Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
04/2008
04/16/2008CN100381437C Compounds, compositions and methods
04/16/2008CN100381428C Quinazolone and quinazolone compound and application thereof
04/16/2008CN100381425C 6-amino-1H-indazole and its pharmaceutical compositions as phosphodiesterase 4 inhibitors, and use thereof
04/16/2008CN100381423C Novel piperidine derivatives as modulators of chemokine receptor CCR5
04/15/2008USRE40245 Gyrase inhibitors and uses thereof
04/15/2008US7358377 Schweinfurthin analogues
04/15/2008US7358364 Substituted carboxylic acids
04/15/2008US7358276 2-Oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
04/15/2008US7358274 Methods for treating or preventing cancer using Benzopyranone Compounds
04/15/2008US7358269 selective to alpha2B and/or alpha2C adrenergic receptors, minimal cardivascular and/or sedatory activity; pain
04/15/2008US7358266 Cyclopropyl and cyclobutyl epothilone analogs
04/15/2008US7358257 sulfonylurea derivatives, sulfonylthiourea derivatives, sulfonylguanidine derivatives, sulfonylcyanoguanidine derivatives, thioacylsulfonamide derivatives, and acylsulfonamide derivatives; effective for prevention and treatment of cardiovascular diseases, antithrombotic agents
04/15/2008US7358249 Heterocyclic compounds having inhibitory activity against HIV integrase
04/15/2008US7358248 treatment of diabetes and/or cancer; useful in the treatment of syndrome X; capable of inhibiting Protein tyrosine phosphatases
04/15/2008US7358239 Treating impaired fundic relaxation; [1(R),[A-(3 alpha ,4 alpha )]]-1-[1-[(3,4-dihydro-2H-1-benzopyran-2-yl)methyl]-3-methoxy-4-piperidinyl]-2(1H)-pyrimidinone
04/15/2008CA2411468C Thrombopoietin mimetics
04/15/2008CA2240107C Novel diphenylarsines
04/10/2008WO2008042639A1 Compounds and compositions as protein kinase inhibitors
04/10/2008WO2008042282A2 Imidazole-4, 5-dicarboxamide derivatives as jak-2 modulators
04/10/2008WO2008040649A2 Pyrazine-2-carboxamide derivatives as cb2 receptor modulators
04/10/2008WO2008040445A1 Novel crystalline modification of 4- (n-methyl-2-chloro-5-pyridylmethylamino) -2,5-dihydrofuran-2-one
04/10/2008WO2008040236A1 Flavones derivatives, preparation methods and uses thereof
04/10/2008WO2008040097A1 Furanone compounds and lactam analogues thereof
04/10/2008WO2008016596A3 Pseudobase benzo [c] phenanthridines with improved efficacy, stability, and safety
04/10/2008WO2007144652A3 Parp inhibitors
04/10/2008WO2007143597A3 Organic compounds
04/10/2008WO2007120824A3 Processes for the synthesis of azetidinone
04/10/2008WO2007110868A3 Heterocyclic compounds and uses thereof in the treatment of sexual disorders
04/10/2008WO2007019180A3 Compounds for binding to eralpha/beta and gpr30, methods of treating disease states and conditions mediated through these receptors and identification thereof
04/10/2008US20080086003 1-[4-amino-3,5-dibromo-N-[[4-(2,3,4,5-tetrahydro-2(1H)-oxo-1,3-benzodiazepin-3-yl)-1-piperidinyl]carbonyl]-D-phenylalanyl]-4-(1-piperidinyl)-piperidine-p-toluenesulphonate or other inorganic organic salts; calcitonin gene related peptide-antagonist; useful for treating headache and migraine
04/10/2008US20080085923 Thrombosis, atherosclerosis, restenosis, hypertension, angina pectoris, arrhythmia, heart failure, and cancer; use with other drugs such as aspirin, clodipogrel, prasugrel, cangrelor, Fragmin; himbacine derivatives
04/10/2008US20080085910 For inflammatory bowel disease; oral administration, bioavailability, pharmacokinetics; 2-(2,6-Dichlorobenzamido)-5-[4-(ethyl-pyrimidin-2-ylamino)phenyl]pent-4-enoic acid methyl ester for example
04/10/2008US20080085894 Alpha-(n-sulfonamido)acetamide derivatives as beta-amyloid inhibitors
04/10/2008CA2664621A1 Pyrazine-2-carboxamide derivatives
04/10/2008CA2663856A1 Jak-2 modulators and methods of use
04/09/2008EP1908760A1 Chromane and thiochromane-3-yl-1,3-dihydroimidazoles as inhibitors of dopamine-beta-hydroxylase and methods of their preparation
04/09/2008EP1908759A2 3,4-dihydro-3-amino-2H-1-benzopyrane and -benzothiopyrane derivatives as dopamine-beta-hydroxylase Inhibitors and methods of their preparation
04/09/2008EP1908752A1 Novel 2-quinolone derivative
04/09/2008EP1907387A1 An oxime derivative and preparations thereof
04/09/2008EP1906964A1 Piperazinone derivatives useful as histamine h3 receptor antagonists and/or inverse agonists
04/09/2008EP1828125B1 Arylpiperazine derivatives and their use as ligangs selective of the dopamine d3 receptor
04/09/2008EP1727793B1 Substituted azetidine compounds as cyclooxygenase-1 - cyclooxygenase-2 inhibitors, and their preparation and use as medicaments
04/09/2008EP1594867B1 Phenylacetamides and their use as glucokinase modulators
04/09/2008EP1461320B1 Enantioselective transformation of alfa,beta-unsaturated ketones using chiral organic catalysts
04/09/2008EP1439837B1 Pyrazolidinone compounds as ligands of the prostaglandin ep2 and/or ep4 receptors
04/09/2008EP1414444B1 Novel imidazolidine derivatives, their preparation and their use as vla-4 antagonists
04/09/2008EP0964864B1 Pyrido 2,3-d pyrimidines and 4-aminopyrimidines as inhibitors of cellular proliferation
04/09/2008CN101160308A Methods of treating cancer and related methods
04/09/2008CN101160306A 苯并咪唑化合物 Benzimidazole compounds
04/09/2008CN101160301A Aminoalkyl-amidomethyl-substituted 2- (4-sulphonylamino) -3-hydroxy-3 , 4-dihydro-2h-cromen-6-yl derivatives and their use as potassium channel blockers
04/09/2008CN101160287A 吡啶基非芳香族含氮杂环-1-羧酸酯衍生物 Pyridyl non-aromatic nitrogen-containing heterocyclic-1-carboxylate derivative
04/09/2008CN101157688A 6-benzyloxy indole-2-formate furfuralcohol ester derivative and preparation method and usage thereof
04/09/2008CN100379727C Substituted pyrazolyl benzenesulfonamides for the treatment of inflamation
04/09/2008CN100379724C Inhibition of pulp and paper yellowing using nitroxides and other coadditives
04/09/2008CN100379415C Hetero biaryl derivatives as matrix metalloproteinase inhibitors
04/08/2008US7355340 Electron transportation; hole blocking properties
04/08/2008US7355054 Indole derivatives
04/08/2008US7355053 1-phenylpyrrolidine-2-one-3-carboxamides
04/08/2008US7355052 Melanocortin receptors; analgesivs; antiinflammatory agents; eating disorders; psycological disorders; anxiolytic agents; antidepressants; anticancer agents; aids; antiarthritic agents
04/08/2008US7355049 Biaryloxymethylarenecarboxylic acids as glycogen synthase activator
04/08/2008US7355046 Chronic obstructive pulmonary dusease; asthma
04/08/2008US7355042 Sleep disorders; side effect reduction
04/08/2008US7354946 Biarylurea derivatives
04/08/2008US7354944 protein kinase B inhibitors; abnormal cell growth, cancer, inflammation, and metabolic disordersp; 3-(3-Fluoro-phenyl)-N-[5-(3-methyl-1H-indazol-5-yl)-[1,3,4]thiadiazol-2-yl]-propane-1,2-diamine
04/08/2008US7354940 2,5-dioxoimidazolidin-4-yl acetamines and analogues as inhibitors of metalloproteinase mmp12
04/08/2008US7354938 4[2(2,4chlorophenyl)pyrazol]-phenyl-cyclopropan; 11-Beta-hydroxysteroid dehydrogenase 1 inhibitor; antidiabrtic agent, obesity, insulin resistance; improved physicochemical (stability) and biological (activity to inhibit HSD1, specificity, bioavailability, metabolism)
04/08/2008US7354936 2-phenylpyran-4-one derivatives
04/08/2008CA2232663C At1-receptor antagonists for preventing and treating postischemic renal failure and for protecting ischemic kidneys
04/08/2008CA2188924C Arylpiperidine and arylpiperazine derivatives and drugs containing the same
04/03/2008WO2008039645A1 Compounds which modulate the cb2 receptor
04/03/2008WO2008038711A1 Oxepin derivative
04/03/2008WO2008038251A2 3-aza-bicyclo[3.1.0]hexane derivatives
04/03/2008WO2008037789A1 Fungicide n-cycloalkyl-carboxamide, thiocarboxamide and n-substituted-carboximidamide derivatives
04/03/2008WO2008037626A1 Quinoline derivatives with 5-ht-binding properties
04/03/2008WO2008018639A3 Glycine transporter inhibitor
04/03/2008WO2008012234A3 Azolylmethyloxiranes, use thereof for controlling plant pathogenic fungi, and agents containing the same
04/03/2008WO2008008776A3 Hepatitis c virus inhibitors
04/03/2008WO2008005955A9 Synthesis of heterocyclic compounds
04/03/2008WO2007145834A3 Benzamide derivatives and uses related thereto
04/03/2008WO2007135565A3 Anti-proliferative compounds deriving from a 3-aryl-coumarine or 3-aryl-quinolin-2-one and uses thereof
04/03/2008WO2007135131A9 Substituted pyrazinone derivatives for use as a medicine
04/03/2008WO2007130429A3 Histone deacetylase and tubulin deacetylase inhibitors
04/03/2008WO2007070359A3 Quinolone based compounds exhibiting prolyl hydroxylase inhibitory activity, and compositions, and uses thereof
04/03/2008US20080081907 5-HT5A serotonin receptor activity; such as (5-Methyl-furan-2-ylmethyl)-(5-phenoxymethyl-quinolin-2-yl)-amine; anxiety, depression, sleep disorders, schizophrenia
04/03/2008US20080081825 5-((2,4-difluorophenyl) {[(1-methyl-4-piperidinyl)oxy]imino}methyl)-1-(2,6-dimethylphenyl)-2(1H)-pyridinone; p38 MAP kinase and tumor necrosis factor inhibitor; inflammatory cytokines or chemokine, respiratory diseases, cardiovascular diseases and bone diseases
04/03/2008US20080081813 Lipid Lowering Biphenylcarboxamides
04/03/2008US20080081807 Arylphenyl-substituted cyclic keto-enols
04/03/2008DE102006046161A1 New crystalline modified 4-((6-chloro-pyridin-3-ylmethyl)-methyl-amin o)-5H-furan-2-one exhibiting reflex positions using copper potassium-alpha-radiation, useful e.g. to combat pest and harmful insects
04/03/2008CA2664345A1 Oxepin derivative
04/03/2008CA2664342A1 New chemical inhibitors of bacterial heptose synthesis, methods for their preparation and biological applications of said inhibitors
04/03/2008CA2664310A1 Compounds which modulate the cb2 receptor
04/03/2008CA2664031A1 Quinoline derivatives with 5-ht-binding properties
04/03/2008CA2662612A1 3-aza-bicyclo[3.1.0]hexane derivatives
04/02/2008EP1905829A2 Templated molecules and methods for using such molecules
04/02/2008EP1905770A1 A process for the preparation of phenyltetrazole compounds
04/02/2008EP1905769A1 Heterocycle-substituted benzimidazole derivative
04/02/2008EP1904487A2 Indole derivatives for the treatment of tuberculosis
04/02/2008EP1904479A2 Novel 2,4-dianilinopyrimidine derivatives, the preparation thereof, their use as medicaments, pharmaceutical compositions and, in particular, as ikk inhibitors
04/02/2008EP1904473A1 Benzoheterocyclylethylcarboxamide derivatives
04/02/2008EP1904465A1 Method of synthesis of imidazole-amino acid derivatives and related compounds