Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
10/2001
10/18/2001US20010031770 Pyridoxal analogues and methods of treatment
10/18/2001US20010031761 Compounds such as camptothecin 20-o-nonanoate; antitumor agents; low toxicity; good absorbability
10/18/2001CA2405089A1 Benzoamide piperidine containing compounds and related compounds
10/17/2001EP1146047A1 3,5-Dioxa-8-aza-tricyclo(5.2.1.00,0)decane-9-methanols, their metal complexes and enantioselective hydrogenation processes
10/17/2001EP1144416A1 Heterocyclically anellated indenochromene derivatives
10/17/2001EP1144415A2 Functionalized heterocycles as chemokine receptor modulators
10/17/2001EP1144405A1 Triazole compounds with dopamine-d3-receptor affinity
10/17/2001EP0942911B1 Benzopyranopyrrole and benzopyranopyridine alpha-1 adrenergic compounds
10/17/2001EP0833818B1 3-acylindoles as cb2 receptor agonists
10/17/2001EP0809643B1 Synthesis of (+)-pancratistatin
10/17/2001EP0652871B1 Benzodiazepine derivatives
10/17/2001CN1317969A Treatment of depression
10/16/2001US6303615 2,3 disubstituded-4(3H)-quinazolinones
10/16/2001US6303609 Used for the inhibition of platelet aggregation, as thrombolytics, and/or for the treatment of thromboembolic disorders
10/11/2001WO2001074821A1 Novel process for producing fused imidazopyridine derivative and novel crystal form
10/11/2001WO2001074820A1 Novel derivatives and analogues of galanthamin
10/11/2001WO2001074770A1 C2 phenyl-substituted cyclic keto-enols used as pesticides and herbicides
10/11/2001WO2001074344A2 Small organic molecule regulators of cell proliferation
10/11/2001WO2001074339A2 A use of galantamine for the treatment of neuropsychiatric behaviour associated with alzheimer's disease
10/11/2001WO2001022951A3 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives for the treatment of multiple sclerosis
10/11/2001US20010029298 Novel intermediates in the synthesis of camptothecin and related compounds and synthesis thereof
10/11/2001US20010029297 Chemical synthesis of spirocyclic piperidines by double ring-closing metathesis
10/11/2001DE10017539A1 New 6-acylamino-4-amino-quinazoline or quinoline derivatives, are tyrosine kinase-mediated signal transduction inhibitors useful e.g. for treating tumors or respiratory or gastrointestinal diseases
10/11/2001DE10016544A1 New phenyl-substituted cyclic keto-enol compounds useful e.g. as insecticides, acaricides, nematocides, acaricides, herbicides, ectoparasiticides, antifouling agents or intermediates
10/11/2001CA2829534A1 C2-phenyl-substituted cyclic keto-enols as pesticides and herbicides
10/11/2001CA2404868A1 C2-phenyl-substituted cyclic keto-enols as pesticides and herbicides
10/11/2001CA2404413A1 Small organic molecule regulators of cell proliferation
10/11/2001CA2403131A1 Novel process for producing fused imidazopyridine derivative and novel crystal form
10/11/2001CA2368966A1 New derivatives and analogues of galanthamine
10/10/2001EP1142889A1 Pyrazole derivatives as anti-inflammatory/analgesic agents
10/10/2001EP1142881A1 Poly(adp-ribose) polymerase inhibitors consisting of pyrimidine derivatives
10/10/2001EP1142587A1 Remedies for pain
10/10/2001EP1141137A1 Water-soluble rhodamine dyes and conjugates thereof
10/10/2001EP1140948A1 Camptothecin analogs and methods of preparation thereof
10/10/2001EP1140944A1 Epothilone derivatives and their use as antitumor agents
10/10/2001EP1140934A1 BENZISOXAZOLES AND PHENONES AS $g(a) 2?-ANTAGONISTS
10/10/2001EP1140930A1 DIBENZO a,g]QUINOLIZINIUM DERIVATIVES AND THE SALTS THEREOF
10/10/2001EP1140924A1 Piperazine derivatives
10/10/2001EP1140908A1 Triazole compounds with dopamine-d3-receptor affinity
10/10/2001EP1140907A1 Triazole compounds with dopamine-d3-receptor affinity
10/10/2001EP1140906A1 Imidazolones and their use in treating benign prostatic hyperplasia and other disorders
10/10/2001EP1140901A2 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors
10/10/2001EP1140898A1 Amide and urea derivatives as 5-ht reuptake inhibitors and as 5-ht1b/1d ligands
10/10/2001EP1140871A1 Thrombin or factor xa inhibitors
10/10/2001EP1140867A1 New beta-amide and beta-sulfonamide carboxylic acid derivatives, their preparation and their use as endothelin receptor antagonists
10/10/2001EP1140862A1 THROMBIN OR FACTOR Xa INHIBITORS
10/10/2001EP1140850A1 Quinolinecarboxamides as antiviral agents
10/10/2001EP1140814A2 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
10/10/2001EP1140768A1 Use of substituted 4-biarylbutyric and 5-biarylpentanoic acid derivatives as matrix metalloprotease inhibitors for the treatment of respiratory diseases
10/10/2001EP1139972A1 Dihydropyrimidines and uses thereof
10/10/2001EP0923566A4 High molecular weight polymer-based prodrugs
10/10/2001CN1317005A Substituted pyrazole derivatives condensed with six-membered heterocyclic rings
10/10/2001CN1072649C Benzoxazepine compounds, their production method and use
10/09/2001US6300316 C-4 substituted macrolide antibiotics
10/04/2001WO2001072757A1 Tricyclic imidazopyridines
10/04/2001WO2001072756A1 Prodrugs of imidazopyridine derivatives
10/04/2001WO2001072755A1 Pyrano[2,3-c]imidazo[-1,2-a]pyridine derivatives for the treatment of gastrointestinal disorders
10/04/2001WO2001072754A1 Alkylated imidazopyridine derivatives
10/04/2001WO2001072753A1 Ketol fatty acid derivatives and plant growth regulating agents
10/04/2001WO2001072696A1 Arthropodicidal carboxanilides
10/04/2001WO2001072309A2 Treatment of cerebrovascular disease
10/04/2001US20010027199 Administering a Tumor Necrosis Factor-alpha inhibitor from the group of metalloproteinase inhibitors, quinolones, corticoids, thalidomide, lazaroides, pentoxyphyllines, hydroxamic and carbocyclic acids; spinal disk hernias
10/04/2001US20010027197 Antiproliverative, -carcinogenic and -tumor agents; mitogenesis-activated protein kinase inhibitors; noncytotoxic; binding with high affinity at the adenosine triphosphate binding site of the kinases
10/04/2001US20010027175 Inhibiting tumor necrosis factor-alpha (TNF-a) for treating nerve conditions such as sciatica by administering antiinflammatory agent etanercept or infliximab
10/04/2001EP1138682A1 Novel water soluble c-ring analogues of 20 (s)-camptothecin
10/04/2001EP1137413A2 Non-peptide antagonists of glp-1 receptor and methods of use
10/04/2001EP1137411A1 Palladium-substituted bacteriochlorophyll derivatives and use thereof
10/04/2001EP0855999B1 1-(1,2-disubstituted piperidinyl)-4-substituted piperidine derivatives as tachykinin receptor antagonists
10/04/2001EP0741712B1 Process for making hiv protease inhibitors
10/04/2001EP0631575B1 Substituted pyrimidines and their use as pesticides
10/04/2001CA2404477A1 Tricyclic imidazopyridines
10/04/2001CA2404474A1 Prodrugs of imidazopyridine derivatives
10/04/2001CA2404466A1 Pyrano[2,3-c]imidazo[-1,2-a]pyridine derivatives for the treatment of gastrointestinal disorders
10/04/2001CA2404460A1 Alkylated imidazopyridine derivatives
10/04/2001CA2404329A1 Treatment of cerebrovascular disease
10/03/2001CN1315954A Substituted benzimidazoles, production and use thereof as agents for combating parasitic protozoas
10/03/2001CN1072221C 3-halo-3-heteroaryl carboxylic acid derivatives, method of preparing them and intermediates
10/02/2001US6297238 3-aryl pyrazoles with 4,5(3,4)-bicyclic ring fusion which are inhibitors of protein kinases particularly tyrosine kinases and serine/threonine kinases
09/2001
09/27/2001WO2001070747A1 Process for producing camptothecin
09/27/2001WO2001070746A1 Furoisoquinoline derivatives, process for producing the same and use thereof
09/27/2001WO2001070745A1 Pyranoindoles for treating glaucoma
09/27/2001WO2001070732A1 Pyrazoline derivatives or tetrahydropyridazine derivatives and medicinal use thereof
09/27/2001WO2001070728A1 2-[nitrogen-heterocyclic]pyrimidone derivatives
09/27/2001WO2001070716A1 A process for the preparation of epothilone analogs and intermediates
09/27/2001WO2001070677A1 Sulphonamido-substituted bridged bicycloalkyl derivatives
09/27/2001WO2001070232A1 Protease inhibitors
09/27/2001WO2001017972A3 Novel herbicides
09/27/2001WO2000012047A3 Enhancement of return to independent living status with a growth hormone secretagogue
09/27/2001US20010025035 Water soluble prodrugs of hindered alcohols
09/27/2001CA2404226A1 Furoisoquinoline derivatives, process for producing the same and use thereof
09/27/2001CA2404206A1 Protease inhibitors
09/26/2001EP1136493A1 2-(Thienopyridinyl)pyrimidone, 2-(furopyridinyl)pyrimidone 2-(isoquinolinyl)pyrimidone, 2-(pyridoindolyl)pyrimidone and 2-(benzofuropyridinyl)pyrimidone derivatives
09/26/2001EP1136477A1 Benzofuran derivatives, process for the preparation of the same and uses thereof
09/26/2001EP1136071A2 Use of glycogen phosphorylase inhibitors
09/26/2001EP1135393A2 Substituted benzofuranoindoles and indenoindoles as novel potassium channel openers
09/26/2001EP1135135A1 Chk1 kinase inhibitors
09/26/2001EP0802922B1 Novel amino acid derivatives, method of producing them and pharmaceutical compositions containing these compounds
09/26/2001CN1314999A Modulating multiple lineage kinase proteins
09/26/2001CN1314345A Novel piperidine-4-sulfamide compound, its preparing method and medicinal composition containing them
09/25/2001US6294566 Imidazoline derivatives and uses thereof