Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
07/2000
07/20/2000WO2000042019A1 6-arylphenanthridines with pde-iv inhibiting activity
07/20/2000WO2000029406A3 Novel isoxazoline fibrinogen receptor antagonists
07/20/2000CA2372197A1 Functionalized heterocycles as chemokine receptor modulators
07/20/2000CA2359990A1 Novel aralkyl amines of spirofuropyridines useful in therapy
07/20/2000CA2359952A1 Triazole compounds with dopamine-d3-receptor affinity
07/20/2000CA2359942A1 Triazole compounds with dopamine-d3-receptor affinity
07/20/2000CA2359416A1 6-arylphenanthridines with pde-iv inhibiting activity
07/19/2000EP1020470A2 Galanthamine derivatives, a process for their preparation and their use as medicaments
07/19/2000EP1020469A2 Galanthamine derivatives, a process for their preparation and their use as medicaments
07/19/2000EP1020468A2 Methods and intermediates for the asymmetric synthesis of camptothecin and camptothecin analogs
07/19/2000EP1020467A1 N-acylamino acid amide compounds and intermediates for preparation thereof
07/19/2000EP1020462A1 Heterocyclic compounds and antitumor agent containing the same as active ingredient
07/19/2000EP1020445A1 Fused pyridine derivatives
07/19/2000EP1019412A1 Biphenyl(thio)amide and biphenylethan(thi)one derivatives, their preparation and their use as 5-ht 1d? receptor antagonists
07/19/2000EP1019410A1 Spiro-piperidine derivatives and their use as tachykinin antagonists
07/19/2000EP1019409A1 Poly(adp-ribose) polymerase ("parp") inhibitors, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damage
07/19/2000EP1019408A1 1,2,3,4-TETRAHYDRO-BENZOFURO 3,2-c]PYRIDINE DERIVATIVES--
07/19/2000EP1019389A2 Epothilone derivatives
07/19/2000EP1019385A1 Aminoaryl oxazolidinone n-oxides
07/19/2000EP1019052A1 Alpha 1a adrenergic receptor antagonists
07/19/2000EP0760819B1 Tricyclic dicarbonyl derivatives
07/19/2000EP0667861B1 2-trifluoromethyl benzimidazole derivatives, their preparation and their use as pesticides
07/19/2000CN1260791A 3-benzylpiperidine
07/18/2000US6090954 Benzimidazole derivatives
07/18/2000US6090837 Substituted hydrochromenopyrroles
07/18/2000US6090820 Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones
07/18/2000US6090818 Indolin-2-one derivatives, method for preparing them and pharmaceutical compositions containing them
07/18/2000US6090808 Dimeric piperidine, tetrahydropyridine and piperazine derivatives
07/13/2000WO2000040561A1 Quinolinecarboxamides as antiviral agents
07/13/2000WO2000040539A1 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors for the treatment of respiratory diseases
07/13/2000WO2000024741A3 Dihydropyridine compounds and their use as potassium channel openers
07/13/2000CA2356053A1 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors for the treatment of respiratory diseases
07/13/2000CA2353636A1 Quinolinecarboxamides as antiviral agents
07/12/2000EP1018514A1 NF-$g(k)B INHIBITORS CONTAINING INDAN DERIVATIVES AS THE ACTIVE INGREDIENT
07/12/2000EP1017676A1 Method for the synthesis of quinoline derivatives
07/12/2000EP1017675A1 Highly lipophilic camptothecin derivatives
07/12/2000EP1017399A1 Camptothecin analogs and methods of preparation thereof
07/12/2000EP1017395A1 Method for treating premenstrual or late luteal phase syndrome
07/12/2000EP0877734B1 Quinoline and quinazoline compounds useful in therapy
07/12/2000EP0731802B1 N-substituted azabicycloalkane derivatives as neuroleptics etc.
07/12/2000EP0642502B1 Fungicidal imidazolinones
07/12/2000CN1259938A Crambescidin compound
07/11/2000US6087510 Method of use of imidazolium cations
07/11/2000US6087495 Salt formation by seeding
07/11/2000US6087370 Methods of treatment using lamellarin-class alkaloids
07/11/2000US6087369 Indole derivatives, process for producing the same and medicinal uses of the same
07/11/2000CA2208569C Novel processes for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof
07/06/2000WO2000039108A1 Thrombin or factor xa inhibitors
07/06/2000WO2000039102A1 THROMBIN OR FACTOR Xa INHIBITORS
07/06/2000WO2000039087A2 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors
07/06/2000WO2000039081A2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
07/06/2000WO2000038720A1 Remedies for pain
07/06/2000WO2000038687A1 Protease inhibitors
07/06/2000WO2000038683A1 THROMBIN OR FACTOR Xa INHIBITORS
07/06/2000CA2358047A1 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds
07/06/2000CA2356671A1 Protease inhibitors
07/06/2000CA2356269A1 Pain control agent
07/06/2000CA2349557A1 Thrombin or factor xa inhibitors
07/06/2000CA2348740A1 Thrombin or factor xa inhibitors
07/06/2000CA2320730A1 Thrombin or factor xa inhibitors
07/05/2000EP1015469A2 Bi- and tri-cyclic nucleoside, nucleotide and oligonucleoide analogues
07/05/2000EP1015458A1 Furopyrrolidine derivatives and their use as serine protease inhibitors
07/05/2000EP1015457A1 1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives as ampa/kainate receptor inhibitors
07/05/2000EP1014973A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
07/05/2000EP0675889B1 Antiallergic triazolo(pyrrolo, thieno or furano)azepine derivatives
07/05/2000EP0565621B1 Method of making camptothecin and camptothecin analogs
07/05/2000CN1259125A Substituted 3-cyano quinolines
07/04/2000US6084095 Including 6-amino-4-(3-bromoanilino)pyrido(3,2-d)pyrimidine; 4-(3-bromoanilino)-6-methylaminopyrido (3,2-d)pyrimidine; and 4-(3-bromoanilino)-6-methylaminopyrido(3,2-d)pyrimidine; useful in treating proliferative diseases such as cancer
07/04/2000US6084094 Oxidative process for preparing narwedine derivatives
07/04/2000US6083956 Optically pure androgen mediator
07/04/2000CA1341044C Benzopyrido piperidine, piperidylidene and peperazine compounds, compositions, methods of manufacture and methods of use
06/2000
06/29/2000WO2000037473A1 Epothilone derivatives and their use as antitumor agents
06/29/2000WO2000037468A1 DIBENZO[a,g]QUINOLIZINIUM DERIVATIVES AND THE SALTS THEREOF
06/29/2000WO2000037466A1 BENZISOXAZOLES AND PHENONES AS α2-ANTAGONISTS
06/29/2000WO2000037456A1 Amide and urea derivatives as 5-ht reuptake inhibitors and as 5-ht1b/1d ligands
06/29/2000WO2000037450A1 NEW β-AMIDE AND β-SULFONAMIDE CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS
06/29/2000WO2000037026A1 Dihydropyrimidines and uses thereof
06/29/2000CA2355861A1 Amide and urea derivatives as 5-ht reuptake inhibitors and as 5-ht1b/1d ligands
06/29/2000CA2355848A1 Dihydropyrimidines and uses thereof
06/29/2000CA2355469A1 Dibenzo[a,g]quinolizinium derivatives and the salts thereof
06/29/2000CA2355251A1 New .beta.-amide and .beta.-sulfonamide carboxylic acid derivatives, their preparation and their use as endothelin receptor antagonists
06/28/2000EP1012145A1 Alkoxy-substituted compounds, methods, and compositions for inhibiting parp activity
06/28/2000EP1011665A1 Heterocyclic agents
06/28/2000EP0808318B1 Tricyclic substituted hexahydrobenz[e]isoindole alpha-1 adrenergic antagonists
06/27/2000US6080852 4,7-dichlororhodamine dyes
06/27/2000US6080776 Used as a microbiocide for crop protection
06/27/2000US6080754 For treatment and prophylaxis of estrogen related syndromes and disorders
06/27/2000US6080752 For treating condition which requires antagonism of a dopamine receptor such as psychtic condition
06/27/2000US6080743 2,3-dioxo-1,2,3,4-tetrahydro-quinoxalinyl derivatives
06/22/2000WO2000035924A1 Camptothecin analogs and methods of preparation thereof
06/22/2000WO2000035915A1 Piperazine derivatives
06/22/2000WO2000035907A1 Imidazolones and their use in treating benign prostatic hyperplasia and other disorders
06/22/2000CA2355202A1 Imidazolones and their use in treating benign prostatic hyperplasia and other disorders
06/22/2000CA2354875A1 Piperazine derivatives
06/21/2000EP1009739A2 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity
06/21/2000EP1009738A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
06/21/2000DE19858779A1 New 3-acylamino-propionic acid and 3-sulfonylamino-propionic acid derivatives useful as endothelin receptor antagonists in treatment of e.g. cardiovascular and renal disorders, migraine and cancer
06/21/2000CN1257506A Spiro-quinuclidine derivatives, their preparation and use
06/21/2000CN1257505A Fused dihydropyrans
06/21/2000CN1257504A Salts of aromatic sulphonic acids