| Patents for C07B 59 - Introduction of isotopes of elements into organic compounds (2,678) |
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| 05/19/2005 | WO2005045850A2 Radioactive arsenic triiodide and use thereof for radioactive markings |
| 05/19/2005 | WO2005044758A1 Process for producing radioactive-fluorine-labeled compound |
| 05/12/2005 | WO2005042441A1 Method and apparatus for the use of [11c] carbon monixide in labeling synthesis by photo-initiated carbonylation |
| 05/11/2005 | EP1337532B1 Compound for chelating a metal, radiopharmaceutical, manufacturing process therefor, and diagnostic kit |
| 05/06/2005 | CA2782783A1 Fused heterocyclic compounds |
| 04/28/2005 | WO2005037853A2 Side chain deuterated amino acids and methods of use |
| 04/28/2005 | WO2005037737A1 Method for the production of [18f] fluoride-marked aromatic l-amino acids |
| 04/28/2005 | US20050089471 A reaction product of an antibody, protein, biomolecule, polysaccharide, or peptidomimetic, a luminescent dye, radionuclide, near infrared dye, a magnetically active isotope, a superparamagnetic particle, or a metal ion, and a linker moiety; diagnosis and monitoring of inflammatory diseases |
| 04/28/2005 | US20050089470 Labeled peptides for lectin-like oxidized low-density lipoprotein receptor (LOX-1) |
| 04/21/2005 | US20050084452 Deuterated hydrogen in protein, radioactive carbon or nitrogen; bioassay of accurate analyzing the structure of the target high molecular weight protein; producing stable isotope-labeled fumaric acid, tartaric acid through esterification, oxidation, hydrolysis; chemical peptide synthesis |
| 04/19/2005 | CA2138150C 4-amino-n-(4-methyl-4-piperidinyl)-2-methoxybenzamides |
| 04/07/2005 | WO2005030677A1 Process for producing radioactive fluorine compound |
| 04/07/2005 | WO2005030676A1 Methods of [11c]-radiolabelling phenothiazine and phenothiazine-like compounds |
| 04/07/2005 | CA2540827A1 Methods of [11c]-radiolabelling phenothiazine and phenothiazine-like compounds |
| 03/29/2005 | US6872381 Such as 1-(5-chloro-2-(2-((2R)-4-(4-fluoro-18F-benzyl)-2-methylpiperazin-1-yl)-2 -oxoethoxy)phenyl)urea for binding chemokine receptors in brain tissue; tomography |
| 03/02/2005 | EP0836609B1 Method and device for synthesising labelled compounds |
| 02/17/2005 | WO2005014479A2 Process for preparing radiolabeled compounds |
| 02/17/2005 | CA2536659A1 Process |
| 02/03/2005 | CA2783275A1 Stable radiopharmaceutical compositions and methods for their preparation |
| 02/03/2005 | CA2533416A1 Heavy-hydrogenated norbornyl (meth)acrylates, process for producing them, polymers thereof and optical members |
| 02/03/2005 | CA2533415A1 Heavy-hydrogenated (meth)acrylates, process for producing them, polymers thereof and optical members |
| 01/27/2005 | WO2004098650A3 Prosthetic groups attached to stannyl polymer in the synthesis of radiopharmaceuticals |
| 01/27/2005 | US20050020679 Enzyme inhibitors for anandamide transporter and pharmacological use with urea, amide, thiourea or other groups |
| 01/20/2005 | CA2532038A1 Compositions and methods for stable isotope labelling of biological compounds |
| 01/19/2005 | EP1181271B1 Naphthalene ureas as glucose uptake enhancers |
| 01/19/2005 | CN1185252C Somatostatin peptides |
| 01/19/2005 | CN1185210C Use of naphthalene-carboxylic acid for preparing a medicament used for treating diseases characterized by amyloid aggregation sedimentation |
| 01/12/2005 | EP1495031A1 Labeled oxazinocarbazoles as diagnostic agents |
| 12/29/2004 | CN1182116C Mutilin derivatives and their use as antibacterials |
| 12/29/2004 | CN1182111C Nitroso compound and use of it as spin catching agent |
| 12/28/2004 | US6835371 Diagnostic and therapeutic piperazine and piperidine compounds and process |
| 12/22/2004 | EP1487763A2 Use of microfabricated devices for radiosynthesis |
| 12/22/2004 | EP1487762A1 Radiofluorination methods |
| 12/16/2004 | WO2004108636A2 Isotopically labeled chemically stable reagents and process for the synthesis thereof |
| 12/16/2004 | US20040253180 Deuterated nifedipine and penicillins; improved bioavailability |
| 12/15/2004 | EP0988263B1 Process for the production of radioiodinated neuroreceptor agents |
| 12/02/2004 | US20040242887 Hypotonic bladder diseases |
| 12/02/2004 | US20040242852 Bifunctional chelating agent for actinium |
| 12/02/2004 | US20040242652 Beta benzyloxyaspartate derivatives with amino group on benzene ring |
| 12/01/2004 | EP1480739A2 Apparatus for synthesis of radiolabeled compounds |
| 11/30/2004 | US6824982 High-throughput-screening method for determining enantioselectivity |
| 11/30/2004 | US6824760 Imaging agents, precursors thereof and methods of manufacture |
| 11/25/2004 | US20040236085 Solid-phase nucleophilic fluorination |
| 11/25/2004 | US20040235910 Mutilin derivatives and their use as antibacterials |
| 11/18/2004 | WO2004100490A2 Device and method for the fluorination of nucleophiles |
| 11/18/2004 | WO2004098650A2 Prosthetic groups attached to stannyl polymer in the synthesis of radiopharmaceuticals |
| 11/18/2004 | US20040230064 Novel labeled resiniferatoxin derivatives |
| 11/16/2004 | US6818200 Modification of the molecular structure of dihydropyridine family drug containing one or more hydrogen atoms by deuterating one or more hydrogen atoms to deuterium atoms; improved activity over the known drug |
| 11/11/2004 | US20040225121 Labeling using deuterium, tritium with catalyst |
| 11/10/2004 | EP1474177A2 Non-invasive diagnostic imaging technology for mitochondria using radiolabeled lipophilic salts |
| 11/04/2004 | DE10316965A1 New technetium-labeled fatty acids based on nitrilo-tris-(alkanethiolato) complexes, useful as stable radioactive tracers for diagnostic imaging of the myocardium |
| 10/26/2004 | CA2185306C Radio-detection method of oxygenation reaction |
| 10/20/2004 | CN1538876A Novel catalytic formulation and its preparation method |
| 10/19/2004 | WO2004069773A1 Irreversible caspase-3 inhibitors as active site probes |
| 10/19/2004 | US6806281 Treatment of cocaine abuse, parkinson's disease |
| 10/19/2004 | CA2514441A1 Irreversible caspase-3 inhibitors as active site probes |
| 10/13/2004 | EP1173184B1 para-BORONOPHENYLALANINE COMPLEXES WITH FRUCTOSE AND RELATED CARBOHYDRATES AND POLYOLS |
| 10/13/2004 | EP0876402B1 Growth hormone secretagogue receptor family |
| 10/07/2004 | US20040197257 reacting carbon dioxide isotope in gas mixture ; forming, trapping carbon monoxide in complex; using pressurized chemical reactor |
| 09/29/2004 | EP0912533B1 Alkylaminobenzothiazole and -benzoxazole derivatives |
| 09/23/2004 | WO2004080492A1 Methods of radiofluorination of biologically active vectors |
| 09/23/2004 | US20040186312 Solid-phase electrophilic fluorination |
| 09/23/2004 | US20040186136 E.g., mono-, poly- or perdeuteriated tolperisone and eperisone; appreciably better pharmacokinetic and/or pharmacodynamic properties than the undeuterated compounds; muscular disorders; muscle relaxants (skeletal); antispasmodic agents; vasodilation |
| 09/23/2004 | US20040184991 Ac-HEHA and related compounds, methods of synthesis and methods of use |
| 09/23/2004 | CA2518889A1 Methods of radiofluorination of biologically active vectors |
| 09/21/2004 | US6794522 Labeling organic compounds with deuterium and tritium using specific catalysts based on group 8 metals containing pentamethylcyclopentadiene ligand; deuterated tetrahydrofuran or diethyl ether for example |
| 09/15/2004 | EP1457482A1 Stable isotope-labeled amino acid, method of integrating the same into target protein, method of nmr structural analysis of protein and process for producing site-selective stable isotope-labeled fumaric acid and tartaric acid |
| 09/15/2004 | EP1165834B1 High throughput screening method for determining enantioselectivity |
| 09/14/2004 | US6790843 C-19-halogen-substituted steroids of the androst-9(11)-ene-series, methods for the production and use thereof |
| 09/08/2004 | CN1527823A Deuterated 3-piperidinopropiophenone and medicaments containing said compounds |
| 09/01/2004 | EP0674530B1 Radiolabeled polyhydric phenol compounds |
| 08/31/2004 | US6784193 Mutilin derivatives and their use as antibacterials |
| 08/26/2004 | US20040167330 Suitable targeting moieties are monoclonal antibodies, their fragments and recombinant derivatives such as single chain antibodies, diabodies, triabodies, humanized, human or chimeric variants but also peptides, aptamers, spiegelmers, nucleotides, anti sense oligomers |
| 08/12/2004 | WO2004010846A3 Design and synthesis of renal dipeptidase inhibitors |
| 08/11/2004 | CN1520315A Solid-phase nucleophilic fluorination |
| 07/29/2004 | DE19949237B4 Vorstufenverbindung für Radiodiagnostika und Verfahren zu ihrer Herstellung Precursor for radio diagnostics and process for their preparation |
| 07/28/2004 | CN1516684A Deuterated N-substituted and alpha-substituted diphenylalkoxy acetic acid amino alkyl esters and medicaments containing these compounds |
| 07/27/2004 | US6767715 Nitroso compounds and their use as spin traps |
| 07/22/2004 | WO2004060831A1 Method of deuterization |
| 07/22/2004 | CA2511885A1 Method of deuteration |
| 07/21/2004 | EP1438299A1 Bifunctional chelating agent for actinium |
| 07/08/2004 | WO2004056725A1 Solid-phase preparation of 18f-labelled amino acids |
| 07/08/2004 | WO2004056724A1 Deuterated catecholamine derivatives and medicaments comprising said compounds |
| 07/08/2004 | DE19744003B4 Kontrastmittel für das Infarkt- und Nekroseimaging Contrast agents for infarction and necrosis |
| 07/01/2004 | WO2003104430A3 Method for obtaining dynamic and structural data pertaining to proteins and protein/ligand complexes |
| 07/01/2004 | DE10261807A1 Deuterierte Catecholaminderivate sowie diese Verbindungen enthaltende Arzneimittel Deuterated catecholamine derivatives and pharmaceutical compositions containing them |
| 06/15/2004 | US6749830 Injecting sample comprising a precursor chemical compound, into injection loop of a high performance liquid chromatograph (hplc); injecting radiolabeling reagent into loop to react and form radiolabeled compound, isolating |
| 06/15/2004 | CA2086426C Process for the preparation of transition metal nitrido complexes |
| 06/03/2004 | WO2004046066A1 Method for deuteration or tritiation of heterocyclic ring |
| 06/03/2004 | CA2506010A1 A method for deuteration of a heterocyclic ring |
| 05/27/2004 | WO2004043496A1 Fluorquinolines labelled with fluorine-18 |
| 05/19/2004 | EP1418950A1 Solid-phase nucleophilic fluorination |
| 05/13/2004 | WO2004029006A3 Process for the preparation of fluorohaloalkanes |
| 05/13/2004 | US20040091422 Aminophosphinic acid derivatives were synthesized as potential inhibitors of renal dipeptidase, an enzyme overexpressed in benign and malignant colon tumors. Several compounds showed potent enzyme-inhibitory activity. These |
| 05/02/2004 | WO2004011400A1 Method of deuterating aromatic ring |
| 04/14/2004 | EP1406879A1 Novel chelating agents and conjugates thereof, their synthesis and use as diagnostic and therapeutic agents |
| 04/14/2004 | EP1406835A1 Method and apparatus for production and use of ?11 c] carbon monoxide in labeling synthesis |
| 04/08/2004 | WO2004029006A2 Process for the preparation of fluorohaloalkanes |
| 04/01/2004 | US20040062714 Synthesis of 17F labeled fluoroalkanes |
| 03/24/2004 | EP1399401A2 Solid-phase electrophilic fluorination |