Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/2008
06/17/2008US7388021 Novel pyridyl or phenyl ureas and analogues; Purinoreceptors inhibitors; 1-(4-tert-butylphenyl)-3-(2-(3-isopropylphenoxy)pyridin-3-yl)urea; for the treatment of a thromboembolic disorders
06/17/2008US7388014 Quinazoline derivatives and therapeutic use thereof
06/17/2008CA2501799C Pyrazole compounds for treatment of neurodegenerative disorders
06/17/2008CA2395193C Pyrrolidine derivatives as cyclic amp-specific phosphodiesterase inhibitors
06/17/2008CA2393749C Substituted 8-arylquinoline phosphodiesterase-4 inhibitors
06/17/2008CA2383114C Substituted 1,2,3,4,5,6-hexahydro-2,6-methano-3-benzazocines and their use as pharmaceutical compositions
06/17/2008CA2276532C Frangible compounds for pathogen inactivation
06/12/2008WO2008070661A1 Substituted pyrimidines as adenosine receptor antagonists
06/12/2008WO2008070447A2 Anti-viral compounds
06/12/2008WO2008069322A1 Metal coordination compound and light-emitting material using the same
06/12/2008WO2008069242A1 Novel bicyclic heterocyclic compound
06/12/2008WO2008068423A2 P<0}{0pyrrol derivatives, preparation and use of the same in therapy<0}
06/12/2008WO2008068268A1 Antibacterial quinoline derivatives
06/12/2008WO2008068157A1 2-aminoquinolines as 5-ht(5a) receptor antagonists
06/12/2008WO2008067687A1 The salts of imidazol-5-carboxylic acid derivatives, preparation methods and use therrof
06/12/2008WO2008067644A1 Inhibitors of hiv replication
06/12/2008US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection
06/12/2008US20080139666 Anti-Inflammatory and Psoriasis Treatment and Protein Kinase Inhibition by Hydroxy Stilbenes and Novel Stilbene Derivatives and Analogues
06/12/2008US20080139627 Heterocyclic amide and imine derivatives, processes for their preparation, compositions comprising them and their use as pesticides
06/12/2008US20080139625 Pyrrolidin-2-One and Piperidin-2-One Derivatives as 11-Beta Hydroxysteroid Dehydrogenase Inhibitors
06/12/2008US20080139622 Decahydronaphthalene Compounds
06/12/2008US20080139619 Novel derivatives of benzimidazale and imidazo-pyridine and their use as medicaments
06/12/2008US20080139566 4-Benzyloxymethyl-2-hydroxymethyl-2-(tetrazol-2-yl)oxetane; DNA and RNA nucleoside polymerase inhibitor; viral, fungal, bacterial, protozoa infections; anticarcinogenic agent: breast cancer
06/12/2008US20080139547 N-Hydroxyalkynylbenzamide (or hydroxamate) derivatives; anticarcinogenic and antiproliferative agents
06/12/2008US20080139546 e.g. 3-(3,4-dihydroquinolin-1(2H)-yl)-N-{[8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinolin-2-yl]methyl}propan-1-amine; modulators of serotonin 5-HT1A receptor activity and/or serotonin reuptake; antidepressant, anxiolytic agent, cognition activator; schizophrenia, sexual disorders
06/12/2008US20080139536 Benzodiazepines for Treating or Preventing Rsv Infection
06/12/2008US20080139523 Oxime-containing macrocyclic acyl guanidines as beta-secretase inhibitors
06/12/2008CA2671749A1 Bicyclic compounds and uses as antidiabetics
06/12/2008CA2669996A1 Pyrrol derivatives, preparation and use of the same in therapy
06/12/2008CA2669590A1 2-aminoquinolines as 5-ht(5a) receptor antagonists
06/12/2008CA2668517A1 Antibacterial quinoline derivatives
06/11/2008EP1930322A1 1-(4-piperidinyl)-1,3-dihydro-2H-benzoxazole-2-one derivatives and related compounds as nociceptin analogs and ORL1 ligands for the treatment of pain
06/11/2008EP1928863A2 Pharmaceutical dosage forms and compositions comprising lecoztan
06/11/2008EP1928862A1 2-aminopyrimidine derivatives as modulators of the histamine h4 receptor activity
06/11/2008EP1928840A1 1h-pyrazole 4-carboxylamides, their preparation and their use as 11beta-hydroxysteroid dehydrogenase
06/11/2008EP1928833A1 Novel quinoline compounds capable of binding at the cb2 receptor
06/11/2008EP1463501B1 Cis-imidazolines as mdm2 inhibitors
06/11/2008EP1313713B1 4-pyrimidinamine derivatives, pharmaceutical compositions and related methods
06/11/2008EP1230235B1 Compounds with antibacterial and antiparasitic properties
06/11/2008CN101198328A Solid pharmaceutical preparation containing (R)-(-)-2-[5-(4-fluorophenyl)-3-pyridylmethylaminomethyl]-chroman
06/11/2008CN100393716C Coumarin derivatives, and their preparing method and use as alpha, receptor agonist
06/11/2008CN100393715C Imidazole deriviatives and their use as peripherally-selective inhibitors of dopamine-beta-hydroxylase
06/11/2008CN100393714C Gyrase inhibitors and uses thereof
06/10/2008US7385063 Method for preparing imidazole derivatives
06/10/2008US7385059 3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dependent kinase and glycogen synthase kinase-3 modulators
06/10/2008US7384962 Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
06/10/2008US7384961 Saturated and unsaturated heteroarylcycloalkylmethyl amines as anti-depressants
06/10/2008US7384958 Quinoline inhibitors of cGMP phosphodiesterase
06/10/2008US7384957 3,4-dihydro-1H-isoquinolin-2-yl-derivatives
06/10/2008US7384947 Treating cancer with anticarcinogenic agents 3-Amino-9-chloro-5,6,7,8-tetrahydro-naphtho[2,3-b]furan-2-yl))-(2-methyl-pyridin-3-yl)-methanone; antiproliferative agents
06/10/2008US7384944 Organ grafting; antiarthritic agents; inflammatory bowel disease
06/10/2008US7384943 Substituted chroman derivatives
06/10/2008CA2429590C Novel crystal forms of atorvastatin hemi-calcium and processes for their preparation as well as novel processes for preparing other forms
06/10/2008CA2238889C Method for selective protection of baccatin derivatives and its application to taxane synthesis
06/05/2008WO2008067390A2 Metabolites of 5-fluoro-8-{4-[4-(6-methoxyquinolin-8-yl)piperazin-1-yl]piperidin-1-yl} quinoline and methods of preparation and uses thereof
06/05/2008WO2008066097A1 Carboxylic acid derivative
06/05/2008WO2008065754A1 Substituted carbinol compound
06/05/2008WO2008065493A1 Pyrazole analogs
06/05/2008WO2008064788A1 Cyclically substituted 3,5-dicyano-2-thiopyridines and use thereof
06/05/2008WO2008043788A3 Novel compounds
06/05/2008US20080132710 Atrasentan hydrochloride crystalline form 2
06/05/2008US20080132562 Tetronic and tetramic acids
06/05/2008US20080132550 4,5-diphenyl-2-amino-4,5-dihydro-imidazole derivatives; antiinflammatory agent, neurodegenerative diseases; inflammatory bowel disease, rheumatoid arthritis and diseases associated with central nervous system, such as Alzheimer's disease
06/05/2008US20080132523 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
06/05/2008US20080132521 Isoquinolinone Derivatives and Their Use As Therapeutic Agents
06/05/2008US20080132504 2, 4-Pyrimidinediamines Useful In The Treatment Of Neoplastic Diseases, Inflammatory And Immune System Disorders
06/05/2008US20080132481 Use of 3-substituted amino-2-carboxy-substituted indoles or benzo(b)thiophenes or esters thereof that modulate T helper (Th) cells; treating allergy, asthma, rhinitis, dermatitis, B-cell lymphomas, tumors and diseases associated with bacterial, rhinovirus or respiratory syncytial virus (RSV) infections
06/05/2008DE19946341B4 Verfahren zur Herstellung substituierter Phenylsulfonylharnstoffe aus Sulfohalogeniden A process for the preparation of substituted phenylsulfonylureas of Sulfohalogeniden
06/05/2008DE19739797B4 Stabilisatorkombination Stabilizer combination
06/05/2008DE102006056740A1 Cyclisch substituierte 3,5-Dicyano-2-thiopyridine und ihre Verwendung Cyclic substituted 3,5-dicyano-2-thiopyridines and their use
06/05/2008DE102006056526A1 Verfahren zur stereoselektiven Synthese von chiralen Epoxiden durch ADH-Reduktion von alpha-Abgangsgruppen-substituierten Ketonen und Cyclisierung Method for the stereoselective synthesis of chiral epoxides by ADH reduction of alpha-leaving group-substituted ketones and cyclization
06/05/2008CA2671080A1 Carboxylic acid derivatives
06/05/2008CA2670105A1 Substituted dihydroimidazoles and their use in the treatment of tumors
06/04/2008EP1927594A1 1,2,3-Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto such as diabetes and hyperglycemia
06/04/2008EP1927589A1 Quinoline derivatives
06/04/2008EP1926734A1 Pyrazolopyridine and pyrazolopyrimidine compounds useful as kinase enzymes modulators
06/04/2008EP1926727A1 4-chromenonyl-1,4-dihydropyridinecarbonitriles and the use thereof
06/04/2008EP1926724A1 Analogs of dehydrophenylahistins and their therapeutic use
06/04/2008EP1926708A1 Biaryl substituted heterocycle inhibitors of lta4h for treating inflammation
06/04/2008EP1592687B1 Benzofurane derivatives and the use of the same as antidepressants and anxiolytics
06/04/2008EP1487817B1 Piperidine derivatives useful as modulators of chemokine receptor activity
06/04/2008EP1343775B1 Piperazine derivatives
06/04/2008EP1237887B1 9-(piperazinylalkyl)carbazoles as bax-modulators
06/04/2008EP1204643B1 Fungicidal heterocyclic aromatic amides and their compositions, methods of use and preparation
06/04/2008CN101193985A Cyanine coloring matter and optical recording medium
06/04/2008CN101193885A Benzofuran derivative as 5-HT6 receptor inhibitor
06/04/2008CN101193880A Exo- and diastereo- selective syntheses of himbacine analogs
06/04/2008CN101193869A Glucocortioid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/04/2008CN101193868A Pyrimidine derivatives for the treatment of GABA B mediated nervous system disorders
06/04/2008CN101193867A N-substituted benzimidazolyl c-Kit inhibitors and combinatorial benzimidazole library
06/04/2008CN101193860A 有机化合物 Organic compounds
06/04/2008CN101193852A Analogs of 4-hydroxyisoleucine and uses thereof
06/04/2008CN101190912A Antiviral compound and preparation method thereof
06/04/2008CN101190894A Fatty acid synthetic enzyme inhibitor and medical preparation use thereof
06/04/2008CN100391944C Indoles useful in the treatment of androgen-receptor related diseases
06/03/2008US7381828 Forming a salt such as a tartrate or mandelate of 6-amino-2,2-dimethyltetrahydro-3aH-cyclopenta[d][1,3]-dioxol-4-yl]oxy}-1-ethanol, chemical intermediates
06/03/2008US7381827 Processes and intermediates
06/03/2008US7381824 Quinoline derivatives
06/03/2008US7381741 In which the amino is substituted by arylmethyl- or heteroarylmethyl- group, e.g., 2-Methoxybenzyl)-(2-phenylpyrrolidin-3-yl)-amine and 5-{[2-(3-Chloro-phenyl)-pyrrolidin-3-ylamino]-methyl}-6-methoxy-3-methyl-1,1a,3,7b-tetrahydro-3-aza-cyclopropa[a]naphalen-2-one; neurokinin 1 (Substance P) inhititors
06/03/2008US7381733 Tropane derivatives having dopamine reuptake inhibitor activity for the treatment of ischemic diseases