Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
02/2001
02/13/2001US6187777 Pyrrolo(3,2-d)pyrimidine derivatives; neuropeptide y and corticotropin releasing factor modulators; dietetics; antidiabetic, antiinflammatory, and antitumor agents
02/13/2001US6187774 Fused heterocyclic compounds and pharmaceutical applications thereof
02/08/2001WO2001055118A1 Benzene-fused heterocycle derivatives and drugs containing the same as the active ingredient
02/08/2001WO2001009372A1 Chemiluminescent substrates of hydrolytic enzymes such as phosphatases
02/08/2001WO2001009139A1 Aromatic esters of camptothecins and methods to treat cancers
02/08/2001WO2001009138A2 Chemokine receptor antagonists and methods of use therefor
02/08/2001WO2001009137A1 Chemokine receptor antagonists and methods of use therefor
02/08/2001WO2001009130A1 TRICYCLIC COMPOUNDS HAVING sPLA2-INHIBITORY ACTIVITIES
02/08/2001WO2001009119A2 Chemokine receptor antagonists
02/08/2001WO2001009101A1 Isoquinoline derivatives, pharmaceutical compositions containing the same, and a process for the preparation of the active substance
02/08/2001WO2001009094A2 Chemokine receptor antagonists and methods of use therefor
02/08/2001WO2001009092A1 Biphenyl-substituted cyclic keto enols as pesticides
02/08/2001WO2001008663A2 Liposomal prodrugs comprising derivatives of camptothecin and methods of treating cancer using these prodrugs
02/08/2001WO2000076984A3 Novel compounds, their use and preparation
02/08/2001CA2391267A1 Chemokine receptor antagonists and methods of use therefor
02/08/2001CA2379660A1 Liposomal prodrugs comprising derivatives of camptothecin and methods of treating cancer using these prodrugs
02/07/2001EP1073655A1 Pharmaceutically available protoberberine salts derivatives, and protoberberine derivatives and salts thereof
02/07/2001EP1073654A1 2,3-olefinic epothilone derivatives
02/07/2001EP1073648A1 12,13-Modified epothilone derivatives
02/07/2001EP1073647A1 12,13-cyclopropane epothilone derivatives
02/07/2001EP1073639A1 Quinoline derivatives
02/07/2001EP1073435A1 Substituted tricyclic pyrazole derivatives with protein kinase activity
02/07/2001EP0799226B1 Tetracyclic spiro compounds, process for their preparation and their use as 5ht1d receptor antagonists
02/07/2001CN1283187A Novel dipydropyridine derivative
02/07/2001CN1282517A Pest controlling agent containing substituted aminoquinazolone or thioketone derivative or its salt as active component
02/07/2001CN1061658C Tricyclic benzazepine vasopression antagonists
02/06/2001US6184379 Rhodamine derivatives and the use thereof
02/06/2001US6184221 Antiarrhythmia agents, antiulcer agents
02/06/2001US6184004 Process for the preparation of galanthamine and its derivatives
02/01/2001WO2001007050A1 Nociceptin receptor orl-1 agonists for use in treating cough
02/01/2001DE19935963A1 Biphenylsubstituierte cyclische Ketoenole Biphenyl-cyclic ketoenols
02/01/2001CA2379398A1 Nociceptin receptor orl-1 agonists for use in treating cough
01/2001
01/31/2001EP1072593A1 Liquid crystalline compound having piperidine ring, liquid crystal composition and liquid crystal display element
01/31/2001EP1071683A1 New compounds
01/31/2001EP1071666A1 Azacycloalkane derivatives, preparation and therapeutic application
01/31/2001EP1071455A1 Terminally-branched polymeric linkers and polymeric conjugates containing the same
01/31/2001EP0746320B1 Hiv protease inhibitors and intermediates
01/31/2001CN1282332A Novel acronycine compounds, preparation method and pharmaceutical compositions containing them
01/31/2001CN1061346C Diazabicycloalkene derivatives and use, and drug composition containing said derivatives
01/30/2001US6180794 Steroids and dehydrohalogenation and amination
01/30/2001US6180640 Di- and tetra-hydroquinoline-indole antimicrobial agents, uses and compositions related thereto
01/25/2001WO2001005795A1 Remedies or preventives for frequent urination or urinary incontinence
01/25/2001WO2001005790A1 New compounds
01/25/2001WO2001005772A1 Pyrazinones, compositions containing such compounds
01/25/2001WO2001005230A1 Alpha-hydroxy-gamma-[[(carbocyclic-or heterocyclic-substituted)amino]carbonyl]alkanamide derivatives and uses thereof
01/25/2001WO2001005228A2 Fungicidal combinations of active substances
01/25/2001DE19933938A1 Fungizide Wirkstoffkombinationen Fungicidal drug combinations
01/25/2001CA2379577A1 Remedies or preventives for frequent urination or urinary incontinence
01/25/2001CA2378202A1 New compounds
01/25/2001CA2375954A1 Alpha-hydroxy-gamma-¬¬(carbocyclic-or heterocyclic-substituted)amino|carbonyl|alkanamide derivatives and uses thereof
01/24/2001EP1070060A1 Heterocyclic glycyl beta-alanine derivatives as vitronectin antagonists
01/24/2001EP1069899A1 Treatment of panic attacks
01/24/2001CN1281459A Piperidine derivatives
01/24/2001CN1281439A 4-Hydroxyquinoline-3-carboxamides and hydrazides as antiviral agents
01/24/2001CN1280825A Sigma-receptor acting medicine containing protopine-type alkaloid
01/23/2001US6177568 Intermediates for the synthesis of camptothecin derivatives
01/23/2001US6177464 Bactericides
01/23/2001US6177445 Substituted isoquinolines as ultra short acting neuromuscular blockers
01/23/2001US6177440 Substituted tricyclics
01/23/2001US6177439 Anticarcinogenic agents; viricides
01/23/2001US6177423 N-(hydroxy or protected hydroxy)-benzo(de)isoquinoline-1,3-dione derivatives; bacterial dna gyrase and dna topoisomerase inhibitors useful for antibacterial agents having reduced drug resistance and reduced side effects
01/23/2001US6177401 Use of organic compounds for the inhibition of Flk-1 mediated vasculogenesis and angiogenesis
01/23/2001US6177379 Containing diels-alder adduct obtained by reacting specified azo compound and conjugated diene
01/18/2001WO2001004122A2 New 2,3-benzodiazepine derivatives
01/18/2001CA2378305A1 New 2,3-benzodiazepine derivatives
01/17/2001EP1069127A1 Microencapsulated lewis acid
01/17/2001EP1069125A2 Carbamate derivatives of 4-amino-3-isoxazolidinones, 3-amino-1-hydroxypyrrolidin-2-ones and 1-amino-1-cyclopropanecarboxylic acid analogs, a process for their preparation and their use as medicaments
01/17/2001EP1069124A1 2-Benzimidazolylamine compounds as ORL1-receptor agonists
01/17/2001EP1068189A1 4,4-disubstituted-3,4-dihydro-2(1h)-quinazolinthione derivatives, their preparation and their use as hiv reverse transcriptase inhibitors
01/17/2001EP0983258A4 N-hydroxy 4-sulfonyl butanamide compounds
01/17/2001CN1280569A 1,2-dihydro-2-oxoquinoline derivatives
01/17/2001CN1280567A Nitrogen-containing tetracyclic compounds
01/16/2001US6174905 As carcinostatic agent to a hematologic malignancy and a solid carcinoma
01/16/2001CA2314008A1 2-benzimidazolylamine compounds as orl1-receptor agonists
01/11/2001WO2001002409A1 Thieno- and furopyrimidine derivatives as a2a-receptor antagonists
01/11/2001WO2001002374A1 Bridged fluorescent dyes, their preparation and their use in assays
01/11/2001WO2001002369A2 Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
01/11/2001CA2376955A1 Bridged fluorescent dyes, their preparation and their use in assays
01/10/2001EP1066258A1 Aryl phenyl substituted cyclic ketoenols
01/10/2001EP1066039A1 Substituted quinazolines and analogs and the use thereof
01/10/2001EP0777655B1 Process for preparing chiral tetracyclic dopaminergic compounds
01/10/2001CN1279687A Bi-and tri-cyclic nucleoside, nucleotide and oligonucleotide analoguse
01/10/2001CN1279682A bicyclic kinase inhibitors
01/10/2001CN1279239A Acridine carboxylic ester compound, preparation and medicinal composition thereof
01/10/2001CN1060478C Substituted pyrazole derivatives
01/10/2001CN1060472C Hydroxamic acid derivatives with tricylic substitution, their preparing methods, medicines containing them and uses thereof
01/09/2001US6172255 Alkoxy-alkyl-substituted 1-H-3-aryl-pyrrolidine-2,4-diones used as herbicides and pesticides
01/09/2001US6172230 Process for the preparation of tetrahydro-indolizines
01/09/2001US6172170 Initiators for radical polymerization
01/09/2001US6172102 Pyrrole derivatives and medicinal composition
01/09/2001US6172092 Fungicides, bactericides for crops; treating plant diseases; applying to wood, leather, plastic
01/09/2001US6172084 Quinoline-indole antimicrobial agents, uses and compositions related thereto
01/09/2001US6172078 Quinolinomorphinane derivatives and medicinal use thereof
01/09/2001US6172077 Tachykinin inhibitors; analgesics, antiinflammatory agents, antiemetics; neuralgia, headaches
01/09/2001US6172074 Imidazopyridines and oxazolopyridines
01/09/2001US6172073 Benzimidazolyloxy alkanamines as serotonin reuptake inhibitors; nicotine and tobacco withdrawal; psychological, eating, brain, gastrointestinal, sleep, and sexual disorders
01/09/2001US6172006 Furyl-pyridone compounds, useful as fungicides and obtained from the fungus Cladobotryum
01/04/2001WO2001000626A1 Hexahydropyrrolo[1,2-c]pyrimidines as antiviral, antifungal and/or antitumor agents
01/04/2001WO2001000615A1 Respiratory syncytial virus replication inhibitors
01/04/2001WO2001000213A1 Src kinase inhibitor compounds