| Patents for C07B 59 - Introduction of isotopes of elements into organic compounds (2,678) |
|---|
| 03/17/2004 | EP1397370A1 B-benzyloxyaspartate derivatives with amino group on benzene ring |
| 03/17/2004 | EP1397327A2 DEUTERATED N-SUBSTITUTED AND $g(a)-SUBSTITUTED DIPHENYLALKOXY ACETIC ACID AMINO ALKYL ESTERS AND MEDICAMENTS CONTAINING THESE COMPOUNDS |
| 03/11/2004 | WO2002102743A9 DEUTERATED N-SUBSTITUTED AND α-SUBSTITUTED DIPHENYLALKOXY ACETIC ACID AMINO ALKYL ESTERS AND MEDICAMENTS CONTAINING THESE COMPOUNDS |
| 03/09/2004 | CA2216423C Ternary radiopharmaceutical complexes |
| 03/04/2004 | US20040043920 Chelate compound of metal and dithiocarbamate; therapy, diagnosis |
| 02/24/2004 | US6696551 225Ac-HEHA and related compounds, methods of synthesis and methods of use |
| 02/19/2004 | WO2003065882A3 Non-invasive diagnostic imaging technology for mitochondria using radiolabeled lipophilic salts |
| 02/19/2004 | US20040033197 Non-invasive diagnostic imaging technology for mitochondria dysfunction using radiolabeled lipophilic salts |
| 02/19/2004 | US20040033196 Synthesis of 17F labeled fluoroalkanes |
| 02/12/2004 | US20040029963 Use of pamoic acid or one of its derivatives, or one of its analogues , for the preparation of a medicament for the treatment of diseases characterised by deposits of amyloid aggregates |
| 02/05/2004 | WO2004010846A2 Design and synthesis of renal dipeptidase inhibitors |
| 02/05/2004 | US20040024307 Para-hydrogen labeled agents and their use in magnetic resonance imaging |
| 02/05/2004 | CA2493773A1 A method of deuteration of an aromatic ring |
| 02/04/2004 | EP0863858B1 Mass-based encoding and qualitative analysis of combinatorial libraries |
| 02/04/2004 | CN1473158A Radiopharmaceuticals for diagnosing alzheimer's disease |
| 01/28/2004 | EP1383752A2 Deuterated 3-piperidinopropiophenone and medicaments containing said compounds |
| 01/21/2004 | EP1381396A2 Tc and re labeled radioactive glycosylated octreotide derivatives |
| 01/13/2004 | US6676926 Radiopharmaceuticals for diagnosing Alzheimer's disease |
| 12/31/2003 | WO2003078358A3 Use of microfabricated devices for radiosynthesis |
| 12/30/2003 | CA2001765C Chelants possessing ortho ligating functionality and complexes thereof |
| 12/18/2003 | WO2003104430A2 Method for obtaining dynamic and structural data pertaining to proteins and protein/ligand complexes |
| 12/18/2003 | WO2003104166A1 Process for deuteration of inert methylene |
| 12/18/2003 | CA2488773A1 Method for obtaining dynamic and structural data pertaining to proteins and protein/ligand complexes |
| 12/09/2003 | US6660246 Ligands and metal complexes thereof |
| 12/04/2003 | WO2003099746A1 Method for the production of 18f-fluorinated alpha acids |
| 11/27/2003 | US20030220234 A cyclosporine A derivative with isotopic or chemical substitution in the amino acid position selected from the group consisting of 1,3, and 9 or combination |
| 11/26/2003 | EP1363954A2 Polymer precursors of radiolabeled compounds, and methods of making and using the same |
| 11/26/2003 | EP0974572B1 Novel process for producing alcohols |
| 11/06/2003 | WO2003064678A3 Apparatus for synthesis of radiolabeled compounds |
| 11/05/2003 | EP1359147A1 4,4-disubstituted-1,4-dihydro-2H-3,1-benzoxazin-2-ones useful as HIV reverse transcriptase inhibitors and processes for making the same |
| 11/04/2003 | CA2123570C Cocaine receptor binding ligands |
| 10/30/2003 | WO2003089438A1 Labeled oxazinocarbazoles as diagnostic agents |
| 10/21/2003 | CA2093896C Hormone labelling with rhenium and technetium |
| 10/16/2003 | US20030194748 Method for labeling with tritium |
| 10/15/2003 | EP1351930A2 Protease inhibitors |
| 10/15/2003 | CN1449375A Use of pamoic acid or one of derivatives or analogs thereof for preparing a medicament used for treating diseases |
| 10/08/2003 | EP0533845B1 USING 5,10,15,20-TETRAKIS(r-CARBOXYPHENYL)PORPHINE FOR DETECTING AND TREATING LUNG CANCER |
| 10/02/2003 | WO2003080544A1 Radiofluorination methods |
| 10/01/2003 | EP1066235B1 Synthetic endogenous cannabinoid analogues and uses thereof |
| 09/25/2003 | WO2003078358A2 Use of microfabricated devices for radiosynthesis |
| 09/17/2003 | CN1121374C Novel trienoic retinoid compounds and method |
| 09/12/2003 | WO2002085418A3 Tc and re labeler radioactive glycosylated octreotide derivatives |
| 09/10/2003 | EP1341795A2 Novel labeled resiniferatoxin derivatives |
| 09/04/2003 | US20030166144 Growth hormone secretagogue receptor family |
| 09/03/2003 | EP0929533B1 4,4-disubstituted-1,4-dihydro-2h-3,1-benzoxazin-2-ones useful as hiv reverse transcriptase inhibitors and intermediates and processes for making the same |
| 09/02/2003 | US6613739 Immunosuppressants |
| 08/27/2003 | EP1337532A2 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit |
| 08/27/2003 | EP0760685B1 Thiolation of proteins for radionuclide-based radioimmunodetection and radioimmunotherapy |
| 08/19/2003 | US6607710 Provide a bisphosphonic acid derivative and said bisphosphonic acid derivative being labeled with a radioactive nuclide, which has properties of rapid accumulation to the bone and rapid urinary excretion. |
| 08/14/2003 | WO2003065882A2 Non-invasive diagnostic imaging technology for mitochondria using radiolabeled lipophilic salts |
| 08/14/2003 | WO2002070020A9 Polymer precursors of radiolabeled compounds, and methods of making and using the same |
| 08/14/2003 | CA2474142A1 Non-invasive diagnostic imaging technology for mitochondria dysfunction using radiolabeled lipophilic salts |
| 08/12/2003 | US6605593 Enhanced efficacy and reduced toxicity |
| 08/07/2003 | WO2003064678A2 Apparatus for synthesis of radiolabeled compounds |
| 08/06/2003 | EP1332138A1 Radiopharmaceuticals for diagnosing alzheimer's disease |
| 07/31/2003 | WO2001034566A3 Protease inhibitors |
| 07/31/2003 | US20030144322 Analogs of cocaine |
| 07/29/2003 | CA2134092C Carboxamide modified polyamine chelators and radioactive complexes thereof for conjugation to antibodies |
| 07/17/2003 | US20030135063 Especially Type II diabetes; stimulating the kinase activity of the insulin receptor; activating the insulin receptor |
| 07/09/2003 | EP1325917A1 Radiolabelled alkylamino-benzothiazole and -benzoxazole derivatives and their use as D4 ligands |
| 07/03/2003 | WO2003053910A1 Stable isotope-labeled amino acid, method of integrating the same into target protein, method of nmr structural analysis of protein and process for producing site-selective stable isotope-labeled fumaric acid and tartaric acid |
| 07/03/2003 | US20030124059 Imaging agents, precursors thereof and methods of manufacture |
| 07/01/2003 | US6585953 Fluorinating a 17F-labeled F2 with an alkane, a substituted or unsubstituted alkene, or a substituted or unsubstituted alkyne in the presence of a metal oxide, especially silver oxide, catalyst |
| 06/05/2003 | US20030103896 Methods of synthesis and use of radiolabelled platinum chemotherapeutic agents |
| 06/04/2003 | EP1315689A1 Synthesis of 17f labeled fluoroalkanes |
| 06/03/2003 | US6574495 Para-hydrogen labelled agents and their use in magnetic resonance imaging |
| 05/30/2003 | WO2002088100A3 Deuterated 3-piperidinopropiophenone and medicaments containing said compounds |
| 05/30/2003 | WO2002070020A3 Polymer precursors of radiolabeled compounds, and methods of making and using the same |
| 05/21/2003 | EP0765166B1 Radiolabeled annexin-galactose conjugates |
| 05/20/2003 | US6565828 Bifunctional chelant for attaching diagnostic metals and therpeutic isotopes to target specific biomolecules; heavy metal detoxification |
| 05/06/2003 | CA2109208C Radiolabeled metal-binding protein for the treatment of arthritis |
| 05/02/2003 | EP1173184A4 Rho-boronophenylalanine complexes with fructose and related carbohydrates and polyols |
| 04/24/2003 | WO2003002489A3 Solid-phase electrophilic fluorination |
| 04/16/2003 | EP1301463A1 Use of pamoic acid or one of its derivatives, or one of its analogues, for the preparation of a medicament for the treatment of diseases characterised by deposits of amyloid aggregates |
| 04/15/2003 | US6548042 Bis-phosphonate compounds |
| 03/27/2003 | WO2003024940A1 Bifunctional chelating agent for actinium |
| 03/19/2003 | EP1023264B1 New marker, production process and use thereof |
| 03/18/2003 | US6534488 32P or 33P-labelled bisphosphonates as radiotherapeutic radiopharmaceuticals. The 32P- or 33P-labelled bisphosphonates, which are chemically identical to the unlabelled agent, are expected to target the lesion site in |
| 03/18/2003 | US6534038 Ternary ligand complexes useful as radiopharmaceuticals |
| 03/13/2003 | WO2002102743A3 DEUTERATED N-SUBSTITUTED AND α-SUBSTITUTED DIPHENYLALKOXY ACETIC ACID AMINO ALKYL ESTERS AND MEDICAMENTS CONTAINING THESE COMPOUNDS |
| 03/12/2003 | CN1401629A Image forming agent, its precursor and preparing process thereof |
| 03/11/2003 | US6531636 Derivatives of 2-archidonoyl glycerol, stable to hydrolysis; ethers derived from long chain fatty alcohols (archidonyl alcohol) bind to the CB1 and CB2 cannabinoid receptors; in vivo effects similar to anandamide and 2-Ara-Gl |
| 03/11/2003 | US6531314 Growth hormone secretagogue receptor family |
| 03/06/2003 | WO2002090298A3 Method for the synthesis of 18f marked compounds which are low in carriers |
| 02/26/2003 | EP1285902A1 Method for labeling with tritium |
| 02/26/2003 | EP0832068B1 Stable reagents for the preparation of radiopharmaceuticals |
| 02/12/2003 | EP1282631A1 Methods of synthesis and use of radiolabelled platinum chemotherapeutic agents |
| 02/11/2003 | US6517811 Compounds for cancer imaging and therapy |
| 02/11/2003 | CA2216851C Radiolabeled peptides for diagnosis and therapy |
| 02/06/2003 | WO2002030937A3 Labeled resiniferatoxin derivatives for use in vanilloid receptor binding assay |
| 02/04/2003 | US6515112 For use in diagnosis and therapy |
| 01/30/2003 | WO2003008394A1 Novel chelating agents and conjugates thereof, their synthesis and use as diagnostic and therapeutic agents |
| 01/23/2003 | WO2001005805A9 Novel c-19-halogen-substituted, 5-substituted, 5-substituted or 6,10 carbocyclically condensed steroids of the androst-9(11)-ene-series, methods for the production and use thereof |
| 01/21/2003 | US6509001 Calcitonin receptor binding reagents |
| 01/09/2003 | WO2003002489A2 Solid-phase electrophilic fluorination |
| 01/09/2003 | WO2003002157A1 Solid-phase nucleophilic fluorination |
| 01/07/2003 | CA2069154C Polypeptides |
| 01/03/2003 | WO2003000698A1 β-BENZYLOXYASPARTATE DERIVATIVES WITH AMINO GROUP ON BENZENE RING |
| 01/02/2003 | EP1268497A1 Ternary ligand complexes useful as radiopharmaceuticals |
| 12/27/2002 | WO2002102743A2 DEUTERATED N-SUBSTITUTED AND α-SUBSTITUTED DIPHENYLALKOXY ACETIC ACID AMINO ALKYL ESTERS AND MEDICAMENTS CONTAINING THESE COMPOUNDS |