Patents for C07B 53 - Asymmetric syntheses (6,231)
10/2001
10/24/2001EP1147075A1 Method for producing l-phenylephrine hydrochloride
10/23/2001US6307067 Palladium and boron co-catalyzed addition of oxygen nucleophiles to vinyl epoxides
10/23/2001US6307057 Catalyze enantioselective reactions, e.g., diels-alder reactions
10/18/2001US20010031892 Stereoselective synthesis starting from (S)-3-hydroxy-4-butyrolactone
10/18/2001US20010031875 Optically active ionic liquid
10/18/2001US20010031858 Coupling of 2-(2-acetylamino-3-(4-amidinophenyl) propionylamino)-2-cyclohexylacetic acid with a 3-(2-amino-2-carbamoylethyl)-1-methylpyridinium salt or a salt thereof; anticoagulants
10/17/2001EP1146047A1 3,5-Dioxa-8-aza-tricyclo(5.2.1.00,0)decane-9-methanols, their metal complexes and enantioselective hydrogenation processes
10/17/2001EP1146036A2 Tamiflu, Gallocarboxylic acid approach
10/17/2001EP1144375A2 Synthesis of oligoketides
10/17/2001EP1144367A1 Alpha-substitution of unprotected beta-amino ester compounds
10/17/2001EP0641330B1 Gaba and l-glutamic acid analogs for antiseizure treatment
10/17/2001CN1317481A Method for preparing 4,5-diamino shikimic acid derivative
10/16/2001US6303796 Chemical intermediates; optically active compounds useful as optical resolution agents; metal-coordinated compounds useful as asymmetric catalysts
10/11/2001WO2001074828A1 Water soluble chiral diphosphines
10/11/2001WO2001074741A2 Catalytic asymmetric desymmetrization of meso compounds
10/11/2001CA2405535A1 Catalytic asymmetric desymmetrization of meso compounds
10/10/2001EP1141374A2 Method for producing optically active 1-amino-4-(hydroxymethyl)-cyclopent-2-ene derivatives
10/10/2001EP1141373A1 Method for the enantioselective reduction of 3,5-dioxocarboxylic acids, their salts and their esters
10/10/2001EP1140956A1 Ligands and complexes for enantioselective hydrogenation
10/10/2001EP1140874A1 Stereoselective synthesis of oxazoline derivative
10/10/2001EP1140842A1 Alkyl esters of 3-(3,4-dihalogenophenyl)-2,6-dioxopiperidine-3-propionic acid useful as intermediates
10/10/2001EP1140818A1 Amidomalonamides and their use as inhibitors of matrix metalloproteinase
10/10/2001EP1140815A1 Novel thio-aminotetralin compounds useful in pain management
10/10/2001EP1140794A1 Novel method for preparing chiral amino acids
10/10/2001EP1140790A1 Novel oxo-aminotetralin compounds useful in pain management
10/10/2001EP1140769A1 Method for producing glyoxylic acid esters or the hydrates thereof
10/10/2001EP1140745A1 Colchinol derivatives as vascular damaging agents
10/04/2001WO2001034612A3 Chiral phosphines, transition metal complexes thereof and uses thereof in asymmetric reactions
10/03/2001CN1316013A Process for preparing optically pure (S)-3,4-dihydroxybutyric acid derivatives
10/03/2001CN1316012A Process for preparing optically pure (S)-3-hydroxy-gamma-butyrolactone
10/03/2001CN1316011A Continuous process for preparing optically pure (S)-3,4-dihydroxybutyric acid derivatives
10/03/2001CN1316010A Continuous process for preparing optically pure (S)-3-hydroxy-gamma-butyrolactone
10/03/2001CN1316008A Process for preparing alpha-(1,4) linked oligosaccharide
10/03/2001CN1315319A Process for preparing ethyl-sulfonylpiperidine derivatives
10/03/2001CN1072227C Optically active diphosphine ligands
09/2001
09/26/2001EP1136475A1 Piperidine and piperazine compounds for use in the treatment of Alzheimer
09/26/2001EP0900214B1 Process for preparation of pyrimidine derivatives
09/26/2001CN1314880A Novel method for preparing optically active alpha-aminonitriles
09/20/2001WO2001068637A2 Method for the preparation of tetrahydrobenzothiepines
09/20/2001WO2001068254A1 Chiral lead catalyst and method of asymmetric aldol reaction
09/19/2001EP1134226A2 Process for producing an optically active ruthenium-phosphine complex and process for producing an optically active alcohol by using the complex
09/13/2001WO2001066509A1 PROCESS FOR PRODUCING α,α-DIFLUORO- β -KETOESTER
09/13/2001WO2000040547A8 α-SUBSTITUTION OF UNPROTECTED β-AMINO ESTER COMPOUNDS
09/12/2001EP1131323A1 Synthesis of acyclic nucleoside derivatives
09/12/2001EP1131313A1 Enantioselective alkylation of tricyclic compounds
09/12/2001EP1131279A1 Industrial process for the production of l-carnitine
09/12/2001EP1131278A1 Process for production of esters
09/12/2001EP1131274A2 Methods for producing chiral aldehydes
09/12/2001EP1131270A1 Process for converting an alcohol to the corresponding fluoride
09/12/2001CN1312805A Benzothiepines having activity as inhibitors of ileal bile acid transport and taurocholate uptake
09/11/2001US6288279 Their preparation process and their use in asymmetrical catalysis. rearranging a diphosphole, reacting the diphosphole with an acetylenic compound to form the diphosphine
09/11/2001US6288272 Reaction of enantiomorphs of amylopectin to linked oligosaccharide, oxidation of oligosaccharide, esterification with alcohol
09/11/2001US6288247 Catalytic multistage process forming a racemic mixture of compounds
09/07/2001WO2001028990A3 Methods of asymmetrically synthesizing enantiomers of casodex, its derivatives and intermediates thereof
09/05/2001EP1129073A2 Process and intermediates for production of donepezil and related compounds
09/04/2001US6284925 Hydrogenation catalysts for hydrogenation of double bonds or imine groups
08/2001
08/29/2001EP1127886A1 Synthesis of 3,6-dialkyl-5,6-dihydro-4-hydroxy-2H-pyran-2one
08/29/2001EP1127872A1 Tamiflu via Diels-Alder
08/29/2001EP1127871A1 New esters derived from substituted phenyl-cyclohexyl compounds
08/29/2001EP1127616A1 Catalyst for asymmetric epoxidation of enones and process for producing optically active epoxide employing it
08/29/2001EP1127061A1 Chiral ligands for asymmetric catalysis
08/29/2001EP1127043A1 Stereoselective process for preparing (cyclo)alkyl phenylglycolic acids
08/29/2001CN1310170A Process for producing 4,5-diamino shikimic acid derivative
08/28/2001USRE37344 For forming complexes with iridium or rhodium which are used for enantioselective hydrogenation catalysts for homogeneous hydrogenation of prochiral unsaturated compounds
08/28/2001US6281390 Chiral diphenyldiphosphines and d-8 metal complexes thereof
08/28/2001US6281379 Halogenating g-amino-b-keto sulfoxide; reacting with acid and alcohol; forming b-amino-a-hydroxy acid compounds
08/23/2001WO2001060777A1 PROCESS FOR OBTAINING 1, 2, 3, 5, 6, 7, 8, 8A-OLTAHYDRO-1, 2, 8, 8TETRAMETHYLNAPHTHALEN-2-YL!ETAN-1-ONE
08/23/2001US20010016669 Novel process and intermediates
08/22/2001EP1124833A1 Diphosphines
08/22/2001CN1309632A Salts of N-tert-butylhydroxylamine
08/22/2001CN1309631A Aminomethylcarboxylic acid derivs
08/21/2001US6278024 As catalysts for assymetric synthesis
08/21/2001US6277997 Hydrogenating asymmetrically 2,5-dihydrofuran derivative in presence of catalyst comprising metal diphosphine complex to produce lactone derivative
08/16/2001WO2001058588A1 Chiral ferrocene phosphines and their use in asymmetric catalytic reactions
08/16/2001WO2000055124A3 Novel compounds and compositions as protease inhibitors
08/16/2001WO2000047551A3 Inhibitors of aspartyl protease
08/16/2001CA2400183A1 Chiral ferrocene phosphines and their use in asymmetric catalytic reactions
08/16/2001CA2399515A1 Process for the preparation of (r)-2-bromo-3-phenyl-propionic acid
08/15/2001CN1069624C Production of derivatives of 4a,5,9,10,11,12,-bexahydro-6H-benzofuro[3a,3,2-ef][2] benzazepine
08/14/2001US6274758 Enantiomorph selectivity
08/09/2001WO2001057232A1 Method for the enzymatic resolution of the racemates of aminomethyl-aryl-cyclohexanol derivatives
08/09/2001DE10004926A1 Verfahren zur enzymatischen Racematspaltung von Aminomethyl-Aryl-Cyclohexanol-Derivaten A process for the enzymatic resolution of aminomethyl-aryl-cyclohexanol derivatives
08/07/2001US6271388 Process for producing oxazolidin-2-one derivative
08/02/2001WO2001055175A2 Process for the preparation of acetyl-amidiniophenylalanyl-cyclohexylglycyl-pyridinioalaninamides
08/02/2001WO2001055097A1 Preparation of nitrogen mustard derivatives
08/02/2001WO2001055090A1 Asymmetric synthesis of pregabalin
08/02/2001WO2001055060A2 Chiral ionic liquids
08/02/2001US20010011074 Antiischemic agents; cardiovascular disorders
08/02/2001DE10003708A1 Neuartige chirale ionische Flüssigkeiten und Verfahren zu ihrer Darstellung in enantiomerenreiner oder enantiomerenangereicherter Form Novel chiral ionic liquids and methods for their representation in enantiomerically pure or enantiomerically enriched form
08/01/2001EP1120162A2 Use of catalysts with a higher molecular weight in an asymmetrical continous hydration reaction, ligands and catalysts
08/01/2001EP1120161A1 High molecular weight ligands for homogeneously soluble asymmetric hydrogenation catalysts, process for their preparation and use thereof
08/01/2001EP1120160A1 Polymeric diphosphine ligands for homogeneously soluble hydrogenation catalysts, process for their preparation and use thereof
08/01/2001EP0941228B1 PROCESS FOR PREPARING MeO-Peg-PROTECTED DIHYDROQUININE OR DIHYDROQUINIDINE DERIVATIVES, DIHYDROQUININE OR DIHYDROQUINIDINE DERIVATIVES AND THEIR USE
07/2001
07/26/2001WO2001053269A1 Acid addition salts of imidazolidinones as reaction catalysts
07/26/2001WO2001053241A1 Chemical transformation of substrates using nonmetallic, organic catalyst compositions
07/26/2001WO2000068183A3 High purity (1r,2s,4r)-(-)-2-[(2'-{n,n-dimethylamino}-ethoxy)]-2-[phenyl]-1,7,7-tri-[methyl]-bicyclo[2.2.1]heptane and pharmaceutically acceptable acid addition salts thereof, process for the preparation of these compounds and medicaments containing them
07/26/2001DE10002976A1 Molekulargewichtsvergrößerte Liganden für asymmetrische homogen lösliche Hydrierkatalysatoren, Verfahren zu deren Herstellung und Verwendung Molecular weight-ligands for asymmetric homogeneous hydrogenation catalysts soluble, to processes for their preparation and use
07/26/2001DE10002975A1 Verwendung von molekulargewichtsvergrößerten Katalysatoren in einem Verfahren zur asymmetrischen kontinuierlichen Hydrierung, neue molekulargewichtsvergrößerte Liganden und Katalysatoren Use of molecular weight-catalysts in a process for the asymmetric hydrogenation continuous, molecular weight-new ligands and catalysts
07/26/2001DE10002973A1 Polymere Diphosphinliganden für homogen lösliche Hydrierkatalysatoren, Verfahren zu deren Herstellung und Verwendung Diphosphine ligands for homogeneous hydrogenation catalysts soluble polymers, processes for their preparation and use
07/26/2001CA2397650A1 Chemical transformation of substrates using nonmetallic, organic catalyst compositions
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