Patents
Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865)
06/2000
06/28/2000CN1053895C Substd. sulfonic acid amide, preparation process and pharmaceutical composition of same
06/27/2000US6080790 Selective and potent inhibitors of phosphodiesterase iv and are useful for the prophylaxis and treatment of inflammatory diseases and the alleviation of conditions associated with central nervous malfunction
06/27/2000US6080773 Benzylamine derivatives which are useful in treating psychiatric disorders
06/22/2000WO2000035883A1 Continuous process for the preparation of optically pure decahydroisoquinolinecarboxamide
06/22/2000WO2000035882A1 1,2,3,4-tetrahydronaphthalenes and their pharmaceutical use
06/22/2000WO2000035860A2 Acyl isothiocyanate resins and their use in solid-supported synthesis of guanidines
06/22/2000WO2000035280A1 Exo-r-mecamylamine formulation and use in treatment
06/22/2000WO2000035279A1 Exo-s-mecamylamine formulation and use in treatment
06/22/2000CA2393442A1 Exo-r-mecamylamine formulation and use in treatment
06/21/2000EP1009758A1 Meta-benzamidine derivatives as serine protease inhibitors
06/21/2000EP1009749A1 Preparation of (s)-n-tert-butyl-1,2,3,4-tetrahydroisoquinoline-3-carboxyamide
06/21/2000EP1009739A2 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity
06/21/2000EP1009405A1 Pyrrolidine and piperidine modulators of chemokine receptor activity
06/21/2000CN1257483A Substituted isoquinolines as ultra short acting neuromuscular blockers
06/15/2000WO2000034268A1 Thiourea inhibitors of herpes viruses
06/15/2000WO2000034260A2 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
06/15/2000WO2000034238A1 Thiourea inhibitors of herpes viruses
06/15/2000WO2000034237A2 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
06/15/2000CA2351403A1 Thiourea inhibitors of herpes viruses
06/15/2000CA2350996A1 Thiourea inhibitors of herpes viruses
06/15/2000CA2350899A1 Acetamide and substituted acetamide-containing thiourea inhibitors of herpes viruses
06/15/2000CA2350833A1 Alpha-methylbenzyl-containing thiourea inhibitors of herpes viruses containing a phenylenediamine group
06/14/2000EP0777645B1 Oxime ethers and their use as pesticides
06/07/2000EP1005459A1 Substituted isoquinolines as anticonvulsivants
06/07/2000EP1005446A1 N-aroylphenylalanine derivatives
06/07/2000CN1255917A Anti-convulsant isoquinolyl-benzamide derivatives
06/06/2000US6071969 Substituted aminoguanidines and methods of use thereof
06/06/2000US6071929 Selective blockers of n-methyl-d-aspartic acid for teatment of nervous system and brain disorders or injuries
06/06/2000US6071906 Inhibits or modulates the inducible isoform of nitric oxide synthase over the the constitutive isoforms; antiarthritic, -diabetic, ischemic, thrombosis agents; cardiovascular disorders; toxic shock syndrome; autoimmune diseases
06/02/2000WO2000031036A1 Novel naphthalene derivatives
05/2000
05/31/2000EP1004306A2 Estrogen agonists/antagonists
05/31/2000CN1255124A Substituted isoquinoline derivatives and their use as anticonulsants
05/31/2000CN1052984C New erythromycin derivative and its preparing process and application in medicine
05/31/2000CN1052976C Substituted benzenesulfonylureas and -thioureas, preparation process and possible uses of pharmaceutical preparation therefor
05/25/2000WO2000029380A1 Tetrahydroisoquinoline derivatives as lhrh antagonists
05/25/2000CA2351187A1 Tetrahydroisoquinoline derivatives as lhrh antagonists
05/24/2000EP1001973A1 Compounds which inhibit leukocyte adhesion mediated by vla-4
05/24/2000CN1254337A N-hydroxy 4-sulfonyl butyramide compounds
05/23/2000US6066650 Inhibitors of microsomal triglyceride transfer protein and method
05/18/2000WO2000027790A1 Mutilin compounds
05/18/2000WO2000004892A3 Coadministration of acat and mmp inhibitors for the treatment of atherosclerotic lesions
05/17/2000EP1000999A1 Compounds for organic el devices and organic el devices
05/17/2000EP1000018A2 Urokinase inhibitors
05/17/2000EP0848701B1 O-benzyl oxime ether derivatives and their use in crop protection compositions
05/17/2000CN1253559A Sulfonyl divalent aryl alpha-hydroxamic acid compounds
05/17/2000CN1253548A HIV protease inhibitors
05/17/2000CN1253547A 1,4-substituted cyclic amine derivatives
05/17/2000CN1253545A Aryl sulfonamides and analogues thereof and their use in treatment of neurodegenerative diseases
05/17/2000CN1253474A Sulfonyl divalent aryl or heteroaryl hydroxamic acid compounds
05/17/2000CN1253133A Method for purifying isoquinoline
05/17/2000CN1253019A Method for preparing medicine composition capable of inhibiting post infective virus proteinase
05/16/2000US6063925 Separation of enantiomers of octahydroisoquinoline
05/16/2000US6063789 Antiinflammatory agents
05/16/2000US6063784 Heteroaryloxyethylamines, method of preparation, application as medicine and pharmaceutical compositions containing them
05/11/2000WO2000025777A1 SUBSTITUTED PHENETHYLSULFONES AND METHOD OF REDUCING TNFαLEVELS
05/10/2000EP0999256A1 Compounds for organic el element and organic el element
05/10/2000EP0999210A1 Process for the purification of isoquinoline
05/10/2000EP0999208A1 Nitrogenous heterocyclic compounds and hyperlipemia remedy containing the same
05/10/2000EP0998451A1 Substituted 3,3-diamino-2-propenenitriles, their preparation and use
05/10/2000CN1252792A Process and intermediates for the preparation of 4'-trifluoromethyl-bipheyl-2-carboxylic acid (1,2,3,4-tetrahydro-isoquinolin-6-yl)-amide
05/10/2000CN1052240C Method for preparing inhibitor of retroinfection viral protease
05/09/2000US6060503 Antiestrogenic, anticarcinogenic stereospecific benzopyran derivative; breast cancer
05/04/2000WO2000024718A1 Serine protease inhibitor
05/04/2000WO2000024717A2 Isoquinoline derivatives
05/04/2000CA2346990A1 Serine protease inhibitor
05/03/2000EP0997147A1 Amino acid derivatives
05/03/2000EP0996439A1 $g(b)-ALKOXYACRYLATES AGAINST MALARIA
05/03/2000CN1252058A Preparation of butylthio-isoquinoline and intermediate thereof
05/03/2000CN1051998C Isoquinolines preparation thereof and its medicinal compositions
05/02/2000US6057358 Amine derivatives, processes for producing them and a use of them as antiarrhythmic drugs
05/02/2000US6057313 Treating central nervous system disorders
04/2000
04/27/2000WO2000023421A1 (SUBSTITUTED)ACYL DIPEPTIDYL INHIBITORS OF THE ICE/ced-3 FAMILY OF CYSTEINE PROTEASES
04/27/2000WO2000023420A1 Aromatic amine derivatives, process for the preparation thereof and agents containing the same
04/27/2000WO2000023078A1 Pharmaceutical compositions containing tetrahydroisoquinoline compounds
04/27/2000CA2348159A1 Aromatic amine derivatives, their production and use
04/27/2000CA2347792A1 (substituted)acyl dipeptidyl inhibitors of the ice/ced-3 family of cysteine proteases
04/26/2000EP0994862A2 Sulphonamide derivatives being 5-ht6 receptor antagonists and process for their preparation
04/26/2000CN1251586A Noval pyrimidine derivatives and process and preparing thereof
04/20/2000WO2000021920A1 Diaminopropionic acid derivatives
04/20/2000WO2000021537A1 Novel indenoisoquinolines as antineoplastic agents
04/13/2000WO2000020413A1 Novel 2-[3-phenyl-2-propenyl]-1,2,3,4-tetrahydroxyisoquinoline derivatives, preparation method and use as fungicides
04/13/2000WO2000002850A3 Sulfonylamino carboxylic acid n-arylamides as guanylate cyclase activators
04/12/2000EP0992502A1 2-(3-Phenyl-2-propenyl)-1,2,3,4-tetrahydro-isochinolin derivatives, process for their preparation and their use as fungicides
04/12/2000EP0992495A1 Process for obtaining quinapryl hydrochloride and solvates useful for isolating and purifying quinapryl hydrochloride
04/12/2000EP0991624A1 Phenylalkyl derivatives with thrombin-inhibiting effect
04/12/2000EP0991619A1 INHIBITORS OF $g(a) 4?$g(b) 1?MEDIATED CELL ADHESION
04/11/2000US6048854 2,3-diaminopropionic acid derivative
04/11/2000CA2016656C Enzyme inhibitors
04/06/2000WO2000018735A1 2-substituted heterocyclic sulfonamides
04/06/2000WO2000018733A1 Heterocyclic 2-substituted ketoamides useful for treating hair loss in mammals
04/06/2000WO2000018724A1 (R)-CHIRAL HALOGENATED 1-SUBSTITUTEDAMINO-(n+1)-ALKANOLS USEFUL FOR INHIBITING CHOLESTERYL ESTER TRANSFER PROTEIN ACTIVITY
04/06/2000WO2000018721A1 Substituted polycyclic aryl and heteroaryl tertiary-heteroalkylamines useful for inhibiting cholesteryl ester transfer protein activity
04/06/2000WO2000018708A1 Transfer hydrogenation process
04/04/2000US6046211 Amidino derivatives useful as nitric oxide synthase inhibitors
04/04/2000US6046210 Antipsychotic agents
04/04/2000US6046191 Combination
03/2000
03/29/2000EP0988280A1 Hydroxamic acid compounds having anticancer and anti-parasitic properties
03/29/2000CN1248968A Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of MIP-1-alpha binding to its CCRI receptor
03/28/2000US6043253 Treatment of diabetes, obesity, lowering triglyceride or cholesterol levels, increasing high density lipoprotein levels or decreasing gut motility, reducing neurogenic inflammation, depression or gastrointestinal disorders
03/28/2000CA2160270C 1,2-ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
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