988280A1 Hydroxamic acid compounds having anticancer and anti-parasitic properties |
03/29/2000 | CN1248968A Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of MIP-1-alpha binding to its CCRI receptor |
03/28/2000 | US6043253 Treatment of diabetes, obesity, lowering triglyceride or cholesterol levels, increasing high density lipoprotein levels or decreasing gut motility, reducing neurogenic inflammation, depression or gastrointestinal disorders |
03/28/2000 | CA2160270C 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same |