Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
09/2001
09/25/2001US6294560 Synthesis of clasto-lactacystin β-lactone and analogs thereof
09/22/2001CA2341344A1 Use of glycogen phosphorylase inhibitors
09/20/2001WO2001068650A1 Perylene-derivative based crystallization modifiers
09/20/2001WO2001068649A1 Novel process for the preparation of a quinoline carboxylic acid derivative having a 7-(4-aminomethyl-3-oxime)pyrrolidine substituent
09/20/2001WO2001068641A1 6-aminoalkyl-dihydropyrimidines and the use thereof as medicaments against viral diseases
09/20/2001WO2001068625A1 Method for the production of spirocyclic tetronic acid derivatives
09/20/2001WO2001068619A1 5-amide substituted diarylamines as mex inhibitors
09/20/2001WO2001068588A1 POLYMER-IMMOBILIZED α-IMINOESTER
09/20/2001WO2001034591A3 Substituted 4h-chromene and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/20/2001DE10013188A1 New hydrogenated perylenetetracarboxylic dianhydride, diimide and anhydride-imide derivatives are used as crystallization modifiers for organic pigments and in perylene pigment formulations
09/20/2001DE10013126A1 New 6-aminoalkyl-dihydropyrimidine-5-carboxylate ester derivatives, useful as antiviral agents having strong activity against hepatitis B virus and low cytotoxicity
09/20/2001CA2403017A1 5-amide substituted diarylamines as mex inhibitors
09/19/2001EP1134217A2 Cosmetic composition containing a furan-naphthoquinone derivative, use therof as dyeing agent, and derivatives
09/19/2001EP1134215A1 2-oxo-imidazolidine-4-carboxylic acid hydroxamine compounds that inhibit matrix metalloproteinases
09/19/2001CN1313859A Preparation of camptothecin and nothapodytine derivatives
09/19/2001CN1313286A S type 4-substituted hydroxypyranoindolidine compound and its derivatives and preparation thereof
09/19/2001CN1071117C Antitussive
09/18/2001US6291684 Process for the preparation of aziridinyl epothilones from oxiranyl epothilones
09/18/2001US6291681 Reacting meso-2,3-bis(benzylamino)succinic acid dialkali metal salt with phenyl chloroformate; acidification, isolating 2-oxo-1,3-dibenzyl-cis-4,5-imidazolidinedicarboxylic acid; heating with acetic anhydride to produce anhydride compound
09/18/2001US6291676 As antiproliferative agent
09/18/2001US6291483 Administering a therapeutically effective amount of berberine or a pharmaceutically acceptable salt thereof
09/18/2001US6291475 Bispidine antiarrhythmic compounds
09/18/2001US6291472 4a, 5a, 8a, 8b-tetrahydro-6H-pyrrolo[3′,4′:4, 5]furo[3,2-b] pyri-dine-6,8(7H)-dione derivatives for control of endoparasites processes for their preparation
09/18/2001US6291470 Indole derivatives process for producing the same and medicinal uses of the same
09/18/2001US6291425 Compounds, methods and pharmaceutical compositions for treating cellular damage, such as neural or cardiovascular tissue damage
09/18/2001CA2236814C Quinoline and quinazoline compounds useful in therapy
09/17/2001CA2341840A1 Cosmetic composition comprising a furan-naphthoquinone derivative, its use as a coloring agent and derivatives
09/13/2001WO2001066544A2 Tricyclic dihydropyrazolone and tricyclic dihydroisoxazolone potassium channel openers
09/13/2001WO2001009138A3 Chemokine receptor antagonists and methods of use therefor
09/13/2001WO1997014683A3 Phenanthridine derivatives, methods of producing them and medicaments containing phenanthridine derivatives
09/13/2001US20010021791 Cyclopropyl phenyl ketone compound
09/13/2001US20010021777 Indane or dihydroindole derivatives
09/13/2001CA2402179A1 Tricyclic dihydropyrazolone and tricyclic dihydroisoxazolone potassium channel openers
09/12/2001EP1131325A1 [pyrrole]naphthopyranes, their preparation, compositions and (co)polymer matrices containing them
09/12/2001EP1131322A2 Dihydropyridine compounds and methods of use
09/12/2001EP1131306A2 Isoxazoline fibrinogen receptor antagonists
09/12/2001EP1131295A1 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
09/12/2001EP0817775B1 Quinazoline derivatives
09/12/2001CN1312804A Macrocyclic analogs and methods of their use and preparation
09/11/2001US6288185 Initiators for radical polymerization
09/11/2001US6288102 Substituted phenylketoenols and their use as pesticides and herbicides
09/11/2001US6288099 Compounds such as 8-bromo-10h-benzo(4,5)furo(3,2-b)indole-1-carboxylic acid used to treat disorders associated with smooth muscle contration such as urinary incontinence and irritable bowl syndrome
09/11/2001US6288084 Administering comounds such as 4-(4-chlorophenyl)-1-(4-(3-methoxyphenyl)-4-(3-pyridinyl)-3 -butenyl)piperidin-4-ol to treat diseases associated with aberrant leukocyte recruitment and/or activation
09/11/2001US6288083 Chemokine receptor antagonists and methods of use therefor
09/11/2001US6288081 Use of 7-(1-aminomethyl-2-oxa-7-aza-bicyclo[3.3.0]oct-7-yl)-quinolone carboxylic acid and naphthyridone carboxylic acid derivatives for treating Helicobacter pylori infections and the gastroduodenal diseases associated therewith
09/11/2001US6288073 Acronycine derivatives, preparation method and pharmaceutical compositions
09/11/2001US6288072 Anticarcinogenic and antitumor agents; leukemia
09/11/2001US6288059 Acylated hetero-alicyclic derivatives
09/11/2001US6288058 Treating muscular, nervous system, psychological and gastrointestinal disorders
09/11/2001US6288057 Physical form of dihydro-2,3-benzodiazepine derivative
09/07/2001WO2001064692A1 Cardioprotective phosphonates and malonates
09/07/2001WO2001064681A2 3-(pyrolyllactone)-2-indolinone compounds as kinase inhibitors
09/07/2001WO2001064670A1 Novel cyclic amide derivatives
09/07/2001WO2001064655A1 2, 4-di(hetero-)arylamino (-oxy)-5-substituted pyrimidines as antineoplastic agents
09/07/2001WO2001064650A2 Synthesis of epothilones, intermediates thereto and analogues thereof
09/07/2001WO2001064635A1 Ningalin b analogs employable for reversing multidrug resistance
09/07/2001WO2001064213A1 Compounds and methods
09/07/2001CA2401800A1 Synthesis of epothilones, intermediates thereto and analogues thereof
09/07/2001CA2401673A1 Ningalin b analogs employable for reversing multidrug resistance
09/07/2001CA2400649A1 3-(pyrolyllactone)-2-indolinone compounds as kinase inhibitors
09/07/2001CA2398685A1 2,4-di(hetero-)arylamino(-oxy)-5-substituted pyrimidines as antineoplastic agents
09/06/2001WO2001064715A2 Memno peptides, a process for their preparation and their use
09/06/2001US20010020114 Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
09/06/2001US20010020101 Process for preparing biotin
09/06/2001US20010020095 High affinity for D4 receptors; treatment of schizophrenia, other psychoses, anxiety disorders, depression, alcohol abuse, impulse control disorders, aggression
09/06/2001US20010020093 Preparation of asymmetric cyclic ureas through a monoacylated diamine intermeidate
09/06/2001US20010020027 Using 1-(4-(1-(4-fluorophenyl)-1H-indole-3-yl)-1-butyl spiro(isobenzofuran-1(3H,4-piperidine)
09/06/2001US20010020021 Metalloprotease inhibitor
09/05/2001EP1130027A1 Memno peptides, process for preparation and use thereof
09/05/2001EP1130021A2 Pyrrolopyridinium derivatives
09/05/2001EP1130016A1 Thiocarbamic acid derivatives
09/05/2001EP1129076A1 Tetrahydroisoquinoline derivatives as lhrh antagonists
09/05/2001CN1311778A Fused-heterocycle dicarboxylic diamide derivatives of salts thereof, herbicides and usage thereof
09/05/2001CN1311777A High affinity ligands for nociceptin receptor ORL-1
09/05/2001CN1311773A Neuropeptide Y5 receptor antagonists
09/05/2001CN1311678A Substituted tricyclic pyrazole derivatives with protein kinase activity
09/05/2001CN1070493C Heterocyclic condensed furanpyranoid ring compound and herbicides
09/04/2001US6284891 Intermediates such as 4-ethyl-1h-pyrano(3,4-c)pyridin-8-one; or 4-ethyl-7-(7-iodo-9-((4-methyl-piperazinyl)methyl) -2,3-dihydro-(1,4)dioxino(2,3-g)quinolin-8-ylmethyl)-1h-pyrano (3,4-c)pyridin-8-one.
09/04/2001US6284769 Nonpeptide kappa opioid receptor antagonists
09/04/2001US6284764 Antiproliferative agent
08/2001
08/30/2001WO2001062761A1 Method of preparing alkaloids using supercritical fluids from plants
08/30/2001WO2001011968A3 Heterocyclic spiro compounds as pesticides
08/30/2001US20010018521 Novel intermediates useful for the preparation of antihistaminic piperidine derivatives
08/30/2001US20010018441 Antiinflammatory agent, immunosuppressant, anticancer agents, antiarthritic agents
08/29/2001EP1127879A1 Preparation of 2-oxo-1,3-dibenzyl-cis-4,5-imidazolidin dicarboxylic acid and its anhydrid
08/29/2001EP1127872A1 Tamiflu via Diels-Alder
08/29/2001EP1127051A2 Tricyclic pyrazole derivatives
08/29/2001EP0828741B1 Spirocyclic and bicyclic diazinyl and carbazinyl oxazolidinones
08/29/2001EP0819108B1 Process for preparing galanthamine derivatives by asymmetric reduction
08/29/2001CN1310721A Medicine nitrate salts
08/29/2001CN1310712A Phenylazole compound, process for producing the same and drugs for hyperlipemia
08/29/2001CN1310706A Inhibitors of phospholipase enzymes
08/29/2001CN1310705A Indole derivatives and their use in the treatment of malignant and other diseases caused by pathological cell proliferation
08/29/2001CN1310702A Nitric ester and nitrate salts of specific drugs
08/29/2001CN1310629A Coadministration of ACAT and MMP inhibitors for the treatment of atherosclerotic lesions
08/29/2001CN1310621A Substituted anilide compounds and methods
08/29/2001CN1310176A Production of cyclic acid
08/29/2001CN1310170A Process for producing 4,5-diamino shikimic acid derivative
08/29/2001CN1309964A Carbazole-alkoloid cell cycle inhibitor, cell death inducer and their preparation
08/28/2001US6281355 Nitrogen-containing tetracyclic compounds