Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
02/2008
02/20/2008EP1581522B1 Flavaxate derivatives as muscarinic receptor antagonists
02/20/2008EP1432417B1 Substituted benzimidazole compounds and their use for the treatment of cancer
02/20/2008EP1427417B1 3-substituted 6,7-dihydroxytetrahydroisoquinoline derivatives for use as antibacterial agents
02/20/2008CN101128458A Tricyclic delta-opioid modulators
02/20/2008CN101128457A 凝血酶受体拮抗剂 Thrombin receptor antagonists
02/20/2008CN101128436A 甘氨酸衍生物及其用途 Glycine derivatives and their use
02/20/2008CN101128434A Amide derivatives
02/20/2008CN101125849A 1,4-pyran derivative and use thereof
02/20/2008CN100369908C New taxane derivatives
02/20/2008CN100369899C Substituted indazoles with anti-cancer activity
02/20/2008CN100369898C Nicotinamide derivates useful as p38 inhibitors
02/19/2008US7332608 Potassium channel modulators; cardiovascular disorders; antiarrhythmia agents; synthesis
02/19/2008US7332518 Carboxamides as fungicides in agriculture
02/19/2008US7332517 1-(1H-indol-3-ylmethyl)-3-(4-nitrophenyl)-5-[2-(4-phenyl-1H-imidazol-2-yl)ethyl]-2thioxo-4imidazolidinone; somastatin receptor affinity; acromegaly, hypophyseal adenomas, endocrine gastroenteropancreatic tumors, as carcinoid syndrome and gastrointestinal bleeding
02/19/2008US7332511 Vanilloid receptor ligands and their use in treatments
02/19/2008US7332509 Used for controlling animal pests, in particular arthropods, such as insects and acarids, and helminths
02/19/2008US7332501 Indol-3-yl-carbonyl-spiro-piperidine derivatives as V1a receptor antagonists
02/19/2008US7332496 Methods of using sodium channel blockers
02/19/2008US7332495 Aralkyl-ketone piperazine derivatives and their uses as new antalgic or ataractic agent
02/19/2008US7332493 [3-Methyl-4-(pyridin-3-yloxy)-phenyl]-(6-piperidin-3-ylethynyl-quinazolin-4-yl)-amine; selective inhibitors of receptor tyrosine kinases and non-receptor tyrosine kinases (eg: Ick, src, abl) or serine/threonine kinases (e.g.: cyclin dependent kinases); carcinoma
02/19/2008US7332490 inhibit smooth muscle cell proliferation by modulating Heparan Sulfate Proteoglycans (HSPGs); inhibit or block glycated protein and Advanced Glycation Endproducts (AGE) produced induction of the signaling-associated inflammatory response in endothelial cells; antiproliferative and antiinflammatory agent
02/19/2008US7332489 Methods and compositions of novel triazine compounds
02/19/2008US7332488 Methods and compositions of novel triazine compounds
02/19/2008US7332487 Nitrogen-containing 5-membered ring compound
02/19/2008US7332484 2,4-pyrimidinediamine compounds and their uses
02/19/2008US7332483 3-(5-benzamido-2-chlorophenyl)-7-methoxy-3,4-dihydroquinazolin-4-one;cytokines (tumor necrosis factor and interleukins) inhibitor; antiinflammatory agent, rheumatoid arthritis, osteoarthritis, psoriasis, chronic obstructive pulmonary disease
02/19/2008US7332481 Thrombopoietin mimetics
02/19/2008US7332260 Naphthopyrans annelated in C5-C6, their preparation and compositions and (CO)polymer matrices containing them
02/19/2008CA2210072C Crop protection products
02/19/2008CA2207100C Pyrimidine derivatives
02/14/2008WO2008019292A2 Compositions and methods for potentiating antibiotic activity
02/14/2008WO2008018639A2 Glycine transporter inhibitor
02/14/2008WO2008017710A1 1h-quinolin-4-one compounds, with affinity for the gaba receptor, processes, uses and compositions
02/14/2008WO2008017685A1 Nitrate esters of piperidines
02/14/2008WO2008017515A1 Nucleosides for suppressing or reducing the development of resistance in cytostatic therapy
02/14/2008WO2008008493A3 Alkyne-substituted pyridone compounds and methods of use
02/14/2008WO2008005954A3 Tryphostin-analogs for the treatment of cell proliferative diseases
02/14/2008WO2008002245A3 Imidazol-pyrimidine derivatives for treatment of diseases related to glycogen synthase kinase (gsk3)
02/14/2008WO2008002244A3 Imidazol-pyrimidine derivatives for treatment of diseases related to glycogen synthase kinase (gsk3)
02/14/2008WO2007139955A8 Triazole compounds that modulate hsp90 activity
02/14/2008WO2007136302A3 Active substances, pharmaceutical composition and a method for the production and use thereof
02/14/2008WO2007110704A3 Macrolide compositions as therapeutic agent
02/14/2008US20080039640 Process for the preparation of nitrile compounds
02/14/2008US20080039622 2,4-pyrimidinediamine compounds and their uses
02/14/2008US20080039505 5-((((2R)-1-(4-((S)-1-hydroxyhexyl)phenyl)-4-methyl-5-oxopyrrolidin-2-yl)methoxy)methyl)thiophene-2-carboxylic acid; glaucoma or ocular hypertension
02/14/2008US20080039502 e.g. N-[4-(4'-Methoxy-biphenyl-4-yloxymethyl)-5-methyl-furan-2-carbonyl]-benzenesulfonamide; prostaglandin E4 receptor antagonist; analgesic, antiinflammatory agent; migraines and headache
02/14/2008US20080039479 Compounds and therapeutical use thereof
02/14/2008US20080039473 Preparation and utility of substituted quinazoline compounds with alpha-adrenergic blocking effects
02/14/2008US20080039465 Triazolyl phenyl benzenesulfonamides
02/14/2008US20080039450 Compounds
02/14/2008US20080039449 [1,4]benzodiazepine derivatives, used for treating osteoarthritis, pancreatitis, glomerulonephritis, rheumatoid arthritis, inflammatory bowel disease, Crohn's disease, psoriasis, graft vs host disease, leukemia, septic shock, multiple sclerosis, and inflammatory bowel disease
02/14/2008US20080039447 CDK-Inhibitory pyrimidines, their production and use as pharmaceutical agents
02/14/2008US20080039442 Compounds With Kv4 Ion Channel Activity
02/14/2008US20080038745 Nucleotide analogs with six-membered rings
02/14/2008DE102006037724A1 Verwendung von Ascorbinsäurederivaten zur Funktionalisierung von Matrices Use of ascorbic acid for the functionalization of matrices
02/14/2008CA2660636A1 Nucleosides, drugs containing these and use thereof
02/14/2008CA2660538A1 Nitrate esters of piperidines
02/14/2008CA2660421A1 1h-quinolin-4-one compounds, with affinity for the gaba receptor, processes, uses and compositions
02/13/2008EP1887003A1 3-[4-heterocyclyl -1,2,3-triazol-1-yl]-n-aryl-benzamides as inhibitors of the cytokines production for the treatment of chronic inflammatory diseases
02/13/2008EP1886996A1 1H-Quinolin-4-one compounds, with affinity for the GABA receptor, processes, uses and compositions
02/13/2008EP1886994A1 Cyclic amine compounds as CCR5 antagonists
02/13/2008EP1885715A1 Selected tetracyclic tetrahydrofuran derivatives containing a cyclic amine side chain
02/13/2008EP1885710A1 Substituted aminopropenyl piperidine or morpholine derivatives as novel inhibitors of histone deacetylase
02/13/2008EP1689741B1 Benzoyl amino pyridyl carboxylic acid derivatives as glucokinase activators
02/13/2008EP1480973B1 1,4-disubstituted benzofused cycloalkyl urea compounds useful in treating cytokine mediated diseases
02/13/2008EP1335908B1 Peroxisome proliferator activated receptor alpha agonists
02/13/2008EP1299390B1 Pyrimidine compounds and their use in the preparation of a triazolo -pyrimidine carba nucleoside
02/13/2008CN101124220A 5-substituted quinoline and isoquinoline derivatives, a process for their production and their use as anti-inflammatory agents
02/13/2008CN101124212A Chroman derivatives and their use as 5-HT receptor ligands
02/13/2008CN101123962A 可诱导一氧化氮合成酶二聚化的抑制剂 Inducible nitric oxide synthase dimerization inhibitor
02/13/2008CN101121711A Pyrazolcarbazone derivatives and application thereof
02/13/2008CN100368415C 6-alkenyl-, 6-alkinyl-and 6-epoxy-epothilone derivatives, process for their production, and their use in pharmaceutical preparations
02/13/2008CN100368404C Substituted alkylaminopyridazinone derivatives, process for the preparation thereof and pharmaceutical composition containing the same
02/12/2008US7329762 Prodrugs of mitotic kinesin inhibitors
02/12/2008US7329753 Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors
02/12/2008US7329683 Moderation of cortisol; non-insulin dependent diabetes; hypotensive agents; using a 1,2,4 triazole compound
02/12/2008US7329680 Heterocycle substituted carboxylic acids
02/12/2008US7329675 Substituted azabicyclic compounds
02/12/2008US7329672 N4-(1,4-Benzoxazin-6-yl)-5-fluoro-N2-[3-(N-methylamino)carbonylmethyleneoxyphenyl]-2,4-pyrimidinediamine or a salt, hydrate, solvate and/or N-oxide; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors
02/12/2008US7329671 N2,N4-bis(3-hydroxyphenyl)-5-fluoro-2,4-pyrimidinediamine or a salt, hydrate, solvate and/or N-oxide; inhibit the IgE and/or IgG receptor signaling cascades that lead to the release of chemical mediators; Syk kinase inhibitors
02/12/2008US7329664 Substituted (7-pyridyl-4-phenylamino-quinazolin-2-yl)-methanol analogues
02/12/2008US7329657 Indazolyl-substituted pyrroline compounds as kinase inhibitors
02/12/2008US7329655 Drugs that inhibit phosphorylation kinases as an antigrowth or antiproliferation agent
02/12/2008US7329318 Methods of crystal precipitation
02/12/2008CA2374737C Novel process for synthesis of heteroaryl-substituted urea compounds
02/12/2008CA2290992C (imidazol-5-yl)methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation
02/12/2008CA2258701C Carboxamide derivatives of pyrrolidine, piperidine and hexahydroazepine for the treatment of thrombosis disorders
02/07/2008WO2008016973A1 2,4-diaminoquinazolines for spinal muscular atrophy
02/07/2008WO2008016762A1 Fluorogenic protein kinase substrates
02/07/2008WO2008016596A2 Pseudobase benzo [c] phenanthridines with improved efficacy, stability, and safety
02/07/2008WO2008016184A1 Alpha-carboline derivatives and methods for preparation thereof
02/07/2008WO2008015525A2 An improved process for the preparation of alfuzosin hydrochloride
02/07/2008WO2008014822A1 6-1h-imidazo-quinazoline and quinolines derivatives, new potent analgesics and anti-inflammatory agents
02/07/2008WO2008014815A1 Amidine derivatives of 2-heteroaryl-quinazolines and quinolines; potent analgesics and anti-inflammatory agents
02/07/2008WO2007144487A3 Dual molecules containing a peroxide derivative, their synthesis and therapeutic uses
02/07/2008WO2007136300A3 Substituted indoles and a method for the production and use thereof
02/07/2008WO2007117778A3 Quinolones useful as inducible nitric oxide synthase inhibitors
02/07/2008US20080033175 Process for preparation of 4-amino-3-quinolinecarbonitriles
02/07/2008US20080033172 Mutagenic Heterocycles
02/07/2008US20080033023 Therapeutic compounds