Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
01/2005
01/20/2005US20050014705 E.g., dimethylcarbamic acid, 2-oxo-3-benzyl-4-methyl-2H-1-benzopyran; affects both the Tumor Necrosis Factor alpha level and transcription activity of NuclearFactor kappa Beta; antiimmunoinflammatory agents and autoimmune properties; antiarthritis agents; rheummatic diseases; osteoporosis; leukemia
01/20/2005US20050014700 Cbi analogues of cc-1065 and the duocarmycins
01/20/2005US20050014650 Delta 1-pyrrolines used as pesticides
01/20/2005US20050014278 Acid-labile isotope-coded extractant (ALICE) and its use in quantitative mass spectrometric analysis of protein mixtures
01/20/2005US20050011411 Anthraquinone, xanthene dyes: coloring ink
01/20/2005DE10329860A1 Sulfonamidderivate polycyclischer Farbstoffe für analytische Anwendungen Sulfonamide derivatives of polycyclic dyes for analytical applications
01/20/2005CA2532056A1 Pyrrole-2, 5-dione derivatives as liver x receptor modulators
01/20/2005CA2531757A1 Benzofuran derivatives and their use in the treatment of microbial infections
01/20/2005CA2531751A1 Pyrazolyl-indole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
01/20/2005CA2530737A1 Cck-1 receptor modulators
01/20/2005CA2530538A1 Thiophenylaminoimidazolines as prostaglandin i2 antagonists
01/20/2005CA2530450A1 5-substituted quinazolinone derivatives
01/20/2005CA2530312A1 Arylamine-substituted quinazolinone compounds
01/20/2005CA2528626A1 Indoles useful in the treatment of inflammation
01/19/2005EP1498411A1 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient
01/19/2005EP1498109A1 Furan derivatives and dyeing composition comprising a furan derivative as coupler
01/19/2005EP1497298A1 Derivatives of 2,2,4-trisubstituted tetrahydrofuran as antifungal agents
01/19/2005EP1497287A1 Quinolinone derivatives
01/19/2005EP1497284A2 Pyrrolidinium derivatives as antagonists of m3 muscarinic receptors
01/19/2005EP1497282A2 Inhibitors of serine protease, particularly hepatitis c virus ns3-ns4 protease
01/19/2005EP1497279A2 Substituted indoles and their use as 5ht-reuptake inhibitors and as 5ht ligands
01/19/2005EP1497240A1 Non-heating clay composites for building materials
01/19/2005EP1496898A2 Tyrosine kinase inhibitors
01/19/2005EP1496894A1 Angiogenesis inhibitors
01/19/2005EP1496892A2 1h-benzo(f)indazol-5-yl derivatives as selective glucocorticoid receptor modulators
01/19/2005EP1395574B1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
01/19/2005EP0958293B1 Nanomolar, non-peptide inhibitors of cathepsin d
01/19/2005CN1568323A Activator for peroxisome proliferator-activated receptor delta
01/19/2005CN1568320A 异羟肟酸衍生物 Hydroxamic acid derivatives
01/19/2005CN1568187A 2H-2, 3-dinitrogen phenodiazine-1-ketone and using method thereof
01/19/2005CN1568185A Compounds effecting glucokinase
01/19/2005CN1566098A Isoquinoline compound, preparation method and application of salt thereof
01/19/2005CN1566096A Prostaglandin agonists and their use to treat bonedisorders
01/19/2005CN1566091A Molindone derivatives and use for preparing antineoplastic medicine thereof
01/19/2005CN1185229C 3-indolyl-4-phenyl-1H-pyrrole-2, 5-dione derivatives as inhibitors of glycogen synthase kinase-3beta
01/19/2005CN1185228C Hydroxyphenyl-piperidin-4-ylidene-methyl-benzamide derivatives for treatment of pain
01/19/2005CN1185227C Novel compounds
01/19/2005CN1185223C Novel Compounds and methods for synthesis and therapy
01/19/2005CN1185216C Fungicides
01/19/2005CN1185213C Azetidine derivatives, preparation and pharmaceutical compositions thereof
01/18/2005US6844441 Hypoglycemic agents; dietetics; gastrointestinal disorders; antidepressants; gastrointestinal disorders; antiinflammatory agents
01/18/2005US6844437 Chemical intermediates; anticholesterol agents, antilipemic agents
01/18/2005US6844344 Depression, anxiety; tobacco or nicotine withdrawal; such as 1-(benzofuran-4-yl)oxy-3-(4-(6-methoxybenzo(b)thiophen-2-yl)piperidinyl)-2 -propanol oxalate
01/13/2005WO2005003131A1 Tricyclic delta opioid modulators
01/13/2005WO2005003124A1 Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
01/13/2005WO2005003123A1 Novel pyridine derivatives as jnk specific inhibitors
01/13/2005WO2005003122A1 5ht4-antagonistic 4-(aminomethyl)-piperidine benzamides
01/13/2005WO2005003121A1 Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5ht4-antagonists
01/13/2005WO2005003103A2 2, 4, 6-tri-substituted 6-membered heterocycles and their use in the treatment of neurodegenerative diseases
01/13/2005WO2005003102A1 Methods of preparation of dehydro-diketopiperazines in liquid phase or of solid supported phase
01/13/2005WO2005003101A2 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005WO2005003100A2 4-arylamino-quinazolines as activators of caspases and inducers of apoptosis
01/13/2005WO2005003099A2 Pyrimidines useful as modulators of voltage-gated ion channels
01/13/2005WO2005003097A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005WO2005003086A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
01/13/2005WO2005002552A2 Benzimidazole derivatives and their use as protein kinases inhibitors
01/13/2005WO2004106329A3 Novel antiinfective compounds and their pharmaceutical compositions
01/13/2005WO2004099192A3 Heterocycle substituted carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
01/13/2005WO2004072047A8 Indoles, benzimidazoles or naphhimidazoles as histone deacetylase (hdac) inhibitors
01/13/2005WO2004064764A3 Substituted alkyl amido piperidines
01/13/2005WO2004052883A3 Process for the separation of enantiomers
01/13/2005WO2004050035A3 Benzimidazoles and analogs thereof as antivirals
01/13/2005US20050009900 3-Substituted with a heterocyclic group, e.g., 2-Chloro-5-[1-(2,3-dihydroxy-propyl)-5-methyl-1H-pyrazol-3-yl]-N-(1-hydroxy-cycloheptylmethyl)-benzamide; treatment of IL-1 mediated disorders, including osteo- and rheumatoid arthritis, allergies, asthma, COPD, cancer, and reperfusion or ischemia in stroke
01/13/2005US20050009894 Benzimidazole derivatives and their use as KDR kinase protein inhibitors
01/13/2005US20050009892 Phenyloxazole derivatives lower blood triglyceride, glucose, insulin; hyperlipidemia, arteriosclerosis, diabetes mellitus, hypertension, obesity; 2-methyl-2-[6-(5-methyl-2-phenyloxazol-4-yl)-(E)-4-hexenyloxy]propionic acid
01/13/2005US20050009876 Indazole compounds, compositions thereof and methods of treatment therewith
01/13/2005US20050009870 3-(amino)sulfonylamino-substituted, e.g., N-(1,6-Dibenzyl-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-benzenesulfonamide and N-(1-Benzyl-2-oxo-6-(thiophen-3-yl)-1,2,3,4-tetrahydroquinolin-3-yl)benzenesulfonamide; eating, metabolic, obesity, cognitive, neurological, pain, inflammatory and psychiatric disorders
01/13/2005US20050009867 Quinoline derivatives and their use as tyrosine kinase inhibitors
01/13/2005US20050009864 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
01/13/2005US20050009860 Tricyclic delta-opioid modulators
01/13/2005US20050009855 1-(hydroxy, oxo, or epoxy)-3-oxo-3'-benzaminocarbonyl-4'-(carboxy or carboxylate)-1,2,3-trihydroindene-2-spiro-2'-tetrahydrofuran derivatives; these compounds interfere with the E1-E2-DNA complex during initiation of DNA replication
01/13/2005US20050009853 Pyrimidine derivatives for the treatment of abnormal cell growth
01/13/2005US20050009850 Quinazoline compounds with therapeutic use
01/13/2005US20050009844 Inhibitors of p38
01/13/2005US20050009840 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer
01/13/2005US20050009838 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
01/13/2005US20050009819 1-Aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands
01/13/2005US20050009818 Therapeutic heterocyclic compounds
01/13/2005US20050009817 Substituted heteroaryls
01/13/2005US20050009815 4-Aminoquinoline compounds
01/13/2005US20050009812 Remedies for stress diseases comprising mitochondrial benzodiazepine receptor antagonists
01/13/2005US20050009809 Acridine derivatives and their use as medicaments
01/13/2005US20050009808 Azabicyclo compound matrix metalloprotease inibitor and skin preparation
01/13/2005US20050009785 Heterocyclic compounds
01/13/2005US20050009730 Sleep disorders; side effect reduction
01/13/2005US20050009076 Conjugate of hormone (thyroxine) and inosine-5'-monophosphate dehydrogenase inhibitor (such as mycophenolic acid)
01/13/2005US20050008968 Basic compound, resist composition and patterning process
01/13/2005CA2531327A1 Compounds and therapeutical use thereof
01/13/2005CA2531061A1 Pyrimidines useful as modulators of voltage-gated ion channels
01/13/2005CA2531050A1 Pharmaceutical compounds
01/13/2005CA2530389A1 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005CA2528119A1 Cis-2,4,5-triaryl-imidazolines
01/12/2005EP1495757A1 Phosphodiesterase iv inhibitor containing pyridylacrylamide derivative
01/12/2005EP1495040A1 Method for synthesizing beta-l-fluoro-2',3'didehydcytidine (beta-l-fd4c)
01/12/2005EP1495018A1 Tricyclic thrombin receptor antagonists
01/12/2005EP1495004A2 Benzenesulfonamide derivatives and their use as dopamine d3 and d2 receptor ligands
01/12/2005EP1495003A1 Fredericamycin derivatives
01/12/2005EP1495002A1 Benzamide derivatives useful as histone deacetylase inhibitors
01/12/2005EP1495001A1 Antibacterial agents
01/12/2005EP1494989A2 Compounds that modulate ppar activity and methods for their preparation