| Patents for C07B 53 - Asymmetric syntheses (6,231) |
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| 07/26/2001 | CA2397644A1 Acid addition salts of imidazolidinones as reaction catalysts |
| 07/25/2001 | EP1117627A1 Transfer hydrogenation process |
| 07/24/2001 | CA2332088A1 Polymeric diphosphine ligands for homogeneously soluble hydrogenation catalysts, process for the production therof and use |
| 07/24/2001 | CA2331993A1 Molecular weight-enlarged ligands for asymmetric, homogeneously soluble hydrogenation catalysts, process for the production thereof and use |
| 07/24/2001 | CA2331872A1 Use of molecular weight-enlarged catalysts in a process for asymmetric, continuous hydrogenation, novel molecular weight-enlarged ligands and catalysts |
| 07/18/2001 | EP1115741A2 Stereoselective process for enalapril |
| 07/18/2001 | EP1115680A1 Allylic substitution reactions |
| 07/17/2001 | US6262278 Reacting water and mixture of stereoisomers of chiral cyclic substrate in the presence of non-racemic chiral catalyst to produce by kinetic resolution stereoisomerically enriched cyclic substrate or stereoisomerically enriched hydrolyzate |
| 07/12/2001 | WO2001049650A1 Novel esters derived from (rr,ss)-2-hydroxybenzoate of 3-(2-dimethylaminomethyl-1-hydroxycyclohexyl)phenyl |
| 07/12/2001 | WO2001049649A1 Process of preparing tolterodine and analogues there of as well as intermediates prepared in the process |
| 07/12/2001 | CA2395976A1 Novel esters derived from (rr,ss)-2-hydroxybenzoate of 3-(2-dimethylaminomethyl-1-hydroxycyclohexyl)phenyl |
| 07/12/2001 | CA2392832A1 Process of preparing tolterodine and analogues there of as well as intermediates prepared in the process |
| 07/11/2001 | EP1114022A1 Process for producing stereoselective nitro compounds |
| 07/11/2001 | EP0821679B1 Asymmetric epoxides, their synthesis and use |
| 07/10/2001 | US6258975 Process for producing optically active 2-hydroxy-4-arylbutyric acid or its ester |
| 07/10/2001 | US6258967 Reacting zinc halide with orgaometallic compounds |
| 07/05/2001 | WO2001047940A1 Benzophenone glycopyranosides, preparation and therapeutic use |
| 07/05/2001 | CA2395561A1 Benzophenone glycopyranosides, preparation and therapeutic use |
| 07/04/2001 | EP1112999A2 Phosphine reduction of azides to amines |
| 07/04/2001 | EP1112240A1 The addition of oxygen nucleophiles to vinyl epoxides |
| 07/04/2001 | EP0748326B1 Optically active diphosphines and method for preparing same by resolution of the racemic mixture |
| 07/03/2001 | US6255493 Transition metal-catalyzed reactions based on chiral amine oxazolinyl ligands |
| 06/28/2001 | WO2001046131A1 Method for making 24(s)-hydroxyvitamin d¿2? |
| 06/28/2001 | WO2001046098A1 1,2-bis(methyl(1,1,3,3-tetramethylbutyl)-phosphino)ethane, process for the preparation thereof, transition metal complexes containing the same as the ligand and uses thereof |
| 06/28/2001 | WO2001045484A2 An improved process for preparing simvastatin |
| 06/28/2001 | WO2000068181A3 Process for preparing (1r,2s,4r) -(-)-2-[(2'- {n,n-dimethylamino} -ethoxy)] -2-[phenyl] -1,7,7-tri- [methyl] -bicyclo [2.2.1] heptane and pharmaceutically acceptable acid addition salts thereof |
| 06/28/2001 | DE10063410A1 New optically active dioxabicyclo-octen-2-one derivatives, useful as intermediates, e.g. for prostaglandins, and their intermediates |
| 06/28/2001 | CA2438477A1 An improved process for preparing simvastatin |
| 06/28/2001 | CA2394624A1 Method for making 24(s)-hydroxyvitamin d2 |
| 06/27/2001 | EP1109819A1 Ferrocene-based diphosphonites for asymmetrical catalysis |
| 06/27/2001 | EP1109777A1 N-hydroxyacylamino compounds, process for their preparation and pharmaceutical compositions containing them |
| 06/27/2001 | EP0855935B1 Chiral solid catalyst, its preparation and its use for the production of substantially enantiomerically pure products |
| 06/27/2001 | CN1301267A Production of optically active phospholanes |
| 06/27/2001 | CN1067681C Asymmetric synthesis of (S)-(+)-N,N-dimethyl-3-(1-naphthyloxyradical)-3-(2-thienyl) propylamine |
| 06/26/2001 | US6251642 Enzymatically converting amylopectin to alpha-(1,4)-linked oligosaccharide, oxidizing basic anion exchange resin to (s)-3,4-dihydroxybutyric acid, esterifying with alcohol and acid catalyst, then cyclizing with acid catalyst |
| 06/21/2001 | WO2000009483A3 Process and intermediates for production of donepezil and related compounds |
| 06/20/2001 | EP1107936A1 Copper-catalysed enantioselective allylic substitution reactions |
| 06/19/2001 | US6248889 Process for converting an alcohol to the corresponding fluoride |
| 06/14/2001 | WO2001042190A1 Method for the stereoselective synthesis of cyclic amino acids |
| 06/14/2001 | WO2001042173A2 Method for the preparation of enantiomerically enriched compounds |
| 06/14/2001 | CA2392761A1 Method for the stereoselective synthesis of cyclic amino acids |
| 06/13/2001 | EP1105400A1 Asymmetric catalysis based on chiral phospholanes |
| 06/13/2001 | EP1105385A2 Water-dispersible or water-soluble d-tocotrienol compounds and methods for making therefor |
| 06/13/2001 | EP1105371A2 Novel aryl sulphonamide amino acid esters and analogues |
| 06/13/2001 | DE19956414A1 Verfahren zur Herstellung von chiralen Aminen durch homogen katalysierte asymmetrische Hydrierung von Enaminen A process for the preparation of chiral amines by homogeneously catalyzed asymmetric hydrogenation of enamines |
| 06/13/2001 | CN1298868A Phosphine reduction method for converting azide into amide |
| 06/07/2001 | WO2001040153A1 PROCESS FOR PREPARING OPTICALLY ACTIVE α-HYDROXY ACIDS AND DERIVATIVES THEREOF |
| 06/07/2001 | WO2001039884A2 Chiral catalysts for asymmetric acylation and related transformations |
| 06/07/2001 | CA2390815A1 Process for preparing optically active .alpha.-hydroxy acids and derivatives thereof |
| 06/06/2001 | EP1104395A1 Stereoselective ring opening reactions |
| 06/05/2001 | US6242386 Drugs formed by hydrolysis of camphor in the presence of metallorganic compounds and basic salts |
| 05/30/2001 | EP1103536A1 Process for the preparation of chiral amines by asymmetric hydrogenation of enamines |
| 05/30/2001 | EP1102744A1 Novel method for preparing optically active alpha-aminonitriles |
| 05/25/2001 | WO2001036359A1 Optically active fluorinated binaphthol derivative |
| 05/23/2001 | EP1100954A1 Continuous process for preparing optically pure (s)-3,4-dihydroxybutyric acid derivatives |
| 05/23/2001 | EP1100953A1 CONTINUOUS PROCESS FOR PREPARING OPTICALLY PURE ($i(S))-3-HYDROXY-GAMA-BUTYROLACTONE |
| 05/23/2001 | EP1100952A1 Process for preparing optically pure (s)-3,4-dihydroxybutyric acid derivatives |
| 05/23/2001 | EP1100951A1 PROCESS FOR PREPARING OPTICALLY PURE ($i(S))-3-HYDROXY-GAMA-BUTYROLACTONE |
| 05/23/2001 | EP1100948A1 Process for preparing alpha-(1,4) linked oligosaccharide |
| 05/23/2001 | EP1100769A1 Aminomethylcarboxylic acid derivatives |
| 05/23/2001 | EP1100768A2 Process for the preparation of r-(-)-carnitine |
| 05/22/2001 | US6235877 Peptido-mimetic compounds containing RGD sequence useful as integrin inhibitors |
| 05/17/2001 | WO2001034612A2 Chiral phosphines, transition metal complexes thereof and uses thereof in asymmetric reactions |
| 05/17/2001 | US20010001309 For treating pathologies related to altered alpha v beta 3 integrin-mediated cell attachment, in particular wherein inhibition of angiogenesis is desired, for example in tumors, also associated with metastasis |
| 05/17/2001 | CA2390998A1 Chiral phosphines, transition metal complexes thereof and uses thereof in asymmetric reactions |
| 05/09/2001 | EP1097116A1 Asymmetric metathesis reactions involving achiral and meso substrates |
| 05/08/2001 | US6229042 Intermediates for the synthesis of enantiomerically pure alpha-lipoic acid; said hydrogenation includes presence of ruthenium-phosphine complex |
| 05/03/2001 | WO2001001569A3 Process for preparing (-)-(1s,4r) n-protected 4-amino-2-cyclopentene-1-carboxylate esters |
| 05/02/2001 | EP1095946A1 Optically active diphosphine compound, production intermediates therefor, transition metal complex containing the compound as ligand and asymmetric hydrogenation catalyst containing the complex |
| 05/02/2001 | EP1095012A1 Novel salts of n-tert-butylhydroxylamine |
| 05/02/2001 | CN1293646A Method for separating diphosphine diastereiosomers |
| 05/01/2001 | US6225341 For inhibiting neuraminidase; for therapy and prophylaxis of virus infection |
| 04/26/2001 | WO2001028990A2 Methods of asymmetrically synthesizing enantiomers of casodex, its derivatives and intermediates thereof |
| 04/26/2001 | CA2387570A1 Methods of asymmetrically synthesizing enantiomers of casodex, its derivatives and intermediates thereof |
| 04/24/2001 | US6222072 Racting imine with hydride reagent in presence of optically active metal compound, wherein hydride reagent is a metal hydride, reagent that undergoes metal exchange, metal trialkoxy hydride complex or metal(tricarboxylic acid)hydride |
| 04/24/2001 | US6222039 Reacting lactone compound containing nitrogen heterocycle with cyclic amine; oxidizing to form carboxylic acid group; introducing hydroxylamine group at hydroxyl of carboxylic acid group |
| 04/24/2001 | US6221639 Process for preparing optically pure(S)-3,4-dihydroxybutyric acid derivatives |
| 04/24/2001 | CA2025458C Iridium complexes, process for their preparation and their use |
| 04/19/2001 | WO2000073274A3 Substituted phenylcyclohexane carboxylic acid amides and their use as adenosine uptake inhibitors |
| 04/18/2001 | EP1091953A1 Novel benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake |
| 04/17/2001 | US6218585 Maintaining borohydride concentration before reduction with borane-tetrahydrofuran complex |
| 04/17/2001 | US6218575 Process for preparing adrenaline |
| 04/12/2001 | WO2001025486A1 Methods for identifying rna binding compounds |
| 04/12/2001 | WO2001025215A2 Method for selectively dissociating cyclic carboxylic acid anhydrides |
| 04/12/2001 | WO2001025188A1 Novel carbamates and ureas |
| 04/12/2001 | WO2001025183A1 Process for preparing carboxylic esters of optically active 1-perfluoroalkylated alcohols, optically active 1-perfluoroalkylated alcohols and process for the preparation thereof |
| 04/12/2001 | DE19947953A1 Verfahren zur selektiven Spaltung cyclischer Carbonsäureanhydride Process for the selective cleavage of cyclic anhydrides |
| 04/12/2001 | CA2386540A1 Novel carbamates and ureas |
| 04/12/2001 | CA2386239A1 Methods for identifying rna binding compounds |
| 04/05/2001 | WO2001023088A1 Catalyst for asymmetric transfer hydrogenation |
| 04/05/2001 | DE19947505A1 Verfahren zur Herstellung organischer Verbindungen im Membranreaktor Process for the preparation of organic compounds in the membrane reactor |
| 04/05/2001 | DE19945737A1 Verfahren zur Hydrierung von organischen Verbindungen enthaltend mindestens eine CC-Doppelbindung A process for the hydrogenation of organic compounds containing at least one CC double bond |
| 04/04/2001 | EP1088587A2 Process for the production of organic compounds in a membrane reactor |
| 04/03/2001 | US6211370 Asymmetric cycloaddition reactions |
| 03/29/2001 | WO2001021625A1 Chiral phosphines, transition metal complexes thereof and uses thereof in asymmetric reactions |
| 03/29/2001 | WO2001021559A1 Method for hydrogenating organic compounds containing at least one c-c double bond |
| 03/27/2001 | US6207868 Based on chiral bidentate phosphine ligands with cyclic ring structures to restrict conformational flexibility, asymmetric synthesis of alcohols by enantioselective hydrogenation of ketones catalyzed by the chiral ligands |
| 03/22/2001 | WO2001019833A1 Thienoisoxazolyl- and thienylpyrrazolyl-phenoxy substituted propyl derivatives useful as d4 antagonists |
| 03/22/2001 | WO2001019787A1 OPTICALLY ACTIVE α-AMINONITRILE AND PROCESS FOR PRODUCING α-AMINO ACID |
| 03/22/2001 | WO2001019761A2 Asymmetric 1,4-reductions of and 1,4-additions to enoates and related systems |