Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
10/2000
10/17/2000US6133296 Substituted pyridyl keto enols
10/17/2000CA2202031C Condensed indan derivatives and salts thereof
10/12/2000WO2000059909A1 Heterocyclic compounds having affinities for serotonin receptors
10/12/2000WO2000059884A1 Pharmaceutically active compounds and methods of use thereof
10/12/2000WO2000059510A1 Aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000WO2000059498A1 Pyrrolidine modulators of chemokine receptor activity
10/12/2000CA2484282A1 Pyrimidine derivatives intermediates for producing aminopyrimidines as sorbitol dehydrogenase inhibitors
10/12/2000CA2369238A1 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/12/2000CA2366858A1 Sorbitol dehydrogenase inhibitors
10/12/2000CA2361734A1 Pharmaceutically active compounds and methods of use thereof
10/12/2000CA2268590A1 Ion channel modulating compounds and uses thereof
10/11/2000EP1043326A1 Steroid receptor modulator compounds and methods
10/11/2000EP1043325A1 Steroid receptor modulator compounds and methods
10/11/2000EP1043315A1 Steroid receptor modulator compounds and methods
10/11/2000EP1043314A1 Novel dihydropyridine derivative
10/11/2000EP1042329A1 Novel farnesyl transferase inhibitors, preparation, pharmaceutical, compositions containing them and use for preparing medicines
10/11/2000EP1042326A1 Novel acronycine derivatives, preparation method and pharmaceutical compositions
10/11/2000EP1042322A1 Kv2.1 ANTAGONISTS
10/11/2000EP1042320A1 New compounds which are p2-purinoceptor 7-transmembrane (tm) g-protein coupled receptor antagonists
10/11/2000EP1042295A1 4-hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
10/11/2000EP1042294A1 Heterocyclic cytotoxic agents
10/11/2000EP1042291A1 Aryl-substituted pyridylalkane, alkene, and alkine carboxamides useful as cytostatic and immunosuppressive agents
10/11/2000EP1042289A1 Indole]naphthopyrans, preparation, compositions and (co)polymer matrices containing them, synthesis intermediates
10/11/2000EP1042288A1 Tripeptidyl peptidase inhibitors
10/11/2000CN1057292C Dicyclic compound, medicinal composition containing same and use thereof
10/10/2000US6130338 Method of producing pyrrolidine derivatives
10/10/2000US6130229 Tricyclic compounds having activity as RAS-FPT inhibitors
10/10/2000US6130227 7-Substituted camptothecin derivatives and methods for inhibiting the growth of tumor cells therewith
10/10/2000US6130101 Fluorescent probes for use in biological samples
10/10/2000US6129119 Flexible tube for lining pipes and ducts as well as method and an apparatus for manufacturing thereof
10/05/2000WO2000058406A1 4,7-dichlororhodamine dyes useful as molecular probes
10/05/2000WO2000058286A2 Method of producing heterocyclic carbamates from aza-heterocyclic compounds and carbon dioxide
10/05/2000WO2000057874A1 A process for the preparation of aziridinyl epothilones from oxiranyl epothilones
10/05/2000WO2000042026B1 Non-peptide glp-1 agonists
10/05/2000WO1999053951A9 Terminally-branched polymeric linkers and polymeric conjugates containing the same
10/05/2000CA2368658A1 A process for the preparation of aziridinyl epothilones from oxiranyl epothilones
10/05/2000CA2361019A1 Process for the preparation of heterocyclic carbamates from aza-heterocycles and carbon dioxide
10/04/2000EP1041074A1 Light-sensitive 4-cyanocoumarin derivatives
10/04/2000EP1041071A1 Methods for the preparation of coumarine derivatives
10/04/2000EP1041066A1 Steroid receptor modulator compounds and methods
10/04/2000EP1040098A1 Integrin receptor antagonists
10/04/2000CN1268948A Optically pure camptothecin analogues, optically pure synthessi intermdidate and method for preparing same
10/04/2000CN1057086C Phenylsulfonyl ureas, process for preparing same, and use as herbicide, herbicide composition contg. same
10/04/2000CN1057083C Tricyclic 1-aminoethylpyrrol derivative
10/03/2000US6127547 Halobenzimidazoles and their use as microbicides
10/03/2000US6127375 A 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthiones for treating viral infection
10/03/2000US6127355 High molecular weight polymer-based prodrugs
09/2000
09/28/2000WO2000056728A1 Tetrahydropyran derivatives and their use as therapeutic agents
09/28/2000WO2000056727A1 Tetrahydropyran derivatives and their use as therapeutic agents
09/28/2000WO2000056337A1 Agents for relieving side effects
09/28/2000WO2000033839B1 Non-peptide antagonists of glp-1 receptor and methods of use
09/28/2000DE19913483A1 Verfahren zur Herstellung von Heterocyclischen Carbamaten aus Aza-Heterocyclen und Kohlendioxid Process for the preparation of heterocyclic carbamates from carbon dioxide and aza heterocycles
09/28/2000CA2367985A1 Tetrahydropyran derivatives and their use as therapeutic agents
09/27/2000EP1038873A2 Benzo(3,4)cyclobuta(1,2-c)pyrrole derivatives as inhibitors of serotonine reuptake
09/27/2000EP1038868A2 Sulfonamides as antiviral agents
09/27/2000EP1037892A1 Piperidine derivatives
09/27/2000EP1037878A2 Metabotropic glutamate receptor antagonists for treating central nervous system diseases
09/27/2000EP1037876A1 Biphenyl derivatives as pharmaceuticals
09/27/2000CN1268133A 2-Aminopyridines containing fused ring substituents as NOS inhibitors
09/26/2000US6124453 Sanglifehrins, immunosuppressant and antiinflammatory compounds
09/26/2000US6124316 Compounds which are specific antagonists of the human NK3 receptor and their use as medicinal products and diagnostic tools
09/26/2000US6124310 Enediyne compounds
09/26/2000US6124306 Treating human immunodeficiency virus infections
09/26/2000US6124292 Antitumor agents
09/26/2000US6123943 NF-KB activity inhibitor
09/21/2000WO2000055158A1 Tricyclic benzoylpyrazole derivatives used as a herbicide
09/21/2000DE19912638A1 Naphthylcarbonsäureamid-substituierte Sulfonamide Naphthylcarbonsäureamid-substituted sulfonamides
09/21/2000CA2367672A1 Tricyclic benzoylpyrazole derivatives used as a herbicide
09/20/2000EP1036076A1 Novel compounds
09/20/2000EP1036072A1 Thrombin receptor antagonists
09/20/2000EP1035848A1 Substituted alkanohydroxamic acids and method of reducing tnf-alpha levels
09/20/2000EP1035824A1 A process for the preparation of ring-opened epothilone intermediates which are useful for the preparation of epothilone analogs
09/20/2000EP1004140A4 A well to substrate photodiode for use in a cmos sensor on a salicide process
09/20/2000CN1056605C Compounds as selective human NK 3-receptor antagonists and their use
09/19/2000US6121451 Anticancer drugs
09/19/2000US6121450 Non-steroidal compounds which are high affinity, high selectivity modulators for steroid receptors
09/19/2000US6121284 Specified 1-(alkyl or cycloalkyl)-2-methyl-3-(alkoxycarbonyl)-4-(substituted pyridyl or aryl)-5-oxo-1,4,5,6,7,8-hexahydroquinoline compounds; treating sickle cell anemia, psychoses, depression
09/19/2000US6121279 Phosphodiesterase inhibitor for treating respiratory system disorders
09/19/2000US6121278 Di-n-heterocyclic compounds, methods, and compositions for inhibiting parp activity
09/19/2000US6120793 Transdermal administering
09/14/2000WO2000053614A1 Method for producing glyco-conjugates of 20(s)-camptothecin
09/14/2000WO2000053608A1 Pyridopyranoazepine derivatives, preparation and therapeutic use
09/14/2000WO2000053607A1 Camptothecin derivatives having antitumor activity
09/14/2000WO2000053606A1 Pyridoxal analogues for vitamin b-6 disorders
09/14/2000WO2000053598A1 Pyran derivatives
09/14/2000CA2366632A1 Method for producing glyco-conjugates of 20(s)-camptothecin
09/14/2000CA2366602A1 Pyridoxal analogues for vitamin b-6 disorders
09/13/2000EP1035114A2 Nitrogen-heterocyclic compounds and process for production thereof
09/13/2000EP1034221A1 Dibenzorhodamine dyes useful as fluorescent labelling agents
09/13/2000EP1034167A1 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
09/13/2000CN1266435A Process for preparing and purifying 9-nitro-20-camptothecin
09/13/2000CN1056374C Tricyclic diazepine vasopression antagonists
09/08/2000WO2000052005A1 Febrifugine and isofebrifugine and processes for the preparation of both
09/07/2000DE19909979A1 Verfahren zur Herstellung von Glycokonjugaten von 20(S)-Camptothecin Process for the preparation of glycoconjugates of 20 (S) -camptothecin
09/06/2000EP1033369A1 5H-PYRANO [2,3-d:6,5-d']DIPYRIMIDINE DERIVATIVES HAVING AN ANTIBACTERIAL, ANTIVIRAL AND IMMUNO-MODULATING ACTIVITY
09/06/2000CN1265661A N-acylamino acid amide compounds and intermediates for preparation thereof
09/06/2000CN1265590A Substituted alkanohydroxamic acid and method of reducing TNF 'alpha' levels
09/05/2000US6114529 Useful for preparing camptothecin derivatives having antitumor activities
09/05/2000US6114374 2-and 2,5-substituted phenylketoenols
09/05/2000US6114360 Pyrrole compounds