Patents
Patents for C07D 405 - Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom (69,397)
06/2008
06/03/2008US7381726 Polymorphic forms of 1-′4-(5-cyanoindol-3-yl)butyl-4-(2-carbamoylbenzofuran-5-yl)piperazine hydrochloride
06/03/2008US7381725 Pyridazine derivatives as ligands for GABA receptors
06/03/2008US7381723 Antiserotonine agents; stroke, brain disorders;trauma; Alzheimer's disease; neurodegenerative disease; schizophrenia; psychological disorders; anxiolytic agents; controlling stresses; eating disorders; sleep disorders; sexual disorders
06/03/2008US7381719 To treat obesity and Related Diseases; oral bioavailablility, oral administration; inhibition of orexigenic effects; side effects reduction; weight loss while maintaining or minimizing the loss of lean muscle mass; 6-[4-(2-Benzylamino-ethyl)-phenoxy]-nicotinamide
06/03/2008US7381537 Use of inhibitors of glutaminyl cyclases for treatment and prevention of disease
06/03/2008CA2435954C Preparation of non-crystalline atorvastatin calcium
06/03/2008CA2401711C Cyclic amide derivatives
06/03/2008CA2389360C Urea derivatives as anti-inflammatory agents
06/03/2008CA2283465C Pesticidal 1-aryl-3-iminopyrazoles
05/2008
05/29/2008WO2008063984A2 Allosteric modulators of the a1 adenosine receptor
05/29/2008WO2008062907A1 Substance capable of inhibiting cytokinin signaling
05/29/2008WO2008062878A1 Novel pyrazole derivative, harmful organism control agent, and use of the control agent
05/29/2008WO2008062770A1 Quinolone derivative or pharmaceutically acceptable salt thereof
05/29/2008WO2008062739A1 Pyrazoles and use thereof as drugs
05/29/2008WO2008062424A2 Substituted 4,5-dihydro-1h-pyrazole derivatives as cannabinoid modulators
05/29/2008WO2008062276A2 Acetylene derivatives as stearoyl coa desaturase inhibitors
05/29/2008WO2008062011A1 Pyrimidylmethyl-sulfonamide compounds useful as fungicides and against arthropods
05/29/2008WO2008061740A1 Pyrimidines and their use as cxcr2 receptor antagonists
05/29/2008WO2008045564A3 Carboxamide compounds and their use as antagonists of the chemokine ccr2 receptor
05/29/2008WO2008040649A3 Pyrazine-2-carboxamide derivatives as cb2 receptor modulators
05/29/2008WO2007146072A3 Process for synthesizing piperazine-piperidine compounds
05/29/2008WO2007072150A3 Piperidine derivatives
05/29/2008US20080125464 Prucalopride n-oxide
05/29/2008US20080125444 Acyclic oximyl hepatitis c protease inhibitors
05/29/2008US20080125441 Spiro and dispiro 1,2,4-trioxolane antimalarials
05/29/2008US20080125438 2-aminothiophene derivatives; {2-Amino-4-[(4-phenylpiperazin-1-yl)methyl]thiophen-3-yl}(4-chlorophenyl)methanone; analgesic for chronic neuropathic pain, cardiac disarrhythmias, angina; neurological disease or injury, sleep disorder, epilepsy, antidepressants
05/29/2008US20080125423 N-methyl-N-(1-methyl-1H-indol-3-ylmethyl)-3-(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-3-yl)acrylamide as an enzyme inhibitor for both Fab I and Fab K which are used in the biosynthesis of fatty acids; enoyl-acyl-carrier protein renamed Fab 1; bactericides; fungicides; Staphylococcus aureus; antibiotics
05/29/2008US20080125422 Use of 5ht4 receptor antagonists in the prophylaxis or treatment of certain cardiovascular conditions
05/29/2008US20080125418 Benzimidazole derivatives and their use as kdr kinase protein inhibitors
05/29/2008US20080124572 A carbazole skeleton to which a diarylamino group bonds via a bonding group as a hole transporting material or a hole injecting material has an enhanced efficiency of light emission and is highly practical; enhances yield in device, improves lifetime
05/29/2008US20080124426 Ketomethionine ketals and derivatives thereof
05/29/2008CA2670143A1 Pyrimidines and their use as cxcr2 receptor antagonists
05/29/2008CA2669275A1 Agent for inhibiting cytokinin signaling
05/29/2008CA2669083A1 5, 6, or 7-substituted-3-(hetero)arylisoquinolinamine derivatives as antitumor agents
05/29/2008CA2668567A1 Pyrimidylmethyl-sulfonamide compounds useful as fungicides and against arthropods
05/28/2008EP1924578A2 6-N-LINKED HETEROCYCLE-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[d]AZEPINES AS 5-HT2C RECEPTOR AGONISTS
05/28/2008EP1924568A1 Quinazoline derivatives useful in cancer treatment
05/28/2008EP1924566A1 Diaminopyrimidines as p2x3 and p2x2/3 modulators
05/28/2008EP1924551A2 Organic compounds
05/28/2008EP1673078B1 Benzylether and benzylamino beta-secretase inhibitors for the treatment of alzheimer's disease
05/28/2008EP1496898B1 Tyrosine kinase inhibitors
05/28/2008EP1485354B1 Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
05/28/2008EP1218360B1 Triazine kinase inhibitors
05/28/2008CN101189229A Synthesis of avrainvillamide, stephacidin B, and analogues thereof
05/28/2008CN101189225A Heteroaryl substituted pyrazinyl-piperazine-piperidines with CXCR3 antagonist activity
05/28/2008CN101189214A Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides
05/28/2008CN101186606A Ampelopsin derivative, synthesizing method thereof and application of the same in preparing antineoplastic medicine
05/28/2008CN100390166C Benzopyran derivatives substituted with a benzimidazole derivative, pharmaceutically acceptable salts thereof, their preparations and pharmaceutical compositions containing them
05/28/2008CN100390164C Isoquinoline compounds and medicinal use thereof
05/28/2008CN100390156C Novel antibacterial compounds, process for their preparation and pharmaceutical compositions containing them
05/28/2008CN100390155C Quinoline and quinoxaline compounds
05/28/2008CN100390154C Quinoline and quinoxaline compounds as PDGF-receptor and/or LCK tyrosine kinase inhibitors
05/28/2008CN100390153C Intermediate for producing novel pyrazine derivatives
05/27/2008US7378532 Anticancer agents; such as succinic acid mono-[5-(1-benzyl-1H-indazol-3-yl)-furan-2-ylmethyl]ester, sodium salt; inhibit cancer cell growth
05/27/2008US7378529 Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
05/27/2008US7378526 Cholinergic ligands at the nicotinic acetylcholine receptors; diseases related to the cholinergic system; neurodegenerative disorders; pain; antiinflammatory; diagnostic or monitoring tools using labelled forms; 3-Phenyletynyl-quinuclidin-2-ene
05/27/2008US7378525 CCR8 inhibitors
05/27/2008US7378518 Vascular conditions such as atherosclerosis, hypercholesterolemia, diabetes, obesity, stroke, demyelination; lowering plasma levels of sterols and/or stanols
05/27/2008US7378431 Amide derivatives as NMDA receptor antagonists
05/27/2008US7378430 inhibitors of cGMP PDE, especially Type 5; erectile dysfunction and sexual disorders; 6-Bromo-N-[(3-chloro-methoxyphenyl)methyl]-2-(2-pyridinyl)-4-quinolinamine
05/27/2008US7378421 Chromenone derivatives
05/27/2008US7378419 3-{[(5,5a,8a,9)-9-(4-hydroxy-3,5-dimethoxyphenyl)-8-oxo-5,5a,6,8,8a,9-hexahydrofuro[3',4':6,7]naphtho[2,3-d][1,3]dioxol-5-yl]amino}-1-methyl-1H-pyrrole-2,5-dione; anticarcinogenic agent; inhibiting catalytic activity of topoisomerase II by stabilization of cleavable complex; better soluble and tolerated
05/27/2008US7378412 Pharmaceutical compounds
05/27/2008US7378375 Substituted pyridine herbicides
05/22/2008WO2008061236A2 Sulfoximines as kinase inhibitors
05/22/2008WO2008060998A1 Indole sulfonamides as sfrp-1 modulators
05/22/2008WO2008060372A2 Thrombin receptor antagonists based on the modified tricyclic unit of himbacine
05/22/2008WO2008060190A2 Ligands of 5-ht6 receptors, a pharmaceutical composition, method for the production and use thereof
05/22/2008WO2008059960A1 Method for producing quarter-pyridine derivative and intermediate of quarter-pyridine derivative
05/22/2008WO2008059867A1 Novel 1,2-dihydroquinoline derivative having (substituted phenyl or substituted heterocyclic) carbonyloxy lower alkyl group and ester-introduced phenyl group as substituents
05/22/2008WO2008059866A1 Novel 1,2-dihydroquinoline derivative having substituted phenylamino lower alkyl group and ester-introduced phenyl group as substituents
05/22/2008WO2008059865A1 Novel 1,2-dihydroquinoline derivative having substituted phenylchalcogeno lower alkyl group and ester-introduced phenyl group as substituents
05/22/2008WO2008059259A2 Anticancer compounds with a benzo ( 1, 2, 4 ) triazin-3yl-amine core
05/22/2008WO2008059214A1 Bisamlde derivatives and use thereof as fatty acid synthase inhibitors
05/22/2008WO2008059130A1 Thionucleosides and pharmaceutical applications
05/22/2008WO2008058402A1 Compounds and methods for treating protein folding disorders
05/22/2008WO2008042282A3 Imidazole-4, 5-dicarboxamide derivatives as jak-2 modulators
05/22/2008WO2008029257A3 Improved method for preparing 1,3-disubstituted pyrrolidine compounds
05/22/2008WO2008021926A3 Modulators of glucocorticoid receptor, and/or ap-1, and/or nf-kb activity and use thereof
05/22/2008WO2008011392A3 Proline urea ccr1 antagonists for the treatment of autoimmune diseases or inflammation
05/22/2008WO2007138431A3 Azabicyclic ether histamine-3 antagonists
05/22/2008US20080119526 Ep2 receptor agonists
05/22/2008US20080119516 2-'4(Phenylamino)-Piperidin-1-Yl!-N-Phenyl-Acetamine Derivatives and Related Compounds as Neuropeptide Y5 (NPY5) Ligands for the Treatment of Obesity
05/22/2008US20080119490 Viral Polymerase Inhibitors
05/22/2008US20080119488 Modulators Of Nuclear Receptors
05/22/2008US20080119487 Novel non-imidazole compounds
05/22/2008US20080119485 Novel Benzofurans and Indols
05/22/2008US20080119484 Novel use of 1-[4-(5-cyanoindol-3-yl)butyl]-4-(2-carbamoyl-benzofuran-5-yl)-piperazine and its physiologically acceptable salts
05/22/2008US20080119477 N-Biaryl and N-Arylheteroaryl Piperazine Derivatives as Modulators of the 5Ht2c Receptor Useful For the Treatment of Disorders Related Thereto
05/22/2008US20080119464 N-(4-piperidin-1-yl-phenyl)-2-[5-(thiaxolidine-3-carbonyl)-pyrrolidin-3-ylidene]-acetamide;antidiabetic agents; hyperglycemia, syndrome X, hyperinsulinemia, obesity, atherosclerosis
05/22/2008CA2669704A1 Sulfoximines as kinase inhibitors
05/22/2008CA2669607A1 Novel 1,2-dihydroquinoline derivative having (substituted phenyl or substituted heterocyclic) carbonyloxy lower alkyl group and ester-introduced phenyl group as substituents
05/22/2008CA2668744A1 Compounds and methods for treating protein folding disorders
05/22/2008CA2668596A1 Novel 1,2-dihydroquinoline derivative having substituted phenylamino lower alkyl group and ester-introduced phenyl group as substituents
05/22/2008CA2668592A1 Novel 1,2-dihydroquinoline derivative having substituted phenylchalcogeno lower alkyl group and ester-introduced phenyl group as substituents
05/22/2008CA2667569A1 Thionucleosides and pharmaceutical applications
05/22/2008CA2666903A1 Thrombin receptor antagonists based on the modified tricyclic unit of himbacine
05/22/2008CA2666685A1 Synthesis of selected stereoisomers of certain substituted alcohols
05/21/2008EP1923391A1 Substituted heterocyclic compounds, method for preparing same and pharmaceutical compositions containing them.
05/21/2008EP1923390A1 Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto