Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726) |
---|
07/20/2000 | WO2000042019A1 6-arylphenanthridines with pde-iv inhibiting activity |
07/20/2000 | WO2000029406A3 Novel isoxazoline fibrinogen receptor antagonists |
07/20/2000 | CA2372197A1 Functionalized heterocycles as chemokine receptor modulators |
07/20/2000 | CA2359990A1 Novel aralkyl amines of spirofuropyridines useful in therapy |
07/20/2000 | CA2359952A1 Triazole compounds with dopamine-d3-receptor affinity |
07/20/2000 | CA2359942A1 Triazole compounds with dopamine-d3-receptor affinity |
07/20/2000 | CA2359416A1 6-arylphenanthridines with pde-iv inhibiting activity |
07/19/2000 | EP1020470A2 Galanthamine derivatives, a process for their preparation and their use as medicaments |
07/19/2000 | EP1020469A2 Galanthamine derivatives, a process for their preparation and their use as medicaments |
07/19/2000 | EP1020468A2 Methods and intermediates for the asymmetric synthesis of camptothecin and camptothecin analogs |
07/19/2000 | EP1020467A1 N-acylamino acid amide compounds and intermediates for preparation thereof |
07/19/2000 | EP1020462A1 Heterocyclic compounds and antitumor agent containing the same as active ingredient |
07/19/2000 | EP1020445A1 Fused pyridine derivatives |
07/19/2000 | EP1019412A1 Biphenyl(thio)amide and biphenylethan(thi)one derivatives, their preparation and their use as 5-ht 1d? receptor antagonists |
07/19/2000 | EP1019410A1 Spiro-piperidine derivatives and their use as tachykinin antagonists |
07/19/2000 | EP1019409A1 Poly(adp-ribose) polymerase ("parp") inhibitors, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damage |
07/19/2000 | EP1019408A1 1,2,3,4-TETRAHYDRO-BENZOFURO 3,2-c]PYRIDINE DERIVATIVES-- |
07/19/2000 | EP1019389A2 Epothilone derivatives |
07/19/2000 | EP1019385A1 Aminoaryl oxazolidinone n-oxides |
07/19/2000 | EP1019052A1 Alpha 1a adrenergic receptor antagonists |
07/19/2000 | EP0760819B1 Tricyclic dicarbonyl derivatives |
07/19/2000 | EP0667861B1 2-trifluoromethyl benzimidazole derivatives, their preparation and their use as pesticides |
07/19/2000 | CN1260791A 3-benzylpiperidine |
07/18/2000 | US6090954 Benzimidazole derivatives |
07/18/2000 | US6090837 Substituted hydrochromenopyrroles |
07/18/2000 | US6090820 Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones |
07/18/2000 | US6090818 Indolin-2-one derivatives, method for preparing them and pharmaceutical compositions containing them |
07/18/2000 | US6090808 Dimeric piperidine, tetrahydropyridine and piperazine derivatives |
07/13/2000 | WO2000040561A1 Quinolinecarboxamides as antiviral agents |
07/13/2000 | WO2000040539A1 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors for the treatment of respiratory diseases |
07/13/2000 | WO2000024741A3 Dihydropyridine compounds and their use as potassium channel openers |
07/13/2000 | CA2356053A1 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors for the treatment of respiratory diseases |
07/13/2000 | CA2353636A1 Quinolinecarboxamides as antiviral agents |
07/12/2000 | EP1018514A1 NF-$g(k)B INHIBITORS CONTAINING INDAN DERIVATIVES AS THE ACTIVE INGREDIENT |
07/12/2000 | EP1017676A1 Method for the synthesis of quinoline derivatives |
07/12/2000 | EP1017675A1 Highly lipophilic camptothecin derivatives |
07/12/2000 | EP1017399A1 Camptothecin analogs and methods of preparation thereof |
07/12/2000 | EP1017395A1 Method for treating premenstrual or late luteal phase syndrome |
07/12/2000 | EP0877734B1 Quinoline and quinazoline compounds useful in therapy |
07/12/2000 | EP0731802B1 N-substituted azabicycloalkane derivatives as neuroleptics etc. |
07/12/2000 | EP0642502B1 Fungicidal imidazolinones |
07/12/2000 | CN1259938A Crambescidin compound |
07/11/2000 | US6087510 Method of use of imidazolium cations |
07/11/2000 | US6087495 Salt formation by seeding |
07/11/2000 | US6087370 Methods of treatment using lamellarin-class alkaloids |
07/11/2000 | US6087369 Indole derivatives, process for producing the same and medicinal uses of the same |
07/11/2000 | CA2208569C Novel processes for preparing intermediates of inhibitors of enkephalinase and angiotensin converting enzyme and intermediates thereof |
07/06/2000 | WO2000039108A1 Thrombin or factor xa inhibitors |
07/06/2000 | WO2000039102A1 THROMBIN OR FACTOR Xa INHIBITORS |
07/06/2000 | WO2000039087A2 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors |
07/06/2000 | WO2000039081A2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds |
07/06/2000 | WO2000038720A1 Remedies for pain |
07/06/2000 | WO2000038687A1 Protease inhibitors |
07/06/2000 | WO2000038683A1 THROMBIN OR FACTOR Xa INHIBITORS |
07/06/2000 | CA2358047A1 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds |
07/06/2000 | CA2356671A1 Protease inhibitors |
07/06/2000 | CA2356269A1 Pain control agent |
07/06/2000 | CA2349557A1 Thrombin or factor xa inhibitors |
07/06/2000 | CA2348740A1 Thrombin or factor xa inhibitors |
07/06/2000 | CA2320730A1 Thrombin or factor xa inhibitors |
07/05/2000 | EP1015469A2 Bi- and tri-cyclic nucleoside, nucleotide and oligonucleoide analogues |
07/05/2000 | EP1015458A1 Furopyrrolidine derivatives and their use as serine protease inhibitors |
07/05/2000 | EP1015457A1 1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives as ampa/kainate receptor inhibitors |
07/05/2000 | EP1014973A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS |
07/05/2000 | EP0675889B1 Antiallergic triazolo(pyrrolo, thieno or furano)azepine derivatives |
07/05/2000 | EP0565621B1 Method of making camptothecin and camptothecin analogs |
07/05/2000 | CN1259125A Substituted 3-cyano quinolines |
07/04/2000 | US6084095 Including 6-amino-4-(3-bromoanilino)pyrido(3,2-d)pyrimidine; 4-(3-bromoanilino)-6-methylaminopyrido (3,2-d)pyrimidine; and 4-(3-bromoanilino)-6-methylaminopyrido(3,2-d)pyrimidine; useful in treating proliferative diseases such as cancer |
07/04/2000 | US6084094 Oxidative process for preparing narwedine derivatives |
07/04/2000 | US6083956 Optically pure androgen mediator |
07/04/2000 | CA1341044C Benzopyrido piperidine, piperidylidene and peperazine compounds, compositions, methods of manufacture and methods of use |
06/29/2000 | WO2000037473A1 Epothilone derivatives and their use as antitumor agents |
06/29/2000 | WO2000037468A1 DIBENZO[a,g]QUINOLIZINIUM DERIVATIVES AND THE SALTS THEREOF |
06/29/2000 | WO2000037466A1 BENZISOXAZOLES AND PHENONES AS α2-ANTAGONISTS |
06/29/2000 | WO2000037456A1 Amide and urea derivatives as 5-ht reuptake inhibitors and as 5-ht1b/1d ligands |
06/29/2000 | WO2000037450A1 NEW β-AMIDE AND β-SULFONAMIDE CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS ENDOTHELIN RECEPTOR ANTAGONISTS |
06/29/2000 | WO2000037026A1 Dihydropyrimidines and uses thereof |
06/29/2000 | CA2355861A1 Amide and urea derivatives as 5-ht reuptake inhibitors and as 5-ht1b/1d ligands |
06/29/2000 | CA2355848A1 Dihydropyrimidines and uses thereof |
06/29/2000 | CA2355469A1 Dibenzo[a,g]quinolizinium derivatives and the salts thereof |
06/29/2000 | CA2355251A1 New .beta.-amide and .beta.-sulfonamide carboxylic acid derivatives, their preparation and their use as endothelin receptor antagonists |
06/28/2000 | EP1012145A1 Alkoxy-substituted compounds, methods, and compositions for inhibiting parp activity |
06/28/2000 | EP1011665A1 Heterocyclic agents |
06/28/2000 | EP0808318B1 Tricyclic substituted hexahydrobenz[e]isoindole alpha-1 adrenergic antagonists |
06/27/2000 | US6080852 4,7-dichlororhodamine dyes |
06/27/2000 | US6080776 Used as a microbiocide for crop protection |
06/27/2000 | US6080754 For treatment and prophylaxis of estrogen related syndromes and disorders |
06/27/2000 | US6080752 For treating condition which requires antagonism of a dopamine receptor such as psychtic condition |
06/27/2000 | US6080743 2,3-dioxo-1,2,3,4-tetrahydro-quinoxalinyl derivatives |
06/22/2000 | WO2000035924A1 Camptothecin analogs and methods of preparation thereof |
06/22/2000 | WO2000035915A1 Piperazine derivatives |
06/22/2000 | WO2000035907A1 Imidazolones and their use in treating benign prostatic hyperplasia and other disorders |
06/22/2000 | CA2355202A1 Imidazolones and their use in treating benign prostatic hyperplasia and other disorders |
06/22/2000 | CA2354875A1 Piperazine derivatives |
06/21/2000 | EP1009739A2 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting parp activity |
06/21/2000 | EP1009738A1 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors |
06/21/2000 | DE19858779A1 New 3-acylamino-propionic acid and 3-sulfonylamino-propionic acid derivatives useful as endothelin receptor antagonists in treatment of e.g. cardiovascular and renal disorders, migraine and cancer |
06/21/2000 | CN1257506A Spiro-quinuclidine derivatives, their preparation and use |
06/21/2000 | CN1257505A Fused dihydropyrans |
06/21/2000 | CN1257504A Salts of aromatic sulphonic acids |