Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726) |
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01/04/2001 | WO2001000206A1 Vla-4 inhibitor compounds |
01/04/2001 | CA2383546A1 Src kinase inhibitor compounds |
01/04/2001 | CA2376785A1 Benzimidazoles and imidazopyridines as respiratory syncytial virus replication inhibitors |
01/04/2001 | CA2376758A1 Hexahydropyrrolo¬1,2-c|pyrimidines as antiviral, antifungal and/or antitumor agents |
01/04/2001 | CA2369308A1 Vla-4 inhibitor compounds |
01/03/2001 | EP1065209A1 Metalloprotease inhibitors, process for their preparation and pharmaceutical compositions containing them |
01/03/2001 | EP1064285A1 Novel cephalotaxane derivatives and process for their preparation |
01/03/2001 | EP0708776B1 Antiallergic imidazoazepines |
01/03/2001 | CN1278823A 1'-[4-[1-(4-Fluorophenyl)-1(H)-indole-3-yl]-1-butyl]-spiro [isobenzofuran-1(3(H),4'-piperidine] hydrohalogenides |
01/03/2001 | CN1278822A 2-phenyl substituted imidazotriazinones as phosphodiesterase inhibitors |
01/03/2001 | CN1278797A Oxo-substituted compouns, process of making, and compositions and methods for inhibiting parp activity |
01/03/2001 | CN1278796A Method for the synthesis of quinoline derivatives |
01/03/2001 | CN1278794A Substituted di-hydroxyl-indol derivatives as protein tyrosine kinase and as protein serine/threenine kinase inhibitors |
01/03/2001 | CN1060175C Method for prepn. of 3-formyl-cephem derivatives |
01/02/2001 | US6169188 Treating cyclooxygenase-2 mediated diseases |
01/02/2001 | US6169097 1-(1,2-Disubstituted piperidinyl)-4-substituted piperidine derivatives |
01/02/2001 | US6169092 3-Ureido-pyridofurans and -pyridothiophenes for the treatment of inflammatory processes |
01/02/2001 | US6169091 Bicyclic heteroaromatic compounds as protein tyrosine kinase inhibitors |
01/02/2001 | US6169090 Heterocyclic compounds and their therapeutic use |
01/02/2001 | US6169080 Highly lipophilic camptothecin derivatives |
01/02/2001 | CA2183313C Novel indane-2-mercaptoacetylamide disulfide derivatives useful as inhibitors of enkephalinase |
01/02/2001 | CA2013449C Antibacterial 5-alkylquinolonecarboxylic acids |
01/02/2001 | CA1341161C Quinolone- and naphthyridone carboxylic acid derivatives, process for their production, antibacterial compositions and feed additives containing them |
12/28/2000 | WO2000078765A2 CHROMENO[4,3,2-de]ISOQUINOLINES AS POTENT DOPAMINE RECEPTOR LIGANDS |
12/28/2000 | WO2000078724A2 Imidazolinderivatives their preparation and their pharmaceutical use |
12/28/2000 | CA2373497A1 Chromeno[4,3,2-de]isoquinolines as potent dopamine receptor ligands |
12/27/2000 | EP1062218A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPases) |
12/27/2000 | EP1062205A2 Inhibitors of phospholipase enzymes |
12/27/2000 | EP0821671B1 Arylsulfonyl hydroxamic acid derivatives as mmp and tnf inhibitors |
12/27/2000 | CN1278251A Novel carboxylic acid derivatives which carry amide side chains, prodn. of same, and use as endothelin receptor antagonists |
12/27/2000 | CN1278249A Biphenyl derivatives as pharmaceuticals |
12/27/2000 | CN1278248A [Indole] naphthopyrans, prepn., compositions and (co) polymer matrics contg. them, synthesis intermediates |
12/26/2000 | US6166209 Piperidine derivatives |
12/26/2000 | US6166034 Spiro piperidine derivatives as 5HT1D receptor antagonists |
12/26/2000 | CA2203494C Energy transfer dyes with enhanced fluorescence |
12/21/2000 | WO2000077010A2 Substituted heterocycle fused gamma-carbolines |
12/21/2000 | WO2000077006A1 Process for the preparation of 1,8-disubstituted-1,3,4,9-tetrahydropyrano (3,4-b)-indole-1-acetic acid esters in a hydroxylic solvent |
12/21/2000 | WO2000077005A1 Naphthopyrans annelated in c5-c6 with a lactam-type c6 ring and compositions and (co)polymer containing them |
12/21/2000 | WO2000077002A1 Substituted heterocycle fused gamma-carbolines |
12/21/2000 | WO2000077001A1 Substituted heterocycle fused gamma-carbolines |
12/21/2000 | WO2000076990A1 New compounds |
12/21/2000 | WO2000076984A2 Novel compounds, their use and preparation |
12/21/2000 | WO2000050426A3 Furo[3, 2-b]pyridines as 5-ht1f agonists |
12/21/2000 | CA2381322A1 Substituted heterocycle fused gamma-carbolines |
12/21/2000 | CA2375860A1 Process for the preparation of 1,8-disubstituted-1,3,4,9-tetrahydropyrano (3,4-b)-indole-1-acetic acid esters in a hydroxylic solvent |
12/21/2000 | CA2375857A1 Naphthopyrans annelated in c5-c6 with a lactam-type c6 ring and compositions and (co)polymer containing them |
12/21/2000 | CA2374239A1 Substituted heterocycle fused gamma-carbolines |
12/21/2000 | CA2373920A1 Substituted heterocycle fused gamma-carbolines |
12/20/2000 | EP1061081A1 7-Oxo-2,3,7,14-tetrahydro-1H-benzo[b]pyrano[3,2-h]acridine carboxylate derivatives, process for their preparation and pharmaceutical compositions containing them |
12/20/2000 | EP1060179A1 Substituted aminomethyl isoxazoline derivatives useful as antimicrobials |
12/20/2000 | EP1060167A1 Novel unsymmetrically substituted carboxylic acid derivatives, method for producing them, and their use as mixed et a?/et b?-receptor antagonists |
12/20/2000 | EP1060163A1 New piperazinyl-substituted pyridylalkane, alkene and alkine carboxamides |
12/20/2000 | EP0714295B1 Fibrinogen receptor antagonists |
12/20/2000 | CN1277613A Poly (ADP-ribose) polymerase ('PARP') inhibitors, methods and pharmaceutical compositions for treating neural or cardiovascular tissue damage |
12/20/2000 | CN1277200A Process for producing hexahydrothiopheno-[3,4-d] imidazole-2,4-diketones compound |
12/19/2000 | US6162798 Cerebrovascular contraction after subarachnoid hemorrhage with quinoline compounds |
12/14/2000 | WO2000075236A1 Extended rhodamine compounds useful as fluorescent labels |
12/14/2000 | WO2000075145A1 Cell adhesion-inhibiting antiinflammatory compounds |
12/14/2000 | WO2000075127A1 Tricyclic fused heterocycle compounds, process for preparing the same and use thereof |
12/14/2000 | CA2390948A1 Cell adhesion-inhibiting antiinflammatory compounds |
12/14/2000 | CA2370013A1 Tricyclic fused heterocycle compounds, process for preparing the same and use thereof |
12/14/2000 | CA2365075A1 Extended rhodamine compounds useful as fluorescent labels |
12/13/2000 | EP1058549A1 THROMBIN OR FACTOR Xa INHIBITORS |
12/13/2000 | CN1276370A Process for preparing anticancer compound, and intermediate |
12/12/2000 | US6160133 Stereospecific biosynthesis of the alcohol by enzymatic reduction of the corresponding aldehyde or ketone using a candida, zygosaccaromyces, or mortierrela microorganism |
12/12/2000 | US6160119 Fused dihydropyrans |
12/12/2000 | US6160003 Antitumor and anticarcinogenic agents |
12/12/2000 | US6160001 Halobenzimidazoles and their use as microbicides |
12/12/2000 | US6159967 such as 1-(2-((2R)-(3,4-dichlorophenyl)-4-(3,4,5-trimethoxybenzoyl) morpholin-2-yl)ethyl)spiro(benzo(c)thiophene-1-(3H), 4'-piperidine)-(2S)-oxide; respiratory disease such as asthma |
12/07/2000 | WO2000073305A1 Preparation of camptothecin and nothapodytine derivatives |
12/07/2000 | WO2000073283A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
12/07/2000 | CA2376024A1 Metabotropic glutamate receptor antagonists and their use for treating central nervous system diseases |
12/07/2000 | CA2340012A1 Preparation of camptothecin and nothapodytine derivatives |
12/06/2000 | EP1057819A1 Phthalazine derivatives and remedies for erectile dysfunction |
12/06/2000 | EP1057814A1 Tetrahydrobenzindole derivatives |
12/06/2000 | EP1056717A1 Arylphenyl-substituted cyclic keto-enols |
12/06/2000 | EP1056451A1 Bicyclic pyrrole derivatives as mcp-1 inhibitors |
12/06/2000 | CN1275979A Isoquinolines as urokinase inhibitors |
12/05/2000 | US6156897 Method for purifying 20(S)-camptothecin |
12/05/2000 | US6156783 Spiroazabicyclic compounds, processes for their preparation, and their pharmaceutical use |
12/05/2000 | US6156772 Indole hormone inhibitors |
12/05/2000 | US6156762 Indolomorphinan derivative and agent for curing and preventing cerebral disorder |
12/05/2000 | US6156757 1,2,3,4-tetrahydro-benzofuro[3,2-C]pyridine derivatives |
12/05/2000 | US6156494 Solid phase synthesis using substrate having regions, each region is an optical fiber having covalently bound reactive groups; fibers are used to direct light, heat or both to compounds tethered to its surface |
11/30/2000 | WO2000071541A1 Optically active quinoline carboxylic acid derivatives having 7-pyrrolidine substitutes causing optical activity and a process for preparing thereof |
11/30/2000 | WO2000071534A1 Heterocyclic substituted aminoazacycles useful as central nervous system agents |
11/30/2000 | WO2000071518A2 Heterocyclic analgesic compounds and their use |
11/30/2000 | WO2000071517A1 Phenoxypropylamine compounds |
11/30/2000 | CA2716369A1 Phenoxypropylamine compounds |
11/30/2000 | CA2373793A1 Heterocyclic substituted aminoazacycles useful as central nervous system agents |
11/30/2000 | CA2372887A1 Heterocyclic analgesic compounds and their use |
11/29/2000 | EP1054887A1 Bicyclic pyridine and pyrimidine derivatives as neuropeptide y receptor antagonists |
11/29/2000 | EP1054870A1 Heterocyclic topoisomerase poisons |
11/29/2000 | EP1054869A1 3,4-dihydroquinoline derivatives as nitrogen monoxide synthase (nos) inhibitors |
11/29/2000 | CN1275124A Phthalazine derivatives and remedies for erectile dysfunction |
11/29/2000 | CN1274723A Dicyclic compound, medicine composition containing the same and use thereof |
11/29/2000 | CN1274718A Novel benzo-[3,4] cyclobutano [1,2-C] pyrroles compound, its prepn. and medicine composition containing the same |
11/29/2000 | CN1274711A New intermediate for preparation of anti-histamine piperidine derivatives |
11/29/2000 | CN1058967C Novel pyridine compounds, processes for their preparation and pharmaceutical compositions thereof |
11/28/2000 | US6153655 Terminally-branched polymeric linkers and polymeric conjugates containing the same |