Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
08/2001
08/28/2001US6281227 Inhibitors of the activity of factor xa.
08/28/2001CA2015996C Bis-(1h-indol-3-yl)-maleinimide derivatives and their use as pharmaceuticals
08/25/2001CA2337620A1 Manufacture of a cyclic acid
08/23/2001WO2001060811A1 Chromene compound
08/23/2001WO2001060803A1 Fused imidazolium derivatives
08/22/2001EP1124828A1 Pyrano, piperidino, and thiopyrano compounds and methods of use
08/22/2001EP1124811A1 2-ureido-thiazole derivatives, process for their preparation, and their use as antitumor agents
08/22/2001EP0785926B1 Carboxylic acid derivatives, their preparation and their use as medicaments
08/22/2001CN1309656A Thioalkyl alpha-substd. pyrimidine compounds
08/22/2001CN1309641A Quinoline derivs.
08/21/2001US6277992 Useful as an intermediate for preparing camptothecin derivatives having antitumor activities
08/21/2001US6277985 As antibiotics; water solubility; in prodrugs
08/21/2001US6277860 Furopyridine antibacterials
08/21/2001US6277536 Heterocyclic compounds
08/21/2001CA2083606C Dialkoxy-pyridinyl-benzimidazole derivatives, process for their preparation and their pharmaceutical use
08/16/2001WO2001058905A1 Synthetic process for an intermediate for ecteinascidin and phthalascidin compounds
08/16/2001WO2001058903A1 Method for producing 2-chloro-benzimidazole derivatives
08/16/2001WO2001058875A2 Substituted 1,2,3,4- tetrahydroquinoline-2-carboxylic acid derivatives
08/16/2001WO2001010842A3 Melanocortin-4 receptor binding compounds and methods of use thereof
08/16/2001WO2001009119A3 Chemokine receptor antagonists
08/16/2001US20010014684 Thieno-pyridine sulfonamides derivatives thereof and related compounds that modulate the activity of endothelin
08/16/2001EP1123297A1 New compounds, their preparation and use
08/16/2001EP1123293A1 Core-extended perylene bisimides
08/16/2001EP1123285A1 Substituted benzopyran analogs for the treatment of inflammation
08/16/2001EP1123099A1 Novel indenoisoquinolines as antineoplastic agents
08/16/2001EP0839137B1 Aromatic acid diamides with antigastrin activity, a method for their preparation and their pharmaceutical use
08/16/2001EP0788498B1 Phenyloxazolidinone antimicrobials
08/16/2001CA2416343A1 Substituted 1,2,3,4-tetrahydroquinoline-2-carboxylic acid derivatives
08/15/2001CN1308631A Heterocyclic derivatives which inhibit factor xa
08/15/2001CN1308622A Biphenyl oxo-acetic acids useful in the treatment of insulin resistance and hyperglycemia
08/15/2001CN1308078A Camptothecin derivative and its preparation
08/15/2001CN1069624C Production of derivatives of 4a,5,9,10,11,12,-bexahydro-6H-benzofuro[3a,3,2-ef][2] benzazepine
08/14/2001US6274587 Tricyclic dihydropyrimidine potassium channel openers
08/14/2001US6274585 Benign prostatic hyperplasia treatment
08/14/2001CA2206824C Inhibitors of rotamase enzyme activity
08/09/2001WO2001057043A1 Method for producing sulfonyl imidazole derivatives by phase transfer catalysis
08/09/2001WO2001014376A8 Novel spiro compounds
08/09/2001US20010012846 A diagnostic tool for assessing the degree to which neurokinin-2 and neurokinin-3 receptor activity(normal, over or underactivity) is implicated in a patient's symptoms
08/09/2001DE10005278A1 Verfahren zur Herstellung von Sulfonyl-imidazol-Derivaten Process for preparing sulphonyl-imidazole derivatives
08/09/2001DE10005277A1 Pure 5,6-alkylenedioxy-2-chloro-benzimidazole preparation in high yield, for use as intermediate for microbicides, especially fungicides, by chlorinating corresponding thione with chlorine in organic diluent
08/08/2001EP1122254A2 4-Sulfonamide piperidine derivatives, method for their preparation and phamaceutical compositions containing them
08/08/2001EP1121122A1 Treatment of depression
08/08/2001EP0815112B1 Process for isolating galanthamine
08/08/2001CN1307580A Syntheses of variety of lamellarin compounds and analogues
08/08/2001CN1069323C Gaseous polymerization method
08/08/2001CN1069317C Novel indane-2-mercaptoacetamide disulfide derivs, useful as inhibitors of enkephaliinase
08/07/2001US6271371 Obtaining narwedine and derivatives thereof in improved yield
08/07/2001US6271342 Sugar-modified cytostatics
08/07/2001US6271253 Cyclooxygenase inhibitors
08/07/2001US6271180 Substituted phenyl keto enols as pesticides and herbicides
08/07/2001CA2213197C Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
08/07/2001CA2015296C Pyranyl cyanoguanidine derivatives
08/02/2001WO2001055122A1 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
08/02/2001WO2001055121A1 Azepine derivatives
08/02/2001WO2001055119A2 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
08/02/2001WO2001054694A1 Tetrahydropyrimidone inhibitors of fatty acid binding protein and method
08/02/2001WO2001005228A3 Fungicidal combinations of active substances
08/02/2001WO2000067801A3 Prodrugs of chemotherapeutic agents with oxaalkanoic acids
08/02/2001US20010011139 Polynucleotides labeled with dibenzorhodamine dyes
08/02/2001US20010011134 Cyclic and heterocyclic N-substituted alpha-iminohydroxamic and -carboxylic acids
08/02/2001US20010011092 High affinity ligands for nociceptin receptor ORL-1
08/02/2001CA2396596A1 Tetrahydropyrimidone inhibitors of fatty acid binding protein and method
08/01/2001EP1119571A2 Tricyclic delta3-piperidines as alpha2-antagonists
08/01/2001EP1119570A1 Tricyclic delta3-piperidines as pharmaceuticals
08/01/2001CN1306510A Optical active tetrahydrobenzindole derivatives
07/2001
07/31/2001US6268508 For crop protection
07/31/2001US6268499 Process and intermediates for preparation of substituted piperidine-epoxides
07/31/2001US6268497 Converting lactol precursor to one of a select number of mixed acetal derivatives, and then treating acetals with a grignard reagent to provide chromenoquinoline compound
07/31/2001US6268375 10, 11-difluoromethylenedioxycamptothecin compounds with topoisomerase I inhibition
07/31/2001US6268369 5-(heterocyclic alkyl)-6-aryl-dihydropyrimidines
07/31/2001US6268358 Compounds for the treatment of Alzheimer's disease
07/31/2001US6268308 Herbicidal S-substituted 1,2,4,6-thiatriazines
07/31/2001US6267606 Removable transceiver module and receptacle
07/31/2001CA2208639C Camptothecin derivatives and its manufacturing method
07/31/2001CA2059305C Hexa-cyclic compound
07/31/2001CA2040774C Compounds formed from o-hydroxyphenyl-1,3,5-triazines and sterically hindered amines
07/26/2001WO2001053299A1 Compounds of the saframycin-ecteinascidin series, uses, and synthesis thereof
07/26/2001WO2001053260A1 Carboxamides useful as inhibitors of microsomal triglyceride transfer protein and of apolipoprotein b secretion
07/26/2001WO2001008663A3 Liposomal prodrugs comprising derivatives of camptothecin and methods of treating cancer using these prodrugs
07/26/2001US20010009919 Tris benzimidazoles; fungicides, anticarcinogenic agents, enzyme inhibitor
07/26/2001US20010009911 Isomers, hydrates, solvates and addition salts in treatment of endothelial dysfunction disease such as atherosclerosis, dyslipidaemia; antidiabetic agents; heart transplantation; inhibition of nitrogen monoxide synthase and oxidative stress
07/26/2001CA2397597A1 Compounds of the saframycin-ecteinascidin series, uses, and synthesis thereof
07/25/2001EP1118322A1 Drugs for improving vesical excretory strength
07/25/2001EP1117659A1 Substituted 3-cyanoquinolines as protein tyrosine kinases inhibitors
07/25/2001EP1117656A1 Grey colouring photochromic fused pyrans
07/25/2001EP1117649A1 Substituted 3-cyanoquinolines as protein tyrosine kinases inhibitors
07/25/2001EP1117297A1 Synthetic analogs of ecteinascidin-743
07/25/2001EP0646117B1 Methods and intermediates for the asymmetric synthesis of camptothecin and camptothecin analogs
07/25/2001CN1305476A 1,3-oxazoline and 1,3-thiazoline derivatives, method for producing the same and their use as pesticides
07/25/2001CN1304930A Arylsulfurylisooximino acid derivative
07/24/2001US6265580 Method for producing pyridine derivatives
07/24/2001US6265418 N-acylamino acid amide compounds and intermediates for preparation thereof
07/24/2001US6265413 Water solubility; anticarcinogenic agents
07/24/2001US6265410 Bicyclic compounds capable of inhibiting tyrosine kinases of the epidermal growth factor receptor family
07/24/2001US6265350 1,3-oxazoline and 1,3-thiazoline derivatives, their preparation, and their use as pesticides
07/24/2001CA2218503C Arylsulfonyl hydroxamic acid derivatives
07/24/2001CA2174033C Novel pyridine compounds; process for preparing the same and pharmaceutical compositions containing them
07/19/2001WO2001051479A2 Tricyclic compounds with antiviral activity
07/19/2001WO2000076984A8 Novel compounds, their use and preparation
07/19/2001US20010008939 Also useful in treating viral infections; antiprotozoa (plasmodium) activity