Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
01/2005
01/12/2005EP1494672A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity
01/12/2005EP1494671A1 1-(4-piperidinyl)benzimidazolones as histamine h3 antagonists
01/12/2005EP1494670A1 Medicine for treating cancer
01/12/2005EP1494668A2 Use of benzimidazole analogs in the treatment of cell proliferation
01/12/2005EP1494663A1 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin k inhibitors for the treatment of bone loss
01/12/2005EP1434773A4 Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
01/12/2005EP1355906B1 2h-1-benzopyran derivatives, processes for their preparation and pharmaceutical compositions thereof
01/12/2005EP0991628B1 QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR P56lck TYROSINE KINASES
01/12/2005CN1564820A Heterocyclic compounds for use in the treatment of disorders of the urinary tract
01/12/2005CN1564814A Triazine compounds, polymers comprising triazine structural units, and processes for the preparation of these polymers
01/12/2005CN1564811A Acylsulfonamides as inhibitors of steroid sulfatase
01/12/2005CN1564685A Pyrrolidinone derivatives
01/12/2005CN1563001A Method for preparing terazosin hydrochloride of optical activity
01/12/2005CN1563000A Xinduo antibiotic, preparation method, and produced pesticide for preventing and curing damage of crop
01/12/2005CN1184206C Prepn process of pyrazole derivative
01/12/2005CN1184204C Piperidine compounds for use as CCR-3 inhibitors
01/12/2005CN1183907C Imidazoline compound, preparing process thereof and pharmaceutical composition contg. same
01/11/2005US6841684 Imidiazoles having reduced side effects
01/11/2005US6841680 2-(Halophenyl)-quinoline derivatives for neuropathic pain; side effect reduction
01/11/2005US6841674 N-heterocyclic derivatives as NOS inhibitors
01/11/2005US6841673 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents
01/11/2005US6841670 Biphenyl-substituted triazines
01/11/2005US6841566 Viral polymerase inhibitors
01/11/2005US6841560 Substituted isoquinoline derivatives and their use as anticonvulsants
01/11/2005US6841552 3a,4,5,9b-tetrahydro-1H-benz[e]indol-2-yl amine-derived neuropeptide Y receptors ligands useful in the treatment of obesity and other disorders
01/06/2005WO2005000839A1 Process for producing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/06/2005WO2005000838A1 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
01/06/2005WO2005000837A1 Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
01/06/2005WO2005000822A1 N-{‘4-substituted piperazine-1-sulfonylmethyl!alkyl}-n-hydroxyfomamide compounds as metalloproteinase inhibitors
01/06/2005WO2005000821A1 Tachykinin receptor antagonists
01/06/2005WO2005000817A2 Diphenylpyridine derivatives, preparation and therapeutic application thereof
01/06/2005WO2005000813A1 Heteroarylamino-phenylketone derivatives and their use as kinase inhibitors
01/06/2005WO2005000811A1 3-aminopyrrolidines as inhibitors of monoamine uptake
01/06/2005WO2005000781A1 Biaryloxymethylarene-carboxylic acids
01/06/2005WO2005000353A1 Serum cholesterol lowering agnet or preventive or therapeutic agent for atherosclerosis
01/06/2005WO2005000305A1 3-aminopiperidines and 3-aminoquinuclidines as inhibitors of monoamine uptake
01/06/2005WO2005000249A2 Preparation of chemical compounds
01/06/2005WO2005000233A2 Novel therapeautic agents for the treatment of cancer, metabolic diseases and skin disorders
01/06/2005WO2004103977A3 Process for the preparation of pyrimidine derivatives
01/06/2005WO2004101528A3 Isoquinoline derivatives and their use as gfat inhibitors
01/06/2005WO2004099193A3 1-aryl-3-(indol-5-yl)-prop-2-en-1-ones, compositions comprising the same and use thereof
01/06/2005WO2004089947A3 Novel compounds having an antibacterial activity
01/06/2005WO2004076445A3 Compounds and methods of treating cell proliferative diseases, retinopathies and arthritis
01/06/2005WO2004037166A3 Therapeutic guanidines
01/06/2005WO2003032912A9 Treatment of cns disorders using cns target modulators
01/06/2005US20050004367 Sulfonamide derivatives
01/06/2005US20050004360 Compounds and methods for modulation of estrogen receptors
01/06/2005US20050004206 suspending crystal strutured or amorphous lipitor in diluents comprising alcohols and/or water mixtures to cause conversion, then separating the diluents; monodispersity
01/06/2005US20050004204 2-Iminopyrrolidine derivatives
01/06/2005US20050004202 Such as 3-[1-(3-methoxypropyl )-1H-indazol-3-yl]-4-[1-(3-pyridinyl )-1H-indol-3-yl]-1H-pyrrole-2,5-dione; protein kinase C and/or glycogen synthase kinase-3 diseases
01/06/2005US20050004200 Pyrazole compounds as integrin receptor antagonists derivatives
01/06/2005US20050004197 Thrombin receptors antagonists; oral efficacy
01/06/2005US20050004180 Conditions mediated by beta chemokine receptor 2, monocyte chemotactic protein 1 and/or their interaction; such as 4-acetyl-5-cyclohexyl-3-amino-1-(4-methylphenyl)-1,5-dihydro-2H-pyrrol-2-one
01/06/2005US20050004176 Pyrazole-amide compounds useful as kinase inhibitors
01/06/2005US20050004166 Imino acid derivatives as inhibitors of matrix metalloproteinases
01/06/2005US20050004162 Piperidinyl indole and tetrohydropyridinyl indole derivatives and method of their use
01/06/2005US20050004152 Thiazole compounds useful as inhibitors of protein kinase
01/06/2005US20050004151 Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators
01/06/2005US20050004149 Pyrimidine compound and medicinal composition thereof
01/06/2005US20050004148 Human immunodeficiency and hepatitis B infections; high activity, low toxicity
01/06/2005US20050004136 Novel amidoalkyl-piperidine and amidoalkyl-piperazine derivatives useful as neurokinin receptor modulators
01/06/2005US20050004133 Inhibiting ligand gated ion channel vanilloid receptor (VR1); pain relievers; such as 6-(3,4-dichloro-phenyl)-N-(2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-nicotinamide
01/06/2005US20050004126 Method of determining potential allosterically-binding matrix metalloproteinase inhibitors
01/06/2005US20050004125 Such as 4-[[4-(1-methyl-1H-imidazol-2-yl)-2-pyrimidinyl]amino]-benzonitrile; bipolar disorder, pain, type 2 diabetes
01/06/2005US20050004124 Synergistic mixture; antidiabetic agents; antiischemic agents
01/06/2005US20050004119 Trypsin like serine protease enzyme inhibitors
01/06/2005US20050004116 Triazole inhibitors of type 2 methionine aminopeptidase
01/06/2005US20050004114 Heterocycle substituted carboxylic acids
01/06/2005US20050004112 C-fms kinase inhibitors
01/06/2005US20050004111 Degenerative joints disease; osteoarthritis
01/06/2005US20050004110 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
01/06/2005US20050004109 Methods and compositions for the treatment and prevention of tumors, tumor-related disorders and cachexia
01/06/2005US20050004104 Methods for the protection of memory and cognition
01/06/2005US20050004103 Vasopressin active material; antidiabetic agents; diuretics; bioavailability
01/06/2005US20050004097 Indole derivatives
01/06/2005US20050004096 Indole derivatives, process for producing the same and drugs containing the same as the active ingredient
01/06/2005US20050004081 Pharmaceutical combinations for the treatment of cancer
01/06/2005US20050004078 Nucleotide analogs with six-membered rings
01/06/2005US20050003232 Quinoxaline derivatives, organic semiconductor device and electroluminescent device
01/06/2005CA2672071A1 Process for preparing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/06/2005CA2531020A1 Cannabinoid receptor modulator
01/06/2005CA2530581A1 Novel therapeautic agents for the treatment of cancer, metabolic diseases and skin disorders
01/06/2005CA2530377A1 Process for preparing 3-acylaminobenzofuran-2-carboxylic acid derivative
01/06/2005CA2529875A1 Biaryloxymethylarene-carboxylic acids
01/06/2005CA2529468A1 N-{[4-substituted piperazine-1-sulfonylmethyl]alkyl}-n-hydroxyfomamide compounds as metalloproteinase inhibitors
01/06/2005CA2528619A1 Diphenylpyridine derivatives, preparation and therapeutic application thereof
01/06/2005CA2526487A1 Heterocyclic methyl sulfone derivative
01/05/2005EP1493743A1 Substituted bipiperidine intermediates and derivatives thereof
01/05/2005EP1493733A2 Fungicidal heterocyclic aromatic amides, their compositions and methods of use
01/05/2005EP1493057A1 Colour photographic recording material
01/05/2005EP1492786A1 Pyridinoylpiperidines as 5-ht1f agonists
01/05/2005EP1492785A1 New compounds
01/05/2005EP1492771A1 Quinoline and isoquinoline derivatives, method for the production thereof and use thereof as anti-inflammatory agents
01/05/2005EP1492765A2 Novel gamma secretase inhibitors
01/05/2005EP1492571A2 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
01/05/2005EP1492568A1 Cancer treatment method comprising administration of an erb-family inhibitor and a raf and/or ras inhibitor
01/05/2005EP1492536A1 4-(n-phenylamino)-quinazolines / quinolines as tyrosine kinase inhibitors
01/05/2005EP1492526A2 Improved prodrugs of cc-1065 analogs
01/05/2005EP1492487A2 Mitotic kinesin inhibitors
01/05/2005EP1226126B1 Pyrimidine derivatives