Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
11/2000
11/28/2000US6153645 Heterocycles as antimicrobial agents
11/28/2000US6153640 For treating depression, panic attacks, obsessive-compulsive disorders, phobias, impulsive disorders, drug abuse or anxiety
11/28/2000US6153614 Piperazinyl pyrimidine dione compounds selective for adrenoceptors
11/23/2000WO2000069862A2 Hemisynthetic method and intermediates thereof
11/23/2000WO2000069844A1 Oligohydroxyl substituted benzofuran-3-yl and pyridofuranylurea derivatives as phosphodiesterase iv inhibitors
11/23/2000WO2000069830A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
11/23/2000WO2000069821A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
11/23/2000WO2000069433A1 Antagonists of gonadotropin releasing hormone
11/23/2000CA2373590A1 Diketodiazacyclic compounds, diazacyclic compounds and combinatorial libraries thereof
11/23/2000CA2372934A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
11/22/2000EP1053472A1 Energy transfer dyes
11/22/2000EP1053240A1 Glucocorticoid-selective antiinflammatory agents
11/22/2000EP1053239A1 Glucocorticoid-selective anti-inflammatory agents
11/22/2000EP1053215A1 Methods for preparing macrocyclic products by ring-closing diine metathesis
11/22/2000EP1052992A1 Cyclic amine modulators of chemokine receptor activity
11/22/2000CN1273974A Camptothecin derviative, its prepn. method and medicinal compsns. containing same
11/22/2000CN1058717C Method of extracting anhydro tetraodotoxin
11/22/2000CN1058716C Water-soluble fluoroethylcamptothecin derivative and process for prodn. thereof
11/21/2000US6150356 Potassium channel inhibitors and method
11/21/2000US6150355 Phenylpiperidine derivative
11/21/2000US6150354 Compounds for the treatment of Alzheimer's disease
11/21/2000US6150343 10-hydroxy-7-substituted silylcamptothecin derivative is used as anticarcinogenic and antitumor agent
11/21/2000US6149215 Durable slings for vehicle frame turnover machines and method of making the slings
11/16/2000WO2000068225A1 Substituted benzimidazole, the production thereof and the use thereof as means against parasitic protozoa
11/16/2000WO2000068196A1 N-substituted dihydropyrrole derivatives
11/16/2000WO2000067801A2 Prodrugs of chemotherapeutic agents with oxaalkanoic acids
11/16/2000WO2000034285A3 Substituted benzofuranoindoles and indenoindoles as novel potassium channel openers
11/16/2000CA2368831A1 Permeable, water soluble, non-irritating prodrugs of chemotherapeutic agents with oxaalkanoic acids
11/15/2000EP1052261A1 Pyran derivatives and use thereof
11/15/2000EP1051418A1 Process for the preparation of substituted 8-azabicyclo [3.2.1]octanes
11/15/2000EP1051403A1 Novel alkanoic acids and their use in medicine, process for their preparation and pharmaceutical compositions containing them
11/15/2000CN1273586A Method for preparation of asymmetric cyclic ureas through monoaylated diamine
11/15/2000CN1273584A Imidazolyl-cyclic acetals
11/15/2000CN1273241A Hydroxy substituted N-alkoxy hindered amine
11/15/2000CN1058495C Polycyclic systems compound and derivatives thereof as neurotransmitter release enhancers useful in the treatment of cognitive disordes and medicine containing them and its use
11/14/2000US6147223 Lactacystin analogs
11/14/2000US6147099 Oxazolidinedione derivatives, their production and use
11/14/2000US6147089 Cholesteryl ester transfer protein inhibitors used to treat diseases which are exacerbated by low levels of hdl cholesterol and/or high levels of ldl-cholesterol and triglycerides, such as atherosclerosis and cardiovascular
11/14/2000US6147083 Novel substituted 1,2-ethanediamine derivatives which antagonize the pharmacological actions of the endogenous neuropeptide tachykinins known as neurokinins, useful for the treatment of asthma, etc.
11/14/2000US6147075 Analgesics; psychological disorders
11/09/2000WO2000066556A1 Indoline derivatives as progesterone antagonists
11/09/2000WO2000066127A1 Novel highly lipophilic camptothecin analogs
11/09/2000WO2000042045A3 Functionalized heterocycles as chemokine receptor modulators
11/09/2000WO2000039087A3 Substituted (aminoiminomethyl or aminomethyl)benzoheteroaryl compounds as factor xa inhibitors
11/09/2000DE19920551A1 Substituierte Benzimidazole, ihre Herstellung und ihre Verwendung als Mittel gegen parasitäre Protozoen Substituted benzimidazoles, their preparation and their use as agents against parasitic protozoa
11/09/2000CA2371638A1 Indoline derivatives as progesterone antagonists
11/08/2000EP1049700A1 Chemokine receptor antagonists and methods of use therefor
11/08/2000EP1049695A1 2-phenyl substituted imidazotriazinones as phosphodiesterase inhibitors
11/08/2000EP1049675A1 Chemokine receptor antagonists and methods of use therefor
11/08/2000EP1049662A1 Inhibitors of alpha4 mediated cell adhesion
11/08/2000CN1272846A 8-substituted-9H-1,3-dioxolo/4,5-h/2,3/benzodiazepine derivatives, as Ampa/kainate receptor inhibitors
11/08/2000CN1272841A Novel lactam metalloprotease inhibitors
11/08/2000CN1058266C 14-substituted marcfortines and derivatives useful as antiparasitic agents and its application
11/07/2000US6143891 Method for preparing camptothecin derivatives
11/07/2000US6143764 Quinoline and quinazoline derivatives inhibiting platelet-derived growth factor receptor autophosphorylation and pharmaceutical compositions containing the same
11/07/2000US6143761 2,3-dihydrofuro [3,2-β]pyridin, preparation and application thereof in therapy
11/07/2000US6143744 Sulfamide-metalloprotease inhibitors
11/07/2000US6143732 Used as antiviral agent against influenza virus
11/07/2000CA2179306C Dopamine receptor ligands
11/02/2000WO2000064987A1 Novel amidopyrylium fluorescence dyes
11/02/2000WO2000064904A1 5,7-bicyclic amidine derivatives useful as nitric oxide synthase inhibitors
11/02/2000WO2000064877A1 2-aminoquinolinecarboxamides: neurokinin receptor ligands
11/02/2000EP1048658A1 Alicyclic acylated heterocyclic derivatives
11/02/2000EP1048655A1 1,2-dihydro-2-oxoquinoline derivatives
11/02/2000EP1048651A1 Nitrogen-containing tetracyclic compounds
11/02/2000EP1047695A1 Novel bispidine antiarrhythmic compounds
11/02/2000EP1047675A1 Chemokine receptor antagonists and methods of use therefor
11/02/2000EP0713489B1 Photochromic heterocyclochromenes
11/02/2000DE19919120A1 Neue Amidopyrylium-Fluoreszenz-Farbstoffe New amidopyrylium fluorescent dyes
11/01/2000CN1058014C New heterocyclic spiro compounds, process for preparation thereof, and pharmaceutical compositions containing them
10/2000
10/31/2000US6140513 Color forming dye precursor, composition containing the same and color forming heat-sensitive recording material
10/31/2000US6140358 Substituted phenyl keto enols as pesticides and herbicides
10/31/2000US6140339 Monomeric and dimeric arylisoquinoline alkaloids and derivatives thereof
10/31/2000US6140336 Spiro[2H-1-benzopyran-2,4'-piperidine]-4(3H)-one derivatives, acid addition salts thereof and pharmaceutical compositions containing them
10/31/2000US6140328 Heterocyclic cytotoxic agents
10/26/2000WO2000062778A1 Cyclic protein tyrosine kinase inhibitors
10/25/2000EP1045837A1 Monomeric and dimeric arylisoquinoline alkaloids and derivatives thereof
10/25/2000CN1271360A 1,3-dioxolo/4,5-Hl/2,3/benzodiazepine derivatives as AMPA/Kainate receptor inhibitors
10/25/2000CN1271355A Heterocyclic compounds and antitumor agent containing the same as active ingredient
10/25/2000CN1271342A Synthesis of clasto-lactacystin-beta-lactone and analogs thereof
10/24/2000US6137002 Glycoprotein IIb/IIIa antagonists
10/24/2000US6136981 Preparation of 4-phenyl-1,2,3,6-tetrahydropyridines
10/24/2000US6136979 Process for preparing a morphinan derivative
10/24/2000US6136978 Camptothecin analogs and methods of preparation thereof
10/24/2000US6136817 Opioid receptor antagonist compounds
10/24/2000US6136800 Steroids
10/24/2000CA2157247C Physical form of dihydro-2,3-benzodiazepine derivative
10/19/2000WO2000061146A1 Camptothecin analogs and methods of preparation thereof
10/18/2000EP1044977A1 Camptothecin derivatives having antitumor activity
10/18/2000EP1044969A2 Processes and intermediates for preparing anti-cancer compounds
10/18/2000EP1044202A1 1'- 4- 1- (4-fluorophenyl)- 1h-indole-3-yl] -1-butyl]-spiro isobenzofuran- 1(3h),4'- piperidine] hydrohalogenides
10/18/2000EP1044197A2 New piperidinyl-substituted pyridylalkane, alkene and alkine carboxamides
10/18/2000EP1043991A1 Treatment for alzheimer's disease
10/18/2000EP0773965B1 Gas phase production of polydienes
10/18/2000CN1270592A Spiroazabicyclic heterocyclic compounds
10/18/2000CN1270589A Epothilone derivatives
10/18/2000CN1270169A Benzopyrane derivatives and preparation thereof
10/18/2000CN1270166A Derivatives of tricyclo-substituted isohydroxyloxime acid
10/17/2000US6133445 Rigidized trimethine cyanine dyes
10/17/2000US6133308 Synthesis of clasto-lactacystin beta-lactone and analogs thereof