Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
10/2004
10/28/2004WO2004058721A3 Pyrazole derivatives modulators of hepatocyte growth factor (scatter factor) activity
10/28/2004WO2004000826A8 Processes for producing epoxytriazole derivative and intermediate therefor
10/28/2004US20040215024 naphthopyrans having an oxygen-containing heterocyclic group F annelated on the i, j, or k side of the naphthopyran ring; have interesting photochromic properties; part of polymer or in polymer matrix; ophthalmic lenses
10/28/2004US20040215017 Such as 2-methylpropyl-(4-bromo-3-fluorophenyl)carbamate
10/28/2004US20040214887 for example, 6,9-Dihydroxy-2,2,13,13-tetramethyl-tetradecanedioic acid, 2,2,13,13-Tetramethyl-tetradecane-1,6,9,14-tetraol, 6,10-Dihydroxy-2,2,14,14-tetramethyl-pentadecanedioic acid; treatment of Alzheimer's Disease, metabolic syndrome disorder, cancer, cardiovascular disease, diabetic nephropathy
10/28/2004US20040214875 Imidazolinylmethyl aralkylsulfonamides
10/28/2004US20040214874 Inhibition of protein-tyrosine kinase cmet to block cancer cell proliferation, oral bioavailibility; 2-(2,6-dichlorophenyl)-4-phenyl-5-(pyrimidin-4yl)-1H-imidazoles
10/28/2004US20040214868 Treatment or prevention of type 2 diabetes; chemical synthesis; 2-[ benzoyl]aminopyridine-5-carboxylate derivatives
10/28/2004US20040214857 Substituted benzimidazoles and imidazo-[4,5]-pyridines
10/28/2004US20040214845 Barbiturates as integrin antagonists and their use for treating inflammatory diseases
10/28/2004US20040214844 N4-acylcytosine nucleosides for treatment of viral infections
10/28/2004US20040214843 Such as spiro(cyclohexane-1-4'-(3',4'-dihydro)quinazolin)-2'(1'H)-one for treatment of T-cell-related diseases, autoimmune diseases, osteoarthritis, multiple sclerosis, osteoporosis, asthma and cancer
10/28/2004US20040214841 Quinazoline derivatives for treatment of tumours
10/28/2004US20040214818 Alzheimer's disease; Parkinson's disease; Huntington's disease; cognition activators; learning enhancement; central nervous system disorders
10/28/2004US20040214817 Diaminotriazoles useful as inhibitors of protein kinases
10/28/2004US20040214814 Pyrazole compounds useful as protein kinase inhibitors
10/28/2004US20040214784 covalent conjugates with mono-, di- , poly- or thiaalkanoic acids; ability to adjust the solubility of steroidal molecules, lipophilicity and bioavailability by altering the structure and length of the acid chain; avoids or reduces the local irritation caused by the parent drug
10/28/2004US20040213264 Service class and destination dominance traffic management
10/28/2004CA2522595A1 Compositions useful as inhibitors of protein kinases
10/28/2004CA2522522A1 Quinazoline compounds
10/28/2004CA2522266A1 Phenylazole compound, production process therefor and antioxidant
10/28/2004CA2522118A1 Compounds that modulate ppar activity and methods of preparation
10/28/2004CA2522084A1 Cyclic amine derivatives and their use in the treatment of inflammation-related disorders mediated by bradykinin
10/28/2004CA2521937A1 Bicyclic compounds having bradykinin receptors affinity and pharmaceutical compositions thereof
10/28/2004CA2521915A1 Alpha substituted carboxylic acid as ppar modulators
10/28/2004CA2520323A1 Tie-2 modulators and methods of use
10/27/2004EP1471068A1 Process for total synthesis of ecteinascidins and intermediates therefor
10/27/2004EP1471064A1 Coumarin derivatives, process for their production and use thereof
10/27/2004EP1471063A1 Compounds and methods of treating cell proliferative diseases, retinopathies and arthritis
10/27/2004EP1471057A1 Pyrimidinylacetic acid derivatives useful for the treatment of diseases mediated by CRTH2
10/27/2004EP1471055A1 6-phenylpyridyl-2-amine derivatives
10/27/2004EP1470143A1 Compounds that inhibit factor xa activity
10/27/2004EP1470137A1 Edg receptor agonists
10/27/2004EP1470121A1 Pyrimidine derivatives as rho-kinase inhibitors
10/27/2004EP1470113A1 Pyrimidinone viral polymerase inhibitors
10/27/2004EP1470112A1 Substituted pyridazinones as inhibitors of p38
10/27/2004EP1469851A1 Melanocortin receptor agonists
10/27/2004EP1212269B1 Methods for preparing n- (aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
10/27/2004EP1073428B1 Dihydroxyphenyl derivatives for hepatoprotection and treatment of liver diseases
10/27/2004EP0960108B1 Matrix metalloproteinase inhibitors
10/27/2004CN1541259A Fluorescent diketopyrrolopyrrole analogues
10/27/2004CN1541215A HIV inhibiting pyrimidines derivatives
10/27/2004CN1541211A Derivatives of N-(arylsulfonyl) beta-aminoacids comprising substituted aminomethyl group, prepn. method thereof and pharmaceutical compsns. contg same
10/27/2004CN1541208A 2-anilino-pyrimidine derivatives as cyclin dependent kinase inhibitors
10/27/2004CN1541203A 4-(phenyl-(piperidin-4-YL)-amino)-benzamide derivatives and their use for treatment of pain, anxiety or gastrointestinal disorders
10/27/2004CN1539825A Compounds useful to treat retroviral infections
10/27/2004CN1172930C PDE IV inhibiting pyridine derivatives
10/27/2004CN1172917C Steroid receptor modulator compounds and methods
10/26/2004US6809199 (Halo-benzo carbonyl)heterocyclo fused phenyl p38 kinase inhibiting agents
10/26/2004US6809113 For therapy of arthritis, asthma, atherosclerosis, diabetic nephropathy, inflammatory bowel disease, crohn's disease, multiple sclerosis, nephritis, pancreatitis, pulmonary fibrosis, psoriasis, restenosis transplant rejection
10/26/2004US6809102 For therapy of proliferative diseases, such as cancer; to interrupt mitosis
10/26/2004US6809100 Hydroxamic acid derivatives
10/26/2004US6809098 Compounds
10/26/2004US6809093 Drug resistance therapy
10/26/2004US6809088 Derivatives of 2-(iminomethyl)amino-phenyl, their preparation, their use as medicaments and the pharmaceutical compositions containing them
10/26/2004CA2295752C Novel process for manufacturing paroxetine solid dispersions
10/26/2004CA2196263C Process for the preparation of 4-oxoimidazolinium salts
10/26/2004CA2023811C Process and intermediates for preparing compounds having a disubstituted acetylene moiety and retinoic acid-like biological activity
10/21/2004WO2004090543A1 Assay method
10/21/2004WO2004089947A2 Novel compounds having an antibacterial activity
10/21/2004WO2004089940A1 Novel heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
10/21/2004WO2004089939A1 Condensed furan derivatives as adenosine antagonists
10/21/2004WO2004089932A1 Substituted pyrazole compounds
10/21/2004WO2004089931A1 Substituted pyrazoles
10/21/2004WO2004089927A1 Novel methods for the treatment of inflammatory diseases
10/21/2004WO2004089925A1 Pi-3 kinase inhibitor prodrugs
10/21/2004WO2004089914A1 Benzenesulphonamide derivatives as herbicides or desiccant/defoliant compounds
10/21/2004WO2004089910A1 1,3,4-substituted pyrazoles for use as 5-ht receptor antagonists in the treatment of psychoses and neurological disorders
10/21/2004WO2004089908A2 3-azabicyclo[3.2.1]octane derivatives
10/21/2004WO2004089903A1 Piperidine derivatives as renin inhibitors for the treatment of hypertension
10/21/2004WO2004089901A2 Phospholipase c inhibitors for use in treating inflammatory disorders
10/21/2004WO2004089894A1 Process for preparing 5-(4-fluorophenyl)-1-[2-((2r,4r)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)ethyl]-2-isopropyl-4-phenyl-1h-pyrrole-3-carboxylic acid phenylamide
10/21/2004WO2004089892A2 Diarylmethyl and related compounds having beta2 andrenergic receptor agonist and muscarinic receptor antagonist activity
10/21/2004WO2004089888A1 Pyrazole compounds
10/21/2004WO2004089373A1 4- (4-(heterocyclylalkoxy}phenyl)-1-(heterocyclyl-carbonyl)piperidine derivatives and related compounds as histamine h3 antagonists for the treatment of neurological diseases such as alzheimer’s
10/21/2004WO2004089370A1 4-phenyl-piperidine compounds and their use as modulators of opioid receptors
10/21/2004WO2004089367A1 Pharmaceutical use of substituted 1,2,4-triazoles
10/21/2004WO2004089363A1 Substituted azabicyclo hexane derivatives as muscarinic receptor antagonists
10/21/2004WO2004089362A1 2-cyanopyrroles and their analogues as ddp-iv inhibitors
10/21/2004WO2004065380A8 1,2,3-trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prpphylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
10/21/2004WO2004058144A3 Antibacterial agents
10/21/2004WO2004056786A3 Pyrimidine derivates for the treatment of abnormal cell growth
10/21/2004WO2004047674A3 Oxyge-containing heterocyclic fused naphthopyrans
10/21/2004US20040209981 Protective coating for food, beverages, drugs; cosmetics; shampoo; radiation resistance
10/21/2004US20040209948 especially naphthalene sulfonamides, used for treating asthma
10/21/2004US20040209940 potent antibacterial activity against various bacteria including drug-resistant strains
10/21/2004US20040209938 Novel 1,3-dihydro-2H-indol-2one derivatives, process for preparing them and pharmaceutical compositions containing them
10/21/2004US20040209936 Compounds that modulate PPAR activity and methods of preparation
10/21/2004US20040209929 Fused heteroaryl carboxylic acids as PPAR agonists
10/21/2004US20040209925 e.g., phenyl ((1S,2R)-1-(3,5-difluorobenzyl)-3-{[(1S)-7-ethyl-1,2,3,4-tetrahydronaphthalen-1-yl]amino}-2-hydroxypropyl)carbamate; inhibitors of the beta-secretase enzyme that are useful in the treatment of Alzheimer's disease and other diseases characterized by deposition of A beta peptide
10/21/2004US20040209922 Pyridine matrix metalloproteinase inhibitors
10/21/2004US20040209915 substituted with an N- (p-hydroxy-alpha-hydroxybenzylaminoalkylpiperidinyloxy- (or -amino-)carbonylamino group; useful for identifying compounds having both beta 2 adrenergic receptor agonist and muscarinic receptor antagonist activity
10/21/2004US20040209914 Aromatic sulfone hydroxamic acids and their use as protease inhibitors
10/21/2004US20040209913 Bicyclic Heteroaromatic Alanines
10/21/2004US20040209912 Substituted isoquinoline derivatives and their use as anticonvulsants
10/21/2004US20040209908 New derivatives of hydantoins, thiohydantoins, pyrimidinediones and thioxopyrimidinones, their preparation processes and their use as medicaments
10/21/2004US20040209904 Substituted quinazoline compounds useful as P38 kinase inhibitors
10/21/2004US20040209894 e.g., 1-(4-chloroanilino)-4-[2-(pyridin-3-yl)-ethyl]-isoquinoline and 5-[4-(tert-butyl)-anilino]-8-[(6-methoxy-pyridin-3-yl)-methyl]-[1,6]naphthyridine
10/21/2004US20040209884 Fused azabicycic compounds that inhibit vanilloid receptor subtype 1(VR1) receptor
10/21/2004US20040209883 Nitrogen-containing heterocyclic compounds and their use as raf inhibitors