Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
11/2004
11/04/2004WO2004094375A2 4 - (3,4 - disubstituted phenyl) - pyrrolidin-2-one compounds as phosphodiesterase 4 inhibitors
11/04/2004WO2004093873A1 2-phenyl-benzimidazol and 2-phenyl-imidazo-`4,5!-pyridine derivatives as checkpoint kinase cds1 (chk2) inhibitors for the treatment of cancer
11/04/2004WO2004093856A2 Combination of a cox-2 inhibitor and an alkylating-type antineoplastic agent for treatment of neoplasia
11/04/2004WO2004093789A2 Use of galr3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods
11/04/2004WO2004087673A3 Migrastatin analogs and uses thereof
11/04/2004WO2004078874A3 Novel dye complexes and use thereof in imaging members and methods
11/04/2004WO2004078747A8 Novel cyanopyridine derivatives useful in the treatment of cancer and other disorders
11/04/2004WO2004074812A3 Library of biphenyl derivatives useful for identifying compounds having both beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity
11/04/2004WO2004069792A8 Quinoline-derived amide modulators of vanilloid vr1 receptor
11/04/2004WO2004060865A3 N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines
11/04/2004WO2004056774A3 Substituted biphenyl-4-carboxylic acid arylamide analogues as capsaicin receptor modulators
11/04/2004WO2004004657A3 Hiv integrase inhibitors
11/04/2004WO2003087044A3 Novel carboxamide compounds for use in mch receptor related disorders
11/04/2004US20040220402 4-(substituted cycloalkylmethyl) imidazole-2-thiones, 4-(substituted cycloalkenylmethyl) imidazole-2-thiones, 4-(substituted cycloalkylmethyl) imidazol-2-ones and 4-(substituted cycloalkenylmethyl) imidazol-2-ones and related compounds
11/04/2004US20040220254 Process for preparing 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl) ethyl]-2-isopropyl-4-phenyl-1H-pyrrole-3-carboxylic acid phenylamide
11/04/2004US20040220253 Synthesis of pyrrole amides
11/04/2004US20040220247 N-[4-(4,5-Dihydro-1H-imidazol-2-yl-amino)-benzyl]-4-methoxy-benzamide and derivatives; prostaglandin inhibitors; urinary tract disease, disease related pain, neuropathic pain, respiratory asthma, allergy
11/04/2004US20040220232 Organometallic reagent reacted with an activated carboxylic acid to produce a ketone which is reacted with carbon disulfide and dihalomethane, further reacting the dithietane product with a secondary amine, and condensing the thioamide with hydrazine; useful as p38 kinase and COX-2 inhibitors
11/04/2004US20040220230 transfroming growth factor antagonist; therapy for urogenital disorders, cardiovascular disorders
11/04/2004US20040220229 insulin resistance; central nervous system disorders; vision defects; anticholesterol agents;antilipemic agents; antiischemic agents
11/04/2004US20040220223 Novel human NK3 receptor-selective antagonist compounds, method for obtaining them and pharmaceutical compositions containing them
11/04/2004US20040220222 Malonamide derivatives
11/04/2004US20040220207 Chemokine receptor binding heterocyclic compounds
11/04/2004US20040220200 Compositions useful as protein kinase inhibitors
11/04/2004US20040220196 antitumor agents; 4-amino-5-fluoro-3-(6-( 4-methylpiperazin-1-yl)1H-benzimidazol-2-yl)-quinolin-2-one
11/04/2004US20040220193 Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound
11/04/2004US20040220191 Substituted N-aryl heterocycles, process for their preparation and their use as medicaments
11/04/2004US20040220188 Alkylidene pyrazolidinedione derivatives
11/04/2004US20040220182 tyrosine kinase inhibitor; antitumor agents
11/04/2004US20040220177 Anticancer agents
11/04/2004US20040220173 central nervous system disorders; psychological disorders; Parkinson's disease; Huntington's disease ; sleep disorders
11/04/2004US20040220171 anticoagulants; immunomoderators; antiinflammatory agents
11/04/2004US20040220148 5-Membered ring heterocycles as inhibitors of leucocyte adhesion and as VLA-4 antagonists
11/04/2004CA2523200A1 Nk-2 antagonist basic linear compounds and formulations containing them
11/04/2004CA2522687A1 Pyrazole derivatives as phosphodiesterase 4 inhibitors
11/04/2004CA2522682A1 Indazole derivatives as jnk inhibitors
11/04/2004CA2522667A1 Combination of a cox-2 inhibitor and an alkylating-type antineoplastic agent for treatment of neoplasia
11/04/2004CA2522631A1 4 - (3,4 - disubstituted phenyl) - pyrrolidin-2-one compounds as phosphodiesterase 4 inhibitors
11/04/2004CA2522562A1 2-phenyl-benzimidazol and 2-phenyl-imidazo-`4,5!-pyridine derivatives as checkpoint kinase cds1 (chk2) inhibitors for the treatment of cancer
11/04/2004CA2518180A1 Isoquinoline-5-sulfonic acid amides as inhibitors of akt (protein kinase b)
11/03/2004EP1473293A1 Chromenon derivatives
11/03/2004EP1472244A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors
11/03/2004EP1472236A1 Method for preparing benzisoxazole methane sulfonyl chloride and its amidation to form zonisamide
11/03/2004EP1472230A2 Ansamycins having improved pharmacological and biological properties
11/03/2004EP1472228A1 Process for the manufacture of hmg-coa reductase inhibitors
11/03/2004EP1472227A2 Process for the manufacture of organic compounds
11/03/2004EP1472225A2 2-piperazine-pyridines useful for treating pain
11/03/2004EP1472223A1 Gamma secretase inhibitors
11/03/2004EP1472222A1 Piperidylcarboxamide derivatives and their use in the treatment of tachykinim-mediated diseases
11/03/2004EP1472216A2 Novel bicyclic hydroxamates as inhibitors of histone deacetylase
11/03/2004EP1472215A2 (oxime)carbamoyl fatty acid amide hydrolase inhibitors
11/03/2004EP1471915A2 2,4-pyrimidinediamine compounds and their uses
11/03/2004EP1471910A2 Substituted quinazolin-4-ylamine analogues as modulators of capsaicin receptors
11/03/2004EP1471786A1 Microbiocidal n-phenyl-n- 4-(4-pyridyl)-2-pyrimidin-2-yl]-amine derivatives
11/03/2004EP1232153B1 Imidazole derivatives and their use as raf kinase inhibitors
11/03/2004EP1206452B1 Novel method for preparing benzoperhydroisoindole compounds
11/03/2004EP0956021B1 L-beta-dioxolane uridine analogs for treating and preventing infections by ebv, vzv and hv-8
11/03/2004EP0942906B1 Compounds useful for inhibition of farnesyl protein transferase
11/03/2004CN1543456A Substituted naphthyl benzofuran derivatives as inhibitors of plasminogen activator inhibitor-1 (PAI-1)
11/03/2004CN1543455A 3-phenoxy-4-pyridazinol derivative and herbicide composition containing the same
11/03/2004CN1543453A 6-(aryl-amido or aryl-amidomethyl)-naphthalen-2-yloxy-acidic derivatives as inhibitors of plasminogen activator inhibitor type-1 (PAI-1)
11/03/2004CN1543346A Novel compounds
11/03/2004CN1542011A Sulphur containing heterocyclic and naphthalimides compound and use thereof
11/03/2004CN1542001A Small molecule inhibitors of rotamase enzyme activity
11/03/2004CN1541532A Herbicidal synergistic composition, and method of controlling weeds
11/03/2004CN1173985C Novel diphenylarsines
11/03/2004CN1173974C Piperidylaminomethyltrifluoromethyl cyclic ether compound as p substance antagonist
11/03/2004CN1173964C Novel benzofuranone derivative and process for producing same
11/03/2004CN1173951C Substituted 1,3-diaryl-2-pyridine-2-yl-3-(pyridine-2-ylamino)-propanol derivatives, methods for their production, pharmaceutical compositions containing the same and their use
11/03/2004CN1173947C 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides
11/03/2004CN1173946C Method for preparing an N-[(aliphatic or aromatic) carbonyl]-2-aminoacetamide compound and a cyclyzed compound
11/02/2004US6812353 Intermediates for central nervous system medications; primary amine functionality
11/02/2004US6812349 Process and intermediates for the preparation of imidazopyridines
11/02/2004US6812243 Indole derivatives and their use for the treatment of malignant and other diseases based on pathological proliferation
11/02/2004US6812235 2-acylamino- beta -alanine derivatives and a pharmaceutically acceptable salt, useful as fibrinogen receptor antagonists
11/02/2004US6812233 Therapeutic nucleosides
11/02/2004US6812225 Pyschological disorders; antidepressants
11/02/2004US6811998 Conjugates of uncompetitive inhibitors of inosine monophosphate dehydrogenase
11/02/2004CA2315614C Pyrazoles
11/02/2004CA2301787C New derivatives of benzo[3,4]cyclobuta[1,2-c]pyrrole, the procedure for preparing them and the pharmaceutical compounds that contain them
11/02/2004CA2296313C 2-aminopyridines containing fused ring substituents as nos inhibitors
11/02/2004CA2129040C Styryl derivatives and processes for their preparation
10/2004
10/28/2004WO2004092196A2 Tie-2 modulators and methods of use
10/28/2004WO2004092164A1 Cyclic amine derivatives and their use in the treatment of inflammation-related disorders mediated by bradykinin
10/28/2004WO2004092163A1 Phenylazole compound, production process, and antioxidant drug
10/28/2004WO2004092154A1 Compositions useful as inhibitors of protein kinases
10/28/2004WO2004092145A1 Alpha substituted carboxylic acid as ppar modulators
10/28/2004WO2004092144A2 Quinazoline compounds useful as p38 kinase inhibitors
10/28/2004WO2004092116A1 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof
10/28/2004WO2004092115A2 Hydroxamates as therapeutic agents
10/28/2004WO2004091605A1 Preventive/remedy for retinal nerve diseases containing alkyl ether derivatives or salts thereof
10/28/2004WO2004091604A1 Compounds that modulate ppar activity and methods of preparation
10/28/2004WO2004091514A2 Cgrp receptor antagonists
10/28/2004WO2004091488A2 Estrogen receptor modulators
10/28/2004WO2004078732B1 N-aryl heteroaromatic products, compositions containing same and use thereof
10/28/2004WO2004078479A3 Imaging system
10/28/2004WO2004078103A3 G-lactam derivatives as prostaglandin agonists
10/28/2004WO2004078030A3 Rhodol derivatives useful as image dyes
10/28/2004WO2004076444A3 Novel hydroxycoumaranone derivatives as antitumor and antimetastatic
10/28/2004WO2004075823A8 Novel benzimidazole and imidazopyridine derivatives and use thereof as a medicament