Patents for C07D 217 - Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems (11,865) |
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04/24/2013 | CN102070525B Tetrahydroisoquinoline derivatives and preparation method and application thereof |
04/24/2013 | CN101550085B Novel organic electroluminescent compounds and organic electroluminescent device using the same |
04/23/2013 | US8426596 Process of producing bleach boosters |
04/23/2013 | CA2552419C Azadecalin glucocorticoid receptor modulators |
04/23/2013 | CA2529257C Methods and compositions for treating amyloid-related diseases |
04/18/2013 | WO2013056060A1 Substituted tetrahydroisoquinoline compounds as factor xia inhibitors |
04/18/2013 | WO2013056034A1 Substituted tetrahydroisoquinoline compounds as factor xia inhibitors |
04/18/2013 | WO2013055984A1 Substituted tetrahydroisoquinoline compounds as factor xia inhibitors |
04/18/2013 | WO2013027196A9 Substituted 2-alkyl-1-oxo-n-phenyl-3-heteroaryl-1,2,3,4- tetrahydroisoquinoline-4-carboxamides for antimalarial therapies |
04/18/2013 | US20130096310 Isoquinoline derivative |
04/18/2013 | US20130096119 Isoquinolin-3-Ylurea Derivatives |
04/18/2013 | US20130096083 Use of isoquinolones for preparing drugs, novel isoquinolones and method for synthesising same |
04/18/2013 | CA2851810A1 Substituted tetrahydroisoquinoline compounds as factor xia inhibitors |
04/17/2013 | CN102234276B Preparation method of optical isomer of stepholidine or its derivative and intermediate used in the method |
04/16/2013 | US8420667 Isoquinolinone derivatives as NK3 antagonists |
04/16/2013 | US8420661 Arylethynyl derivatives |
04/10/2013 | EP2578571A1 Isoquinoline modulators of ATP-binding cassette transporters |
04/10/2013 | EP2576514A1 Substituted isoquinolines and their use as tubulin polymerization inhibitors |
04/10/2013 | CN103038218A Condensed ring pyridine compound |
04/09/2013 | US8415474 One-pot preparation of hexahydroisoquinolines from dihydroisoquinolines |
04/04/2013 | WO2013047751A1 Production method for 3,4-dihydroisoquinoline derivative |
04/04/2013 | WO2013047750A1 Production methods for 3,4-dihydroisoquinoline derivatives, and production intermediates for same |
04/03/2013 | CN101516834B Isoserine derivatives for use as coagulation factor IXa inhibitors |
04/03/2013 | CN101516833B Tartrate derivatives for use as coagulation factor IXa inhibitors |
04/02/2013 | CA2616373C Octahydroisoquinoline compounds as opioid receptor modulators |
04/02/2013 | CA2564085C Heterocyclic amide compound and use thereof as an mmp-13 inhibitor |
03/28/2013 | WO2012162513A3 Alcohol-, diol-, and carbohydrate-substituted indenoisoquinolines as topoisomerase i inhibitors |
03/27/2013 | CN103003244A Salt and solvates of a tetrahydroisoquinoline derivative |
03/27/2013 | CN101442909B Bicycloheteroaryl compounds as P2X7 modulators and uses thereof |
03/21/2013 | WO2013038136A1 BI-AROMATIC AND TRI-AROMATIC COMPOUNDS AS NADPH OXIDASE 2 (Nox2) INHIBITORS |
03/20/2013 | CN102977016A Nitrogen-containing heteroaryl compounds and their use in increasing endogeneous erythropoietin |
03/20/2013 | CN102977015A Nitrogen-containing heteroaryl compounds and their use in increasing endogeneous erythropoietin |
03/20/2013 | CN101588803B Intermediate duration neuromuscular blocking agents and antagonists thereof |
03/20/2013 | CN101573338B Cycloalkylamine substituted isoquinolone and isoquinolinone derivatives |
03/19/2013 | US8399493 Pyridinone derivatives and their use as positive allosteric modulators of mGluR2-receptors |
03/19/2013 | US8399482 6-substituted isoquinolines and isoquinolinones |
03/19/2013 | US8399481 Compounds |
03/19/2013 | CA2524027C Immunosuppressant compounds and compositions |
03/14/2013 | WO2013021398A3 A process for preparation of mivacurium chloride |
03/12/2013 | US8394831 Carbonylamino-derivatives as novel inhibitors of histone deacetylase |
03/12/2013 | US8394825 Compound |
03/07/2013 | WO2013031930A1 Imine derivative |
03/07/2013 | WO2013030358A1 Glycine b antagonists |
03/07/2013 | WO2013003315A3 Methods for preparing isoquinolines |
03/07/2013 | US20130059882 8-Phenylisoquinolines And Pharmaceutical Composition Used In Treatment For Sepsis |
03/07/2013 | US20130059852 Compounds for treating disease, for administering, and for pharmaceutical compositions |
03/06/2013 | CN102958914A 1-phenyl-substituted heterocyclyl derivatives and their use as prostaglandin D2 receptor modulators |
03/06/2013 | CN102952146A Heterocyclic compound, organic light-emitting device, and flat display device |
03/06/2013 | CN101679273B 1-substituted tetrahydroisoquinoline compound |
03/05/2013 | US8389730 Compositions and methods for the treatment of disease associated with TRP-P8 expression |
03/05/2013 | US8389570 Hydroxamates as therapeutic agents |
03/05/2013 | US8389553 4-carboxybenzylamino derivatives as histone deacetylase inhibitors |
02/28/2013 | WO2013027196A1 Substituted 2-alkyl-1-oxo-n-phenyl-3-heteroaryl-1,2,3,4- tetrahydroisoquinoline-4-carboxamides for antimalarial therapies |
02/28/2013 | WO2013027168A1 Novel heterocyclic compounds as bromodomain inhibitors |
02/28/2013 | US20130053348 Certain chemical entities, compositions, and methods |
02/28/2013 | CA2846507A1 Substituted 2-alkyl-1-oxo-n-phenyl-3-heteroaryl-1,2,3,4- tetrahydroisoquinoline-4-carboxamides for antimalarial therapies |
02/26/2013 | US8383094 Hepatitis C virus inhibitors |
02/20/2013 | EP2559455A1 Heteroaryl derivatives as DGAT1 inhibitors |
02/20/2013 | CN101595094B Cycloalkylamine substituted isoquinolone derivatives |
02/14/2013 | US20130041154 Process for producing cisatracurium and associated intermediates |
02/13/2013 | CN102161664B Photoreaction-based synthesis method of spiro isoquinoline polycyclic heterocyclic compounds |
02/12/2013 | US8372864 1-oxo-isoindoline-4-carboxamide and 1-oxo-1,2,3,4-tetrahydroisoquinoline-5-carboxamide derivatives, preparation and therapeutic use thereof |
02/07/2013 | WO2013017654A1 Novel estrogen receptor ligands |
02/07/2013 | CA2842719A1 Novel estrogen receptor ligands |
02/06/2013 | EP2552893A1 Antibacterial isoquinolin-3-ylurea derivatives |
02/05/2013 | US8367832 Crystalline forms of Nelfinavir mesylate |
02/05/2013 | US8367701 Crystalline pharmaceutical and methods of preparation and use thereof |
02/05/2013 | US8367700 Substituted 4-(1.2,3,4-tetrahydroisoquinolin-2-yl)-4-oxobutyric acid amide as KCNQ2/3 modulators |
02/05/2013 | US8367699 Tetrahydro-isoquinolines |
02/05/2013 | CA2526872C Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor |
01/31/2013 | WO2013013609A1 Polymorphic forms of compounds as prolyl hydroxylase inhibitor, and uses thereof |
01/31/2013 | US20130028843 Kallikrein 7 modulators |
01/31/2013 | CA2842730A1 Polymorphic forms of compounds as prolyl hydroxylase inhibitor, and uses thereof |
01/30/2013 | CN102898370A Cis-atracurium besilate for injection |
01/29/2013 | US8362264 Compositions and methods for the treatment of disease associated with Trp-p8 expression |
01/23/2013 | EP2548618A2 Organic compounds |
01/22/2013 | US8357807 Isoquinolinium compounds useful in the preparation of cisatracurium and associated intermediates |
01/22/2013 | US8357806 Process for synthesizing substituted isoquinolines |
01/22/2013 | US8357699 6-aminoisoquinoline compounds |
01/17/2013 | WO2013007371A2 Kinetic resolution of chiral amines |
01/16/2013 | EP2546239A1 6-amino isoquinolins compounds and methods for making the same |
01/16/2013 | EP2546238A1 6-amino isoquinolins compounds and methods for making the same |
01/16/2013 | EP2546237A1 7-amino isoquinolins compounds and methods for making the same |
01/16/2013 | CN102875466A Isoquinolinone derivatives, and preparation method and medical purpose thereof |
01/16/2013 | CN102875465A Method for preparing 7-bromoisoquinoline |
01/16/2013 | CN102875413A 免疫抑制剂化合物及组合物 Immunosuppressant compounds and compositions |
01/16/2013 | CN102872915A Iron catalyst system for preparation of pyridine derivatives and its application |
01/10/2013 | WO2013005157A1 Sulfone derivatives and their use as pkm2 modulators for the treatment of cancer |
01/10/2013 | WO2013005049A1 N- (2 -aminophenyl) benzamide derivatives as histone deacetylase inhibitors |
01/10/2013 | US20130012536 Modulators of atp-binding cassette transporters |
01/09/2013 | EP2542530A2 Process for the preparation of 2-(cyclohexylmethyl)-n-{2- [(2s)-1-methylpyrrolidin-2-yl]ethyl}-1, 2, 3, 4- tetrahydroisoquinoline-7-sulfonamide |
01/09/2013 | EP2542239A1 Use of isoquinolones for preparing drugs, novel isoquinolones and method for synthesising same |
01/09/2013 | CN102863380A Preparation method of 1-alkynyl-2-aryl-1,2,3,4-tetrahydroisoquinoline compound |
01/08/2013 | US8350039 Substituted isoquinoline derivatives, pharmaceutical compositions, and methods of use as beta-secretase inhibitors |
01/08/2013 | US8350038 Fluorescence quencher molecules |
01/08/2013 | US8349868 Azaquinolones that inhibit prolyl hydroxylase |
01/03/2013 | WO2013003315A2 Methods for preparing isoquinolines |
01/03/2013 | WO2013002357A1 Hiv replication inhibitor |
01/03/2013 | WO2013000651A1 Fluorinated arylalkylaminocarboxamide derivatives |
01/03/2013 | US20130005965 Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin |